Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kcal/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Microsomal glutathione S-transferase 1 (Homo sapiens (Human)) | BDBM50422689 (640/359 | CEFUROXIME) | UniProtKB/SwissProt GoogleScholar AffyNet | Purchase DrugBank MCE KEGG MMDB PC cid PC sid PDB UniChem Similars | Article PubMed | 3.24E+4 | n/a | 5.64E+4 | n/a | n/a | n/a | n/a | 6.5 | n/a |
Ondokuz Mayis University | Assay Description Enzymatic activity was determined spectrophotometrically by measuring the conjugation of CDNB with GSH. The 1 ml assay mixture contained 0.5 mM CDNB,... | J Enzyme Inhib Med Chem 28: 824-9 (2013) Article DOI: 10.3109/14756366.2012.688042 BindingDB Entry DOI: 10.7270/Q21J98P4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Microsomal glutathione S-transferase 1 (Homo sapiens (Human)) | BDBM50049707 ((6R,7R)-7-{2-(2-Amino-thiazol-4-yl)-2-[(Z)-methoxy...) | UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL DrugBank MCE KEGG PC cid PC sid UniChem Patents Similars | Article PubMed | 3.54E+4 | n/a | 6.18E+4 | n/a | n/a | n/a | n/a | 6.5 | n/a |
Ondokuz Mayis University | Assay Description Enzymatic activity was determined spectrophotometrically by measuring the conjugation of CDNB with GSH. The 1 ml assay mixture contained 0.5 mM CDNB,... | J Enzyme Inhib Med Chem 28: 824-9 (2013) Article DOI: 10.3109/14756366.2012.688042 BindingDB Entry DOI: 10.7270/Q21J98P4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Microsomal glutathione S-transferase 1 (Homo sapiens (Human)) | BDBM237182 (Ceftizoxime) | UniProtKB/SwissProt GoogleScholar AffyNet | Purchase DrugBank MCE KEGG PC cid PC sid UniChem | Article PubMed | 1.65E+5 | n/a | 2.78E+5 | n/a | n/a | n/a | n/a | 6.5 | n/a |
Ondokuz Mayis University | Assay Description Enzymatic activity was determined spectrophotometrically by measuring the conjugation of CDNB with GSH. The 1 ml assay mixture contained 0.5 mM CDNB,... | J Enzyme Inhib Med Chem 28: 824-9 (2013) Article DOI: 10.3109/14756366.2012.688042 BindingDB Entry DOI: 10.7270/Q21J98P4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Microsomal glutathione S-transferase 1 (Homo sapiens (Human)) | BDBM50390999 (CEFOPERAZONE) | UniProtKB/SwissProt GoogleScholar AffyNet | Purchase MCE KEGG PC cid PC sid UniChem Similars | Article PubMed | 2.67E+5 | n/a | 4.84E+5 | n/a | n/a | n/a | n/a | 6.5 | n/a |
Ondokuz Mayis University | Assay Description Enzymatic activity was determined spectrophotometrically by measuring the conjugation of CDNB with GSH. The 1 ml assay mixture contained 0.5 mM CDNB,... | J Enzyme Inhib Med Chem 28: 824-9 (2013) Article DOI: 10.3109/14756366.2012.688042 BindingDB Entry DOI: 10.7270/Q21J98P4 | |||||||||||
More data for this Ligand-Target Pair |