Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kcal/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Adenylate kinase 2, mitochondrial (Homo sapiens (Human)) | BDBM50367071 (CHEMBL607736) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | PubMed | 4.70E+6 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Ability to inhibit Escherichia coli adenylate kinase II, activity expressed as Inhibition constant | J Med Chem 25: 382-6 (1982) BindingDB Entry DOI: 10.7270/Q24F1R9V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenylate kinase 2, mitochondrial (Homo sapiens (Human)) | BDBM50367065 (CHEMBL608643) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | PubMed | 6.70E+6 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Ability to inhibit Escherichia coli adenylate kinase II, activity expressed as Inhibition constant | J Med Chem 25: 382-6 (1982) BindingDB Entry DOI: 10.7270/Q24F1R9V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenylate kinase 2, mitochondrial (Homo sapiens (Human)) | BDBM50367072 (CHEMBL3350534 | CHEMBL610134) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | PubMed | 6.80E+6 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Ability to inhibit Escherichia coli adenylate kinase II, activity expressed as Inhibition constant | J Med Chem 25: 382-6 (1982) BindingDB Entry DOI: 10.7270/Q24F1R9V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenylate kinase 2, mitochondrial (Homo sapiens (Human)) | BDBM50367070 (CHEMBL609238) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | PubMed | 7.30E+6 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Ability to inhibit Escherichia coli adenylate kinase II, activity expressed as Inhibition constant | J Med Chem 25: 382-6 (1982) BindingDB Entry DOI: 10.7270/Q24F1R9V | |||||||||||
More data for this Ligand-Target Pair |