Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kcal/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Sliding-clamp-loader large/small subunit (Enterobacteria phage T4 (Bacteriophage T4)) | BDBM36319 (5-nitro-indolyl- 2'-deoxyriboside triphosphate...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | KEGG MMDB PC cid PC sid PDB UniChem Similars | Article PubMed | 4.80E+3 | -7.25 | n/a | n/a | n/a | n/a | n/a | 7.5 | 25 |
Case Western Reserve University | Assay Description ATPase assay contained 10 mM Mg2+, 1uM 13/20 DNA, 500uM (r)NTP or (d)NTP, 500 nM gp45, and 500 nM gp44/62 in T4 buffer. ATPase activity was measured ... | ACS Chem Biol 5: 183-94 (2010) Article DOI: 10.1021/cb900218c BindingDB Entry DOI: 10.7270/Q26M356K | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sliding-clamp-loader large/small subunit (Enterobacteria phage T4 (Bacteriophage T4)) | BDBM36324 (6-nitro-indolyl- 2'-deoxyriboside triphosphate...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | KEGG PC cid PC sid UniChem Similars | Article PubMed | 5.10E+3 | -7.21 | n/a | n/a | n/a | n/a | n/a | 7.5 | 25 |
Case Western Reserve University | Assay Description ATPase assay contained 10 mM Mg2+, 1uM 13/20 DNA, 500uM (r)NTP or (d)NTP, 500 nM gp45, and 500 nM gp44/62 in T4 buffer. ATPase activity was measured ... | ACS Chem Biol 5: 183-94 (2010) Article DOI: 10.1021/cb900218c BindingDB Entry DOI: 10.7270/Q26M356K | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sliding-clamp-loader large/small subunit (Enterobacteria phage T4 (Bacteriophage T4)) | BDBM36321 (5-cyclohexene-indolyl- 2'-deoxyriboside tripho...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | KEGG PC cid PC sid UniChem Similars | Article PubMed | 1.00E+4 | -6.82 | n/a | n/a | n/a | n/a | n/a | 7.5 | 25 |
Case Western Reserve University | Assay Description ATPase assay contained 10 mM Mg2+, 1uM 13/20 DNA, 500uM (r)NTP or (d)NTP, 500 nM gp45, and 500 nM gp44/62 in T4 buffer. ATPase activity was measured ... | ACS Chem Biol 5: 183-94 (2010) Article DOI: 10.1021/cb900218c BindingDB Entry DOI: 10.7270/Q26M356K | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sliding-clamp-loader large/small subunit (Enterobacteria phage T4 (Bacteriophage T4)) | BDBM36312 (ATP{gamma}S | adenosine 5'-O-(3-thiotriphospha...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | Purchase PC cid PC sid UniChem Similars | Article PubMed | 2.89E+4 | -6.19 | n/a | n/a | n/a | n/a | n/a | 7.5 | 25 |
Case Western Reserve University | Assay Description ATPase assay contained 10 mM Mg2+, 1uM 13/20 DNA, 500uM (r)NTP or (d)NTP, 500 nM gp45, and 500 nM gp44/62 in T4 buffer. ATPase activity was measured ... | ACS Chem Biol 5: 183-94 (2010) Article DOI: 10.1021/cb900218c BindingDB Entry DOI: 10.7270/Q26M356K | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sliding-clamp-loader large/small subunit (Enterobacteria phage T4 (Bacteriophage T4)) | BDBM36323 (4-nitro-indolyl- 2'-deoxyriboside triphosphate...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | KEGG PC cid PC sid UniChem Similars | Article PubMed | 3.42E+4 | -6.09 | n/a | n/a | n/a | n/a | n/a | 7.5 | 25 |
Case Western Reserve University | Assay Description ATPase assay contained 10 mM Mg2+, 1uM 13/20 DNA, 500uM (r)NTP or (d)NTP, 500 nM gp45, and 500 nM gp44/62 in T4 buffer. ATPase activity was measured ... | ACS Chem Biol 5: 183-94 (2010) Article DOI: 10.1021/cb900218c BindingDB Entry DOI: 10.7270/Q26M356K | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sliding-clamp-loader large/small subunit (Enterobacteria phage T4 (Bacteriophage T4)) | BDBM36318 (5-carboxylate-indolyl- 2'-deoxyriboside tripho...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | KEGG PC cid PC sid UniChem Similars | Article PubMed | 3.70E+4 | -6.04 | n/a | n/a | n/a | n/a | n/a | 7.5 | 25 |
Case Western Reserve University | Assay Description ATPase assay contained 10 mM Mg2+, 1uM 13/20 DNA, 500uM (r)NTP or (d)NTP, 500 nM gp45, and 500 nM gp44/62 in T4 buffer. ATPase activity was measured ... | ACS Chem Biol 5: 183-94 (2010) Article DOI: 10.1021/cb900218c BindingDB Entry DOI: 10.7270/Q26M356K | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sliding-clamp-loader large/small subunit (Enterobacteria phage T4 (Bacteriophage T4)) | BDBM36322 (5-phenyl-indolyl- 2'-deoxyriboside triphosphat...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | KEGG PC cid PC sid UniChem Similars | Article PubMed | 4.20E+4 | -5.97 | n/a | n/a | n/a | n/a | n/a | 7.5 | 25 |
Case Western Reserve University | Assay Description ATPase assay contained 10 mM Mg2+, 1uM 13/20 DNA, 500uM (r)NTP or (d)NTP, 500 nM gp45, and 500 nM gp44/62 in T4 buffer. ATPase activity was measured ... | ACS Chem Biol 5: 183-94 (2010) Article DOI: 10.1021/cb900218c BindingDB Entry DOI: 10.7270/Q26M356K | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sliding-clamp-loader large/small subunit (Enterobacteria phage T4 (Bacteriophage T4)) | BDBM36320 (5-cyclohexyl-indolyl- 2'-deoxyriboside triphos...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | KEGG PC cid PC sid UniChem Similars | Article PubMed | 4.75E+4 | -5.89 | n/a | n/a | n/a | n/a | n/a | 7.5 | 25 |
Case Western Reserve University | Assay Description ATPase assay contained 10 mM Mg2+, 1uM 13/20 DNA, 500uM (r)NTP or (d)NTP, 500 nM gp45, and 500 nM gp44/62 in T4 buffer. ATPase activity was measured ... | ACS Chem Biol 5: 183-94 (2010) Article DOI: 10.1021/cb900218c BindingDB Entry DOI: 10.7270/Q26M356K | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sliding-clamp-loader large/small subunit (Enterobacteria phage T4 (Bacteriophage T4)) | BDBM36316 (5-ethyl-indolyl- 2'-deoxyriboside triphosphate...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | KEGG PC cid PC sid UniChem Similars | Article PubMed | 8.15E+4 | -5.57 | n/a | n/a | n/a | n/a | n/a | 7.5 | 25 |
Case Western Reserve University | Assay Description ATPase assay contained 10 mM Mg2+, 1uM 13/20 DNA, 500uM (r)NTP or (d)NTP, 500 nM gp45, and 500 nM gp44/62 in T4 buffer. ATPase activity was measured ... | ACS Chem Biol 5: 183-94 (2010) Article DOI: 10.1021/cb900218c BindingDB Entry DOI: 10.7270/Q26M356K | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sliding-clamp-loader large/small subunit (Enterobacteria phage T4 (Bacteriophage T4)) | BDBM36315 (5-fluoro-indolyl- 2'-deoxyriboside triphosphat...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | KEGG PC cid PC sid UniChem Similars | Article PubMed | <2.00E+5 | <-5.04 | n/a | n/a | n/a | n/a | n/a | 7.5 | 25 |
Case Western Reserve University | Assay Description ATPase assay contained 10 mM Mg2+, 1uM 13/20 DNA, 500uM (r)NTP or (d)NTP, 500 nM gp45, and 500 nM gp44/62 in T4 buffer. ATPase activity was measured ... | ACS Chem Biol 5: 183-94 (2010) Article DOI: 10.1021/cb900218c BindingDB Entry DOI: 10.7270/Q26M356K | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sliding-clamp-loader large/small subunit (Enterobacteria phage T4 (Bacteriophage T4)) | BDBM36314 (5-amino-indolyl- 2'-deoxyriboside triphosphate...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | KEGG PC cid PC sid UniChem Similars | Article PubMed | <2.00E+5 | <-5.04 | n/a | n/a | n/a | n/a | n/a | 7.5 | 25 |
Case Western Reserve University | Assay Description ATPase assay contained 10 mM Mg2+, 1uM 13/20 DNA, 500uM (r)NTP or (d)NTP, 500 nM gp45, and 500 nM gp44/62 in T4 buffer. ATPase activity was measured ... | ACS Chem Biol 5: 183-94 (2010) Article DOI: 10.1021/cb900218c BindingDB Entry DOI: 10.7270/Q26M356K | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sliding-clamp-loader large/small subunit (Enterobacteria phage T4 (Bacteriophage T4)) | BDBM36313 (dITP | indolyl- 2'-deoxyriboside triphosphate) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | KEGG PC cid PC sid UniChem Similars | Article PubMed | <2.00E+5 | <-5.04 | n/a | n/a | n/a | n/a | n/a | 7.5 | 25 |
Case Western Reserve University | Assay Description ATPase assay contained 10 mM Mg2+, 1uM 13/20 DNA, 500uM (r)NTP or (d)NTP, 500 nM gp45, and 500 nM gp44/62 in T4 buffer. ATPase activity was measured ... | ACS Chem Biol 5: 183-94 (2010) Article DOI: 10.1021/cb900218c BindingDB Entry DOI: 10.7270/Q26M356K | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sliding-clamp-loader large/small subunit (Enterobacteria phage T4 (Bacteriophage T4)) | BDBM36317 (5-ethylene-indolyl- 2'-deoxyriboside triphosph...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | KEGG PC cid PC sid UniChem Similars | Article PubMed | <2.00E+5 | <-5.04 | n/a | n/a | n/a | n/a | n/a | 7.5 | 25 |
Case Western Reserve University | Assay Description ATPase assay contained 10 mM Mg2+, 1uM 13/20 DNA, 500uM (r)NTP or (d)NTP, 500 nM gp45, and 500 nM gp44/62 in T4 buffer. ATPase activity was measured ... | ACS Chem Biol 5: 183-94 (2010) Article DOI: 10.1021/cb900218c BindingDB Entry DOI: 10.7270/Q26M356K | |||||||||||
More data for this Ligand-Target Pair |