Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kcal/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Histamine H1 receptor (Cavia porcellus (domestic guinea pig)) | BDBM50007538 (8-(2-Azetidin-1-yl-ethyl)-3-chloro-6-methyl-7,8-di...) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 0.260 | n/a | n/a | n/a | n/a | n/a | n/a |
A. H. Robins Company, Inc. Curated by ChEMBL | Assay Description Inhibition of [3H]-mepyramine binding to the histamine receptor in guinea pig cortex | J Med Chem 34: 1314-28 (1991) BindingDB Entry DOI: 10.7270/Q23F4NMG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine H1 receptor (Cavia porcellus (domestic guinea pig)) | BDBM22567 (3H]pyrilamine | CHEMBL511 | Dorantamin | Mepyramin...) | UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL DrugBank MCE KEGG PC cid PC sid PDB UniChem Patents Similars | Article PubMed | n/a | n/a | 1.5 | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Inc. Curated by ChEMBL | Assay Description Inhibition of guinea pig histamine H1 receptor | Bioorg Med Chem 18: 7675-99 (2010) Article DOI: 10.1016/j.bmc.2010.07.034 BindingDB Entry DOI: 10.7270/Q2DF6S69 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine H1 receptor (Cavia porcellus (domestic guinea pig)) | BDBM50131441 (9,13b-dihydro-1H-dibenzo[c,f]imidazo[1,5-a]azepin-...) | UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL DrugBank MCE PC cid PC sid UniChem Patents | PubMed | n/a | n/a | 1.58 | n/a | n/a | n/a | n/a | n/a | n/a |
Vrije Universiteit Curated by ChEMBL | Assay Description Potency against histamine H1 receptor on guinea pig ileum | J Med Chem 38: 3351-60 (1995) BindingDB Entry DOI: 10.7270/Q2ZW1N49 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine H1 receptor (Cavia porcellus (domestic guinea pig)) | BDBM50007542 (3-Chloro-8-(2-dimethylamino-ethyl)-6-methyl-7,8-di...) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 1.90 | n/a | n/a | n/a | n/a | n/a | n/a |
A. H. Robins Company, Inc. Curated by ChEMBL | Assay Description Inhibition of [3H]-mepyramine binding to the histamine receptor in guinea pig cortex | J Med Chem 34: 1314-28 (1991) BindingDB Entry DOI: 10.7270/Q23F4NMG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine H1 receptor (Cavia porcellus (domestic guinea pig)) | BDBM50019624 (1-(2-Ethoxy-ethyl)-2-(4-methyl-[1,4]diazepan-1-yl)...) | UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL DrugBank MCE KEGG PC cid PC sid UniChem Patents Similars | PubMed | n/a | n/a | 6.10 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description In vitro inhibition of histamine-induced contractions in guinea pig ileum | J Med Chem 29: 1178-83 (1987) BindingDB Entry DOI: 10.7270/Q2QR4XPC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine H1 receptor (Cavia porcellus (domestic guinea pig)) | BDBM50019595 (2-(4-Methyl-piperazin-1-yl)-1-(2-phenoxy-ethyl)-1H...) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | n/a | n/a | 6.90 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description In vitro inhibition of histamine-induced contractions in guinea pig ileum | J Med Chem 29: 1178-83 (1987) BindingDB Entry DOI: 10.7270/Q2QR4XPC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine H1 receptor (Cavia porcellus (domestic guinea pig)) | BDBM50019605 (1-(2-Ethoxy-ethyl)-2-(4-pentyl-[1,4]diazepan-1-yl)...) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 7.40 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description In vitro inhibition of histamine-induced contractions in guinea pig ileum | J Med Chem 29: 1178-83 (1987) BindingDB Entry DOI: 10.7270/Q2QR4XPC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine H1 receptor (Cavia porcellus (domestic guinea pig)) | BDBM50017371 (1-[4-(3-{4-[Bis-(4-fluoro-phenyl)-hydroxy-methyl]-...) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL MCE PC cid PC sid UniChem Patents Similars | PubMed | n/a | n/a | 8 | n/a | n/a | n/a | n/a | n/a | n/a |
A.H. Robins Company Curated by ChEMBL | Assay Description Inhibitory activity of the compound against Tritiated [3H]- mepyramine binding to histamine H1 receptor in guinea pig cerebral cortex | J Med Chem 32: 105-18 (1989) BindingDB Entry DOI: 10.7270/Q2WM1CD6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine H1 receptor (Cavia porcellus (domestic guinea pig)) | BDBM50019644 (1-(2-Ethoxy-ethyl)-2-(4-propyl-[1,4]diazepan-1-yl)...) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 8.40 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description In vitro inhibition of histamine-induced contractions in guinea pig ileum | J Med Chem 29: 1178-83 (1987) BindingDB Entry DOI: 10.7270/Q2QR4XPC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine H1 receptor (Cavia porcellus (domestic guinea pig)) | BDBM50019643 (2-(4-Butyl-[1,4]diazepan-1-yl)-1-(2-ethoxy-ethyl)-...) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 8.40 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description In vitro inhibition of histamine-induced contractions in guinea pig ileum | J Med Chem 29: 1178-83 (1987) BindingDB Entry DOI: 10.7270/Q2QR4XPC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine H1 receptor (Cavia porcellus (domestic guinea pig)) | BDBM50019602 (1-(2-Ethoxy-ethyl)-2-(4-hexyl-piperazin-1-yl)-1H-b...) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 8.60 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description In vitro inhibition of histamine-induced contractions in guinea pig ileum | J Med Chem 29: 1178-83 (1987) BindingDB Entry DOI: 10.7270/Q2QR4XPC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine H1 receptor (Cavia porcellus (domestic guinea pig)) | BDBM35938 (1-(p-chlorophenyl)-1-(2-pyridyl)-3-N,N-dimethylpro...) | UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL DrugBank MCE KEGG PC cid PC sid UniChem Patents Similars | PubMed | n/a | n/a | 8.80 | n/a | n/a | n/a | n/a | n/a | n/a |
A. H. Robins Company, Inc. Curated by ChEMBL | Assay Description Inhibition of [3H]-mepyramine binding to the Histamine H1 receptor in guinea pig cortex | J Med Chem 34: 1314-28 (1991) BindingDB Entry DOI: 10.7270/Q23F4NMG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine H1 receptor (Cavia porcellus (domestic guinea pig)) | BDBM76863 (3-[3-(4-benzhydrylpiperazin-1-yl)propyl]-1H-benzim...) | UniProtKB/SwissProt GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem | PubMed | n/a | n/a | 9 | n/a | n/a | n/a | n/a | n/a | n/a |
A.H. Robins Company Curated by ChEMBL | Assay Description Inhibitory activity of the compound against Tritiated [3H]- mepyramine binding to Histamine H1 receptor in guinea pig cerebral cortex | J Med Chem 32: 105-18 (1989) BindingDB Entry DOI: 10.7270/Q2WM1CD6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine H1 receptor (Cavia porcellus (domestic guinea pig)) | BDBM50019628 (2-(4-Methyl-[1,4]diazepan-1-yl)-1-(2-phenoxy-ethyl...) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | n/a | n/a | 9.10 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description In vitro inhibition of histamine-induced contractions in guinea pig ileum | J Med Chem 29: 1178-83 (1987) BindingDB Entry DOI: 10.7270/Q2QR4XPC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine H1 receptor (Cavia porcellus (domestic guinea pig)) | BDBM50019609 (2-(4-Methyl-[1,4]diazepan-1-yl)-1-(2-prop-2-ynylox...) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | n/a | n/a | 9.90 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description In vitro inhibition of histamine-induced contractions in guinea pig ileum | J Med Chem 29: 1178-83 (1987) BindingDB Entry DOI: 10.7270/Q2QR4XPC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine H1 receptor (Cavia porcellus (domestic guinea pig)) | BDBM50019636 (2-(4-Methyl-piperazin-1-yl)-1-(2-vinyloxy-ethyl)-1...) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 10 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description In vitro inhibition of histamine-induced contractions in guinea pig ileum | J Med Chem 29: 1178-83 (1987) BindingDB Entry DOI: 10.7270/Q2QR4XPC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine H1 receptor (Cavia porcellus (domestic guinea pig)) | BDBM50019607 (1-(2-Ethoxy-ethyl)-2-(4-methyl-piperazin-1-yl)-1H-...) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | n/a | n/a | 10 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description In vitro inhibition of histamine-induced contractions in guinea pig ileum | J Med Chem 29: 1178-83 (1987) BindingDB Entry DOI: 10.7270/Q2QR4XPC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine H1 receptor (Cavia porcellus (domestic guinea pig)) | BDBM50019618 (1-(2-Allyloxy-ethyl)-2-(4-methyl-[1,4]diazepan-1-y...) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | n/a | n/a | 10 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description In vitro inhibition of histamine-induced contractions in guinea pig ileum | J Med Chem 29: 1178-83 (1987) BindingDB Entry DOI: 10.7270/Q2QR4XPC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine H1 receptor (Cavia porcellus (domestic guinea pig)) | BDBM50019614 (1-(2-Butoxy-ethyl)-2-(4-methyl-[1,4]diazepan-1-yl)...) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 10 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description In vitro inhibition of histamine-induced contractions in guinea pig ileum | J Med Chem 29: 1178-83 (1987) BindingDB Entry DOI: 10.7270/Q2QR4XPC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine H1 receptor (Cavia porcellus (domestic guinea pig)) | BDBM50089149 (2-Benzyl-9-phenyl-2,3,4,4a-tetrahydro-1H-indeno[2,...) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 11 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Bath Curated by ChEMBL | Assay Description In vitro antagonistic activity at the Histamine H1 receptor in guinea pig ileum | Bioorg Med Chem Lett 10: 1277-9 (2000) BindingDB Entry DOI: 10.7270/Q2T152VB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine H1 receptor (Cavia porcellus (domestic guinea pig)) | BDBM50019629 (1-(2-Ethoxy-ethyl)-2-piperazin-1-yl-1H-benzoimidaz...) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | n/a | n/a | 11 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description In vitro inhibition of histamine-induced contractions in guinea pig ileum | J Med Chem 29: 1178-83 (1987) BindingDB Entry DOI: 10.7270/Q2QR4XPC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine H1 receptor (Cavia porcellus (domestic guinea pig)) | BDBM50019596 (2-(4-Methyl-piperazin-1-yl)-1-(2-prop-2-ynyloxy-et...) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | n/a | n/a | 12 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description In vitro inhibition of histamine-induced contractions in guinea pig ileum | J Med Chem 29: 1178-83 (1987) BindingDB Entry DOI: 10.7270/Q2QR4XPC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine H1 receptor (Cavia porcellus (domestic guinea pig)) | BDBM35938 (1-(p-chlorophenyl)-1-(2-pyridyl)-3-N,N-dimethylpro...) | UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL DrugBank MCE KEGG PC cid PC sid UniChem Patents Similars | PubMed | n/a | n/a | 12 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description In vitro inhibition of histamine-induced contractions in guinea pig ileum | J Med Chem 29: 1178-83 (1987) BindingDB Entry DOI: 10.7270/Q2QR4XPC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine H1 receptor (Cavia porcellus (domestic guinea pig)) | BDBM50019634 (1-(2-Methoxy-ethyl)-2-(4-methyl-piperazin-1-yl)-1H...) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 13 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description In vitro inhibition of histamine-induced contractions in guinea pig ileum | J Med Chem 29: 1178-83 (1987) BindingDB Entry DOI: 10.7270/Q2QR4XPC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine H1 receptor (Cavia porcellus (domestic guinea pig)) | BDBM50019597 (2-(4-Butyl-piperazin-1-yl)-1-(2-ethoxy-ethyl)-1H-b...) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 15 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description In vitro inhibition of histamine-induced contractions in guinea pig ileum | J Med Chem 29: 1178-83 (1987) BindingDB Entry DOI: 10.7270/Q2QR4XPC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine H1 receptor (Cavia porcellus (domestic guinea pig)) | BDBM50019625 (2-(4-Benzyl-[1,4]diazepan-1-yl)-1-(2-ethoxy-ethyl)...) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 15 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description In vitro inhibition of histamine-induced contractions in guinea pig ileum | J Med Chem 29: 1178-83 (1987) BindingDB Entry DOI: 10.7270/Q2QR4XPC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine H1 receptor (Cavia porcellus (domestic guinea pig)) | BDBM50019631 (1-(2-Ethoxy-ethyl)-2-(4-propyl-piperazin-1-yl)-1H-...) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 16 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description In vitro inhibition of histamine-induced contractions in guinea pig ileum | J Med Chem 29: 1178-83 (1987) BindingDB Entry DOI: 10.7270/Q2QR4XPC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine H1 receptor (Cavia porcellus (domestic guinea pig)) | BDBM50019630 (1-(2-Ethoxy-ethyl)-2-(4-ethyl-[1,4]diazepan-1-yl)-...) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 16 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description In vitro inhibition of histamine-induced contractions in guinea pig ileum | J Med Chem 29: 1178-83 (1987) BindingDB Entry DOI: 10.7270/Q2QR4XPC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine H1 receptor (Cavia porcellus (domestic guinea pig)) | BDBM50019611 (2-(4-Methyl-[1,4]diazepan-1-yl)-1-(2-propoxy-ethyl...) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | n/a | n/a | 16 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description In vitro inhibition of histamine-induced contractions in guinea pig ileum | J Med Chem 29: 1178-83 (1987) BindingDB Entry DOI: 10.7270/Q2QR4XPC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine H1 receptor (Cavia porcellus (domestic guinea pig)) | BDBM50089150 (2-Ethyl-9-phenyl-2,3,4,9-tetrahydro-1H-indeno[2,1-...) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 17 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Bath Curated by ChEMBL | Assay Description In vitro antagonistic activity at the Histamine H1 receptor in guinea pig ileum | Bioorg Med Chem Lett 10: 1277-9 (2000) BindingDB Entry DOI: 10.7270/Q2T152VB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine H1 receptor (Cavia porcellus (domestic guinea pig)) | BDBM50019617 (1-(2-Allyloxy-ethyl)-2-(4-methyl-piperazin-1-yl)-1...) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | n/a | n/a | 17 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description In vitro inhibition of histamine-induced contractions in guinea pig ileum | J Med Chem 29: 1178-83 (1987) BindingDB Entry DOI: 10.7270/Q2QR4XPC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine H1 receptor (Cavia porcellus (domestic guinea pig)) | BDBM50019616 (1-Benzyl-2-(4-methyl-piperazin-1-yl)-1H-benzoimida...) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | n/a | n/a | 17 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description In vitro inhibition of histamine-induced contractions in guinea pig ileum | J Med Chem 29: 1178-83 (1987) BindingDB Entry DOI: 10.7270/Q2QR4XPC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine H1 receptor (Cavia porcellus (domestic guinea pig)) | BDBM50019635 (1-(2-Ethoxy-ethyl)-2-(4-ethyl-piperazin-1-yl)-1H-b...) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | n/a | n/a | 18 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description In vitro inhibition of histamine-induced contractions in guinea pig ileum | J Med Chem 29: 1178-83 (1987) BindingDB Entry DOI: 10.7270/Q2QR4XPC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine H1 receptor (Cavia porcellus (domestic guinea pig)) | BDBM50019619 (2-(4-Methyl-piperazin-1-yl)-1-propoxymethyl-1H-ben...) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | PubMed | n/a | n/a | 18 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description In vitro inhibition of histamine-induced contractions in guinea pig ileum | J Med Chem 29: 1178-83 (1987) BindingDB Entry DOI: 10.7270/Q2QR4XPC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine H1 receptor (Cavia porcellus (domestic guinea pig)) | BDBM50019626 (2-(4-Methyl-piperazin-1-yl)-1-pentyl-1H-benzoimida...) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 19 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description In vitro inhibition of histamine-induced contractions in guinea pig ileum | J Med Chem 29: 1178-83 (1987) BindingDB Entry DOI: 10.7270/Q2QR4XPC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine H1 receptor (Cavia porcellus (domestic guinea pig)) | BDBM50019593 (1-(2-Ethylsulfanyl-ethyl)-2-(4-methyl-piperazin-1-...) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | PubMed | n/a | n/a | 19 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description In vitro inhibition of histamine-induced contractions in guinea pig ileum | J Med Chem 29: 1178-83 (1987) BindingDB Entry DOI: 10.7270/Q2QR4XPC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine H1 receptor (Cavia porcellus (domestic guinea pig)) | BDBM50019599 (2-(4-Methyl-piperazin-1-yl)-1-(2-propoxy-ethyl)-1H...) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | n/a | n/a | 20 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description In vitro inhibition of histamine-induced contractions in guinea pig ileum | J Med Chem 29: 1178-83 (1987) BindingDB Entry DOI: 10.7270/Q2QR4XPC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine H1 receptor (Cavia porcellus (domestic guinea pig)) | BDBM50089148 (((3R,4S)-1-Ethyl-4-hydroxy-4-phenyl-piperidin-3-yl...) | UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 23 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Bath Curated by ChEMBL | Assay Description In vitro antagonistic activity at the Histamine H1 receptor in guinea pig ileum | Bioorg Med Chem Lett 10: 1277-9 (2000) BindingDB Entry DOI: 10.7270/Q2T152VB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine H1 receptor (Cavia porcellus (domestic guinea pig)) | BDBM50007536 (CHEMBL24517 | [3-(5-Chloro-pyridin-2-yl)-3-pyridin...) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 24 | n/a | n/a | n/a | n/a | n/a | n/a |
A. H. Robins Company, Inc. Curated by ChEMBL | Assay Description Inhibition of [3H]-mepyramine binding to the Histamine H1 receptor in guinea pig cortex | J Med Chem 34: 1314-28 (1991) BindingDB Entry DOI: 10.7270/Q23F4NMG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine H1 receptor (Cavia porcellus (domestic guinea pig)) | BDBM50019639 (2-[1,4]Diazepan-1-yl-1-(2-ethoxy-ethyl)-1H-benzoim...) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | n/a | n/a | 25 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description In vitro inhibition of histamine-induced contractions in guinea pig ileum | J Med Chem 29: 1178-83 (1987) BindingDB Entry DOI: 10.7270/Q2QR4XPC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine H1 receptor (Cavia porcellus (domestic guinea pig)) | BDBM50019632 (1-Hexyl-2-(4-methyl-piperazin-1-yl)-1H-benzoimidaz...) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 26 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description In vitro inhibition of histamine-induced contractions in guinea pig ileum | J Med Chem 29: 1178-83 (1987) BindingDB Entry DOI: 10.7270/Q2QR4XPC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine H1 receptor (Cavia porcellus (domestic guinea pig)) | BDBM50089146 (((3R,4S)-4-Hydroxy-1-methyl-4-phenyl-piperidin-3-y...) | UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 26 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Bath Curated by ChEMBL | Assay Description In vitro antagonistic activity at the Histamine H1 receptor in guinea pig ileum | Bioorg Med Chem Lett 10: 1277-9 (2000) BindingDB Entry DOI: 10.7270/Q2T152VB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine H1 receptor (Cavia porcellus (domestic guinea pig)) | BDBM50019627 (2-(4-Benzyl-piperazin-1-yl)-1-(2-ethoxy-ethyl)-1H-...) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | n/a | n/a | 27 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description In vitro inhibition of histamine-induced contractions in guinea pig ileum | J Med Chem 29: 1178-83 (1987) BindingDB Entry DOI: 10.7270/Q2QR4XPC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine H1 receptor (Cavia porcellus (domestic guinea pig)) | BDBM50089144 (2-Methyl-9-phenyl-2,3,4,4a-tetrahydro-1H-indeno[2,...) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 28 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Bath Curated by ChEMBL | Assay Description In vitro antagonistic activity at the Histamine H1 receptor in guinea pig ileum | Bioorg Med Chem Lett 10: 1277-9 (2000) BindingDB Entry DOI: 10.7270/Q2T152VB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine H1 receptor (Cavia porcellus (domestic guinea pig)) | BDBM50156861 (2-(2-(4-(1-((5-chlorothiophen-2-yl)methyl)-6-fluor...) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 28 | n/a | n/a | n/a | n/a | n/a | n/a |
Rhône-Poulenc Rorer Curated by ChEMBL | Assay Description Displacement of [3H]mepyramine from histamine H1 receptor in guinea pig cerebellum membranes | J Med Chem 47: 6326-37 (2004) Article DOI: 10.1021/jm0498203 BindingDB Entry DOI: 10.7270/Q2HM57XC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine H1 receptor (Cavia porcellus (domestic guinea pig)) | BDBM50007539 (8-(2-Dimethylamino-ethyl)-6-methyl-7,8-dihydro-6H-...) | UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Patents Similars | PubMed | n/a | n/a | 30 | n/a | n/a | n/a | n/a | n/a | n/a |
A. H. Robins Company, Inc. Curated by ChEMBL | Assay Description Inhibition of [3H]-mepyramine binding to the histamine receptor in guinea pig cortex | J Med Chem 34: 1314-28 (1991) BindingDB Entry DOI: 10.7270/Q23F4NMG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine H1 receptor (Cavia porcellus (domestic guinea pig)) | BDBM50019601 (1-(2-Ethoxy-ethyl)-2-(4-pentyl-piperazin-1-yl)-1H-...) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 30 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description In vitro inhibition of histamine-induced contractions in guinea pig ileum | J Med Chem 29: 1178-83 (1987) BindingDB Entry DOI: 10.7270/Q2QR4XPC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine H1 receptor (Cavia porcellus (domestic guinea pig)) | BDBM50019592 (1-(2-Ethoxy-ethyl)-2-(4-phenethyl-piperazin-1-yl)-...) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 31 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description In vitro inhibition of histamine-induced contractions in guinea pig ileum | J Med Chem 29: 1178-83 (1987) BindingDB Entry DOI: 10.7270/Q2QR4XPC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine H1 receptor (Cavia porcellus (domestic guinea pig)) | BDBM50156893 (2-(2-{4-[1-(2-Ethoxy-ethyl)-1H-indol-3-yl]-piperid...) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 34 | n/a | n/a | n/a | n/a | n/a | n/a |
Rhône-Poulenc Rorer Curated by ChEMBL | Assay Description Displacement of [3H]mepyramine from histamine H1 receptor in guinea pig cerebellum membranes | J Med Chem 47: 6326-37 (2004) Article DOI: 10.1021/jm0498203 BindingDB Entry DOI: 10.7270/Q2HM57XC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine H1 receptor (Cavia porcellus (domestic guinea pig)) | BDBM22567 (3H]pyrilamine | CHEMBL511 | Dorantamin | Mepyramin...) | UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL DrugBank MCE KEGG PC cid PC sid PDB UniChem Patents Similars | PubMed | n/a | n/a | 34 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Bath Curated by ChEMBL | Assay Description In vitro antagonistic activity at the Histamine H1 receptor in guinea pig ileum | Bioorg Med Chem Lett 10: 1277-9 (2000) BindingDB Entry DOI: 10.7270/Q2T152VB | |||||||||||
More data for this Ligand-Target Pair |
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