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Compile Data Set for Download or QSAR

Found 32 hits with Last Name = 'ghidini' and Initial = 'e'   
Target/Host
(Institution)
LigandTarget/Host
Links
Ligand
Links
Trg + Lig
Links
Ki
nM
ΔG°
kJ/mole
IC50
nM
Kd
nM
EC50/IC50
nM
koff
s-1
kon
M-1s-1
pHTemp
°C
cAMP-specific 3',5'-cyclic phosphodiesterase 4B


(Homo sapiens (Human))
BDBM50246909
PNG
(CHEMBL4075951)
PDB

UniProtKB/SwissProt

antibodypedia
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
PubMed
n/an/a 2.80n/an/an/an/an/an/a



Chiesi Farmaceutici S.p.A.

Curated by ChEMBL




J Med Chem 60: 10026-10046 (2017)


Article DOI: 10.1021/acs.jmedchem.7b01044
More data for this
Ligand-Target Pair
cAMP-specific 3',5'-cyclic phosphodiesterase 4B


(Homo sapiens (Human))
BDBM50246908
PNG
(CHEMBL4093768)
PDB

UniProtKB/SwissProt

antibodypedia
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
PubMed
n/an/a 8.80n/an/an/an/an/an/a



Chiesi Farmaceutici S.p.A.

Curated by ChEMBL




J Med Chem 60: 10026-10046 (2017)


Article DOI: 10.1021/acs.jmedchem.7b01044
More data for this
Ligand-Target Pair
3',5'-cyclic phosphodiesterase


(Homo sapiens (Human))
BDBM50246909
PNG
(CHEMBL4075951)
PDB
MMDB

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UniChem
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n/an/a 660n/an/an/an/an/an/a



Chiesi Farmaceutici S.p.A.

Curated by ChEMBL




J Med Chem 60: 10026-10046 (2017)


Article DOI: 10.1021/acs.jmedchem.7b01044
More data for this
Ligand-Target Pair
cAMP and cAMP-inhibited cGMP 3',5'-cyclic phosphodiesterase 10A


(Homo sapiens (Human))
BDBM50246909
PNG
(CHEMBL4075951)
PDB
MMDB

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UniChem
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n/an/a 810n/an/an/an/an/an/a



Chiesi Farmaceutici S.p.A.

Curated by ChEMBL




J Med Chem 60: 10026-10046 (2017)


Article DOI: 10.1021/acs.jmedchem.7b01044
More data for this
Ligand-Target Pair
Acetylcholinesterase


(Tetronarce californica (Pacific electric ray) (Tor...)
BDBM11683
PNG
((3aS,8aS)-1,3a,8-trimethyl-5-[(methylcarbamoyl)oxy...)
Show SMILES [H][C@@]12N(C)c3ccc(OC(=O)NC)cc3[C@]1(C)CC[N+]2(C)[O-] |r|
Show InChI InChI=1S/C15H21N3O3/c1-15-7-8-18(4,20)13(15)17(3)12-6-5-10(9-11(12)15)21-14(19)16-2/h5-6,9,13H,7-8H2,1-4H3,(H,16,19)/t13-,15-,18?/m0/s1
PDB
MMDB

UniProtKB/SwissProt

B.MOAD
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UniChem
Article
PubMed
n/an/a 1.74E+3n/an/an/an/a8.022



Istituto di Cristallografia



Assay Description
The cholinesterase assays were performed using colorimetric method reported by Ellman. Enzyme activity was determined by measuring the absorbance at ...


J Med Chem 49: 5051-8 (2006)


Article DOI: 10.1021/jm060293s
BindingDB Entry DOI: 10.7270/Q2DN439P
More data for this
Ligand-Target Pair
3',5'-cyclic phosphodiesterase


(Homo sapiens (Human))
BDBM50246908
PNG
(CHEMBL4093768)
PDB
MMDB

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UniChem
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n/an/a 3.46E+3n/an/an/an/an/an/a



Chiesi Farmaceutici S.p.A.

Curated by ChEMBL




J Med Chem 60: 10026-10046 (2017)


Article DOI: 10.1021/acs.jmedchem.7b01044
More data for this
Ligand-Target Pair
Phosphodiesterase 8


(Homo sapiens (Human))
BDBM50246909
PNG
(CHEMBL4075951)
PDB
MMDB

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n/an/a 3.56E+3n/an/an/an/an/an/a



Chiesi Farmaceutici S.p.A.

Curated by ChEMBL




J Med Chem 60: 10026-10046 (2017)


Article DOI: 10.1021/acs.jmedchem.7b01044
More data for this
Ligand-Target Pair
cAMP and cAMP-inhibited cGMP 3',5'-cyclic phosphodiesterase 10A


(Homo sapiens (Human))
BDBM50246908
PNG
(CHEMBL4093768)
PDB
MMDB

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UniChem
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n/an/a 4.03E+3n/an/an/an/an/an/a



Chiesi Farmaceutici S.p.A.

Curated by ChEMBL




J Med Chem 60: 10026-10046 (2017)


Article DOI: 10.1021/acs.jmedchem.7b01044
More data for this
Ligand-Target Pair
Acetylcholinesterase


(Tetronarce californica (Pacific electric ray) (Tor...)
BDBM11685
PNG
((3aS,8aS)-1,3a,8-trimethyl-5-{[(2-methylphenyl)car...)
Show SMILES [H][C@@]12N(C)c3ccc(OC(=O)Nc4ccccc4C)cc3[C@]1(C)CC[N+]2(C)[O-] |r|
Show InChI InChI=1S/C21H25N3O3/c1-14-7-5-6-8-17(14)22-20(25)27-15-9-10-18-16(13-15)21(2)11-12-24(4,26)19(21)23(18)3/h5-10,13,19H,11-12H2,1-4H3,(H,22,25)/t19-,21-,24?/m0/s1
PDB
MMDB

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UniChem
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n/an/a 4.04E+3n/an/an/an/a8.022



Istituto di Cristallografia



Assay Description
The cholinesterase assays were performed using colorimetric method reported by Ellman. Enzyme activity was determined by measuring the absorbance at ...


J Med Chem 49: 5051-8 (2006)


Article DOI: 10.1021/jm060293s
BindingDB Entry DOI: 10.7270/Q2DN439P
More data for this
Ligand-Target Pair
3',5'-cyclic phosphodiesterase


(Homo sapiens (Human))
BDBM50246909
PNG
(CHEMBL4075951)
PDB
MMDB

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UniChem
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n/an/a 4.61E+3n/an/an/an/an/an/a



Chiesi Farmaceutici S.p.A.

Curated by ChEMBL




J Med Chem 60: 10026-10046 (2017)


Article DOI: 10.1021/acs.jmedchem.7b01044
More data for this
Ligand-Target Pair
Acetylcholinesterase


(Tetronarce californica (Pacific electric ray) (Tor...)
BDBM11684
PNG
((3aS,8aS)-1,3a,8-trimethyl-1-oxido-5-[(phenylcarba...)
Show SMILES [H][C@@]12N(C)c3ccc(OC(=O)Nc4ccccc4)cc3[C@]1(C)CC[N+]2(C)[O-] |r|
Show InChI InChI=1S/C20H23N3O3/c1-20-11-12-23(3,25)18(20)22(2)17-10-9-15(13-16(17)20)26-19(24)21-14-7-5-4-6-8-14/h4-10,13,18H,11-12H2,1-3H3,(H,21,24)/t18-,20-,23?/m0/s1
PDB
MMDB

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UniChem
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n/an/a 4.74E+3n/an/an/an/a8.022



Istituto di Cristallografia



Assay Description
The cholinesterase assays were performed using colorimetric method reported by Ellman. Enzyme activity was determined by measuring the absorbance at ...


J Med Chem 49: 5051-8 (2006)


Article DOI: 10.1021/jm060293s
BindingDB Entry DOI: 10.7270/Q2DN439P
More data for this
Ligand-Target Pair
Acetylcholinesterase


(Tetronarce californica (Pacific electric ray) (Tor...)
BDBM11686
PNG
((-)-O-[(2-ethylphenyl)carbamoyl]geneseroline | (3a...)
Show SMILES [H][C@@]12N(C)c3ccc(OC(=O)Nc4ccccc4CC)cc3[C@]1(C)CC[N+]2(C)[O-] |r|
Show InChI InChI=1S/C22H27N3O3/c1-5-15-8-6-7-9-18(15)23-21(26)28-16-10-11-19-17(14-16)22(2)12-13-25(4,27)20(22)24(19)3/h6-11,14,20H,5,12-13H2,1-4H3,(H,23,26)/t20-,22-,25?/m0/s1
PDB
MMDB

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PDB
UniChem
PDB
Article
PubMed
n/an/a 5.12E+3n/an/an/an/a8.022



Istituto di Cristallografia



Assay Description
The cholinesterase assays were performed using colorimetric method reported by Ellman. Enzyme activity was determined by measuring the absorbance at ...


J Med Chem 49: 5051-8 (2006)


Article DOI: 10.1021/jm060293s
BindingDB Entry DOI: 10.7270/Q2DN439P
More data for this
Ligand-Target Pair
3D
3D Structure (crystal)
Acetylcholinesterase


(Tetronarce californica (Pacific electric ray) (Tor...)
BDBM11689
PNG
((3aS,8aS)-1,3a,8-trimethyl-5-{[(3-methylphenyl)car...)
Show SMILES [H][C@@]12N(C)c3ccc(OC(=O)Nc4cccc(C)c4)cc3[C@]1(C)CC[N+]2(C)[O-] |r|
Show InChI InChI=1S/C21H25N3O3/c1-14-6-5-7-15(12-14)22-20(25)27-16-8-9-18-17(13-16)21(2)10-11-24(4,26)19(21)23(18)3/h5-9,12-13,19H,10-11H2,1-4H3,(H,22,25)/t19-,21-,24?/m0/s1
PDB
MMDB

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UniChem
Article
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n/an/a 5.13E+3n/an/an/an/a8.022



Istituto di Cristallografia



Assay Description
The cholinesterase assays were performed using colorimetric method reported by Ellman. Enzyme activity was determined by measuring the absorbance at ...


J Med Chem 49: 5051-8 (2006)


Article DOI: 10.1021/jm060293s
BindingDB Entry DOI: 10.7270/Q2DN439P
More data for this
Ligand-Target Pair
3',5'-cyclic phosphodiesterase


(Homo sapiens (Human))
BDBM50246909
PNG
(CHEMBL4075951)
Reactome pathway
KEGG

UniProtKB/SwissProt

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antibodypedia
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PC cid
PC sid
UniChem
Article
PubMed
n/an/a 6.21E+3n/an/an/an/an/an/a



Chiesi Farmaceutici S.p.A.

Curated by ChEMBL




J Med Chem 60: 10026-10046 (2017)


Article DOI: 10.1021/acs.jmedchem.7b01044
More data for this
Ligand-Target Pair
Phosphodiesterase 1A (PDE1A)


(Homo sapiens (Human))
BDBM50246909
PNG
(CHEMBL4075951)
KEGG

UniProtKB/SwissProt

DrugBank
antibodypedia
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
PubMed
n/an/a 7.40E+3n/an/an/an/an/an/a



Chiesi Farmaceutici S.p.A.

Curated by ChEMBL




J Med Chem 60: 10026-10046 (2017)


Article DOI: 10.1021/acs.jmedchem.7b01044
More data for this
Ligand-Target Pair
Acetylcholinesterase


(Tetronarce californica (Pacific electric ray) (Tor...)
BDBM11691
PNG
((3aS,8aS)-1,3a,8-trimethyl-5-{[(4-methylphenyl)car...)
Show SMILES [H][C@@]12N(C)c3ccc(OC(=O)Nc4ccc(C)cc4)cc3[C@]1(C)CC[N+]2(C)[O-] |r|
Show InChI InChI=1S/C21H25N3O3/c1-14-5-7-15(8-6-14)22-20(25)27-16-9-10-18-17(13-16)21(2)11-12-24(4,26)19(21)23(18)3/h5-10,13,19H,11-12H2,1-4H3,(H,22,25)/t19-,21-,24?/m0/s1
PDB
MMDB

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n/an/a 7.61E+3n/an/an/an/a8.022



Istituto di Cristallografia



Assay Description
The cholinesterase assays were performed using colorimetric method reported by Ellman. Enzyme activity was determined by measuring the absorbance at ...


J Med Chem 49: 5051-8 (2006)


Article DOI: 10.1021/jm060293s
BindingDB Entry DOI: 10.7270/Q2DN439P
More data for this
Ligand-Target Pair
Acetylcholinesterase


(Tetronarce californica (Pacific electric ray) (Tor...)
BDBM11687
PNG
((3aS,8aS)-1,3a,8-trimethyl-1-oxido-5-({[2-(propan-...)
Show SMILES [H][C@@]12N(C)c3ccc(OC(=O)Nc4ccccc4C(C)C)cc3[C@]1(C)CC[N+]2(C)[O-] |r|
Show InChI InChI=1S/C23H29N3O3/c1-15(2)17-8-6-7-9-19(17)24-22(27)29-16-10-11-20-18(14-16)23(3)12-13-26(5,28)21(23)25(20)4/h6-11,14-15,21H,12-13H2,1-5H3,(H,24,27)/t21-,23-,26?/m0/s1
PDB
MMDB

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UniChem
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n/an/a 8.38E+3n/an/an/an/a8.022



Istituto di Cristallografia



Assay Description
The cholinesterase assays were performed using colorimetric method reported by Ellman. Enzyme activity was determined by measuring the absorbance at ...


J Med Chem 49: 5051-8 (2006)


Article DOI: 10.1021/jm060293s
BindingDB Entry DOI: 10.7270/Q2DN439P
More data for this
Ligand-Target Pair
Acetylcholinesterase


(Tetronarce californica (Pacific electric ray) (Tor...)
BDBM11688
PNG
((3aS,8aS)-1,3a,8-trimethyl-1-oxido-5-{[(2-propylph...)
Show SMILES [H][C@@]12N(C)c3ccc(OC(=O)Nc4ccccc4CCC)cc3[C@]1(C)CC[N+]2(C)[O-] |r|
Show InChI InChI=1S/C23H29N3O3/c1-5-8-16-9-6-7-10-19(16)24-22(27)29-17-11-12-20-18(15-17)23(2)13-14-26(4,28)21(23)25(20)3/h6-7,9-12,15,21H,5,8,13-14H2,1-4H3,(H,24,27)/t21-,23-,26?/m0/s1
PDB
MMDB

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UniChem
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n/an/a 8.44E+3n/an/an/an/a8.022



Istituto di Cristallografia



Assay Description
The cholinesterase assays were performed using colorimetric method reported by Ellman. Enzyme activity was determined by measuring the absorbance at ...


J Med Chem 49: 5051-8 (2006)


Article DOI: 10.1021/jm060293s
BindingDB Entry DOI: 10.7270/Q2DN439P
More data for this
Ligand-Target Pair
Acetylcholinesterase


(Tetronarce californica (Pacific electric ray) (Tor...)
BDBM11693
PNG
((3aS,8aS)-5-{[(3,5-dimethylphenyl)carbamoyl]oxy}-1...)
Show SMILES [H][C@@]12N(C)c3ccc(OC(=O)Nc4cc(C)cc(C)c4)cc3[C@]1(C)CC[N+]2(C)[O-] |r|
Show InChI InChI=1S/C22H27N3O3/c1-14-10-15(2)12-16(11-14)23-21(26)28-17-6-7-19-18(13-17)22(3)8-9-25(5,27)20(22)24(19)4/h6-7,10-13,20H,8-9H2,1-5H3,(H,23,26)/t20-,22-,25?/m0/s1
PDB
MMDB

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UniChem
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n/an/a 8.58E+3n/an/an/an/a8.022



Istituto di Cristallografia



Assay Description
The cholinesterase assays were performed using colorimetric method reported by Ellman. Enzyme activity was determined by measuring the absorbance at ...


J Med Chem 49: 5051-8 (2006)


Article DOI: 10.1021/jm060293s
BindingDB Entry DOI: 10.7270/Q2DN439P
More data for this
Ligand-Target Pair
Acetylcholinesterase


(Tetronarce californica (Pacific electric ray) (Tor...)
BDBM11690
PNG
((3aS,8aS)-5-{[(3-ethylphenyl)carbamoyl]oxy}-1,3a,8...)
Show SMILES [H][C@@]12N(C)c3ccc(OC(=O)Nc4cccc(CC)c4)cc3[C@]1(C)CC[N+]2(C)[O-] |r|
Show InChI InChI=1S/C22H27N3O3/c1-5-15-7-6-8-16(13-15)23-21(26)28-17-9-10-19-18(14-17)22(2)11-12-25(4,27)20(22)24(19)3/h6-10,13-14,20H,5,11-12H2,1-4H3,(H,23,26)/t20-,22-,25?/m0/s1
PDB
MMDB

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UniChem
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n/an/a 9.80E+3n/an/an/an/a8.022



Istituto di Cristallografia



Assay Description
The cholinesterase assays were performed using colorimetric method reported by Ellman. Enzyme activity was determined by measuring the absorbance at ...


J Med Chem 49: 5051-8 (2006)


Article DOI: 10.1021/jm060293s
BindingDB Entry DOI: 10.7270/Q2DN439P
More data for this
Ligand-Target Pair
3',5'-cyclic phosphodiesterase


(Homo sapiens (Human))
BDBM50246908
PNG
(CHEMBL4093768)
PDB
MMDB

Reactome pathway
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UniChem
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n/an/a 1.39E+4n/an/an/an/an/an/a



Chiesi Farmaceutici S.p.A.

Curated by ChEMBL




J Med Chem 60: 10026-10046 (2017)


Article DOI: 10.1021/acs.jmedchem.7b01044
More data for this
Ligand-Target Pair
Phosphodiesterase 8


(Homo sapiens (Human))
BDBM50246908
PNG
(CHEMBL4093768)
PDB
MMDB

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UniChem
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n/an/a 1.70E+4n/an/an/an/an/an/a



Chiesi Farmaceutici S.p.A.

Curated by ChEMBL




J Med Chem 60: 10026-10046 (2017)


Article DOI: 10.1021/acs.jmedchem.7b01044
More data for this
Ligand-Target Pair
Phosphodiesterase 1A (PDE1A)


(Homo sapiens (Human))
BDBM50246908
PNG
(CHEMBL4093768)
KEGG

UniProtKB/SwissProt

DrugBank
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UniChem
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n/an/a 2.56E+4n/an/an/an/an/an/a



Chiesi Farmaceutici S.p.A.

Curated by ChEMBL




J Med Chem 60: 10026-10046 (2017)


Article DOI: 10.1021/acs.jmedchem.7b01044
More data for this
Ligand-Target Pair
Phosphodiesterase 11A


(Homo sapiens (Human))
BDBM50246908
PNG
(CHEMBL4093768)
KEGG

UniProtKB/SwissProt

DrugBank
antibodypedia
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PC cid
PC sid
UniChem
Article
PubMed
n/an/a>3.00E+4n/an/an/an/an/an/a



Chiesi Farmaceutici S.p.A.

Curated by ChEMBL




J Med Chem 60: 10026-10046 (2017)


Article DOI: 10.1021/acs.jmedchem.7b01044
More data for this
Ligand-Target Pair
3',5'-cyclic phosphodiesterase


(Homo sapiens (Human))
BDBM50246908
PNG
(CHEMBL4093768)
PDB
MMDB

KEGG

UniProtKB/SwissProt

B.MOAD
DrugBank
antibodypedia
GoogleScholar
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PC cid
PC sid
UniChem
Article
PubMed
n/an/a>3.00E+4n/an/an/an/an/an/a



Chiesi Farmaceutici S.p.A.

Curated by ChEMBL




J Med Chem 60: 10026-10046 (2017)


Article DOI: 10.1021/acs.jmedchem.7b01044
More data for this
Ligand-Target Pair
3',5'-cyclic phosphodiesterase


(Homo sapiens (Human))
BDBM50246909
PNG
(CHEMBL4075951)
PDB
MMDB

Reactome pathway
KEGG

UniProtKB/SwissProt

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UniChem
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n/an/a>3.00E+4n/an/an/an/an/an/a



Chiesi Farmaceutici S.p.A.

Curated by ChEMBL




J Med Chem 60: 10026-10046 (2017)


Article DOI: 10.1021/acs.jmedchem.7b01044
More data for this
Ligand-Target Pair
3',5'-cyclic phosphodiesterase


(Homo sapiens (Human))
BDBM50246908
PNG
(CHEMBL4093768)
PDB
MMDB

Reactome pathway
KEGG

UniProtKB/SwissProt

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UniChem
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n/an/a>3.00E+4n/an/an/an/an/an/a



Chiesi Farmaceutici S.p.A.

Curated by ChEMBL




J Med Chem 60: 10026-10046 (2017)


Article DOI: 10.1021/acs.jmedchem.7b01044
More data for this
Ligand-Target Pair
3',5'-cyclic phosphodiesterase


(Homo sapiens (Human))
BDBM50246908
PNG
(CHEMBL4093768)
Reactome pathway
KEGG

UniProtKB/SwissProt

DrugBank
antibodypedia
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
PubMed
n/an/a>3.00E+4n/an/an/an/an/an/a



Chiesi Farmaceutici S.p.A.

Curated by ChEMBL




J Med Chem 60: 10026-10046 (2017)


Article DOI: 10.1021/acs.jmedchem.7b01044
More data for this
Ligand-Target Pair
Phosphodiesterase 11A


(Homo sapiens (Human))
BDBM50246909
PNG
(CHEMBL4075951)
KEGG

UniProtKB/SwissProt

DrugBank
antibodypedia
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
PubMed
n/an/a>3.00E+4n/an/an/an/an/an/a



Chiesi Farmaceutici S.p.A.

Curated by ChEMBL




J Med Chem 60: 10026-10046 (2017)


Article DOI: 10.1021/acs.jmedchem.7b01044
More data for this
Ligand-Target Pair
3',5'-cyclic phosphodiesterase


(Homo sapiens (Human))
BDBM50246909
PNG
(CHEMBL4075951)
PDB
MMDB

KEGG

UniProtKB/SwissProt

B.MOAD
DrugBank
antibodypedia
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
PubMed
n/an/a>3.00E+4n/an/an/an/an/an/a



Chiesi Farmaceutici S.p.A.

Curated by ChEMBL




J Med Chem 60: 10026-10046 (2017)


Article DOI: 10.1021/acs.jmedchem.7b01044
More data for this
Ligand-Target Pair
Acetylcholinesterase


(Tetronarce californica (Pacific electric ray) (Tor...)
BDBM11692
PNG
((3aS,8aS)-5-{[(2,6-dimethylphenyl)carbamoyl]oxy}-1...)
Show SMILES [H][C@@]12N(C)c3ccc(OC(=O)Nc4c(C)cccc4C)cc3[C@]1(C)CC[N+]2(C)[O-] |r|
Show InChI InChI=1S/C22H27N3O3/c1-14-7-6-8-15(2)19(14)23-21(26)28-16-9-10-18-17(13-16)22(3)11-12-25(5,27)20(22)24(18)4/h6-10,13,20H,11-12H2,1-5H3,(H,23,26)/t20-,22-,25?/m0/s1
PDB
MMDB

UniProtKB/SwissProt

B.MOAD
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
PubMed
n/an/a 1.86E+5n/an/an/an/a8.022



Istituto di Cristallografia



Assay Description
The cholinesterase assays were performed using colorimetric method reported by Ellman. Enzyme activity was determined by measuring the absorbance at ...


J Med Chem 49: 5051-8 (2006)


Article DOI: 10.1021/jm060293s
BindingDB Entry DOI: 10.7270/Q2DN439P
More data for this
Ligand-Target Pair
Acetylcholinesterase


(Tetronarce californica (Pacific electric ray) (Tor...)
BDBM11682
PNG
(2,3-dihydroxybutanedioic acid; 3-[(1S)-1-(dimethyl...)
Show SMILES CCN(C)C(=O)Oc1cccc(c1)[C@H](C)N(C)C |r|
Show InChI InChI=1S/C14H22N2O2/c1-6-16(5)14(17)18-13-9-7-8-12(10-13)11(2)15(3)4/h7-11H,6H2,1-5H3/t11-/m0/s1
PDB
MMDB

UniProtKB/SwissProt

B.MOAD
GoogleScholar
AffyNet 
Purchase

DrugBank
KEGG
PC cid
PC sid
UniChem
Article
PubMed
n/an/a 1.87E+5n/an/an/an/a8.022



Istituto di Cristallografia



Assay Description
The cholinesterase assays were performed using colorimetric method reported by Ellman. Enzyme activity was determined by measuring the absorbance at ...


J Med Chem 49: 5051-8 (2006)


Article DOI: 10.1021/jm060293s
BindingDB Entry DOI: 10.7270/Q2DN439P
More data for this
Ligand-Target Pair