Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kcal/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Bombesin receptor subtype-3 (RAT) | BDBM50336889 ((2S)-1,1,1-trifluoro-2-[4-(1H-pyrazol-1-yl)phenyl]...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 2.20 | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Agonist activity at rat BRS-3 expressed in HEK293AEQ cells assessed as induction of intracellular calcium mobilization by aequorin bioluminescence as... | ACS Med Chem Lett 2: 43-47 (2011) Article DOI: 10.1021/ml100196d BindingDB Entry DOI: 10.7270/Q26D5T81 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bombesin receptor subtype-3 (RAT) | BDBM50317453 (CHEMBL1098836 | N-(7-benzyl-5-(piperidin-1-yl)-6,7...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 63 | n/a | n/a | n/a | n/a |
AMRI Curated by ChEMBL | Assay Description Agonist activity at rat BRS3 expressed in HEK293AEQ cells after 10 mins by aequorin bioluminescence assay | Bioorg Med Chem Lett 20: 2785-9 (2010) Article DOI: 10.1016/j.bmcl.2010.03.065 BindingDB Entry DOI: 10.7270/Q2NZ88K4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bombesin receptor subtype-3 (RAT) | BDBM50317454 (CHEMBL1096193 | N-(7-benzyl-5-(piperidin-1-yl)-6,7...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 99 | n/a | n/a | n/a | n/a |
AMRI Curated by ChEMBL | Assay Description Agonist activity at rat BRS3 expressed in HEK293AEQ cells after 10 mins by aequorin bioluminescence assay | Bioorg Med Chem Lett 20: 2785-9 (2010) Article DOI: 10.1016/j.bmcl.2010.03.065 BindingDB Entry DOI: 10.7270/Q2NZ88K4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bombesin receptor subtype-3 (RAT) | BDBM50317455 (CHEMBL1099123 | N-(7-benzyl-5-(piperidin-1-yl)-6,7...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 123 | n/a | n/a | n/a | n/a |
AMRI Curated by ChEMBL | Assay Description Agonist activity at rat BRS3 expressed in HEK293AEQ cells after 10 mins by aequorin bioluminescence assay | Bioorg Med Chem Lett 20: 2785-9 (2010) Article DOI: 10.1016/j.bmcl.2010.03.065 BindingDB Entry DOI: 10.7270/Q2NZ88K4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bombesin receptor subtype-3 (RAT) | BDBM50317456 (CHEMBL1099122 | N-(7-benzyl-5-(piperidin-1-yl)-6,7...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 129 | n/a | n/a | n/a | n/a |
AMRI Curated by ChEMBL | Assay Description Agonist activity at rat BRS3 expressed in HEK293AEQ cells after 10 mins by aequorin bioluminescence assay | Bioorg Med Chem Lett 20: 2785-9 (2010) Article DOI: 10.1016/j.bmcl.2010.03.065 BindingDB Entry DOI: 10.7270/Q2NZ88K4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bombesin receptor subtype-3 (RAT) | BDBM50313710 (4'-(2-(5-butyl-1H-imidazol-2-yl)-5-hydroxypentyl)b...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 174 | n/a | n/a | n/a | n/a |
Merck Research Laboratories Curated by ChEMBL | Assay Description Agonistic activity at rat BRS3 expressed in HEK293AEO at 10 uM by aequorin bioluminescence assay | Bioorg Med Chem Lett 20: 1913-7 (2010) Article DOI: 10.1016/j.bmcl.2010.01.154 BindingDB Entry DOI: 10.7270/Q2M045KD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bombesin receptor subtype-3 (RAT) | BDBM50317447 (CHEMBL1099135 | N-(7-benzyl-5-(piperidin-1-yl)-6,7...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 212 | n/a | n/a | n/a | n/a |
AMRI Curated by ChEMBL | Assay Description Agonist activity at rat BRS3 expressed in HEK293AEQ cells after 10 mins by aequorin bioluminescence assay | Bioorg Med Chem Lett 20: 2785-9 (2010) Article DOI: 10.1016/j.bmcl.2010.03.065 BindingDB Entry DOI: 10.7270/Q2NZ88K4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bombesin receptor subtype-3 (RAT) | BDBM50317466 (7-(2-chlorobenzyl)-5-(piperidin-1-yl)-6,7,8,9-tetr...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 342 | n/a | n/a | n/a | n/a |
AMRI Curated by ChEMBL | Assay Description Agonist activity at rat BRS3 expressed in HEK293AEQ cells after 10 mins by aequorin bioluminescence assay | Bioorg Med Chem Lett 20: 2785-9 (2010) Article DOI: 10.1016/j.bmcl.2010.03.065 BindingDB Entry DOI: 10.7270/Q2NZ88K4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bombesin receptor subtype-3 (RAT) | BDBM50317467 (5-(Piperidin-1-yl)-7-(pyridin-2-ylmethyl)-6,7,8,9-...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 346 | n/a | n/a | n/a | n/a |
AMRI Curated by ChEMBL | Assay Description Agonist activity at rat BRS3 expressed in HEK293AEQ cells after 10 mins by aequorin bioluminescence assay | Bioorg Med Chem Lett 20: 2785-9 (2010) Article DOI: 10.1016/j.bmcl.2010.03.065 BindingDB Entry DOI: 10.7270/Q2NZ88K4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bombesin receptor subtype-3 (RAT) | BDBM50317448 (7-Benzyl-5-(piperidin-1-yl)-6,7,8,9-tetrahydro-3H-...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 380 | n/a | n/a | n/a | n/a |
AMRI Curated by ChEMBL | Assay Description Agonist activity at rat BRS3 expressed in HEK293AEQ cells after 10 mins by aequorin bioluminescence assay | Bioorg Med Chem Lett 20: 2785-9 (2010) Article DOI: 10.1016/j.bmcl.2010.03.065 BindingDB Entry DOI: 10.7270/Q2NZ88K4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bombesin receptor subtype-3 (RAT) | BDBM50317462 (7-(benzo[d][1,3]dioxol-5-ylmethyl)-5-(piperidin-1-...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 402 | n/a | n/a | n/a | n/a |
AMRI Curated by ChEMBL | Assay Description Agonist activity at rat BRS3 expressed in HEK293AEQ cells after 10 mins by aequorin bioluminescence assay | Bioorg Med Chem Lett 20: 2785-9 (2010) Article DOI: 10.1016/j.bmcl.2010.03.065 BindingDB Entry DOI: 10.7270/Q2NZ88K4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bombesin receptor subtype-3 (RAT) | BDBM50317451 (CHEMBL1098838 | N-(7-benzyl-5-(piperidin-1-yl)-6,7...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 413 | n/a | n/a | n/a | n/a |
AMRI Curated by ChEMBL | Assay Description Agonist activity at rat BRS3 expressed in HEK293AEQ cells after 10 mins by aequorin bioluminescence assay | Bioorg Med Chem Lett 20: 2785-9 (2010) Article DOI: 10.1016/j.bmcl.2010.03.065 BindingDB Entry DOI: 10.7270/Q2NZ88K4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bombesin receptor subtype-3 (RAT) | BDBM50317452 (CHEMBL1098837 | N-(7-Benzyl-5-(piperidin-1-yl)-6,7...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 433 | n/a | n/a | n/a | n/a |
AMRI Curated by ChEMBL | Assay Description Agonist activity at rat BRS3 expressed in HEK293AEQ cells after 10 mins by aequorin bioluminescence assay | Bioorg Med Chem Lett 20: 2785-9 (2010) Article DOI: 10.1016/j.bmcl.2010.03.065 BindingDB Entry DOI: 10.7270/Q2NZ88K4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bombesin receptor subtype-3 (RAT) | BDBM50317446 (7-benzyl-N-ethyl-5-(piperidin-1-yl)-6,7,8,9-tetrah...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 471 | n/a | n/a | n/a | n/a |
AMRI Curated by ChEMBL | Assay Description Agonist activity at rat BRS3 expressed in HEK293AEQ cells after 10 mins by aequorin bioluminescence assay | Bioorg Med Chem Lett 20: 2785-9 (2010) Article DOI: 10.1016/j.bmcl.2010.03.065 BindingDB Entry DOI: 10.7270/Q2NZ88K4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bombesin receptor subtype-3 (RAT) | BDBM50317476 (7-benzyl-5-(4-fluoropiperidin-1-yl)-6,7,8,9-tetrah...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 481 | n/a | n/a | n/a | n/a |
AMRI Curated by ChEMBL | Assay Description Agonist activity at rat BRS3 expressed in HEK293AEQ cells after 10 mins by aequorin bioluminescence assay | Bioorg Med Chem Lett 20: 2785-9 (2010) Article DOI: 10.1016/j.bmcl.2010.03.065 BindingDB Entry DOI: 10.7270/Q2NZ88K4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bombesin receptor subtype-3 (RAT) | BDBM50317445 (7-benzyl-N-neopentyl-5-(piperidin-1-yl)-6,7,8,9-te...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 680 | n/a | n/a | n/a | n/a |
AMRI Curated by ChEMBL | Assay Description Agonist activity at rat BRS3 expressed in HEK293AEQ cells after 10 mins by aequorin bioluminescence assay | Bioorg Med Chem Lett 20: 2785-9 (2010) Article DOI: 10.1016/j.bmcl.2010.03.065 BindingDB Entry DOI: 10.7270/Q2NZ88K4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bombesin receptor subtype-3 (RAT) | BDBM50317443 (1-(1-amino-7-benzyl-5-(piperidin-1-yl)-6,7,8,9-tet...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 759 | n/a | n/a | n/a | n/a |
AMRI Curated by ChEMBL | Assay Description Agonist activity at rat BRS3 expressed in HEK293AEQ cells after 10 mins by aequorin bioluminescence assay | Bioorg Med Chem Lett 20: 2785-9 (2010) Article DOI: 10.1016/j.bmcl.2010.03.065 BindingDB Entry DOI: 10.7270/Q2NZ88K4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bombesin receptor subtype-3 (RAT) | BDBM50317477 (7-benzyl-5-(4-methylpiperidin-1-yl)-6,7,8,9-tetrah...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 854 | n/a | n/a | n/a | n/a |
AMRI Curated by ChEMBL | Assay Description Agonist activity at rat BRS3 expressed in HEK293AEQ cells after 10 mins by aequorin bioluminescence assay | Bioorg Med Chem Lett 20: 2785-9 (2010) Article DOI: 10.1016/j.bmcl.2010.03.065 BindingDB Entry DOI: 10.7270/Q2NZ88K4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bombesin receptor subtype-3 (RAT) | BDBM50317449 (7-benzyl-5-(pyrrolidin-1-yl)-6,7,8,9-tetrahydro-3H...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 965 | n/a | n/a | n/a | n/a |
AMRI Curated by ChEMBL | Assay Description Agonist activity at rat BRS3 expressed in HEK293AEQ cells after 10 mins by aequorin bioluminescence assay | Bioorg Med Chem Lett 20: 2785-9 (2010) Article DOI: 10.1016/j.bmcl.2010.03.065 BindingDB Entry DOI: 10.7270/Q2NZ88K4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bombesin receptor subtype-3 (RAT) | BDBM50317459 (7-neopentyl-5-(piperidin-1-yl)-6,7,8,9-tetrahydro-...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 1.06E+3 | n/a | n/a | n/a | n/a |
AMRI Curated by ChEMBL | Assay Description Agonist activity at rat BRS3 expressed in HEK293AEQ cells after 10 mins by aequorin bioluminescence assay | Bioorg Med Chem Lett 20: 2785-9 (2010) Article DOI: 10.1016/j.bmcl.2010.03.065 BindingDB Entry DOI: 10.7270/Q2NZ88K4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bombesin receptor subtype-3 (RAT) | BDBM50317450 (5-(azepan-1-yl)-7-benzyl-6,7,8,9-tetrahydro-3H-pyr...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 1.44E+3 | n/a | n/a | n/a | n/a |
AMRI Curated by ChEMBL | Assay Description Agonist activity at rat BRS3 expressed in HEK293AEQ cells after 10 mins by aequorin bioluminescence assay | Bioorg Med Chem Lett 20: 2785-9 (2010) Article DOI: 10.1016/j.bmcl.2010.03.065 BindingDB Entry DOI: 10.7270/Q2NZ88K4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bombesin receptor subtype-3 (RAT) | BDBM50317475 (7-benzyl-5-morpholino-6,7,8,9-tetrahydro-3H-pyrazo...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 3.56E+3 | n/a | n/a | n/a | n/a |
AMRI Curated by ChEMBL | Assay Description Agonist activity at rat BRS3 expressed in HEK293AEQ cells after 10 mins by aequorin bioluminescence assay | Bioorg Med Chem Lett 20: 2785-9 (2010) Article DOI: 10.1016/j.bmcl.2010.03.065 BindingDB Entry DOI: 10.7270/Q2NZ88K4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bombesin receptor subtype-3 (RAT) | BDBM50415868 (CHEMBL1199153) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 3.86E+3 | n/a | n/a | n/a | n/a |
AMRI Curated by ChEMBL | Assay Description Agonist activity at rat BRS3 expressed in HEK293AEQ cells after 10 mins by aequorin bioluminescence assay | Bioorg Med Chem Lett 20: 2785-9 (2010) Article DOI: 10.1016/j.bmcl.2010.03.065 BindingDB Entry DOI: 10.7270/Q2NZ88K4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bombesin receptor subtype-3 (RAT) | BDBM50317444 (7-benzyl-3-methyl-5-(piperidin-1-yl)-6,7,8,9-tetra...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 6.06E+3 | n/a | n/a | n/a | n/a |
AMRI Curated by ChEMBL | Assay Description Agonist activity at rat BRS3 expressed in HEK293AEQ cells after 10 mins by aequorin bioluminescence assay | Bioorg Med Chem Lett 20: 2785-9 (2010) Article DOI: 10.1016/j.bmcl.2010.03.065 BindingDB Entry DOI: 10.7270/Q2NZ88K4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bombesin receptor subtype-3 (RAT) | BDBM50317471 (7-benzyl-N5-isopropyl-6,7,8,9-tetrahydro-3H-pyrazo...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 7.65E+3 | n/a | n/a | n/a | n/a |
AMRI Curated by ChEMBL | Assay Description Agonist activity at rat BRS3 expressed in HEK293AEQ cells after 10 mins by aequorin bioluminescence assay | Bioorg Med Chem Lett 20: 2785-9 (2010) Article DOI: 10.1016/j.bmcl.2010.03.065 BindingDB Entry DOI: 10.7270/Q2NZ88K4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bombesin receptor subtype-3 (RAT) | BDBM50317458 (7-phenethyl-5-(piperidin-1-yl)-6,7,8,9-tetrahydro-...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 7.91E+3 | n/a | n/a | n/a | n/a |
AMRI Curated by ChEMBL | Assay Description Agonist activity at rat BRS3 expressed in HEK293AEQ cells after 10 mins by aequorin bioluminescence assay | Bioorg Med Chem Lett 20: 2785-9 (2010) Article DOI: 10.1016/j.bmcl.2010.03.065 BindingDB Entry DOI: 10.7270/Q2NZ88K4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bombesin receptor subtype-3 (RAT) | BDBM50317472 (7-benzyl-N5,N5-dimethyl-6,7,8,9-tetrahydro-3H-pyra...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 8.95E+3 | n/a | n/a | n/a | n/a |
AMRI Curated by ChEMBL | Assay Description Agonist activity at rat BRS3 expressed in HEK293AEQ cells after 10 mins by aequorin bioluminescence assay | Bioorg Med Chem Lett 20: 2785-9 (2010) Article DOI: 10.1016/j.bmcl.2010.03.065 BindingDB Entry DOI: 10.7270/Q2NZ88K4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bombesin receptor subtype-3 (RAT) | BDBM50317473 (7-benzyl-5-(4-methylpiperazin-1-yl)-6,7,8,9-tetrah...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 1.00E+4 | n/a | n/a | n/a | n/a |
AMRI Curated by ChEMBL | Assay Description Agonist activity at rat BRS3 expressed in HEK293AEQ cells after 10 mins by aequorin bioluminescence assay | Bioorg Med Chem Lett 20: 2785-9 (2010) Article DOI: 10.1016/j.bmcl.2010.03.065 BindingDB Entry DOI: 10.7270/Q2NZ88K4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bombesin receptor subtype-3 (RAT) | BDBM50317474 (7-benzyl-5-(piperazin-1-yl)-6,7,8,9-tetrahydro-3H-...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 1.00E+4 | n/a | n/a | n/a | n/a |
AMRI Curated by ChEMBL | Assay Description Agonist activity at rat BRS3 expressed in HEK293AEQ cells after 10 mins by aequorin bioluminescence assay | Bioorg Med Chem Lett 20: 2785-9 (2010) Article DOI: 10.1016/j.bmcl.2010.03.065 BindingDB Entry DOI: 10.7270/Q2NZ88K4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bombesin receptor subtype-3 (RAT) | BDBM50317478 (5-(azocan-1-yl)-7-benzyl-6,7,8,9-tetrahydro-3H-pyr...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 1.00E+4 | n/a | n/a | n/a | n/a |
AMRI Curated by ChEMBL | Assay Description Agonist activity at rat BRS3 expressed in HEK293AEQ cells after 10 mins by aequorin bioluminescence assay | Bioorg Med Chem Lett 20: 2785-9 (2010) Article DOI: 10.1016/j.bmcl.2010.03.065 BindingDB Entry DOI: 10.7270/Q2NZ88K4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bombesin receptor subtype-3 (RAT) | BDBM50317460 (7-isobutyl-5-(piperidin-1-yl)-6,7,8,9-tetrahydro-3...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 1.00E+4 | n/a | n/a | n/a | n/a |
AMRI Curated by ChEMBL | Assay Description Agonist activity at rat BRS3 expressed in HEK293AEQ cells after 10 mins by aequorin bioluminescence assay | Bioorg Med Chem Lett 20: 2785-9 (2010) Article DOI: 10.1016/j.bmcl.2010.03.065 BindingDB Entry DOI: 10.7270/Q2NZ88K4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bombesin receptor subtype-3 (RAT) | BDBM50317469 (7-benzyl-N5-phenyl-6,7,8,9-tetrahydro-3H-pyrazolo[...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 1.00E+4 | n/a | n/a | n/a | n/a |
AMRI Curated by ChEMBL | Assay Description Agonist activity at rat BRS3 expressed in HEK293AEQ cells after 10 mins by aequorin bioluminescence assay | Bioorg Med Chem Lett 20: 2785-9 (2010) Article DOI: 10.1016/j.bmcl.2010.03.065 BindingDB Entry DOI: 10.7270/Q2NZ88K4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bombesin receptor subtype-3 (RAT) | BDBM50378777 (CHEMBL1204083) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a |
AMRI Curated by ChEMBL | Assay Description Agonist activity at rat BRS3 expressed in HEK293AEQ cells after 10 mins by aequorin bioluminescence assay | Bioorg Med Chem Lett 20: 2785-9 (2010) Article DOI: 10.1016/j.bmcl.2010.03.065 BindingDB Entry DOI: 10.7270/Q2NZ88K4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bombesin receptor subtype-3 (RAT) | BDBM50317457 (7-(4-Fluorobenzoyl)-5-(piperidin-1-yl)-6,7,8,9-tet...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a |
AMRI Curated by ChEMBL | Assay Description Agonist activity at rat BRS3 expressed in HEK293AEQ cells after 10 mins by aequorin bioluminescence assay | Bioorg Med Chem Lett 20: 2785-9 (2010) Article DOI: 10.1016/j.bmcl.2010.03.065 BindingDB Entry DOI: 10.7270/Q2NZ88K4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bombesin receptor subtype-3 (RAT) | BDBM50317464 (7-(4-methoxybenzyl)-5-(piperidin-1-yl)-6,7,8,9-tet...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 1.00E+4 | n/a | n/a | n/a | n/a |
AMRI Curated by ChEMBL | Assay Description Agonist activity at rat BRS3 expressed in HEK293AEQ cells after 10 mins by aequorin bioluminescence assay | Bioorg Med Chem Lett 20: 2785-9 (2010) Article DOI: 10.1016/j.bmcl.2010.03.065 BindingDB Entry DOI: 10.7270/Q2NZ88K4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bombesin receptor subtype-3 (RAT) | BDBM50317463 (5-(piperidin-1-yl)-7-(3-(trifluoromethyl)benzyl)-6...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 1.00E+4 | n/a | n/a | n/a | n/a |
AMRI Curated by ChEMBL | Assay Description Agonist activity at rat BRS3 expressed in HEK293AEQ cells after 10 mins by aequorin bioluminescence assay | Bioorg Med Chem Lett 20: 2785-9 (2010) Article DOI: 10.1016/j.bmcl.2010.03.065 BindingDB Entry DOI: 10.7270/Q2NZ88K4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bombesin receptor subtype-3 (RAT) | BDBM50317461 (7-(cyclohexylmethyl)-5-(piperidin-1-yl)-6,7,8,9-te...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 1.00E+4 | n/a | n/a | n/a | n/a |
AMRI Curated by ChEMBL | Assay Description Agonist activity at rat BRS3 expressed in HEK293AEQ cells after 10 mins by aequorin bioluminescence assay | Bioorg Med Chem Lett 20: 2785-9 (2010) Article DOI: 10.1016/j.bmcl.2010.03.065 BindingDB Entry DOI: 10.7270/Q2NZ88K4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bombesin receptor subtype-3 (RAT) | BDBM50317470 (7-benzyl-N5-cyclohexyl-6,7,8,9-tetrahydro-3H-pyraz...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 1.00E+4 | n/a | n/a | n/a | n/a |
AMRI Curated by ChEMBL | Assay Description Agonist activity at rat BRS3 expressed in HEK293AEQ cells after 10 mins by aequorin bioluminescence assay | Bioorg Med Chem Lett 20: 2785-9 (2010) Article DOI: 10.1016/j.bmcl.2010.03.065 BindingDB Entry DOI: 10.7270/Q2NZ88K4 | |||||||||||
More data for this Ligand-Target Pair |