Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kcal/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Small conductance calcium-activated potassium channel protein 1/2/3 (Rattus norvegicus-RAT-Rattus norvegicus (Rat)) | BDBM392076 (US10301272, Example 7/9) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 0.0120 | n/a | n/a | n/a | n/a | n/a | n/a |
Phenex Pharmaceuticals AG Curated by ChEMBL | Assay Description Displacement of [125I]apamin from rat brain SkCa channel after 60 mins by scintillation counting analysis | Bioorg Med Chem Lett 28: 1446-1455 (2018) Article DOI: 10.1016/j.bmcl.2018.03.093 BindingDB Entry DOI: 10.7270/Q27W6FPC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Small conductance calcium-activated potassium channel protein 1/2/3 (Rattus norvegicus-RAT-Rattus norvegicus (Rat)) | BDBM50155248 (CHEMBL3774478) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 0.0160 | n/a | n/a | n/a | n/a | n/a | n/a |
Jagiellonian University Medical College Curated by ChEMBL | Assay Description Displacement of [125I]apamin from rat cerebral cortex small conductance calcium-activated potassium channel | Bioorg Med Chem 24: 1793-810 (2016) Article DOI: 10.1016/j.bmc.2016.03.006 BindingDB Entry DOI: 10.7270/Q2J67JS7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Small conductance calcium-activated potassium channel protein 1 (RAT) | BDBM50260153 (Apamin | CHEMBL525408 | Octadecapeptide venom) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 0.0240 | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Inc. Curated by ChEMBL | Assay Description Inhibition of rat SK Calcium channel | Bioorg Med Chem 18: 7675-99 (2010) Article DOI: 10.1016/j.bmc.2010.07.034 BindingDB Entry DOI: 10.7270/Q2DF6S69 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Small conductance calcium-activated potassium channel protein 1/2/3 (Rattus norvegicus-RAT-Rattus norvegicus (Rat)) | BDBM50092131 (1,7-diazonia-15,21-diazapentacyclo[20.6.2.27,14.08...) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 2 | n/a | n/a | n/a | n/a | n/a | n/a |
Aristotelian University of Thessaloniki Curated by ChEMBL | Assay Description Inhibition of after hyperpolarization (AHP) of cultured rat sympathetic neurons as SKCa channel blocking activity | Bioorg Med Chem Lett 14: 4231-5 (2004) Article DOI: 10.1016/j.bmcl.2004.06.011 BindingDB Entry DOI: 10.7270/Q2FF3W4T | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Small conductance calcium-activated potassium channel protein 1/2/3 (Rattus norvegicus-RAT-Rattus norvegicus (Rat)) | BDBM50061977 (17,25-diazonia-2,9-diazaheptacyclo[23.6.2.24,7.210...) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 3 | n/a | n/a | n/a | n/a | n/a | n/a |
University College London Curated by ChEMBL | Assay Description The blocking of apamin-sensitive [Ca2+]-activated K+ (SKCa) channel was assessed by the compounds ability to inhibit the after-hyperpolarization in c... | J Med Chem 43: 420-31 (2000) Article DOI: 10.1021/jm9902537 BindingDB Entry DOI: 10.7270/Q21V5HQ2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Small conductance calcium-activated potassium channel protein 1/2/3 (Rattus norvegicus-RAT-Rattus norvegicus (Rat)) | BDBM50061977 (17,25-diazonia-2,9-diazaheptacyclo[23.6.2.24,7.210...) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 3 | n/a | n/a | n/a | n/a | n/a | n/a |
Aristotelian University of Thessaloniki Curated by ChEMBL | Assay Description Inhibition of after hyperpolarization (AHP) of cultured rat sympathetic neurons as SKCa channel blocking activity | Bioorg Med Chem Lett 14: 4231-5 (2004) Article DOI: 10.1016/j.bmcl.2004.06.011 BindingDB Entry DOI: 10.7270/Q2FF3W4T | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Small conductance calcium-activated potassium channel protein 1/2/3 (Rattus norvegicus-RAT-Rattus norvegicus (Rat)) | BDBM50474856 (CHEMBL184300) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 9 | n/a | n/a | n/a | n/a | n/a | n/a |
Aristotelian University of Thessaloniki Curated by ChEMBL | Assay Description Inhibition of after hyperpolarization (AHP) of cultured rat sympathetic neurons as SKCa channel blocking activity | Bioorg Med Chem Lett 14: 4231-5 (2004) Article DOI: 10.1016/j.bmcl.2004.06.011 BindingDB Entry DOI: 10.7270/Q2FF3W4T | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Small conductance calcium-activated potassium channel protein 1/2/3 (Rattus norvegicus-RAT-Rattus norvegicus (Rat)) | BDBM50474870 (CHEMBL185146) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 10 | n/a | n/a | n/a | n/a | n/a | n/a |
Aristotelian University of Thessaloniki Curated by ChEMBL | Assay Description Inhibition of after hyperpolarization (AHP) of cultured rat sympathetic neurons as SKCa channel blocking activity | Bioorg Med Chem Lett 14: 4231-5 (2004) Article DOI: 10.1016/j.bmcl.2004.06.011 BindingDB Entry DOI: 10.7270/Q2FF3W4T | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Small conductance calcium-activated potassium channel protein 1/2/3 (Rattus norvegicus-RAT-Rattus norvegicus (Rat)) | BDBM50474869 (CHEMBL181911) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 12 | n/a | n/a | n/a | n/a | n/a | n/a |
Aristotelian University of Thessaloniki Curated by ChEMBL | Assay Description Inhibition of after hyperpolarization (AHP) of cultured rat sympathetic neurons as SKCa channel blocking activity | Bioorg Med Chem Lett 14: 4231-5 (2004) Article DOI: 10.1016/j.bmcl.2004.06.011 BindingDB Entry DOI: 10.7270/Q2FF3W4T | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Small conductance calcium-activated potassium channel protein 1/2/3 (Rattus norvegicus-RAT-Rattus norvegicus (Rat)) | BDBM50474865 (CHEMBL183644) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 15 | n/a | n/a | n/a | n/a | n/a | n/a |
Aristotelian University of Thessaloniki Curated by ChEMBL | Assay Description Inhibition of after hyperpolarization (AHP) of cultured rat sympathetic neurons as SKCa channel blocking activity | Bioorg Med Chem Lett 14: 4231-5 (2004) Article DOI: 10.1016/j.bmcl.2004.06.011 BindingDB Entry DOI: 10.7270/Q2FF3W4T | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Small conductance calcium-activated potassium channel protein 1/2/3 (Rattus norvegicus-RAT-Rattus norvegicus (Rat)) | BDBM50474867 (CHEMBL184858) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 16 | n/a | n/a | n/a | n/a | n/a | n/a |
Aristotelian University of Thessaloniki Curated by ChEMBL | Assay Description Inhibition of after hyperpolarization (AHP) of cultured rat sympathetic neurons as SKCa channel blocking activity | Bioorg Med Chem Lett 14: 4231-5 (2004) Article DOI: 10.1016/j.bmcl.2004.06.011 BindingDB Entry DOI: 10.7270/Q2FF3W4T | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Small conductance calcium-activated potassium channel protein 1/2/3 (Rattus norvegicus-RAT-Rattus norvegicus (Rat)) | BDBM50473100 (CHEMBL344807) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 25 | n/a | n/a | n/a | n/a | n/a | n/a |
University College London Curated by ChEMBL | Assay Description The blocking of apamin-sensitive [Ca2+]-activated K+ (SKCa) channel was assessed by the compounds ability to inhibit the after-hyperpolarization in c... | J Med Chem 43: 420-31 (2000) Article DOI: 10.1021/jm9902537 BindingDB Entry DOI: 10.7270/Q21V5HQ2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Small conductance calcium-activated potassium channel protein 1/2/3 (Rattus norvegicus-RAT-Rattus norvegicus (Rat)) | BDBM50474866 (CHEMBL181912) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 25 | n/a | n/a | n/a | n/a | n/a | n/a |
Aristotelian University of Thessaloniki Curated by ChEMBL | Assay Description Inhibition of after hyperpolarization (AHP) of cultured rat sympathetic neurons as SKCa channel blocking activity | Bioorg Med Chem Lett 14: 4231-5 (2004) Article DOI: 10.1016/j.bmcl.2004.06.011 BindingDB Entry DOI: 10.7270/Q2FF3W4T | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Small conductance calcium-activated potassium channel protein 1/2/3 (Rattus norvegicus-RAT-Rattus norvegicus (Rat)) | BDBM50473103 (CHEMBL430146) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 28 | n/a | n/a | n/a | n/a | n/a | n/a |
University College London Curated by ChEMBL | Assay Description The blocking of apamin-sensitive [Ca2+]-activated K+ (SKCa) channel was assessed by the compounds ability to inhibit the after-hyperpolarization in c... | J Med Chem 43: 420-31 (2000) Article DOI: 10.1021/jm9902537 BindingDB Entry DOI: 10.7270/Q21V5HQ2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Small conductance calcium-activated potassium channel protein 1/2/3 (Rattus norvegicus-RAT-Rattus norvegicus (Rat)) | BDBM50473103 (CHEMBL430146) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 28 | n/a | n/a | n/a | n/a | n/a | n/a |
Aristotelian University of Thessaloniki Curated by ChEMBL | Assay Description Inhibition of after hyperpolarization (AHP) of cultured rat sympathetic neurons as SKCa channel blocking activity | Bioorg Med Chem Lett 14: 4231-5 (2004) Article DOI: 10.1016/j.bmcl.2004.06.011 BindingDB Entry DOI: 10.7270/Q2FF3W4T | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Small conductance calcium-activated potassium channel protein 1/2/3 (Rattus norvegicus-RAT-Rattus norvegicus (Rat)) | BDBM50474868 (CHEMBL184891) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 30 | n/a | n/a | n/a | n/a | n/a | n/a |
Aristotelian University of Thessaloniki Curated by ChEMBL | Assay Description Inhibition of after hyperpolarization (AHP) of cultured rat sympathetic neurons as SKCa channel blocking activity | Bioorg Med Chem Lett 14: 4231-5 (2004) Article DOI: 10.1016/j.bmcl.2004.06.011 BindingDB Entry DOI: 10.7270/Q2FF3W4T | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Small conductance calcium-activated potassium channel protein 1/2/3 (Rattus norvegicus-RAT-Rattus norvegicus (Rat)) | BDBM50474871 (CHEMBL182716) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 31 | n/a | n/a | n/a | n/a | n/a | n/a |
Aristotelian University of Thessaloniki Curated by ChEMBL | Assay Description Inhibition of after hyperpolarization (AHP) of cultured rat sympathetic neurons as SKCa channel blocking activity | Bioorg Med Chem Lett 14: 4231-5 (2004) Article DOI: 10.1016/j.bmcl.2004.06.011 BindingDB Entry DOI: 10.7270/Q2FF3W4T | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Small conductance calcium-activated potassium channel protein 1/2/3 (Rattus norvegicus-RAT-Rattus norvegicus (Rat)) | BDBM50474863 (CHEMBL360624) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 35 | n/a | n/a | n/a | n/a | n/a | n/a |
Aristotelian University of Thessaloniki Curated by ChEMBL | Assay Description Inhibition of after hyperpolarization (AHP) of cultured rat sympathetic neurons as SKCa channel blocking activity | Bioorg Med Chem Lett 14: 4231-5 (2004) Article DOI: 10.1016/j.bmcl.2004.06.011 BindingDB Entry DOI: 10.7270/Q2FF3W4T | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Small conductance calcium-activated potassium channel protein 1/2/3 (Rattus norvegicus-RAT-Rattus norvegicus (Rat)) | BDBM50474872 (CHEMBL1180184) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 40 | n/a | n/a | n/a | n/a | n/a | n/a |
Aristotelian University of Thessaloniki Curated by ChEMBL | Assay Description Inhibition of after hyperpolarization (AHP) of cultured rat sympathetic neurons as SKCa channel blocking activity | Bioorg Med Chem Lett 14: 4231-5 (2004) Article DOI: 10.1016/j.bmcl.2004.06.011 BindingDB Entry DOI: 10.7270/Q2FF3W4T | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Small conductance calcium-activated potassium channel protein 1/2/3 (Rattus norvegicus-RAT-Rattus norvegicus (Rat)) | BDBM50474858 (CHEMBL186139) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 60 | n/a | n/a | n/a | n/a | n/a | n/a |
Aristotelian University of Thessaloniki Curated by ChEMBL | Assay Description Inhibition of after hyperpolarization (AHP) of cultured rat sympathetic neurons as SKCa channel blocking activity | Bioorg Med Chem Lett 14: 4231-5 (2004) Article DOI: 10.1016/j.bmcl.2004.06.011 BindingDB Entry DOI: 10.7270/Q2FF3W4T | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Small conductance calcium-activated potassium channel protein 1/2/3 (Rattus norvegicus-RAT-Rattus norvegicus (Rat)) | BDBM50473097 (CHEMBL136488) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 60 | n/a | n/a | n/a | n/a | n/a | n/a |
University College London Curated by ChEMBL | Assay Description The blocking of apamin-sensitive [Ca2+]-activated K+ (SKCa) channel was assessed by the compounds ability to inhibit the after-hyperpolarization in c... | J Med Chem 43: 420-31 (2000) Article DOI: 10.1021/jm9902537 BindingDB Entry DOI: 10.7270/Q21V5HQ2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Small conductance calcium-activated potassium channel protein 1/2/3 (Rattus norvegicus-RAT-Rattus norvegicus (Rat)) | BDBM50150389 (17,23-diazonia-2,9-diazahexacyclo[21.6.2.24,7.210,...) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 60 | n/a | n/a | n/a | n/a | n/a | n/a |
Aristotelian University of Thessaloniki Curated by ChEMBL | Assay Description Inhibition of after hyperpolarization (AHP) of cultured rat sympathetic neurons as SKCa channel blocking activity | Bioorg Med Chem Lett 14: 4231-5 (2004) Article DOI: 10.1016/j.bmcl.2004.06.011 BindingDB Entry DOI: 10.7270/Q2FF3W4T | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Small conductance calcium-activated potassium channel protein 1/2/3 (Rattus norvegicus-RAT-Rattus norvegicus (Rat)) | BDBM50474859 (CHEMBL185258) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 65 | n/a | n/a | n/a | n/a | n/a | n/a |
Aristotelian University of Thessaloniki Curated by ChEMBL | Assay Description Inhibition of after hyperpolarization (AHP) of cultured rat sympathetic neurons as SKCa channel blocking activity | Bioorg Med Chem Lett 14: 4231-5 (2004) Article DOI: 10.1016/j.bmcl.2004.06.011 BindingDB Entry DOI: 10.7270/Q2FF3W4T | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Small conductance calcium-activated potassium channel protein 1/2/3 (Rattus norvegicus-RAT-Rattus norvegicus (Rat)) | BDBM50473106 (CHEMBL137175) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 70 | n/a | n/a | n/a | n/a | n/a | n/a |
Aristotelian University of Thessaloniki Curated by ChEMBL | Assay Description Inhibition of after hyperpolarization (AHP) of cultured rat sympathetic neurons as SKCa channel blocking activity | Bioorg Med Chem Lett 14: 4231-5 (2004) Article DOI: 10.1016/j.bmcl.2004.06.011 BindingDB Entry DOI: 10.7270/Q2FF3W4T | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Small conductance calcium-activated potassium channel protein 1/2/3 (Rattus norvegicus-RAT-Rattus norvegicus (Rat)) | BDBM50473106 (CHEMBL137175) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 70 | n/a | n/a | n/a | n/a | n/a | n/a |
University College London Curated by ChEMBL | Assay Description The blocking of apamin-sensitive [Ca2+]-activated K+ (SKCa) channel was assessed by the compounds ability to inhibit the after-hyperpolarization in c... | J Med Chem 43: 420-31 (2000) Article DOI: 10.1021/jm9902537 BindingDB Entry DOI: 10.7270/Q21V5HQ2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Small conductance calcium-activated potassium channel protein 1/2/3 (Rattus norvegicus-RAT-Rattus norvegicus (Rat)) | BDBM50084848 (BIs-cyclo(4N-pentyl-1-(4-methylbenzyl)-4-quinolini...) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 80 | n/a | n/a | n/a | n/a | n/a | n/a |
University College London Curated by ChEMBL | Assay Description The blocking of apamin-sensitive [Ca2+]-activated K+ (SKCa) channel was assessed by the compounds ability to inhibit the after-hyperpolarization in c... | J Med Chem 43: 420-31 (2000) Article DOI: 10.1021/jm9902537 BindingDB Entry DOI: 10.7270/Q21V5HQ2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Small conductance calcium-activated potassium channel protein 1/2/3 (Rattus norvegicus-RAT-Rattus norvegicus (Rat)) | BDBM50473094 (CHEMBL137155) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 90 | n/a | n/a | n/a | n/a | n/a | n/a |
University College London Curated by ChEMBL | Assay Description The blocking of apamin-sensitive [Ca2+]-activated K+ (SKCa) channel was assessed by the compounds ability to inhibit the after-hyperpolarization in c... | J Med Chem 43: 420-31 (2000) Article DOI: 10.1021/jm9902537 BindingDB Entry DOI: 10.7270/Q21V5HQ2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Small conductance calcium-activated potassium channel protein 1/2/3 (Rattus norvegicus-RAT-Rattus norvegicus (Rat)) | BDBM50473098 (CHEMBL342213) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 100 | n/a | n/a | n/a | n/a | n/a | n/a |
University College London Curated by ChEMBL | Assay Description The blocking of apamin-sensitive [Ca2+]-activated K+ (SKCa) channel was assessed by the compounds ability to inhibit the after-hyperpolarization in c... | J Med Chem 43: 420-31 (2000) Article DOI: 10.1021/jm9902537 BindingDB Entry DOI: 10.7270/Q21V5HQ2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Small conductance calcium-activated potassium channel protein 1/2/3 (Rattus norvegicus-RAT-Rattus norvegicus (Rat)) | BDBM50084852 (1,14-diazonia-22,33-diazaheptacyclo[32.6.2.214,21....) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 110 | n/a | n/a | n/a | n/a | n/a | n/a |
University College London Curated by ChEMBL | Assay Description The blocking of apamin-sensitive [Ca2+]-activated K+ (SKCa) channel was assessed by the compounds ability to inhibit the after-hyperpolarization in c... | J Med Chem 43: 420-31 (2000) Article DOI: 10.1021/jm9902537 BindingDB Entry DOI: 10.7270/Q21V5HQ2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Small conductance calcium-activated potassium channel protein 1/2/3 (Rattus norvegicus-RAT-Rattus norvegicus (Rat)) | BDBM50473099 (CHEMBL140380) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 120 | n/a | n/a | n/a | n/a | n/a | n/a |
University College London Curated by ChEMBL | Assay Description The blocking of apamin-sensitive [Ca2+]-activated K+ (SKCa) channel was assessed by the compounds ability to inhibit the after-hyperpolarization in c... | J Med Chem 43: 420-31 (2000) Article DOI: 10.1021/jm9902537 BindingDB Entry DOI: 10.7270/Q21V5HQ2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Small conductance calcium-activated potassium channel protein 1/2/3 (Rattus norvegicus-RAT-Rattus norvegicus (Rat)) | BDBM50474857 (CHEMBL185106) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 130 | n/a | n/a | n/a | n/a | n/a | n/a |
Aristotelian University of Thessaloniki Curated by ChEMBL | Assay Description Inhibition of after hyperpolarization (AHP) of cultured rat sympathetic neurons as SKCa channel blocking activity | Bioorg Med Chem Lett 14: 4231-5 (2004) Article DOI: 10.1016/j.bmcl.2004.06.011 BindingDB Entry DOI: 10.7270/Q2FF3W4T | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Small conductance calcium-activated potassium channel protein 1/2/3 (Rattus norvegicus-RAT-Rattus norvegicus (Rat)) | BDBM50473107 (CHEMBL341700) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 130 | n/a | n/a | n/a | n/a | n/a | n/a |
Aristotelian University of Thessaloniki Curated by ChEMBL | Assay Description Inhibition of after hyperpolarization (AHP) of cultured rat sympathetic neurons as SKCa channel blocking activity | Bioorg Med Chem Lett 14: 4231-5 (2004) Article DOI: 10.1016/j.bmcl.2004.06.011 BindingDB Entry DOI: 10.7270/Q2FF3W4T | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Small conductance calcium-activated potassium channel protein 1/2/3 (Rattus norvegicus-RAT-Rattus norvegicus (Rat)) | BDBM50473107 (CHEMBL341700) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 130 | n/a | n/a | n/a | n/a | n/a | n/a |
University College London Curated by ChEMBL | Assay Description The blocking of apamin-sensitive [Ca2+]-activated K+ (SKCa) channel was assessed by the compounds ability to inhibit the after-hyperpolarization in c... | J Med Chem 43: 420-31 (2000) Article DOI: 10.1021/jm9902537 BindingDB Entry DOI: 10.7270/Q21V5HQ2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Small conductance calcium-activated potassium channel protein 1/2/3 (Rattus norvegicus-RAT-Rattus norvegicus (Rat)) | BDBM50474862 (CHEMBL425707) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 150 | n/a | n/a | n/a | n/a | n/a | n/a |
Aristotelian University of Thessaloniki Curated by ChEMBL | Assay Description Inhibition of after hyperpolarization (AHP) of cultured rat sympathetic neurons as SKCa channel blocking activity | Bioorg Med Chem Lett 14: 4231-5 (2004) Article DOI: 10.1016/j.bmcl.2004.06.011 BindingDB Entry DOI: 10.7270/Q2FF3W4T | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Small conductance calcium-activated potassium channel protein 1/2/3 (Rattus norvegicus-RAT-Rattus norvegicus (Rat)) | BDBM50474873 (CHEMBL185137) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 150 | n/a | n/a | n/a | n/a | n/a | n/a |
Aristotelian University of Thessaloniki Curated by ChEMBL | Assay Description Inhibition of after hyperpolarization (AHP) of cultured rat sympathetic neurons as SKCa channel blocking activity | Bioorg Med Chem Lett 14: 4231-5 (2004) Article DOI: 10.1016/j.bmcl.2004.06.011 BindingDB Entry DOI: 10.7270/Q2FF3W4T | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Small conductance calcium-activated potassium channel protein 1/2/3 (Rattus norvegicus-RAT-Rattus norvegicus (Rat)) | BDBM50084849 (Bis-quinolinium cyclophane analogue | CHEMBL258254...) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 150 | n/a | n/a | n/a | n/a | n/a | n/a |
University College London Curated by ChEMBL | Assay Description The blocking of apamin-sensitive [Ca2+]-activated K+ (SKCa) channel was assessed by the compounds ability to inhibit the after-hyperpolarization in c... | J Med Chem 43: 420-31 (2000) Article DOI: 10.1021/jm9902537 BindingDB Entry DOI: 10.7270/Q21V5HQ2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Small conductance calcium-activated potassium channel protein 1/2/3 (Rattus norvegicus-RAT-Rattus norvegicus (Rat)) | BDBM50473102 (CHEMBL137266) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 150 | n/a | n/a | n/a | n/a | n/a | n/a |
University College London Curated by ChEMBL | Assay Description The blocking of apamin-sensitive [Ca2+]-activated K+ (SKCa) channel was assessed by the compounds ability to inhibit the after-hyperpolarization in c... | J Med Chem 43: 420-31 (2000) Article DOI: 10.1021/jm9902537 BindingDB Entry DOI: 10.7270/Q21V5HQ2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Small conductance calcium-activated potassium channel protein 1/2/3 (Rattus norvegicus-RAT-Rattus norvegicus (Rat)) | BDBM50084839 (Bis-quinolinium cyclophane analogue | CHEMBL6266 |...) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 170 | n/a | n/a | n/a | n/a | n/a | n/a |
University College London Curated by ChEMBL | Assay Description The blocking of apamin-sensitive [Ca2+]-activated K+ (SKCa) channel was assessed by the compounds ability to inhibit the after-hyperpolarization in c... | J Med Chem 43: 420-31 (2000) Article DOI: 10.1021/jm9902537 BindingDB Entry DOI: 10.7270/Q21V5HQ2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Small conductance calcium-activated potassium channel protein 1/2/3 (Rattus norvegicus-RAT-Rattus norvegicus (Rat)) | BDBM50084851 (Bis-quinolinium cyclophane analogue | CHEMBL266885...) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 180 | n/a | n/a | n/a | n/a | n/a | n/a |
University College London Curated by ChEMBL | Assay Description The blocking of apamin-sensitive [Ca2+]-activated K+ (SKCa) channel was assessed by the compounds ability to inhibit the after-hyperpolarization in c... | J Med Chem 43: 420-31 (2000) Article DOI: 10.1021/jm9902537 BindingDB Entry DOI: 10.7270/Q21V5HQ2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Small conductance calcium-activated potassium channel protein 1/2/3 (Rattus norvegicus-RAT-Rattus norvegicus (Rat)) | BDBM50054105 ((Z)-1.1'-[stilbene-4,4'-diylbis(methylene)]bis(4-a...) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 190 | n/a | n/a | n/a | n/a | n/a | n/a |
University College London Curated by ChEMBL | Assay Description The blocking of apamin-sensitive [Ca2+]-activated K+ (SKCa) channel was assessed by the compounds ability to inhibit the after-hyperpolarization in c... | J Med Chem 43: 420-31 (2000) Article DOI: 10.1021/jm9902537 BindingDB Entry DOI: 10.7270/Q21V5HQ2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Small conductance calcium-activated potassium channel protein 1/2/3 (Rattus norvegicus-RAT-Rattus norvegicus (Rat)) | BDBM50474864 (CHEMBL119859) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 190 | n/a | n/a | n/a | n/a | n/a | n/a |
Aristotelian University of Thessaloniki Curated by ChEMBL | Assay Description Inhibition of after hyperpolarization (AHP) of cultured rat sympathetic neurons as SKCa channel blocking activity | Bioorg Med Chem Lett 14: 4231-5 (2004) Article DOI: 10.1016/j.bmcl.2004.06.011 BindingDB Entry DOI: 10.7270/Q2FF3W4T | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Small conductance calcium-activated potassium channel protein 1/2/3 (Rattus norvegicus-RAT-Rattus norvegicus (Rat)) | BDBM50473108 (CHEMBL137116) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 210 | n/a | n/a | n/a | n/a | n/a | n/a |
University College London Curated by ChEMBL | Assay Description The blocking of apamin-sensitive [Ca2+]-activated K+ (SKCa) channel was assessed by the compounds ability to inhibit the after-hyperpolarization in c... | J Med Chem 43: 420-31 (2000) Article DOI: 10.1021/jm9902537 BindingDB Entry DOI: 10.7270/Q21V5HQ2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Small conductance calcium-activated potassium channel protein 1/2/3 (Rattus norvegicus-RAT-Rattus norvegicus (Rat)) | BDBM50473111 (CHEMBL137256) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 250 | n/a | n/a | n/a | n/a | n/a | n/a |
University College London Curated by ChEMBL | Assay Description The blocking of apamin-sensitive [Ca2+]-activated K+ (SKCa) channel was assessed by the compounds ability to inhibit the after-hyperpolarization in c... | J Med Chem 43: 420-31 (2000) Article DOI: 10.1021/jm9902537 BindingDB Entry DOI: 10.7270/Q21V5HQ2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Small conductance calcium-activated potassium channel protein 1/2/3 (Rattus norvegicus-RAT-Rattus norvegicus (Rat)) | BDBM50473109 (CHEMBL136303) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 260 | n/a | n/a | n/a | n/a | n/a | n/a |
University College London Curated by ChEMBL | Assay Description The blocking of apamin-sensitive [Ca2+]-activated K+ (SKCa) channel was assessed by the compounds ability to inhibit the after-hyperpolarization in c... | J Med Chem 43: 420-31 (2000) Article DOI: 10.1021/jm9902537 BindingDB Entry DOI: 10.7270/Q21V5HQ2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Small conductance calcium-activated potassium channel protein 1/2/3 (Rattus norvegicus-RAT-Rattus norvegicus (Rat)) | BDBM50474861 (CHEMBL185230) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 260 | n/a | n/a | n/a | n/a | n/a | n/a |
Aristotelian University of Thessaloniki Curated by ChEMBL | Assay Description Inhibition of after hyperpolarization (AHP) of cultured rat sympathetic neurons as SKCa channel blocking activity | Bioorg Med Chem Lett 14: 4231-5 (2004) Article DOI: 10.1016/j.bmcl.2004.06.011 BindingDB Entry DOI: 10.7270/Q2FF3W4T | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Small conductance calcium-activated potassium channel protein 1/2/3 (Rattus norvegicus-RAT-Rattus norvegicus (Rat)) | BDBM50473096 (CHEMBL434234) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 280 | n/a | n/a | n/a | n/a | n/a | n/a |
University College London Curated by ChEMBL | Assay Description The blocking of apamin-sensitive [Ca2+]-activated K+ (SKCa) channel was assessed by the compounds ability to inhibit the after-hyperpolarization in c... | J Med Chem 43: 420-31 (2000) Article DOI: 10.1021/jm9902537 BindingDB Entry DOI: 10.7270/Q21V5HQ2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Small conductance calcium-activated potassium channel protein 1/2/3 (Rattus norvegicus-RAT-Rattus norvegicus (Rat)) | BDBM50054098 (1,1'-[biphenyl-3,3'-diylbis(methylene)]-bis(4-amin...) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 290 | n/a | n/a | n/a | n/a | n/a | n/a |
University College London Curated by ChEMBL | Assay Description The blocking of apamin-sensitive [Ca2+]-activated K+ (SKCa) channel was assessed by the compounds ability to inhibit the after-hyperpolarization in c... | J Med Chem 43: 420-31 (2000) Article DOI: 10.1021/jm9902537 BindingDB Entry DOI: 10.7270/Q21V5HQ2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Small conductance calcium-activated potassium channel protein 1/2/3 (Rattus norvegicus-RAT-Rattus norvegicus (Rat)) | BDBM50084846 (1-[7-(4-amino-1-quinoliniumylmethyl)-9H-2-fluoreny...) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 310 | n/a | n/a | n/a | n/a | n/a | n/a |
University College London Curated by ChEMBL | Assay Description The blocking of apamin-sensitive [Ca2+]-activated K+ (SKCa) channel was assessed by the compounds ability to inhibit the after-hyperpolarization in c... | J Med Chem 43: 420-31 (2000) Article DOI: 10.1021/jm9902537 BindingDB Entry DOI: 10.7270/Q21V5HQ2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Small conductance calcium-activated potassium channel protein 1/2/3 (Rattus norvegicus-RAT-Rattus norvegicus (Rat)) | BDBM50473105 (CHEMBL133311) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 360 | n/a | n/a | n/a | n/a | n/a | n/a |
University College London Curated by ChEMBL | Assay Description The blocking of apamin-sensitive [Ca2+]-activated K+ (SKCa) channel was assessed by the compounds ability to inhibit the after-hyperpolarization in c... | J Med Chem 43: 420-31 (2000) Article DOI: 10.1021/jm9902537 BindingDB Entry DOI: 10.7270/Q21V5HQ2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Small conductance calcium-activated potassium channel protein 1/2/3 (Rattus norvegicus-RAT-Rattus norvegicus (Rat)) | BDBM50054103 (1,1'-[biphenyl-4,4'-diylbis(methylene)]-bis(4-amin...) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 380 | n/a | n/a | n/a | n/a | n/a | n/a |
University College London Curated by ChEMBL | Assay Description The blocking of apamin-sensitive [Ca2+]-activated K+ (SKCa) channel was assessed by the compounds ability to inhibit the after-hyperpolarization in c... | J Med Chem 43: 420-31 (2000) Article DOI: 10.1021/jm9902537 BindingDB Entry DOI: 10.7270/Q21V5HQ2 | |||||||||||
More data for this Ligand-Target Pair |
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