Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kcal/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Bcl-2-related protein A1 (Homo sapiens (Human)) | BDBM50558852 (CHEMBL4747465) | PDB MMDB NCI pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 6.5 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Binding affinity to human Bcl2A1 incubated for 2 hrs by FBid based competitive FP assay | Citation and Details Article DOI: 10.1021/acs.jmedchem.8b00010 BindingDB Entry DOI: 10.7270/Q28S4TMJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bcl-2-related protein A1 (Homo sapiens (Human)) | BDBM50558851 (CHEMBL4782684) | PDB MMDB NCI pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 6.60 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Binding affinity to human Bcl2A1 incubated for 2 hrs by FBid based competitive FP assay | Citation and Details Article DOI: 10.1021/acs.jmedchem.8b00010 BindingDB Entry DOI: 10.7270/Q28S4TMJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bcl-2-related protein A1 (Homo sapiens (Human)) | BDBM50210070 (CHEMBL3883565) | PDB MMDB NCI pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 8.5 | n/a | n/a | n/a | n/a | n/a | n/a |
The University of Queensland Curated by ChEMBL | Assay Description Inhibition of FITC-betaA-DIIRNIARHLAQVGDSMRSI-NH2 binding to recombinant human Bcl2A1 (1 to 152 residues) BH3 binding site expressed in Escherichia c... | ACS Med Chem Lett 8: 22-26 (2017) Article DOI: 10.1021/acsmedchemlett.6b00395 BindingDB Entry DOI: 10.7270/Q2NS0WWV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bcl-2-related protein A1 (Homo sapiens (Human)) | BDBM50558856 (CHEMBL4791348) | PDB MMDB NCI pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 13 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Binding affinity to human Bcl2A1 incubated for 2 hrs by FBid based competitive FP assay | Citation and Details Article DOI: 10.1021/acs.jmedchem.8b00010 BindingDB Entry DOI: 10.7270/Q28S4TMJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bcl-2-related protein A1 (Homo sapiens (Human)) | BDBM50558854 (CHEMBL4755711) | PDB MMDB NCI pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 14 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Binding affinity to human Bcl2A1 incubated for 2 hrs by FBid based competitive FP assay | Citation and Details Article DOI: 10.1021/acs.jmedchem.8b00010 BindingDB Entry DOI: 10.7270/Q28S4TMJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bcl-2-related protein A1 (Homo sapiens (Human)) | BDBM50587033 (CHEMBL5075478) | PDB MMDB NCI pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 18 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of human Bfl-1 (1 to 149 residues) expressed in Rosetta-gami (DE3) using biotinylated-BH3 peptide as substrate measured after 2 hrs by DEL... | Citation and Details Article DOI: 10.1021/acs.jmedchem.1c00005 BindingDB Entry DOI: 10.7270/Q2CZ3C3Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bcl-2-related protein A1 (Homo sapiens (Human)) | BDBM50558857 (CHEMBL4752520) | PDB MMDB NCI pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 20 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Binding affinity to human Bcl2A1 incubated for 2 hrs by FBid based competitive FP assay | Citation and Details Article DOI: 10.1021/acs.jmedchem.8b00010 BindingDB Entry DOI: 10.7270/Q28S4TMJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bcl-2-related protein A1 (Homo sapiens (Human)) | BDBM333146 (Compound I | US10196404, Example 1 | US10196404, E...) | PDB MMDB NCI pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | Purchase MCE PC cid PC sid PDB UniChem | Article PubMed | n/a | n/a | >20 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Citation and Details Article DOI: 10.1016/j.bmcl.2020.127717 BindingDB Entry DOI: 10.7270/Q2MW2N34 | ||||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bcl-2-related protein A1 (Homo sapiens (Human)) | BDBM50558853 (CHEMBL4465826) | PDB MMDB NCI pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 31 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Binding affinity to human Bcl2A1 incubated for 2 hrs by FBid based competitive FP assay | Citation and Details Article DOI: 10.1021/acs.jmedchem.8b00010 BindingDB Entry DOI: 10.7270/Q28S4TMJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bcl-2-related protein A1 (Homo sapiens (Human)) | BDBM50558855 (CHEMBL4740212) | PDB MMDB NCI pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 55 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Binding affinity to human Bcl2A1 incubated for 2 hrs by FBid based competitive FP assay | Citation and Details Article DOI: 10.1021/acs.jmedchem.8b00010 BindingDB Entry DOI: 10.7270/Q28S4TMJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bcl-2-related protein A1 (Homo sapiens (Human)) | BDBM50210069 (CHEMBL3884841) | PDB MMDB NCI pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 110 | n/a | n/a | n/a | n/a | n/a | n/a |
The University of Queensland Curated by ChEMBL | Assay Description Inhibition of FITC-betaA-DIIRNIARHLAQVGDSMRSI-NH2 binding to recombinant human Bcl2A1 (1 to 152 residues) BH3 binding site expressed in Escherichia c... | ACS Med Chem Lett 8: 22-26 (2017) Article DOI: 10.1021/acsmedchemlett.6b00395 BindingDB Entry DOI: 10.7270/Q2NS0WWV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bcl-2-related protein A1 (Homo sapiens (Human)) | BDBM50330250 (5,5'-Dibenzyl-6,6',7,7'-tetrahydroxy-3,3'-dimethyl...) | PDB MMDB NCI pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 122 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Maryland Curated by ChEMBL | Assay Description Inhibition of FITC-labeled Bim BH3 binding to GST-tagged Bcl2A1 (unknown origin) preincubated for 2 mins followed by FITC-Bim-BH3 addition measured a... | J Med Chem 60: 821-838 (2017) Article DOI: 10.1021/acs.jmedchem.5b01888 BindingDB Entry DOI: 10.7270/Q2ZC85BP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bcl-2-related protein A1 (Homo sapiens (Human)) | BDBM39156 (3-chloranyl-1-(3,4-dichlorophenyl)-4-[4-(2-hydroxy...) | PDB MMDB NCI pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 240 | n/a | n/a | n/a | n/a | n/a | n/a |
Human BioMolecular Research Institute Curated by ChEMBL | Assay Description Inhibition of N-terminal FITC BH3 peptide binding to GST-tagged Bfl1 by fluorescence polarization assay | Bioorg Med Chem Lett 20: 6560-4 (2010) Article DOI: 10.1016/j.bmcl.2010.09.046 BindingDB Entry DOI: 10.7270/Q27D2VCZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bcl-2-related protein A1 (Homo sapiens (Human)) | BDBM50587038 (CHEMBL5090086) | PDB MMDB NCI pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | >250 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of human Bfl-1 (1 to 149 residues) expressed in Rosetta-gami (DE3) using biotinylated-BH3 peptide as substrate measured after 2 hrs by DEL... | Citation and Details Article DOI: 10.1021/acs.jmedchem.1c00005 BindingDB Entry DOI: 10.7270/Q2CZ3C3Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bcl-2-related protein A1 (Homo sapiens (Human)) | BDBM50313364 ((2S,3R,4R,5S,6R)-2-(3-(4-ethylbenzyl)-4-methylphen...) | PDB MMDB NCI pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 250 | n/a | n/a | n/a | n/a | n/a | n/a |
Human BioMolecular Research Institute Curated by ChEMBL | Assay Description Inhibition of N-terminal FITC BH3 peptide binding to GST-tagged Bfl1 by fluorescence polarization assay | Bioorg Med Chem Lett 20: 6560-4 (2010) Article DOI: 10.1016/j.bmcl.2010.09.046 BindingDB Entry DOI: 10.7270/Q27D2VCZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bcl-2-related protein A1 (Homo sapiens (Human)) | BDBM39124 (3-chloranyl-1-(3,4-dichlorophenyl)-4-(dimethylamin...) | PDB MMDB NCI pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 300 | n/a | n/a | n/a | n/a | n/a | n/a |
Human BioMolecular Research Institute Curated by ChEMBL | Assay Description Inhibition of N-terminal FITC BH3 peptide binding to GST-tagged Bfl1 by fluorescence polarization assay | Bioorg Med Chem Lett 20: 6560-4 (2010) Article DOI: 10.1016/j.bmcl.2010.09.046 BindingDB Entry DOI: 10.7270/Q27D2VCZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bcl-2-related protein A1 (Homo sapiens (Human)) | BDBM39146 (3-chloranyl-1-(3,4-dichlorophenyl)-4-[4-[2-(2-hydr...) | PDB MMDB NCI pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 300 | n/a | n/a | n/a | n/a | n/a | n/a |
Human BioMolecular Research Institute Curated by ChEMBL | Assay Description Inhibition of N-terminal FITC BH3 peptide binding to GST-tagged Bfl1 by fluorescence polarization assay | Bioorg Med Chem Lett 20: 6560-4 (2010) Article DOI: 10.1016/j.bmcl.2010.09.046 BindingDB Entry DOI: 10.7270/Q27D2VCZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bcl-2-related protein A1 (Homo sapiens (Human)) | BDBM39124 (3-chloranyl-1-(3,4-dichlorophenyl)-4-(dimethylamin...) | PDB MMDB NCI pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 400 | n/a | n/a | n/a | n/a | n/a | n/a |
Human BioMolecular Research Institute Curated by ChEMBL | Assay Description Inhibition of N-terminal FITC BH3 peptide binding to GST-tagged Bfl1 by time resolved-FRET assay | Bioorg Med Chem Lett 20: 6560-4 (2010) Article DOI: 10.1016/j.bmcl.2010.09.046 BindingDB Entry DOI: 10.7270/Q27D2VCZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bcl-2-related protein A1 (Homo sapiens (Human)) | BDBM31809 (Apogossypol derivative, 8k) | PDB MMDB NCI pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 400 | n/a | n/a | n/a | n/a | n/a | 25 |
Burnham Institute for Medical Research | Assay Description FPAs were performed using various concentrations of GST-Bcl-2 family proteins, incubated with FITC-conjugated peptide substrates in the presence of i... | J Med Chem 52: 4511-23 (2009) Article DOI: 10.1021/jm900472s BindingDB Entry DOI: 10.7270/Q247486S | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bcl-2-related protein A1 (Homo sapiens (Human)) | BDBM39146 (3-chloranyl-1-(3,4-dichlorophenyl)-4-[4-[2-(2-hydr...) | PDB MMDB NCI pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 400 | n/a | n/a | n/a | n/a | n/a | n/a |
Human BioMolecular Research Institute Curated by ChEMBL | Assay Description Inhibition of N-terminal FITC BH3 peptide binding to GST-tagged Bfl1 by time resolved-FRET assay | Bioorg Med Chem Lett 20: 6560-4 (2010) Article DOI: 10.1016/j.bmcl.2010.09.046 BindingDB Entry DOI: 10.7270/Q27D2VCZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bcl-2-related protein A1 (Homo sapiens (Human)) | BDBM50587036 (CHEMBL5091695) | PDB MMDB NCI pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | >400 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of human Bfl-1 (1 to 149 residues) expressed in Rosetta-gami (DE3) using biotinylated-BH3 peptide as substrate measured after 2 hrs by DEL... | Citation and Details Article DOI: 10.1021/acs.jmedchem.1c00005 BindingDB Entry DOI: 10.7270/Q2CZ3C3Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bcl-2-related protein A1 (Homo sapiens (Human)) | BDBM31810 (Apogossypol derivative, 8r) | PDB MMDB NCI pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | Purchase PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 420 | n/a | n/a | n/a | n/a | n/a | n/a |
Sanford-Burnham Medical Research Institute Curated by ChEMBL | Assay Description Displacement of FITC-labeled Bak BH3 peptide from Bfl-1 after 30 mins by fluorescence polarization assay | J Med Chem 53: 4166-76 (2010) Article DOI: 10.1021/jm1001265 BindingDB Entry DOI: 10.7270/Q2FF3T97 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bcl-2-related protein A1 (Homo sapiens (Human)) | BDBM50313335 (6-(cyclohexylamino)-N-(4-sulfamoylphenyl)pyrimidin...) | PDB MMDB NCI pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 450 | n/a | n/a | n/a | n/a | n/a | n/a |
Human BioMolecular Research Institute Curated by ChEMBL | Assay Description Inhibition of N-terminal FITC BH3 peptide binding to GST-tagged Bfl1 by time resolved-FRET assay | Bioorg Med Chem Lett 20: 6560-4 (2010) Article DOI: 10.1016/j.bmcl.2010.09.046 BindingDB Entry DOI: 10.7270/Q27D2VCZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bcl-2-related protein A1 (Homo sapiens (Human)) | BDBM31805 (Apogossypol derivative, 8n) | PDB MMDB NCI pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 550 | n/a | n/a | n/a | n/a | n/a | 25 |
Burnham Institute for Medical Research | Assay Description FPAs were performed using various concentrations of GST-Bcl-2 family proteins, incubated with FITC-conjugated peptide substrates in the presence of i... | J Med Chem 52: 4511-23 (2009) Article DOI: 10.1021/jm900472s BindingDB Entry DOI: 10.7270/Q247486S | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bcl-2-related protein A1 (Homo sapiens (Human)) | BDBM39147 (3-chloranyl-1-(3,4-dichlorophenyl)-4-[(3R)-3-methy...) | PDB MMDB NCI pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 600 | n/a | n/a | n/a | n/a | n/a | n/a |
Human BioMolecular Research Institute Curated by ChEMBL | Assay Description Inhibition of N-terminal FITC BH3 peptide binding to GST-tagged Bfl1 by fluorescence polarization assay | Bioorg Med Chem Lett 20: 6560-4 (2010) Article DOI: 10.1016/j.bmcl.2010.09.046 BindingDB Entry DOI: 10.7270/Q27D2VCZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bcl-2-related protein A1 (Homo sapiens (Human)) | BDBM34194 (3-chloranyl-1-(3,4-dichlorophenyl)-4-(4-methylpipe...) | PDB MMDB NCI pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | Purchase PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 600 | n/a | n/a | n/a | n/a | n/a | n/a |
Human BioMolecular Research Institute Curated by ChEMBL | Assay Description Inhibition of N-terminal FITC BH3 peptide binding to GST-tagged Bfl1 by fluorescence polarization assay | Bioorg Med Chem Lett 20: 6560-4 (2010) Article DOI: 10.1016/j.bmcl.2010.09.046 BindingDB Entry DOI: 10.7270/Q27D2VCZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bcl-2-related protein A1 (Homo sapiens (Human)) | BDBM50316672 ((R)-1,1',6,6',7,7'-Hexahydroxy-3,3'-dimethyl-N5-((...) | PDB MMDB NCI pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 620 | n/a | n/a | n/a | n/a | n/a | n/a |
Sanford-Burnham Medical Research Institute Curated by ChEMBL | Assay Description Displacement of FITC-labeled Bak BH3 peptide from Bfl-1 after 30 mins by fluorescence polarization assay | J Med Chem 53: 4166-76 (2010) Article DOI: 10.1021/jm1001265 BindingDB Entry DOI: 10.7270/Q2FF3T97 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bcl-2-related protein A1 (Homo sapiens (Human)) | BDBM39156 (3-chloranyl-1-(3,4-dichlorophenyl)-4-[4-(2-hydroxy...) | PDB MMDB NCI pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 620 | n/a | n/a | n/a | n/a | n/a | n/a |
Human BioMolecular Research Institute Curated by ChEMBL | Assay Description Inhibition of N-terminal FITC BH3 peptide binding to GST-tagged Bfl1 by time resolved-FRET assay | Bioorg Med Chem Lett 20: 6560-4 (2010) Article DOI: 10.1016/j.bmcl.2010.09.046 BindingDB Entry DOI: 10.7270/Q27D2VCZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bcl-2-related protein A1 (Homo sapiens (Human)) | BDBM50316672 ((R)-1,1',6,6',7,7'-Hexahydroxy-3,3'-dimethyl-N5-((...) | PDB MMDB NCI pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 620 | n/a | n/a | n/a | n/a | n/a | n/a |
Sanford-Burnham Medical Research Institute Curated by ChEMBL | Assay Description Displacement of FITC-labeled Bak BH3 peptide from Bfl-1 after 30 mins by fluorescence polarization assay | J Med Chem 53: 4166-76 (2010) Article DOI: 10.1021/jm1001265 BindingDB Entry DOI: 10.7270/Q2FF3T97 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bcl-2-related protein A1 (Homo sapiens (Human)) | BDBM142756 (US8937193, 6i) | PDB MMDB NCI pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 650 | n/a | n/a | n/a | n/a | n/a | 25 |
Sanford-Burnham Medical Research Institute US Patent | Assay Description A Bak BH3 peptide (F-BakBH3) (GQVGRQLAIIGDDINR (SEQ ID NO:1)) was labeled at the N-terminus with fluorescein isothiocyanate (FITC) (Molecular Probes)... | US Patent US8937193 (2015) BindingDB Entry DOI: 10.7270/Q20C4TG4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bcl-2-related protein A1 (Homo sapiens (Human)) | BDBM50330250 (5,5'-Dibenzyl-6,6',7,7'-tetrahydroxy-3,3'-dimethyl...) | PDB MMDB NCI pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 650 | n/a | n/a | n/a | n/a | n/a | n/a |
Sanford-Burnham Medical Research Institute Curated by ChEMBL | Assay Description Displacement of F-BakBH3 from Bfl-1 after 30 mins by fluorescence polarization assay | J Med Chem 53: 8000-11 (2010) Article DOI: 10.1021/jm100746q BindingDB Entry DOI: 10.7270/Q22N52H7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bcl-2-related protein A1 (Homo sapiens (Human)) | BDBM31811 (Apogossypol derivative, 8s) | PDB MMDB NCI pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 670 | n/a | n/a | n/a | n/a | n/a | 25 |
Burnham Institute for Medical Research | Assay Description FPAs were performed using various concentrations of GST-Bcl-2 family proteins, incubated with FITC-conjugated peptide substrates in the presence of i... | J Med Chem 52: 4511-23 (2009) Article DOI: 10.1021/jm900472s BindingDB Entry DOI: 10.7270/Q247486S | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bcl-2-related protein A1 (Homo sapiens (Human)) | BDBM142749 (US8937193, 7) | PDB MMDB NCI pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 690 | n/a | n/a | n/a | n/a | n/a | 25 |
Sanford-Burnham Medical Research Institute US Patent | Assay Description A Bak BH3 peptide (F-BakBH3) (GQVGRQLAIIGDDINR (SEQ ID NO:1)) was labeled at the N-terminus with fluorescein isothiocyanate (FITC) (Molecular Probes)... | US Patent US8937193 (2015) BindingDB Entry DOI: 10.7270/Q20C4TG4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bcl-2-related protein A1 (Homo sapiens (Human)) | BDBM39149 (3-chloranyl-1-(3,4-dichlorophenyl)-4-[4-[(E)-3-phe...) | PDB MMDB NCI pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 690 | n/a | n/a | n/a | n/a | n/a | n/a |
Human BioMolecular Research Institute Curated by ChEMBL | Assay Description Inhibition of N-terminal FITC BH3 peptide binding to GST-tagged Bfl1 by time resolved-FRET assay | Bioorg Med Chem Lett 20: 6560-4 (2010) Article DOI: 10.1016/j.bmcl.2010.09.046 BindingDB Entry DOI: 10.7270/Q27D2VCZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bcl-2-related protein A1 (Homo sapiens (Human)) | BDBM50330257 (6,6',7,7'-Tetrahydroxy-3,3'-dimethyl-5,5'-bis(2-ph...) | PDB MMDB NCI pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 690 | n/a | n/a | n/a | n/a | n/a | n/a |
Sanford-Burnham Medical Research Institute Curated by ChEMBL | Assay Description Displacement of F-BakBH3 from Bfl-1 after 30 mins by fluorescence polarization assay | J Med Chem 53: 8000-11 (2010) Article DOI: 10.1021/jm100746q BindingDB Entry DOI: 10.7270/Q22N52H7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bcl-2-related protein A1 (Homo sapiens (Human)) | BDBM50330256 (5,5'-Bis(4-chlorobenzyl)-6,6',7,7''-tetrahydroxy-3...) | PDB MMDB NCI pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 700 | n/a | n/a | n/a | n/a | n/a | n/a |
Sanford-Burnham Medical Research Institute Curated by ChEMBL | Assay Description Displacement of F-BakBH3 from Bfl-1 after 30 mins by fluorescence polarization assay | J Med Chem 53: 8000-11 (2010) Article DOI: 10.1021/jm100746q BindingDB Entry DOI: 10.7270/Q22N52H7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bcl-2-related protein A1 (Homo sapiens (Human)) | BDBM142757 (US8937193, 6l) | PDB MMDB NCI pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 700 | n/a | n/a | n/a | n/a | n/a | 25 |
Sanford-Burnham Medical Research Institute US Patent | Assay Description A Bak BH3 peptide (F-BakBH3) (GQVGRQLAIIGDDINR (SEQ ID NO:1)) was labeled at the N-terminus with fluorescein isothiocyanate (FITC) (Molecular Probes)... | US Patent US8937193 (2015) BindingDB Entry DOI: 10.7270/Q20C4TG4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bcl-2-related protein A1 (Homo sapiens (Human)) | BDBM50330258 (6,6',7,7'-Tetrahydroxy-3,3'-dimethyl-1,1',4,4'-tet...) | PDB MMDB NCI pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 710 | n/a | n/a | n/a | n/a | n/a | n/a |
Sanford-Burnham Medical Research Institute Curated by ChEMBL | Assay Description Displacement of F-BakBH3 from Bfl-1 after 30 mins by fluorescence polarization assay | J Med Chem 53: 8000-11 (2010) Article DOI: 10.1021/jm100746q BindingDB Entry DOI: 10.7270/Q22N52H7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bcl-2-related protein A1 (Homo sapiens (Human)) | BDBM142746 (US8937193, 8a) | PDB MMDB NCI pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 710 | n/a | n/a | n/a | n/a | n/a | 25 |
Sanford-Burnham Medical Research Institute US Patent | Assay Description A Bak BH3 peptide (F-BakBH3) (GQVGRQLAIIGDDINR (SEQ ID NO:1)) was labeled at the N-terminus with fluorescein isothiocyanate (FITC) (Molecular Probes)... | US Patent US8937193 (2015) BindingDB Entry DOI: 10.7270/Q20C4TG4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bcl-2-related protein A1 (Homo sapiens (Human)) | BDBM31810 (Apogossypol derivative, 8r) | PDB MMDB NCI pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | Purchase PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 730 | n/a | n/a | n/a | n/a | n/a | 25 |
Burnham Institute for Medical Research | Assay Description FPAs were performed using various concentrations of GST-Bcl-2 family proteins, incubated with FITC-conjugated peptide substrates in the presence of i... | J Med Chem 52: 4511-23 (2009) Article DOI: 10.1021/jm900472s BindingDB Entry DOI: 10.7270/Q247486S | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bcl-2-related protein A1 (Homo sapiens (Human)) | BDBM50316671 ((S)-1,(R)-1,1',6,6',7,7'-Hexahydroxy-3,3'-dimethyl...) | PDB MMDB NCI pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | Purchase PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 750 | n/a | n/a | n/a | n/a | n/a | n/a |
Sanford-Burnham Medical Research Institute Curated by ChEMBL | Assay Description Displacement of FITC-labeled Bak BH3 peptide from Bfl-1 after 30 mins by fluorescence polarization assay | J Med Chem 53: 4166-76 (2010) Article DOI: 10.1021/jm1001265 BindingDB Entry DOI: 10.7270/Q2FF3T97 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bcl-2-related protein A1 (Homo sapiens (Human)) | BDBM50316671 ((S)-1,(R)-1,1',6,6',7,7'-Hexahydroxy-3,3'-dimethyl...) | PDB MMDB NCI pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | Purchase PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 750 | n/a | n/a | n/a | n/a | n/a | n/a |
Sanford-Burnham Medical Research Institute Curated by ChEMBL | Assay Description Displacement of FITC-labeled Bak BH3 peptide from Bfl-1 after 30 mins by fluorescence polarization assay | J Med Chem 53: 4166-76 (2010) Article DOI: 10.1021/jm1001265 BindingDB Entry DOI: 10.7270/Q2FF3T97 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bcl-2-related protein A1 (Homo sapiens (Human)) | BDBM34194 (3-chloranyl-1-(3,4-dichlorophenyl)-4-(4-methylpipe...) | PDB MMDB NCI pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | Purchase PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 800 | n/a | n/a | n/a | n/a | n/a | n/a |
Human BioMolecular Research Institute Curated by ChEMBL | Assay Description Inhibition of N-terminal FITC BH3 peptide binding to GST-tagged Bfl1 by time resolved-FRET assay | Bioorg Med Chem Lett 20: 6560-4 (2010) Article DOI: 10.1016/j.bmcl.2010.09.046 BindingDB Entry DOI: 10.7270/Q27D2VCZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bcl-2-related protein A1 (Homo sapiens (Human)) | BDBM39147 (3-chloranyl-1-(3,4-dichlorophenyl)-4-[(3R)-3-methy...) | PDB MMDB NCI pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 800 | n/a | n/a | n/a | n/a | n/a | n/a |
Human BioMolecular Research Institute Curated by ChEMBL | Assay Description Inhibition of N-terminal FITC BH3 peptide binding to GST-tagged Bfl1 by time resolved-FRET assay | Bioorg Med Chem Lett 20: 6560-4 (2010) Article DOI: 10.1016/j.bmcl.2010.09.046 BindingDB Entry DOI: 10.7270/Q27D2VCZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bcl-2-related protein A1 (Homo sapiens (Human)) | BDBM50313335 (6-(cyclohexylamino)-N-(4-sulfamoylphenyl)pyrimidin...) | PDB MMDB NCI pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 800 | n/a | n/a | n/a | n/a | n/a | n/a |
Human BioMolecular Research Institute Curated by ChEMBL | Assay Description Inhibition of N-terminal FITC BH3 peptide binding to GST-tagged Bfl1 by fluorescence polarization assay | Bioorg Med Chem Lett 20: 6560-4 (2010) Article DOI: 10.1016/j.bmcl.2010.09.046 BindingDB Entry DOI: 10.7270/Q27D2VCZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bcl-2-related protein A1 (Homo sapiens (Human)) | BDBM39143 (3-chloranyl-1-(2-chlorophenyl)-4-(4-methylpiperazi...) | PDB MMDB NCI pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 1.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Human BioMolecular Research Institute Curated by ChEMBL | Assay Description Inhibition of N-terminal FITC BH3 peptide binding to GST-tagged Bfl1 by time resolved-FRET assay | Bioorg Med Chem Lett 20: 6560-4 (2010) Article DOI: 10.1016/j.bmcl.2010.09.046 BindingDB Entry DOI: 10.7270/Q27D2VCZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bcl-2-related protein A1 (Homo sapiens (Human)) | BDBM50313365 ((2R,3R,4S,5S,6R)-2-(3-(4-ethylbenzyl)-4-methylbenz...) | PDB MMDB NCI pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Human BioMolecular Research Institute Curated by ChEMBL | Assay Description Inhibition of N-terminal FITC BH3 peptide binding to GST-tagged Bfl1 by time resolved-FRET assay | Bioorg Med Chem Lett 20: 6560-4 (2010) Article DOI: 10.1016/j.bmcl.2010.09.046 BindingDB Entry DOI: 10.7270/Q27D2VCZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bcl-2-related protein A1 (Homo sapiens (Human)) | BDBM50587037 (CHEMBL5082279) | PDB MMDB NCI pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | >1.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of human Bfl-1 (1 to 149 residues) expressed in Rosetta-gami (DE3) using biotinylated-BH3 peptide as substrate measured after 2 hrs by DEL... | Citation and Details Article DOI: 10.1021/acs.jmedchem.1c00005 BindingDB Entry DOI: 10.7270/Q2CZ3C3Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bcl-2-related protein A1 (Homo sapiens (Human)) | BDBM50313363 (3-(4-(6-(cyclohexyl(cyclopropylmethyl)amino)pyrimi...) | PDB MMDB NCI pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 1.10E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Human BioMolecular Research Institute Curated by ChEMBL | Assay Description Inhibition of N-terminal FITC BH3 peptide binding to GST-tagged Bfl1 by time resolved-FRET assay | Bioorg Med Chem Lett 20: 6560-4 (2010) Article DOI: 10.1016/j.bmcl.2010.09.046 BindingDB Entry DOI: 10.7270/Q27D2VCZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bcl-2-related protein A1 (Homo sapiens (Human)) | BDBM39162 (3-chloranyl-1-(3,4-dichlorophenyl)-4-[4-(3-methoxy...) | PDB MMDB NCI pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.20E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Human BioMolecular Research Institute Curated by ChEMBL | Assay Description Inhibition of N-terminal FITC BH3 peptide binding to GST-tagged Bfl1 by fluorescence polarization assay | Bioorg Med Chem Lett 20: 6560-4 (2010) Article DOI: 10.1016/j.bmcl.2010.09.046 BindingDB Entry DOI: 10.7270/Q27D2VCZ | |||||||||||
More data for this Ligand-Target Pair |
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