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Compile Data Set for Download or QSAR

Found 232 hits of ec50 data for polymerid = 4371   
Target/Host
(Institution)
LigandTarget/Host
Links
Ligand
Links
Trg + Lig
Links
Ki
nM
ΔG°
kcal/mole
IC50
nM
Kd
nM
EC50/IC50
nM
koff
s-1
kon
M-1s-1
pHTemp
°C
TGF-beta receptor type I


(Homo sapiens (Human))
BDBM50238071
PNG
(CHEMBL4079857)
PDB

KEGG

UniProtKB/SwissProt

B.MOAD
antibodypedia
GoogleScholar
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PC cid
PC sid
UniChem

Patents

n/an/an/an/a 6.30n/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
TGF-beta receptor type I


(Homo sapiens (Human))
BDBM50238082
PNG
(CHEMBL4102696)
PDB

KEGG

UniProtKB/SwissProt

B.MOAD
antibodypedia
GoogleScholar
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PC cid
PC sid
UniChem

Patents

n/an/an/an/a 7.90n/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
TGF-beta receptor type I


(Homo sapiens (Human))
BDBM50238072
PNG
(CHEMBL4104104)
PDB

KEGG

UniProtKB/SwissProt

B.MOAD
antibodypedia
GoogleScholar
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PC cid
PC sid
UniChem

Patents

n/an/an/an/a 7.90n/an/an/an/a


TBA

Assay Description
Binding affinity against cytidine deaminase of mouse kidney


Citation and Details
More data for this
Ligand-Target Pair
TGF-beta receptor type I


(Homo sapiens (Human))
BDBM50238084
PNG
(CHEMBL4085333)
PDB

KEGG

UniProtKB/SwissProt

B.MOAD
antibodypedia
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PC sid
UniChem

Patents

n/an/an/an/a 7.90n/an/an/an/a


TBA

Assay Description
Concentration required for 50% inhibition of Angiotensin I converting enzyme


Citation and Details
More data for this
Ligand-Target Pair
TGF-beta receptor type I


(Homo sapiens (Human))
BDBM346269
PNG
(US10202377, Compound 1)
PDB

KEGG

UniProtKB/SwissProt

B.MOAD
antibodypedia
GoogleScholar
AffyNet 
UniChem
Article
n/an/an/an/a 9n/an/an/an/a



Boehringer Ingelheim Pharmaceuticals Inc.





J Med Chem 46: 4676-86 (2003)

More data for this
Ligand-Target Pair
TGF-beta receptor type I


(Homo sapiens (Human))
BDBM346383
PNG
(US10202377, Compound 1350)
PDB

KEGG

UniProtKB/SwissProt

B.MOAD
antibodypedia
GoogleScholar
AffyNet 
UniChem
Article
n/an/an/an/a 9n/an/an/an/a



Boehringer Ingelheim Pharmaceuticals Inc.





J Med Chem 46: 4676-86 (2003)

More data for this
Ligand-Target Pair
TGF-beta receptor type I


(Homo sapiens (Human))
BDBM346279
PNG
(US10202377, Compound 55)
PDB

KEGG

UniProtKB/SwissProt

B.MOAD
antibodypedia
GoogleScholar
AffyNet 
UniChem
Article
n/an/an/an/a 9n/an/an/an/a



Boehringer Ingelheim Pharmaceuticals Inc.





J Med Chem 46: 4676-86 (2003)

More data for this
Ligand-Target Pair
TGF-beta receptor type I


(Homo sapiens (Human))
BDBM346283
PNG
(US10202377, Compound 82)
PDB

KEGG

UniProtKB/SwissProt

B.MOAD
antibodypedia
GoogleScholar
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UniChem
Article
n/an/an/an/a 9n/an/an/an/a



Boehringer Ingelheim Pharmaceuticals Inc.





J Med Chem 46: 4676-86 (2003)

More data for this
Ligand-Target Pair
TGF-beta receptor type I


(Homo sapiens (Human))
BDBM346285
PNG
(US10202377, Compound 90)
PDB

KEGG

UniProtKB/SwissProt

B.MOAD
antibodypedia
GoogleScholar
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UniChem
Article
n/an/an/an/a 9n/an/an/an/a



Boehringer Ingelheim Pharmaceuticals Inc.





J Med Chem 46: 4676-86 (2003)

More data for this
Ligand-Target Pair
TGF-beta receptor type I


(Homo sapiens (Human))
BDBM346286
PNG
(US10202377, Compound 93)
PDB

KEGG

UniProtKB/SwissProt

B.MOAD
antibodypedia
GoogleScholar
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UniChem
Article
n/an/an/an/a 9n/an/an/an/a



Boehringer Ingelheim Pharmaceuticals Inc.





J Med Chem 46: 4676-86 (2003)

More data for this
Ligand-Target Pair
TGF-beta receptor type I


(Homo sapiens (Human))
BDBM346287
PNG
(US10202377, Compound 101)
PDB

KEGG

UniProtKB/SwissProt

B.MOAD
antibodypedia
GoogleScholar
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UniChem
Article
n/an/an/an/a 9n/an/an/an/a



Boehringer Ingelheim Pharmaceuticals Inc.





J Med Chem 46: 4676-86 (2003)

More data for this
Ligand-Target Pair
TGF-beta receptor type I


(Homo sapiens (Human))
BDBM346294
PNG
(US10202377, Compound 154)
PDB

KEGG

UniProtKB/SwissProt

B.MOAD
antibodypedia
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UniChem
Article
n/an/an/an/a 9n/an/an/an/a



Boehringer Ingelheim Pharmaceuticals Inc.





J Med Chem 46: 4676-86 (2003)

More data for this
Ligand-Target Pair
TGF-beta receptor type I


(Homo sapiens (Human))
BDBM346296
PNG
(US10202377, Compound 169)
PDB

KEGG

UniProtKB/SwissProt

B.MOAD
antibodypedia
GoogleScholar
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UniChem
Article
n/an/an/an/a 9n/an/an/an/a



Boehringer Ingelheim Pharmaceuticals Inc.





J Med Chem 46: 4676-86 (2003)

More data for this
Ligand-Target Pair
TGF-beta receptor type I


(Homo sapiens (Human))
BDBM346298
PNG
(US10202377, Compound 181)
PDB

KEGG

UniProtKB/SwissProt

B.MOAD
antibodypedia
GoogleScholar
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UniChem
Article
n/an/an/an/a 9n/an/an/an/a



Boehringer Ingelheim Pharmaceuticals Inc.





J Med Chem 46: 4676-86 (2003)

More data for this
Ligand-Target Pair
TGF-beta receptor type I


(Homo sapiens (Human))
BDBM346300
PNG
(US10202377, Compound 190)
PDB

KEGG

UniProtKB/SwissProt

B.MOAD
antibodypedia
GoogleScholar
AffyNet 
UniChem
Article
n/an/an/an/a 9n/an/an/an/a



Boehringer Ingelheim Pharmaceuticals Inc.





J Med Chem 46: 4676-86 (2003)

More data for this
Ligand-Target Pair
TGF-beta receptor type I


(Homo sapiens (Human))
BDBM346301
PNG
(US10202377, Compound 196)
PDB

KEGG

UniProtKB/SwissProt

B.MOAD
antibodypedia
GoogleScholar
AffyNet 
UniChem
Article
n/an/an/an/a 9n/an/an/an/a



Boehringer Ingelheim Pharmaceuticals Inc.





J Med Chem 46: 4676-86 (2003)

More data for this
Ligand-Target Pair
TGF-beta receptor type I


(Homo sapiens (Human))
BDBM346302
PNG
(US10202377, Compound 202)
PDB

KEGG

UniProtKB/SwissProt

B.MOAD
antibodypedia
GoogleScholar
AffyNet 
UniChem
Article
n/an/an/an/a 9n/an/an/an/a



Boehringer Ingelheim Pharmaceuticals Inc.





J Med Chem 46: 4676-86 (2003)

More data for this
Ligand-Target Pair
TGF-beta receptor type I


(Homo sapiens (Human))
BDBM346308
PNG
(US10202377, Compound 234)
PDB

KEGG

UniProtKB/SwissProt

B.MOAD
antibodypedia
GoogleScholar
AffyNet 
UniChem
Article
n/an/an/an/a 9n/an/an/an/a



Boehringer Ingelheim Pharmaceuticals Inc.





J Med Chem 46: 4676-86 (2003)

More data for this
Ligand-Target Pair
TGF-beta receptor type I


(Homo sapiens (Human))
BDBM346313
PNG
(US10202377, Compound 265)
PDB

KEGG

UniProtKB/SwissProt

B.MOAD
antibodypedia
GoogleScholar
AffyNet 
UniChem
Article
n/an/an/an/a 9n/an/an/an/a



Boehringer Ingelheim Pharmaceuticals Inc.





J Med Chem 46: 4676-86 (2003)

More data for this
Ligand-Target Pair
TGF-beta receptor type I


(Homo sapiens (Human))
BDBM346314
PNG
(US10202377, Compound 268)
PDB

KEGG

UniProtKB/SwissProt

B.MOAD
antibodypedia
GoogleScholar
AffyNet 
UniChem
Article
n/an/an/an/a 9n/an/an/an/a



Boehringer Ingelheim Pharmaceuticals Inc.





J Med Chem 46: 4676-86 (2003)

More data for this
Ligand-Target Pair
TGF-beta receptor type I


(Homo sapiens (Human))
BDBM346316
PNG
(US10202377, Compound 271)
PDB

KEGG

UniProtKB/SwissProt

B.MOAD
antibodypedia
GoogleScholar
AffyNet 
UniChem
Article
n/an/an/an/a 9n/an/an/an/a



Boehringer Ingelheim Pharmaceuticals Inc.





J Med Chem 46: 4676-86 (2003)

More data for this
Ligand-Target Pair
TGF-beta receptor type I


(Homo sapiens (Human))
BDBM346317
PNG
(US10202377, Compound 277)
PDB

KEGG

UniProtKB/SwissProt

B.MOAD
antibodypedia
GoogleScholar
AffyNet 
UniChem
Article
n/an/an/an/a 9n/an/an/an/a



Boehringer Ingelheim Pharmaceuticals Inc.





J Med Chem 46: 4676-86 (2003)

More data for this
Ligand-Target Pair
TGF-beta receptor type I


(Homo sapiens (Human))
BDBM346319
PNG
(US10202377, Compound 283)
PDB

KEGG

UniProtKB/SwissProt

B.MOAD
antibodypedia
GoogleScholar
AffyNet 
UniChem
Article
n/an/an/an/a 9n/an/an/an/a



Boehringer Ingelheim Pharmaceuticals Inc.





J Med Chem 46: 4676-86 (2003)

More data for this
Ligand-Target Pair
TGF-beta receptor type I


(Homo sapiens (Human))
BDBM346320
PNG
(US10202377, Compound 288)
PDB

KEGG

UniProtKB/SwissProt

B.MOAD
antibodypedia
GoogleScholar
AffyNet 
UniChem
Article
n/an/an/an/a 9n/an/an/an/a



Boehringer Ingelheim Pharmaceuticals Inc.





J Med Chem 46: 4676-86 (2003)

More data for this
Ligand-Target Pair
TGF-beta receptor type I


(Homo sapiens (Human))
BDBM346321
PNG
(US10202377, Compound 292)
PDB

KEGG

UniProtKB/SwissProt

B.MOAD
antibodypedia
GoogleScholar
AffyNet 
UniChem
Article
n/an/an/an/a 9n/an/an/an/a



Boehringer Ingelheim Pharmaceuticals Inc.





J Med Chem 46: 4676-86 (2003)

More data for this
Ligand-Target Pair
TGF-beta receptor type I


(Homo sapiens (Human))
BDBM346322
PNG
(US10202377, Compound 294)
PDB

KEGG

UniProtKB/SwissProt

B.MOAD
antibodypedia
GoogleScholar
AffyNet 
UniChem
Article
n/an/an/an/a 9n/an/an/an/a



Boehringer Ingelheim Pharmaceuticals Inc.





J Med Chem 46: 4676-86 (2003)

More data for this
Ligand-Target Pair
TGF-beta receptor type I


(Homo sapiens (Human))
BDBM346324
PNG
(US10202377, Compound 298)
PDB

KEGG

UniProtKB/SwissProt

B.MOAD
antibodypedia
GoogleScholar
AffyNet 
UniChem
Article
n/an/an/an/a 9n/an/an/an/a



Boehringer Ingelheim Pharmaceuticals Inc.





J Med Chem 46: 4676-86 (2003)

More data for this
Ligand-Target Pair
TGF-beta receptor type I


(Homo sapiens (Human))
BDBM346333
PNG
(US10202377, Compound 325)
PDB

KEGG

UniProtKB/SwissProt

B.MOAD
antibodypedia
GoogleScholar
AffyNet 
UniChem
Article
n/an/an/an/a 9n/an/an/an/a



Boehringer Ingelheim Pharmaceuticals Inc.





J Med Chem 46: 4676-86 (2003)

More data for this
Ligand-Target Pair
TGF-beta receptor type I


(Homo sapiens (Human))
BDBM346336
PNG
(US10202377, Compound 337)
PDB

KEGG

UniProtKB/SwissProt

B.MOAD
antibodypedia
GoogleScholar
AffyNet 
UniChem
Article
n/an/an/an/a 9n/an/an/an/a



Boehringer Ingelheim Pharmaceuticals Inc.





J Med Chem 46: 4676-86 (2003)

More data for this
Ligand-Target Pair
TGF-beta receptor type I


(Homo sapiens (Human))
BDBM346341
PNG
(US10202377, Compound 367)
PDB

KEGG

UniProtKB/SwissProt

B.MOAD
antibodypedia
GoogleScholar
AffyNet 
UniChem
Article
n/an/an/an/a 9n/an/an/an/a



Boehringer Ingelheim Pharmaceuticals Inc.





J Med Chem 46: 4676-86 (2003)

More data for this
Ligand-Target Pair
TGF-beta receptor type I


(Homo sapiens (Human))
BDBM346343
PNG
(US10202377, Compound 379)
PDB

KEGG

UniProtKB/SwissProt

B.MOAD
antibodypedia
GoogleScholar
AffyNet 
UniChem
Article
n/an/an/an/a 9n/an/an/an/a



Boehringer Ingelheim Pharmaceuticals Inc.





J Med Chem 46: 4676-86 (2003)

More data for this
Ligand-Target Pair
TGF-beta receptor type I


(Homo sapiens (Human))
BDBM346351
PNG
(US10202377, Compound 421)
PDB

KEGG

UniProtKB/SwissProt

B.MOAD
antibodypedia
GoogleScholar
AffyNet 
UniChem
Article
n/an/an/an/a 9n/an/an/an/a



Boehringer Ingelheim Pharmaceuticals Inc.





J Med Chem 46: 4676-86 (2003)

More data for this
Ligand-Target Pair
TGF-beta receptor type I


(Homo sapiens (Human))
BDBM346353
PNG
(US10202377, Compound 427)
PDB

KEGG

UniProtKB/SwissProt

B.MOAD
antibodypedia
GoogleScholar
AffyNet 
UniChem
Article
n/an/an/an/a 9n/an/an/an/a



Boehringer Ingelheim Pharmaceuticals Inc.





J Med Chem 46: 4676-86 (2003)

More data for this
Ligand-Target Pair
TGF-beta receptor type I


(Homo sapiens (Human))
BDBM346354
PNG
(US10202377, Compound 433)
PDB

KEGG

UniProtKB/SwissProt

B.MOAD
antibodypedia
GoogleScholar
AffyNet 
UniChem
Article
n/an/an/an/a 9n/an/an/an/a



Boehringer Ingelheim Pharmaceuticals Inc.





J Med Chem 46: 4676-86 (2003)

More data for this
Ligand-Target Pair
TGF-beta receptor type I


(Homo sapiens (Human))
BDBM346356
PNG
(US10202377, Compound 439)
PDB

KEGG

UniProtKB/SwissProt

B.MOAD
antibodypedia
GoogleScholar
AffyNet 
UniChem
Article
n/an/an/an/a 9n/an/an/an/a



Boehringer Ingelheim Pharmaceuticals Inc.





J Med Chem 46: 4676-86 (2003)

More data for this
Ligand-Target Pair
TGF-beta receptor type I


(Homo sapiens (Human))
BDBM346357
PNG
(US10202377, Compound 442)
PDB

KEGG

UniProtKB/SwissProt

B.MOAD
antibodypedia
GoogleScholar
AffyNet 
UniChem
Article
n/an/an/an/a 9n/an/an/an/a



Boehringer Ingelheim Pharmaceuticals Inc.





J Med Chem 46: 4676-86 (2003)

More data for this
Ligand-Target Pair
TGF-beta receptor type I


(Homo sapiens (Human))
BDBM346358
PNG
(US10202377, Compound 448)
PDB

KEGG

UniProtKB/SwissProt

B.MOAD
antibodypedia
GoogleScholar
AffyNet 
UniChem
Article
n/an/an/an/a 9n/an/an/an/a



Boehringer Ingelheim Pharmaceuticals Inc.





J Med Chem 46: 4676-86 (2003)

More data for this
Ligand-Target Pair
TGF-beta receptor type I


(Homo sapiens (Human))
BDBM346365
PNG
(US10202377, Compound 939)
PDB

KEGG

UniProtKB/SwissProt

B.MOAD
antibodypedia
GoogleScholar
AffyNet 
UniChem
Article
n/an/an/an/a 9n/an/an/an/a



Boehringer Ingelheim Pharmaceuticals Inc.





J Med Chem 46: 4676-86 (2003)

More data for this
Ligand-Target Pair
TGF-beta receptor type I


(Homo sapiens (Human))
BDBM346379
PNG
(US10202377, Compound 953)
PDB

KEGG

UniProtKB/SwissProt

B.MOAD
antibodypedia
GoogleScholar
AffyNet 
UniChem
Article
n/an/an/an/a 9n/an/an/an/a



Boehringer Ingelheim Pharmaceuticals Inc.





J Med Chem 46: 4676-86 (2003)

More data for this
Ligand-Target Pair
TGF-beta receptor type I


(Homo sapiens (Human))
BDBM346271
PNG
(US10202377, Compound 13)
PDB

KEGG

UniProtKB/SwissProt

B.MOAD
antibodypedia
GoogleScholar
AffyNet 
UniChem
Article
n/an/an/an/a 9n/an/an/an/a



Boehringer Ingelheim Pharmaceuticals Inc.





J Med Chem 46: 4676-86 (2003)

More data for this
Ligand-Target Pair
TGF-beta receptor type I


(Homo sapiens (Human))
BDBM346272
PNG
(US10202377, Compound 20)
PDB

KEGG

UniProtKB/SwissProt

B.MOAD
antibodypedia
GoogleScholar
AffyNet 
UniChem
Article
n/an/an/an/a 10n/an/an/an/a



Boehringer Ingelheim Pharmaceuticals Inc.





J Med Chem 46: 4676-86 (2003)

More data for this
Ligand-Target Pair
TGF-beta receptor type I


(Homo sapiens (Human))
BDBM50238070
PNG
(CHEMBL4069101)
PDB

KEGG

UniProtKB/SwissProt

B.MOAD
antibodypedia
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem

Patents

n/an/an/an/a 13n/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
TGF-beta receptor type I


(Homo sapiens (Human))
BDBM346342
PNG
(US10202377, Compound 373)
PDB

KEGG

UniProtKB/SwissProt

B.MOAD
antibodypedia
GoogleScholar
AffyNet 
UniChem
Article
n/an/an/an/a 14n/an/an/an/a



Boehringer Ingelheim Pharmaceuticals Inc.





J Med Chem 46: 4676-86 (2003)

More data for this
Ligand-Target Pair
TGF-beta receptor type I


(Homo sapiens (Human))
BDBM50238095
PNG
(CHEMBL4082868)
PDB

KEGG

UniProtKB/SwissProt

B.MOAD
antibodypedia
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
n/an/an/an/a 16n/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
TGF-beta receptor type I


(Homo sapiens (Human))
BDBM346270
PNG
(US10202377, Compound 7)
PDB

KEGG

UniProtKB/SwissProt

B.MOAD
antibodypedia
GoogleScholar
AffyNet 
UniChem
Article
n/an/an/an/a 17n/an/an/an/a



Boehringer Ingelheim Pharmaceuticals Inc.





J Med Chem 46: 4676-86 (2003)

More data for this
Ligand-Target Pair
TGF-beta receptor type I


(Homo sapiens (Human))
BDBM21513
PNG
(7-[3-(1-methylpyrrolidin-2-yl)propoxy]-4-[2-(pyrid...)
Show SMILES CN1CCCC1CCCOc1ccc2c(ccnc2c1)-c1c2CCCn2nc1-c1ccccn1
Show InChI InChI=1S/C28H31N5O/c1-32-16-4-7-20(32)8-6-18-34-21-11-12-22-23(13-15-30-25(22)19-21)27-26-10-5-17-33(26)31-28(27)24-9-2-3-14-29-24/h2-3,9,11-15,19-20H,4-8,10,16-18H2,1H3
PDB

KEGG

UniProtKB/SwissProt

B.MOAD
antibodypedia
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
PubMed
n/an/a 72n/a 17n/an/a7.530



Lilly Research Laboratories



Assay Description
The kinase activity was assayed by the autophosphorylation reaction of ALK5 (T204D) in the presence of 4 uM ATP and [33P]-gamma-ATP. After incubation...


J Med Chem 51: 2302-2306 (2008)

More data for this
Ligand-Target Pair
TGF-beta receptor type I


(Homo sapiens (Human))
BDBM35941
PNG
(4-pyridinoxy-2-anilinopyridine-based compound, 5)
Show SMILES COc1cc(Nc2cc(Oc3ccc(C)nc3-c3ccccn3)ccn2)cc(OC)c1OC
Show InChI InChI=1S/C25H24N4O4/c1-16-8-9-20(24(28-16)19-7-5-6-11-26-19)33-18-10-12-27-23(15-18)29-17-13-21(30-2)25(32-4)22(14-17)31-3/h5-15H,1-4H3,(H,27,29)
PDB

KEGG

UniProtKB/SwissProt

B.MOAD
antibodypedia
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
PubMed
n/an/a 13n/a 20n/an/a7.423



AstraZeneca



Assay Description
A fluorescence polarization assay was used to assess the ALK5 binding capacity and biochemical activity of compounds. ALK5 protein was added to each ...


J Med Chem 52: 7901-5 (2009)

More data for this
Ligand-Target Pair
TGF-beta receptor type I


(Homo sapiens (Human))
BDBM50238056
PNG
(CHEMBL4060987)
PDB

KEGG

UniProtKB/SwissProt

B.MOAD
antibodypedia
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
n/an/an/an/a 20n/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
TGF-beta receptor type I


(Homo sapiens (Human))
BDBM50238058
PNG
(CHEMBL4087735)
PDB

KEGG

UniProtKB/SwissProt

B.MOAD
antibodypedia
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
n/an/an/an/a 20n/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
TGF-beta receptor type I


(Homo sapiens (Human))
BDBM346345
PNG
(US10202377, Compound 385)
PDB

KEGG

UniProtKB/SwissProt

B.MOAD
antibodypedia
GoogleScholar
AffyNet 
UniChem
Article
n/an/an/an/a 20n/an/an/an/a



Boehringer Ingelheim Pharmaceuticals Inc.





J Med Chem 46: 4676-86 (2003)

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Ligand-Target Pair
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