Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kcal/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Substance-K receptor (HAMSTER) | BDBM50366377 (CHEMBL334721 | MEN-10627) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article | n/a | n/a | 0.0790 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Tested for binding affinity of compound against [125I]NKA binding to neurokinin-2 (NK-2) receptor in hamster urinary bladder | Bioorg Med Chem Lett 7: 31-36 (1997) Article DOI: 10.1016/S0960-894X(96)00570-7 BindingDB Entry DOI: 10.7270/Q2KD1ZDC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Substance-K receptor (HAMSTER) | BDBM50001435 (3-Amino-N-[1-(1-{1-[2-(1-{[(1-carbamoyl-2-phenyl-e...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 1 | n/a | n/a | n/a | n/a | n/a | n/a |
Marion Merrell Dow Research Institute Curated by ChEMBL | Assay Description Competitive inhibition of [125I]NKA binding to hamster urinary bladder Tachykinin receptor 2 | J Med Chem 35: 3949-55 (1992) BindingDB Entry DOI: 10.7270/Q2FF3SZB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Substance-K receptor (HAMSTER) | BDBM50001447 (CHEMBL217406 | His-Lys-Thr-Asp-Ser-Phe-Val-Gly-Leu...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL KEGG PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 1 | n/a | n/a | n/a | n/a | n/a | n/a |
Marion Merrell Dow Research Institute Curated by ChEMBL | Assay Description Competitive inhibition of [125I]NKA binding to hamster urinary bladder Tachykinin receptor 2 | J Med Chem 35: 3949-55 (1992) BindingDB Entry DOI: 10.7270/Q2FF3SZB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Substance-K receptor (HAMSTER) | BDBM50079412 ((NKB)Asp-Met-His-Asp-Phe-Phe-Val-Gly-Leu-Met-NH2 |...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 3.60 | n/a | n/a | n/a | n/a | n/a | n/a |
Cambridge University Forvie Site Curated by ChEMBL | Assay Description Inhibitory activity against Tachykinin receptor 2 in membranes prepared from hamster urinary bladder labeled with [125 I] NKA | J Med Chem 39: 1664-75 (1996) Article DOI: 10.1021/jm950892r BindingDB Entry DOI: 10.7270/Q2CJ8F4R | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Substance-K receptor (HAMSTER) | BDBM50001451 (3-Amino-N-(1-{1-[1-({[1-(1-carbamoyl-3-methylsulfa...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 6 | n/a | n/a | n/a | n/a | n/a | n/a |
Marion Merrell Dow Research Institute Curated by ChEMBL | Assay Description Competitive inhibition of [125I]NKA binding to hamster urinary bladder Tachykinin receptor 2 | J Med Chem 35: 3949-55 (1992) BindingDB Entry DOI: 10.7270/Q2FF3SZB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Substance-K receptor (HAMSTER) | BDBM50001437 (3-Amino-N-[1-(1-{1-[({1-[(1-carbamoyl-2-phenyl-eth...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 9 | n/a | n/a | n/a | n/a | n/a | n/a |
Marion Merrell Dow Research Institute Curated by ChEMBL | Assay Description Competitive inhibition of [125I]NKA binding to hamster urinary bladder Tachykinin receptor 2 | J Med Chem 35: 3949-55 (1992) BindingDB Entry DOI: 10.7270/Q2FF3SZB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Substance-K receptor (HAMSTER) | BDBM50001455 (3-Amino-N-(1-{1-[1-(2-{1-[(1-carbamoyl-2-phenyl-et...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 10 | n/a | n/a | n/a | n/a | n/a | n/a |
Marion Merrell Dow Research Institute Curated by ChEMBL | Assay Description Competitive inhibition of [125I]NKA binding to hamster urinary bladder Tachykinin receptor 2 | J Med Chem 35: 3949-55 (1992) BindingDB Entry DOI: 10.7270/Q2FF3SZB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Substance-K receptor (HAMSTER) | BDBM50079412 ((NKB)Asp-Met-His-Asp-Phe-Phe-Val-Gly-Leu-Met-NH2 |...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 18 | n/a | n/a | n/a | n/a | n/a | n/a |
Marion Merrell Dow Research Institute Curated by ChEMBL | Assay Description Competitive inhibition of [125I]NKA binding to hamster urinary bladder Tachykinin receptor 2 | J Med Chem 35: 3949-55 (1992) BindingDB Entry DOI: 10.7270/Q2FF3SZB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Substance-K receptor (HAMSTER) | BDBM50001440 (3-Amino-N-[1-(1-{1-[({1-[(1-carbamoyl-3-methylsulf...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 50 | n/a | n/a | n/a | n/a | n/a | n/a |
Marion Merrell Dow Research Institute Curated by ChEMBL | Assay Description Competitive inhibition of [125I]NKA binding to hamster urinary bladder Tachykinin receptor 2 | J Med Chem 35: 3949-55 (1992) BindingDB Entry DOI: 10.7270/Q2FF3SZB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Substance-K receptor (HAMSTER) | BDBM50001454 (3-Amino-N-{1-[1-(1-{[(1-{[(1-carbamoyl-3-methyl-bu...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 103 | n/a | n/a | n/a | n/a | n/a | n/a |
Marion Merrell Dow Research Institute Curated by ChEMBL | Assay Description Competitive inhibition of [125I]NKA binding to hamster urinary bladder Tachykinin receptor 2 | J Med Chem 35: 3949-55 (1992) BindingDB Entry DOI: 10.7270/Q2FF3SZB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Substance-K receptor (HAMSTER) | BDBM50001442 (3-Amino-N-(1-{1-[1-(2-{1-[(1-carbamoyl-3-methyl-bu...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 108 | n/a | n/a | n/a | n/a | n/a | n/a |
Marion Merrell Dow Research Institute Curated by ChEMBL | Assay Description Competitive inhibition of [125I]NKA binding to hamster urinary bladder Tachykinin receptor 2 | J Med Chem 35: 3949-55 (1992) BindingDB Entry DOI: 10.7270/Q2FF3SZB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Substance-K receptor (HAMSTER) | BDBM50001443 (3-Amino-N-[1-(1-{1-[({1-[(1-carbamoyl-3-methyl-but...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 115 | n/a | n/a | n/a | n/a | n/a | n/a |
Marion Merrell Dow Research Institute Curated by ChEMBL | Assay Description Competitive inhibition of [125I]NKA binding to hamster urinary bladder Tachykinin receptor 2 | J Med Chem 35: 3949-55 (1992) BindingDB Entry DOI: 10.7270/Q2FF3SZB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Substance-K receptor (HAMSTER) | BDBM50001449 (3-Amino-N-(1-{1-[1-({[1-(1-carbamoyl-3-methyl-buty...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 136 | n/a | n/a | n/a | n/a | n/a | n/a |
Marion Merrell Dow Research Institute Curated by ChEMBL | Assay Description Competitive inhibition of [125I]NKA binding to hamster urinary bladder Tachykinin receptor 2 | J Med Chem 35: 3949-55 (1992) BindingDB Entry DOI: 10.7270/Q2FF3SZB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Substance-K receptor (HAMSTER) | BDBM50001450 ((SP)Arg-Pro-Lys-Pro-Gln-Gln-Phe-Phe-Gly-Leu-Met-NH...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 148 | n/a | n/a | n/a | n/a | n/a | n/a |
Marion Merrell Dow Research Institute Curated by ChEMBL | Assay Description Competitive inhibition of [125I]NKA binding to hamster urinary bladder Tachykinin receptor 2 | J Med Chem 35: 3949-55 (1992) BindingDB Entry DOI: 10.7270/Q2FF3SZB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Substance-K receptor (HAMSTER) | BDBM50001444 (3-Amino-N-{1-[1-(1-{[(1-{[(1-carbamoyl-3-methyl-bu...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 162 | n/a | n/a | n/a | n/a | n/a | n/a |
Marion Merrell Dow Research Institute Curated by ChEMBL | Assay Description Competitive inhibition of [125I]NKA binding to hamster urinary bladder Tachykinin receptor 2 | J Med Chem 35: 3949-55 (1992) BindingDB Entry DOI: 10.7270/Q2FF3SZB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Substance-K receptor (HAMSTER) | BDBM50001438 (3-Amino-N-{1-[1-(1-{[(1-{[(1-carbamoyl-3-methyl-bu...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 193 | n/a | n/a | n/a | n/a | n/a | n/a |
Marion Merrell Dow Research Institute Curated by ChEMBL | Assay Description Competitive inhibition of [125I]NKA binding to hamster urinary bladder Tachykinin receptor 2 | J Med Chem 35: 3949-55 (1992) BindingDB Entry DOI: 10.7270/Q2FF3SZB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Substance-K receptor (HAMSTER) | BDBM50001453 (3-Amino-N-{1-[1-(1-{[(1-{[(1-carbamoyl-3-methyl-bu...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 277 | n/a | n/a | n/a | n/a | n/a | n/a |
Marion Merrell Dow Research Institute Curated by ChEMBL | Assay Description Competitive inhibition of [125I]NKA binding to hamster urinary bladder Tachykinin receptor 2 | J Med Chem 35: 3949-55 (1992) BindingDB Entry DOI: 10.7270/Q2FF3SZB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Substance-K receptor (HAMSTER) | BDBM50283253 ((S)-2-[2-((S)-2-{(S)-2-[(S)-2-((S)-2-Acetylamino-4...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article | n/a | n/a | 637 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Concentration producing half-maximal inhibition of specific binding of. [125I]-Neurokinin A to NK-2 receptors in the hamster urinary bladder | Bioorg Med Chem Lett 4: 2263-2266 (1994) Article DOI: 10.1016/0960-894X(94)85022-4 BindingDB Entry DOI: 10.7270/Q2959HHG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Substance-K receptor (HAMSTER) | BDBM50050641 (CHEMBL45340 | PD-161182 | [(R)-2-(2,3-Difluoro-phe...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article | n/a | n/a | 790 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Compound was tested for binding affinity towards Tachykinin receptor 2 binding sites in membranes prepared from hamster urinary bladder using [125I]n... | Bioorg Med Chem Lett 5: 1773-1778 (1995) Article DOI: 10.1016/0960-894X(95)00313-I BindingDB Entry DOI: 10.7270/Q2QF8TCH | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Substance-K receptor (HAMSTER) | BDBM50050641 (CHEMBL45340 | PD-161182 | [(R)-2-(2,3-Difluoro-phe...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 790 | n/a | n/a | n/a | n/a | n/a | n/a |
Cambridge University Forvie Site Curated by ChEMBL | Assay Description Inhibitory activity against Tachykinin receptor 2 in membranes prepared from hamster urinary bladder labeled with [125 I] NKA | J Med Chem 39: 1664-75 (1996) Article DOI: 10.1021/jm950892r BindingDB Entry DOI: 10.7270/Q2CJ8F4R | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Substance-K receptor (HAMSTER) | BDBM50283250 ((S)-2-[2-((S)-2-{(S)-2-[(S)-2-((S)-2-Acetylamino-4...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article | n/a | n/a | 1.37E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Concentration producing half-maximal inhibition of specific binding of. [125I]-Neurokinin A to NK-2 receptors in the hamster urinary bladder | Bioorg Med Chem Lett 4: 2263-2266 (1994) Article DOI: 10.1016/0960-894X(94)85022-4 BindingDB Entry DOI: 10.7270/Q2959HHG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Substance-K receptor (HAMSTER) | BDBM50050652 (CHEMBL47146 | PD-160946 | [(R)-2-(2-Fluoro-phenyl)...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article | n/a | n/a | 1.50E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Compound was tested for binding affinity towards Tachykinin receptor 2 binding sites in membranes prepared from hamster urinary bladder using [125I]n... | Bioorg Med Chem Lett 5: 1773-1778 (1995) Article DOI: 10.1016/0960-894X(95)00313-I BindingDB Entry DOI: 10.7270/Q2QF8TCH | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Substance-K receptor (HAMSTER) | BDBM50050652 (CHEMBL47146 | PD-160946 | [(R)-2-(2-Fluoro-phenyl)...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.50E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Cambridge University Forvie Site Curated by ChEMBL | Assay Description Inhibitory activity against Tachykinin receptor 2 in membranes prepared from hamster urinary bladder labeled with [125 I] NKA | J Med Chem 39: 1664-75 (1996) Article DOI: 10.1021/jm950892r BindingDB Entry DOI: 10.7270/Q2CJ8F4R | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Substance-K receptor (HAMSTER) | BDBM50283257 ((S)-2-[2-((S)-2-{(S)-2-[(S)-2-((S)-2-Acetylamino-4...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article | n/a | n/a | 1.62E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Concentration producing half-maximal inhibition of specific binding of. [125I]-Neurokinin A to NK-2 receptors in the hamster urinary bladder | Bioorg Med Chem Lett 4: 2263-2266 (1994) Article DOI: 10.1016/0960-894X(94)85022-4 BindingDB Entry DOI: 10.7270/Q2959HHG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Substance-K receptor (HAMSTER) | BDBM50001441 (4-(1-{1-[1-({[1-(1-Carbamoyl-3-methyl-butylcarbamo...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 1.65E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Marion Merrell Dow Research Institute Curated by ChEMBL | Assay Description Competitive inhibition of [125I]NKA binding to hamster urinary bladder Tachykinin receptor 2 | J Med Chem 35: 3949-55 (1992) BindingDB Entry DOI: 10.7270/Q2FF3SZB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Substance-K receptor (HAMSTER) | BDBM50283255 ((S)-2-[(5-Oxo-pyrrolidine-2-carbonyl)-amino]-penta...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article | n/a | n/a | 2.90E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Concentration producing half-maximal inhibition of specific binding of. [125I]-Neurokinin A to NK-2 receptors in the hamster urinary bladder | Bioorg Med Chem Lett 4: 2263-2266 (1994) Article DOI: 10.1016/0960-894X(94)85022-4 BindingDB Entry DOI: 10.7270/Q2959HHG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Substance-K receptor (HAMSTER) | BDBM50289801 (CHEMBL292766 | [(S)-2-(1H-Indol-3-yl)-1-phenethylc...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Similars | Article | n/a | n/a | 3.27E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Concentration required for binding affinity to neurokinin (NK2) receptor in hamster urinary bladder | Bioorg Med Chem Lett 7: 1957-1962 (1997) Article DOI: 10.1016/S0960-894X(97)00346-6 BindingDB Entry DOI: 10.7270/Q28W3DSG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Substance-K receptor (HAMSTER) | BDBM50283252 ((S)-2-[2-((S)-2-{(S)-2-[(S)-2-((S)-2-Amino-4-carba...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Similars | Article | n/a | n/a | 3.29E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Concentration producing half-maximal inhibition of specific binding of. [125I]-Neurokinin A to NK-2 receptors in the hamster urinary bladder | Bioorg Med Chem Lett 4: 2263-2266 (1994) Article DOI: 10.1016/0960-894X(94)85022-4 BindingDB Entry DOI: 10.7270/Q2959HHG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Substance-K receptor (HAMSTER) | BDBM50282774 (CHEMBL295301 | {(S)-1-[(R)-1-(8-Carbamoyl-octylcar...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article | n/a | n/a | 5.02E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Binding affinity for NK2 receptor binding sites in membranes prepared from hamster urinary bladder by using [125I]NKA as radioligand | Bioorg Med Chem Lett 4: 1679-1684 (1994) Article DOI: 10.1016/S0960-894X(00)80360-1 BindingDB Entry DOI: 10.7270/Q22V2GMG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Substance-K receptor (HAMSTER) | BDBM50283777 (BDBM50284761 | CHEMBL295022 | CHEMBL32248 | [1-(1-...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article | n/a | n/a | 5.20E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Binding affinity towards Tachykinin receptor 2 using [125I]iodohistidyl-NKA (0.1 nM)) as radioligand | Bioorg Med Chem Lett 5: 1445-1450 (1995) Article DOI: 10.1016/0960-894X(95)00254-Q BindingDB Entry DOI: 10.7270/Q2GX4C27 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Substance-K receptor (HAMSTER) | BDBM50289293 (1N-[1-carbamoyl-2-phenyl-(1S)-ethyl]-2-amino-3-(1H...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article | n/a | n/a | 5.20E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Tested for binding affinity of compound against [125I]NKA binding to neurokinin-2 (NK-2) receptor in hamster urinary bladder | Bioorg Med Chem Lett 7: 31-36 (1997) Article DOI: 10.1016/S0960-894X(96)00570-7 BindingDB Entry DOI: 10.7270/Q2KD1ZDC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Substance-K receptor (HAMSTER) | BDBM50001448 (3-Amino-N-[1-(1-{1-[({[1-(1-carbamoyl-3-methyl-but...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 5.66E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Marion Merrell Dow Research Institute Curated by ChEMBL | Assay Description Competitive inhibition of [125I]NKA binding to hamster urinary bladder Tachykinin receptor 2 | J Med Chem 35: 3949-55 (1992) BindingDB Entry DOI: 10.7270/Q2FF3SZB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Substance-K receptor (HAMSTER) | BDBM50282782 (CHEMBL297327 | {(S)-1-[(R)-1-(8-Hydroxy-octylcarba...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article | n/a | n/a | 6.16E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Binding affinity for NK2 receptor binding sites in membranes prepared from hamster urinary bladder by using [125I]NKA as radioligand | Bioorg Med Chem Lett 4: 1679-1684 (1994) Article DOI: 10.1016/S0960-894X(00)80360-1 BindingDB Entry DOI: 10.7270/Q22V2GMG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Substance-K receptor (HAMSTER) | BDBM50050642 (CHEMBL296014 | {(S)-1-[(R)-1-(8-Hydroxy-octylcarba...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 6.16E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Cambridge University Forvie Site Curated by ChEMBL | Assay Description Inhibitory activity against Tachykinin receptor 2 in membranes prepared from hamster urinary bladder labeled with [125 I] NKA | J Med Chem 39: 1664-75 (1996) Article DOI: 10.1021/jm950892r BindingDB Entry DOI: 10.7270/Q2CJ8F4R | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Substance-K receptor (HAMSTER) | BDBM50050649 (CHEMBL444832 | {(S)-1-[(R)-1-Methyl-2-phenyl-1-(7-...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article | n/a | n/a | 6.54E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Binding affinity for NK2 receptor binding sites in membranes prepared from hamster urinary bladder by using [125I]NKA as radioligand | Bioorg Med Chem Lett 4: 1679-1684 (1994) Article DOI: 10.1016/S0960-894X(00)80360-1 BindingDB Entry DOI: 10.7270/Q22V2GMG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Substance-K receptor (HAMSTER) | BDBM50050649 (CHEMBL444832 | {(S)-1-[(R)-1-Methyl-2-phenyl-1-(7-...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 6.54E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Cambridge University Forvie Site Curated by ChEMBL | Assay Description Inhibitory activity against Tachykinin receptor 2 in membranes prepared from hamster urinary bladder labeled with [125 I] NKA | J Med Chem 39: 1664-75 (1996) Article DOI: 10.1021/jm950892r BindingDB Entry DOI: 10.7270/Q2CJ8F4R | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Substance-K receptor (HAMSTER) | BDBM50283960 (1-Benzyl-3-(1H-indol-3-ylmethyl)-piperidin-4-one |...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article | n/a | n/a | 6.80E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Binding affinity towards Tachykinin receptor 2 in hamster urinary bladder using [125I]-Neurokinin A as radioligand; Value ranges from 4.6-9.0 uM | Bioorg Med Chem Lett 4: 525-530 (1994) Article DOI: 10.1016/0960-894X(94)80030-8 BindingDB Entry DOI: 10.7270/Q2BV7GKD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Substance-K receptor (HAMSTER) | BDBM50283964 (3-Benzyl-1-(3-1H-indol-3-yl-propionyl)-piperidin-4...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article | n/a | n/a | 6.90E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Binding affinity towards Tachykinin receptor 2 in hamster urinary bladder using [125I]-Neurokinin A as radioligand; Value ranges from 2.6-11 uM | Bioorg Med Chem Lett 4: 525-530 (1994) Article DOI: 10.1016/0960-894X(94)80030-8 BindingDB Entry DOI: 10.7270/Q2BV7GKD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Substance-K receptor (HAMSTER) | BDBM50001452 (3-Amino-N-(2-{1-[1-({[1-(1-carbamoyl-3-methyl-buty...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Marion Merrell Dow Research Institute Curated by ChEMBL | Assay Description Competitive inhibition of [125I]NKA binding to hamster urinary bladder Tachykinin receptor 2 | J Med Chem 35: 3949-55 (1992) BindingDB Entry DOI: 10.7270/Q2FF3SZB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Substance-K receptor (HAMSTER) | BDBM50001436 (3-Amino-N-{1-[1-(1-{2-[1-(1-carbamoyl-3-methyl-but...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Marion Merrell Dow Research Institute Curated by ChEMBL | Assay Description Competitive inhibition of [125I]NKA binding to hamster urinary bladder Tachykinin receptor 2 | J Med Chem 35: 3949-55 (1992) BindingDB Entry DOI: 10.7270/Q2FF3SZB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Substance-K receptor (HAMSTER) | BDBM50001446 (3-Amino-N-(1-{1-benzyl-2-[1-({[1-(1-carbamoyl-3-me...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Marion Merrell Dow Research Institute Curated by ChEMBL | Assay Description Competitive inhibition of [125I]NKA binding to hamster urinary bladder Tachykinin receptor 2 | J Med Chem 35: 3949-55 (1992) BindingDB Entry DOI: 10.7270/Q2FF3SZB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Substance-K receptor (HAMSTER) | BDBM50284763 (1-(3-Benzyl-pyrrolidin-1-yl)-2-(1H-indol-3-yl)-eth...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Similars | Article | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Binding affinity towards Tachykinin receptor 2 using [125I]iodohistidyl-NKA (0.1 nM)) as radioligand | Bioorg Med Chem Lett 5: 1445-1450 (1995) Article DOI: 10.1016/0960-894X(95)00254-Q BindingDB Entry DOI: 10.7270/Q2GX4C27 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Substance-K receptor (HAMSTER) | BDBM50366377 (CHEMBL334721 | MEN-10627) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Binding affinity towards Tachykinin receptor 2 using [125I]iodohistidyl-NKA (0.1 nM)) as radioligand | Bioorg Med Chem Lett 5: 1445-1450 (1995) Article DOI: 10.1016/0960-894X(95)00254-Q BindingDB Entry DOI: 10.7270/Q2GX4C27 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Substance-K receptor (HAMSTER) | BDBM50000040 (((2S,3S)-2-Benzhydryl-1-aza-bicyclo[2.2.2]oct-3-yl...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Patents Similars | PubMed | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer, Inc. Curated by ChEMBL | Assay Description Inhibitory activity against [125I]-neurokinin binding to Tachykinin receptor 2 in hamster urinary bladder | J Med Chem 35: 2591-600 (1992) BindingDB Entry DOI: 10.7270/Q2SJ1JJF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Substance-K receptor (HAMSTER) | BDBM50001439 (3-Amino-N-(1-{1-[1-({[1-benzyl-2-(1-carbamoyl-3-me...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Marion Merrell Dow Research Institute Curated by ChEMBL | Assay Description Competitive inhibition of [125I]NKA binding to hamster urinary bladder Tachykinin receptor 2 | J Med Chem 35: 3949-55 (1992) BindingDB Entry DOI: 10.7270/Q2FF3SZB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Substance-K receptor (HAMSTER) | BDBM50284764 (CHEMBL36402 | L-659874 | {(S)-2-[(S)-2-{(S)-2-[(S)...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article | n/a | n/a | 1.98E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Binding affinity towards Tachykinin receptor 2 using [125I]iodohistidyl-NKA (0.1 nM)) as radioligand | Bioorg Med Chem Lett 5: 1445-1450 (1995) Article DOI: 10.1016/0960-894X(95)00254-Q BindingDB Entry DOI: 10.7270/Q2GX4C27 | |||||||||||
More data for this Ligand-Target Pair |