Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kcal/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Voltage-dependent L-type calcium channel subunit alpha-1C (RAT) | BDBM50283421 (((E)-Azacyclotridec-1-en-2-yl)-(2,2-diphenyl-penty...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article | n/a | n/a | n/a | n/a | 34 | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Binding of [3H]-nitrendipine to calcium channel in rat heart membranes | Bioorg Med Chem Lett 4: 351-354 (1994) Article DOI: 10.1016/S0960-894X(01)80143-8 BindingDB Entry DOI: 10.7270/Q2R78F5H | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Voltage-dependent L-type calcium channel subunit alpha-1C (RAT) | BDBM50283420 (((E)-Azacyclotridec-1-en-2-yl)-((1S,2S)-2-phenyl-c...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article | n/a | n/a | n/a | n/a | 61 | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Binding of [3H]-nitrendipine to calcium channel in rat heart membranes | Bioorg Med Chem Lett 4: 351-354 (1994) Article DOI: 10.1016/S0960-894X(01)80143-8 BindingDB Entry DOI: 10.7270/Q2R78F5H | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Voltage-dependent L-type calcium channel subunit alpha-1C (RAT) | BDBM50283420 (((E)-Azacyclotridec-1-en-2-yl)-((1S,2S)-2-phenyl-c...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article | n/a | n/a | n/a | n/a | 61 | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Binding of [3H]-nitrendipine to calcium channel in rat heart membranes was determined | Bioorg Med Chem Lett 4: 351-354 (1994) Article DOI: 10.1016/S0960-894X(01)80143-8 BindingDB Entry DOI: 10.7270/Q2R78F5H | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Voltage-dependent L-type calcium channel subunit alpha-1C (RAT) | BDBM50516235 (CHEMBL4563408) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a |
RTI International Curated by ChEMBL | Assay Description Displacement of [3H]nitrendipine from rat brain Cav1.2 dihydropyridine site after 90 mins by scintillation counting analysis | J Med Chem 62: 6330-6345 (2019) Article DOI: 10.1021/acs.jmedchem.9b00727 BindingDB Entry DOI: 10.7270/Q24F1V3D | |||||||||||
More data for this Ligand-Target Pair |