Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kcal/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Proprotein convertase subtilisin/kexin type 7 (Homo sapiens (Human)) | BDBM50349829 (CHEMBL1813183) | KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 462 | n/a | n/a | n/a | n/a | n/a | n/a |
Universidade Estadual Paulista Curated by ChEMBL | Assay Description Inhibition of recombinant type 8 subtilisin using Arg-Glu-(EDANS)- Ser-Gln-Asn-Tyr-Pro-Ile-Val-Gln-Lys-(DALBCYL)-Arg fluorogenic substrate preincubat... | J Nat Prod 74: 1353-7 (2011) Article DOI: 10.1021/np1005983 BindingDB Entry DOI: 10.7270/Q2PZ596S | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Proprotein convertase subtilisin/kexin type 7 (Homo sapiens (Human)) | BDBM35525 (3,3''''-methylenebis(4-hydroxy-coumarin | 3,3''''-...) | KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL DrugBank MCE KEGG MMDB PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.30E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Universidade Estadual Paulista Curated by ChEMBL | Assay Description Inhibition of recombinant type 8 subtilisin using Arg-Glu-(EDANS)- Ser-Gln-Asn-Tyr-Pro-Ile-Val-Gln-Lys-(DALBCYL)-Arg fluorogenic substrate preincubat... | J Nat Prod 74: 1353-7 (2011) Article DOI: 10.1021/np1005983 BindingDB Entry DOI: 10.7270/Q2PZ596S | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Proprotein convertase subtilisin/kexin type 7 (Homo sapiens (Human)) | BDBM50343352 (2-hydroxy-3-(3-oxo-1-phenylbutyl)-4H-chromen-4-one...) | KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL DrugBank KEGG PC cid PC sid PDB UniChem Similars | Article PubMed | n/a | n/a | 2.46E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Universidade Estadual Paulista Curated by ChEMBL | Assay Description Inhibition of recombinant type 8 subtilisin using Arg-Glu-(EDANS)- Ser-Gln-Asn-Tyr-Pro-Ile-Val-Gln-Lys-(DALBCYL)-Arg fluorogenic substrate preincubat... | J Nat Prod 74: 1353-7 (2011) Article DOI: 10.1021/np1005983 BindingDB Entry DOI: 10.7270/Q2PZ596S | |||||||||||
More data for this Ligand-Target Pair |