BindingDB PrimarySearch

Found 83 hits of ki for UniProtKB: P28838
Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kcal/mole	IC50 nM	Kd nM	EC50/IC50 nM	k_off s^-1	k_on M^-1s^-1	pH	Temp °C
Cytosol aminopeptidase (Homo sapiens (Human))	BDBM23971 ((2S)-2-[(2S,3R)-3-amino-2-hydroxy-4-phenylbutanami...) Show SMILES Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	Purchase CHEMBL MCE MMDB PC cid PC sid PDB UniChem Patents Similars	Article PubMed	0.600	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Wroclaw University of Technology Curated by ChEMBL					Assay Description Binding affinity for cytosolic leucine aminopeptidase (LAP) from porcine kidney				J Med Chem 46: 2641-55 (2003) Article DOI: 10.1021/jm030795v BindingDB Entry DOI: 10.7270/Q27P903F
Wroclaw University of Technology Curated by ChEMBL					More data for this Ligand-Target Pair
Cytosol aminopeptidase (Homo sapiens (Human))	BDBM23971 ((2S)-2-[(2S,3R)-3-amino-2-hydroxy-4-phenylbutanami...) Show SMILES Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	Purchase CHEMBL MCE MMDB PC cid PC sid PDB UniChem Patents Similars	PubMed	20	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
University of Wisconsin Curated by ChEMBL					Assay Description Inhibitory activity against Leucine aminopeptidase				J Med Chem 31: 2193-9 (1988) BindingDB Entry DOI: 10.7270/Q2Z038RM
University of Wisconsin Curated by ChEMBL					More data for this Ligand-Target Pair
Cytosol aminopeptidase (Homo sapiens (Human))	BDBM50017478 (Amastatin \| CHEMBL28650 \| Leu[1psi,CHOHCONH]ValVal...) Show SMILES Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	Purchase CHEMBL MCE KEGG MMDB PC cid PC sid UniChem Patents Similars	MMDB Article PubMed	30	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Wroclaw University of Technology Curated by ChEMBL					Assay Description Binding affinity for cytosolic leucine aminopeptidase (LAP) from porcine kidney				J Med Chem 46: 2641-55 (2003) Article DOI: 10.1021/jm030795v BindingDB Entry DOI: 10.7270/Q27P903F
Wroclaw University of Technology Curated by ChEMBL					More data for this Ligand-Target Pair
Cytosol aminopeptidase (Homo sapiens (Human))	BDBM50225458 ((2S)-3-[(R)-[(1S)-1-amino-3-phenylpropyl](hydroxy)...) Show SMILES Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL MMDB PC cid PC sid UniChem Similars	Article PubMed	45	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Wroc£?aw University of Technology Curated by ChEMBL					Assay Description Inhibition of pig kidney cytosolic leucine aminopeptidase				Bioorg Med Chem Lett 18: 1550-4 (2008) Article DOI: 10.1016/j.bmcl.2008.01.107 BindingDB Entry DOI: 10.7270/Q28K78TP
Wroc£?aw University of Technology Curated by ChEMBL					More data for this Ligand-Target Pair
Cytosol aminopeptidase (Homo sapiens (Human))	BDBM50457478 (CHEMBL4208547) Show SMILES CC1(C)OB(OC1(C)C)C(N)Cc1ccccc1 Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	50	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Jadavpur University Curated by ChEMBL					Assay Description Inhibition of LAP (unknown origin)				J Med Chem 61: 6468-6490 (2018) Article DOI: 10.1021/acs.jmedchem.7b00782 BindingDB Entry DOI: 10.7270/Q28S4SHS
Jadavpur University Curated by ChEMBL					More data for this Ligand-Target Pair
Cytosol aminopeptidase (Homo sapiens (Human))	BDBM50129685 (2-Amino-4-methyl-pentanal \| CHEMBL88476) Show SMILES CC(C)CC(N)C=O Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Patents Similars	Article PubMed	60	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Wroclaw University of Technology Curated by ChEMBL					Assay Description Binding affinity for cytosolic leucine aminopeptidase (LAP) from porcine kidney				J Med Chem 46: 2641-55 (2003) Article DOI: 10.1021/jm030795v BindingDB Entry DOI: 10.7270/Q27P903F
Wroclaw University of Technology Curated by ChEMBL					More data for this Ligand-Target Pair
Cytosol aminopeptidase (Homo sapiens (Human))	BDBM50129683 (2-[(1-Amino-3-methyl-butyl)-hydroxy-phosphinoylmet...) Show SMILES CC(C)CC(CP(O)(O)C(=N)CC(C)C)C(O)=O Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	65	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Wroclaw University of Technology Curated by ChEMBL					Assay Description Binding affinity for cytosolic leucine aminopeptidase (LAP) from porcine kidney				J Med Chem 46: 2641-55 (2003) Article DOI: 10.1021/jm030795v BindingDB Entry DOI: 10.7270/Q27P903F
Wroclaw University of Technology Curated by ChEMBL					More data for this Ligand-Target Pair
Cytosol aminopeptidase (Homo sapiens (Human))	BDBM50129683 (2-[(1-Amino-3-methyl-butyl)-hydroxy-phosphinoylmet...) Show SMILES CC(C)CC(CP(O)(O)C(=N)CC(C)C)C(O)=O Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	65	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Wroclaw University of Technology Curated by ChEMBL					Assay Description Inhibition of LAP				J Med Chem 54: 5955-80 (2011) Article DOI: 10.1021/jm200587f BindingDB Entry DOI: 10.7270/Q2PV6MGF
Wroclaw University of Technology Curated by ChEMBL					More data for this Ligand-Target Pair
Cytosol aminopeptidase (Homo sapiens (Human))	BDBM50129683 (2-[(1-Amino-3-methyl-butyl)-hydroxy-phosphinoylmet...) Show SMILES CC(C)CC(CP(O)(O)C(=N)CC(C)C)C(O)=O Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	65	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Wroclaw University of Technology Curated by ChEMBL					Assay Description Binding affinity for cytosolic leucine aminopeptidase (LAP) from porcine kidney				J Med Chem 46: 2641-55 (2003) Article DOI: 10.1021/jm030795v BindingDB Entry DOI: 10.7270/Q27P903F
Wroclaw University of Technology Curated by ChEMBL					More data for this Ligand-Target Pair
Cytosol aminopeptidase (Homo sapiens (Human))	BDBM50129684 (3-[(1-amino-3-phenyl-propyl)-hydroxy-phosphinoyl]-...) Show SMILES Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	66	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Wroc£?aw University of Technology Curated by ChEMBL					Assay Description Inhibition of pig kidney cytosolic leucine aminopeptidase				Bioorg Med Chem Lett 18: 1550-4 (2008) Article DOI: 10.1016/j.bmcl.2008.01.107 BindingDB Entry DOI: 10.7270/Q28K78TP
Wroc£?aw University of Technology Curated by ChEMBL					More data for this Ligand-Target Pair
Cytosol aminopeptidase (Homo sapiens (Human))	BDBM50129684 (3-[(1-amino-3-phenyl-propyl)-hydroxy-phosphinoyl]-...) Show SMILES Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	66	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Wroclaw University of Technology Curated by ChEMBL					Assay Description Binding affinity for cytosolic leucine aminopeptidase (LAP) from porcine kidney				J Med Chem 46: 2641-55 (2003) Article DOI: 10.1021/jm030795v BindingDB Entry DOI: 10.7270/Q27P903F
Wroclaw University of Technology Curated by ChEMBL					More data for this Ligand-Target Pair
Cytosol aminopeptidase (Homo sapiens (Human))	BDBM50129681 (3-[(1-Amino-3-phenyl-propyl)-hydroxy-phosphinoyl]-...) Show SMILES Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	67	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Wroclaw University of Technology Curated by ChEMBL					Assay Description Binding affinity for cytosolic leucine aminopeptidase (LAP) from porcine kidney				J Med Chem 46: 2641-55 (2003) Article DOI: 10.1021/jm030795v BindingDB Entry DOI: 10.7270/Q27P903F
Wroclaw University of Technology Curated by ChEMBL					More data for this Ligand-Target Pair
Cytosol aminopeptidase (Homo sapiens (Human))	BDBM50129682 (2-[(1-Amino-3-phenyl-propyl)-hydroxy-phosphinoylme...) Show SMILES CC(C)CC(CP(O)(O)C(=N)CCc1ccccc1)C(O)=O Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	74	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Wroclaw University of Technology Curated by ChEMBL					Assay Description Binding affinity for cytosolic leucine aminopeptidase (LAP) from porcine kidney				J Med Chem 46: 2641-55 (2003) Article DOI: 10.1021/jm030795v BindingDB Entry DOI: 10.7270/Q27P903F
Wroclaw University of Technology Curated by ChEMBL					More data for this Ligand-Target Pair
Cytosol aminopeptidase (Homo sapiens (Human))	BDBM50089610 ((Z)-(S)-5-Amino-7-methyl-4-oxo-oct-2-enoic acid me...) Show SMILES COC(=O)CCC(=O)C(=N)CC(C)C Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem	PubMed	76	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
The Queen's University of Belfast Curated by ChEMBL					Assay Description Inhibitory activity of the compound against leucine aminopeptidase				Bioorg Med Chem Lett 10: 1481-2 (2000) BindingDB Entry DOI: 10.7270/Q2BV7FVK
The Queen's University of Belfast Curated by ChEMBL					More data for this Ligand-Target Pair
Cytosol aminopeptidase (Homo sapiens (Human))	BDBM50027041 (2-(3-Amino-2-hydroxy-5-methyl-hexanoylamino)-4-met...) Show SMILES Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	PubMed	120	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA Curated by ChEMBL					Assay Description Compound was evaluated for the inhibition of Leucine aminopeptidase and the inhibition constant was determined after preincubating the enzyme and inh...				J Med Chem 27: 417-22 (1984) BindingDB Entry DOI: 10.7270/Q280535G
TBA Curated by ChEMBL					More data for this Ligand-Target Pair
Cytosol aminopeptidase (Homo sapiens (Human))	BDBM50017478 (Amastatin \| CHEMBL28650 \| Leu[1psi,CHOHCONH]ValVal...) Show SMILES Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	Purchase CHEMBL MCE KEGG MMDB PC cid PC sid UniChem Patents Similars	MMDB PubMed	200	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA Curated by ChEMBL					Assay Description Effect of inhibitor structure on the slow binding inhibition of Leucine aminopeptidase was determined and the Ki was reported which is = k2/k1				J Med Chem 27: 417-22 (1984) BindingDB Entry DOI: 10.7270/Q280535G
TBA Curated by ChEMBL					More data for this Ligand-Target Pair
Cytosol aminopeptidase (Homo sapiens (Human))	BDBM50017478 (Amastatin \| CHEMBL28650 \| Leu[1psi,CHOHCONH]ValVal...) Show SMILES Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	Purchase CHEMBL MCE KEGG MMDB PC cid PC sid UniChem Patents Similars	MMDB PubMed	220	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA Curated by ChEMBL					Assay Description Effect of inhibitor structure on the slow binding inhibition of aminopeptidase M was determined and Ki* was reported which is obtained by the equatio...				J Med Chem 27: 417-22 (1984) BindingDB Entry DOI: 10.7270/Q280535G
TBA Curated by ChEMBL					More data for this Ligand-Target Pair
Cytosol aminopeptidase (Homo sapiens (Human))	BDBM50316047 (1-amino-2-methylbutylphosphonic acid monophenylest...) Show SMILES CC(C)CC(N)P(O)(=O)Oc1ccccc1 Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	230	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Wroclaw University of Technology Curated by ChEMBL					Assay Description Inhibition of leucine aminopeptidase				Bioorg Med Chem 18: 2930-6 (2010) Article DOI: 10.1016/j.bmc.2010.02.056 BindingDB Entry DOI: 10.7270/Q2FN16C0
Wroclaw University of Technology Curated by ChEMBL					More data for this Ligand-Target Pair
Cytosol aminopeptidase (Homo sapiens (Human))	BDBM50024594 ((R)-1-Ammonium-3-methyl-butane-1-phosphonic acid a...) Show SMILES CC(C)C[C@H]([NH3+])P(O)([O-])=O Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	Purchase CHEMBL PC cid PC sid UniChem Similars	PubMed	230	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA Curated by ChEMBL					Assay Description Inhibition of Leucine aminopeptidase isolated from porcine kidney.				J Med Chem 30: 1603-9 (1987) BindingDB Entry DOI: 10.7270/Q2W66MCD
TBA Curated by ChEMBL					More data for this Ligand-Target Pair
Cytosol aminopeptidase (Homo sapiens (Human))	BDBM50129679 ((1-Amino-3-methyl-butyl)-phosphonic acid \| 1-amino...) Show SMILES CC(C)CC(N)P(O)(O)=O Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	Purchase CHEMBL PC cid PC sid PDB UniChem Patents Similars	Article PubMed	230	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Wroclaw University of Technology Curated by ChEMBL					Assay Description Inhibition of leucine aminopeptidase				Bioorg Med Chem 18: 2930-6 (2010) Article DOI: 10.1016/j.bmc.2010.02.056 BindingDB Entry DOI: 10.7270/Q2FN16C0
Wroclaw University of Technology Curated by ChEMBL					More data for this Ligand-Target Pair
Cytosol aminopeptidase (Homo sapiens (Human))	BDBM50129679 ((1-Amino-3-methyl-butyl)-phosphonic acid \| 1-amino...) Show SMILES CC(C)CC(N)P(O)(O)=O Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	Purchase CHEMBL PC cid PC sid PDB UniChem Patents Similars	Article PubMed	230	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Wroclaw University of Technology Curated by ChEMBL					Assay Description Binding affinity for cytosolic leucine aminopeptidase (LAP) from porcine kidney				J Med Chem 46: 2641-55 (2003) Article DOI: 10.1021/jm030795v BindingDB Entry DOI: 10.7270/Q27P903F
Wroclaw University of Technology Curated by ChEMBL					More data for this Ligand-Target Pair
Cytosol aminopeptidase (Homo sapiens (Human))	BDBM50234656 ((R)-3-[((R)-1-amino-3-phenyl-propyl)-hydroxy-phosp...) Show SMILES Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	271	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Wroc£?aw University of Technology Curated by ChEMBL					Assay Description Inhibition of pig kidney cytosolic leucine aminopeptidase				Bioorg Med Chem Lett 18: 1550-4 (2008) Article DOI: 10.1016/j.bmcl.2008.01.107 BindingDB Entry DOI: 10.7270/Q28K78TP
Wroc£?aw University of Technology Curated by ChEMBL					More data for this Ligand-Target Pair
Cytosol aminopeptidase (Homo sapiens (Human))	BDBM50022747 (2-(3-Amino-2-hydroxy-4-phenyl-thiobutyrylamino)-4-...) Show SMILES Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	PubMed	330	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
University of Wisconsin Curated by ChEMBL					Assay Description Inhibitory activity against Leucine aminopeptidase				J Med Chem 31: 2193-9 (1988) BindingDB Entry DOI: 10.7270/Q2Z038RM
University of Wisconsin Curated by ChEMBL					More data for this Ligand-Target Pair
Cytosol aminopeptidase (Homo sapiens (Human))	BDBM50129677 (3-[(1-Amino-3-methyl-butyl)-hydroxy-phosphinoyl]-p...) Show SMILES CC(C)CC(=N)P(O)(O)CCC(O)=O Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem	Article PubMed	330	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Wroclaw University of Technology Curated by ChEMBL					Assay Description Binding affinity for cytosolic leucine aminopeptidase (LAP) from porcine kidney				J Med Chem 46: 2641-55 (2003) Article DOI: 10.1021/jm030795v BindingDB Entry DOI: 10.7270/Q27P903F
Wroclaw University of Technology Curated by ChEMBL					More data for this Ligand-Target Pair
Cytosol aminopeptidase (Homo sapiens (Human))	BDBM50024596 ((R)-1-Ammonium-2-phenyl-ethanephosphonic acid anio...) Show SMILES [NH3+][C@@H](Cc1ccccc1)P(O)([O-])=O Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	Purchase CHEMBL PC cid PC sid PDB UniChem Similars	PubMed	420	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA Curated by ChEMBL					Assay Description Inhibition of Leucine aminopeptidase isolated from porcine kidney.				J Med Chem 30: 1603-9 (1987) BindingDB Entry DOI: 10.7270/Q2W66MCD
TBA Curated by ChEMBL					More data for this Ligand-Target Pair
Cytosol aminopeptidase (Homo sapiens (Human))	BDBM50316048 (1-amino-2-phenylethylphosphonic acid monophenyl es...) Show SMILES NC(Cc1ccccc1)P(O)(=O)Oc1ccccc1 Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem	Article PubMed	420	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Wroclaw University of Technology Curated by ChEMBL					Assay Description Inhibition of leucine aminopeptidase				Bioorg Med Chem 18: 2930-6 (2010) Article DOI: 10.1016/j.bmc.2010.02.056 BindingDB Entry DOI: 10.7270/Q2FN16C0
Wroclaw University of Technology Curated by ChEMBL					More data for this Ligand-Target Pair
Cytosol aminopeptidase (Homo sapiens (Human))	BDBM50024592 ((S)-1-Ammonium-2-phenyl-ethanephosphonic acid anio...) Show SMILES [NH3+][C@H](Cc1ccccc1)P(O)([O-])=O Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	Purchase CHEMBL PC cid PC sid UniChem Similars	Article PubMed	420	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Wroclaw University of Technology Curated by ChEMBL					Assay Description Inhibition of leucine aminopeptidase				Bioorg Med Chem 18: 2930-6 (2010) Article DOI: 10.1016/j.bmc.2010.02.056 BindingDB Entry DOI: 10.7270/Q2FN16C0
Wroclaw University of Technology Curated by ChEMBL					More data for this Ligand-Target Pair
Cytosol aminopeptidase (Homo sapiens (Human))	BDBM50024590 (1-Ammonium-octane-1-phosphonic acid anion \| CHEMBL...) Show SMILES CCCCCCCC([NH3+])P(O)([O-])=O Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	PubMed	470	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA Curated by ChEMBL					Assay Description Compound was tested for inhibition of Leucine aminopeptidase isolated from porcine kidney; Inhibitor exhibits slow-binding behavior(k on <=1000Me-1Se...				J Med Chem 30: 1603-9 (1987) BindingDB Entry DOI: 10.7270/Q2W66MCD
TBA Curated by ChEMBL					More data for this Ligand-Target Pair
Cytosol aminopeptidase (Homo sapiens (Human))	BDBM50027043 (3-Amino-2-hydroxy-N-(3-methyl-butyl)-4-phenyl-buty...) Show SMILES CC(C)CCNC(=O)[C@H](O)[C@@H](N)Cc1ccccc1 Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	PubMed	500	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA Curated by ChEMBL					Assay Description Compound was evaluated for the inhibition of Leucine aminopeptidase from porcine kidney and the inhibition constant was determined after preincubatin...				J Med Chem 27: 417-22 (1984) BindingDB Entry DOI: 10.7270/Q280535G
TBA Curated by ChEMBL					More data for this Ligand-Target Pair
Cytosol aminopeptidase (Homo sapiens (Human))	BDBM50008431 (3-Amino-2-hydroxy-N-(3-methyl-butyl)-4-phenyl-buty...) Show SMILES CC(C)CCNC(=O)[C@@H](O)[C@H](N)Cc1ccccc1 Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Patents Similars	PubMed	510	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
University of Wisconsin Curated by ChEMBL					Assay Description Inhibitory activity against Leucine aminopeptidase				J Med Chem 31: 2193-9 (1988) BindingDB Entry DOI: 10.7270/Q2Z038RM
University of Wisconsin Curated by ChEMBL					More data for this Ligand-Target Pair
Cytosol aminopeptidase (Homo sapiens (Human))	BDBM50022751 (2-(3-Amino-2-mercapto-4-phenyl-butyrylamino)-4-met...) Show SMILES Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL KEGG PC cid PC sid UniChem Similars	PubMed	550	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
University of Wisconsin Curated by ChEMBL					Assay Description Inhibitory activity against Aminopeptidase M				J Med Chem 31: 2193-9 (1988) BindingDB Entry DOI: 10.7270/Q2Z038RM
University of Wisconsin Curated by ChEMBL					More data for this Ligand-Target Pair
Cytosol aminopeptidase (Homo sapiens (Human))	BDBM50027042 (3-Amino-2-hydroxy-5-methyl-hexanoic acid {2-methyl...) Show SMILES Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	PubMed	890	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA Curated by ChEMBL					Assay Description Compound was evaluated for the inhibition of Leucine aminopeptidase and the inhibition constant was determined after preincubating the enzyme and in...				J Med Chem 27: 417-22 (1984) BindingDB Entry DOI: 10.7270/Q280535G
TBA Curated by ChEMBL					More data for this Ligand-Target Pair
Cytosol aminopeptidase (Homo sapiens (Human))	BDBM50225458 ((2S)-3-[(R)-[(1S)-1-amino-3-phenylpropyl](hydroxy)...) Show SMILES Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL MMDB PC cid PC sid UniChem Similars	Article PubMed	988	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Wroc£?aw University of Technology Curated by ChEMBL					Assay Description Inhibition of pig kidney cytosolic leucine aminopeptidase				Bioorg Med Chem Lett 18: 1550-4 (2008) Article DOI: 10.1016/j.bmcl.2008.01.107 BindingDB Entry DOI: 10.7270/Q28K78TP
Wroc£?aw University of Technology Curated by ChEMBL					More data for this Ligand-Target Pair
Cytosol aminopeptidase (Homo sapiens (Human))	BDBM50024601 (1-Ammonium-hexane-1-phosphonic acid anion \| 1-amin...) Show SMILES CCCCCC([NH3+])P(O)([O-])=O Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	Purchase CHEMBL PC cid PC sid UniChem Similars	PubMed	1.00E+3	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA Curated by ChEMBL					Assay Description Inhibition of Leucine aminopeptidase isolated from porcine kidney.				J Med Chem 30: 1603-9 (1987) BindingDB Entry DOI: 10.7270/Q2W66MCD
TBA Curated by ChEMBL					More data for this Ligand-Target Pair
Cytosol aminopeptidase (Homo sapiens (Human))	BDBM50022751 (2-(3-Amino-2-mercapto-4-phenyl-butyrylamino)-4-met...) Show SMILES Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL KEGG PC cid PC sid UniChem Similars	PubMed	1.00E+3	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
University of Wisconsin Curated by ChEMBL					Assay Description Inhibitory activity against Leucine aminopeptidase				J Med Chem 31: 2193-9 (1988) BindingDB Entry DOI: 10.7270/Q2Z038RM
University of Wisconsin Curated by ChEMBL					More data for this Ligand-Target Pair
Cytosol aminopeptidase (Homo sapiens (Human))	BDBM50024602 (1-Ammonium-2-methyl-propane-1-phosphonic acid anio...) Show SMILES CC(C)C([NH3+])P(O)([O-])=O Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	Purchase CHEMBL PC cid PC sid UniChem Similars	PubMed	1.20E+3	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA Curated by ChEMBL					Assay Description Compound was tested for inhibition of Leucine aminopeptidase isolated from porcine kidney; Inhibitor exhibits slow-binding behavior(k on <=1000Me-1Se...				J Med Chem 30: 1603-9 (1987) BindingDB Entry DOI: 10.7270/Q2W66MCD
TBA Curated by ChEMBL					More data for this Ligand-Target Pair
Cytosol aminopeptidase (Homo sapiens (Human))	BDBM50027046 (2-[2-(3-Amino-2-hydroxy-5-methyl-hexanoylamino)-3-...) Show SMILES Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	PubMed	1.24E+3	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA Curated by ChEMBL					Assay Description Compound was evaluated for the inhibition of Leucine aminopeptidase and the inhibition constant was determined after preincubating the enzyme and inh...				J Med Chem 27: 417-22 (1984) BindingDB Entry DOI: 10.7270/Q280535G
TBA Curated by ChEMBL					More data for this Ligand-Target Pair
Cytosol aminopeptidase (Homo sapiens (Human))	BDBM50457469 (CHEMBL4213478) Show SMILES CC(C)CC(N)B1OC(C)(C)C(C)(C)O1 Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	Purchase PC cid PC sid UniChem	Article PubMed	1.30E+3	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Jadavpur University Curated by ChEMBL					Assay Description Inhibition of LAP (unknown origin)				J Med Chem 61: 6468-6490 (2018) Article DOI: 10.1021/acs.jmedchem.7b00782 BindingDB Entry DOI: 10.7270/Q28S4SHS
Jadavpur University Curated by ChEMBL					More data for this Ligand-Target Pair
Cytosol aminopeptidase (Homo sapiens (Human))	BDBM50024604 (1-Ammonium-propane-1-phosphonic acid anion \| 1-ami...) Show SMILES CCC([NH3+])P(O)([O-])=O Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	Purchase CHEMBL PC cid PC sid UniChem Similars	PubMed	3.60E+3	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA Curated by ChEMBL					Assay Description Compound was tested for inhibition of Leucine aminopeptidase isolated from porcine kidney; Inhibitor exhibits slow-binding behavior(k on <=1000Me-1Se...				J Med Chem 30: 1603-9 (1987) BindingDB Entry DOI: 10.7270/Q2W66MCD
TBA Curated by ChEMBL					More data for this Ligand-Target Pair
Cytosol aminopeptidase (Homo sapiens (Human))	BDBM50022742 (3-Amino-2-hydroxy-N-(3-methyl-butyl)-4-phenyl-thio...) Show SMILES CC(C)CCNC(=S)[C@@H](O)[C@H](N)Cc1ccccc1 Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem	PubMed	4.40E+3	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
University of Wisconsin Curated by ChEMBL					Assay Description Inhibitory activity against Leucine aminopeptidase				J Med Chem 31: 2193-9 (1988) BindingDB Entry DOI: 10.7270/Q2Z038RM
University of Wisconsin Curated by ChEMBL					More data for this Ligand-Target Pair
Cytosol aminopeptidase (Homo sapiens (Human))	BDBM50129680 (CHEMBL423870 \| {[hydroxy(1-hydroxy-3-methylbutyl)p...) Show SMILES CC(C)CC(O)P([O-])(=O)NCC([O-])=O Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem	Article PubMed	4.88E+3	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Wroclaw University of Technology Curated by ChEMBL					Assay Description Binding affinity for cytosolic leucine aminopeptidase (LAP) from porcine kidney				J Med Chem 46: 2641-55 (2003) Article DOI: 10.1021/jm030795v BindingDB Entry DOI: 10.7270/Q27P903F
Wroclaw University of Technology Curated by ChEMBL					More data for this Ligand-Target Pair
Cytosol aminopeptidase (Homo sapiens (Human))	BDBM50234656 ((R)-3-[((R)-1-amino-3-phenyl-propyl)-hydroxy-phosp...) Show SMILES Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	8.80E+3	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Wroc£?aw University of Technology Curated by ChEMBL					Assay Description Inhibition of pig kidney cytosolic leucine aminopeptidase				Bioorg Med Chem Lett 18: 1550-4 (2008) Article DOI: 10.1016/j.bmcl.2008.01.107 BindingDB Entry DOI: 10.7270/Q28K78TP
Wroc£?aw University of Technology Curated by ChEMBL					More data for this Ligand-Target Pair
Cytosol aminopeptidase (Homo sapiens (Human))	BDBM50024592 ((S)-1-Ammonium-2-phenyl-ethanephosphonic acid anio...) Show SMILES [NH3+][C@H](Cc1ccccc1)P(O)([O-])=O Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	Purchase CHEMBL PC cid PC sid UniChem Similars	PubMed	1.54E+4	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA Curated by ChEMBL					Assay Description Inhibition of Leucine aminopeptidase isolated from porcine kidney.				J Med Chem 30: 1603-9 (1987) BindingDB Entry DOI: 10.7270/Q2W66MCD
TBA Curated by ChEMBL					More data for this Ligand-Target Pair
Cytosol aminopeptidase (Homo sapiens (Human))	BDBM50046325 ((S)-2-((2S,3S)-3-Amino-2-hydroxy-4-phenyl-butyryla...) Show SMILES Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	Purchase CHEMBL MMDB PC cid PC sid PDB UniChem Patents Similars	PubMed	1.70E+4	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA Curated by ChEMBL					Assay Description Compound was evaluated for the inhibition of Leucine aminopeptidase and the inhibition constant was determined after preincubating the enzyme and inh...				J Med Chem 27: 417-22 (1984) BindingDB Entry DOI: 10.7270/Q280535G
TBA Curated by ChEMBL					More data for this Ligand-Target Pair
Cytosol aminopeptidase (Homo sapiens (Human))	BDBM50367209 (BESTATIN HYDROCHLORIDE \| Ubenimex) Show SMILES Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	Purchase MCE PC cid PC sid PDB UniChem Similars	PubMed	2.00E+4	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA Curated by ChEMBL					Assay Description Compound was evaluated for the inhibition of Leucine aminopeptidase and the inhibition constant was determined after preincubating the enzyme and inh...				J Med Chem 27: 417-22 (1984) BindingDB Entry DOI: 10.7270/Q280535G
TBA Curated by ChEMBL					More data for this Ligand-Target Pair
Cytosol aminopeptidase (Homo sapiens (Human))	BDBM50027045 (2-{2-[2-(3-Amino-2-hydroxy-5-methyl-hexanoylamino)...) Show SMILES Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	Purchase CHEMBL KEGG PC cid PC sid UniChem Similars	PubMed	2.00E+4	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA Curated by ChEMBL					Assay Description Effect of inhibitor structure on the slow binding inhibition of Aminopeptidase M from porcine kidney was determined and the Ki was reported which is ...				J Med Chem 27: 417-22 (1984) BindingDB Entry DOI: 10.7270/Q280535G
TBA Curated by ChEMBL					More data for this Ligand-Target Pair
Cytosol aminopeptidase (Homo sapiens (Human))	BDBM50017478 (Amastatin \| CHEMBL28650 \| Leu[1psi,CHOHCONH]ValVal...) Show SMILES Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	Purchase CHEMBL MCE KEGG MMDB PC cid PC sid UniChem Patents Similars	MMDB PubMed	2.00E+4	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA Curated by ChEMBL					Assay Description Effect of inhibitor structure on the slow binding inhibition of aminopeptidase M was determined and the Ki was reported which is = k2/k1				J Med Chem 27: 417-22 (1984) BindingDB Entry DOI: 10.7270/Q280535G
TBA Curated by ChEMBL					More data for this Ligand-Target Pair
Cytosol aminopeptidase (Homo sapiens (Human))	BDBM50027045 (2-{2-[2-(3-Amino-2-hydroxy-5-methyl-hexanoylamino)...) Show SMILES Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	Purchase CHEMBL KEGG PC cid PC sid UniChem Similars	PubMed	<2.30E+4	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA Curated by ChEMBL					Assay Description Compound was evaluated for the inhibition of Aminopeptidase M (AP-M) and the inhibition constant was determined after preincubating the enzyme and in...				J Med Chem 27: 417-22 (1984) BindingDB Entry DOI: 10.7270/Q280535G
TBA Curated by ChEMBL					More data for this Ligand-Target Pair
Cytosol aminopeptidase (Homo sapiens (Human))	BDBM50022754 (3-Amino-2-mercapto-N-(3-methyl-butyl)-4-phenyl-but...) Show SMILES CC(C)CCNC(=O)[C@H](S)[C@@H](N)Cc1ccccc1 Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL KEGG PC cid PC sid UniChem Similars	PubMed	2.60E+4	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
University of Wisconsin Curated by ChEMBL					Assay Description Inhibitory activity against Leucine aminopeptidase				J Med Chem 31: 2193-9 (1988) BindingDB Entry DOI: 10.7270/Q2Z038RM
University of Wisconsin Curated by ChEMBL					More data for this Ligand-Target Pair
Cytosol aminopeptidase (Homo sapiens (Human))	BDBM50105577 (CHEMBL3597446) Show SMILES Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem	Article PubMed	3.00E+4	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Universit£ de Haute Alsace Curated by ChEMBL					Assay Description Inhibition of cytosolic leucine aminopeptidase (unknown origin)				Bioorg Med Chem 23: 3192-207 (2015) Article DOI: 10.1016/j.bmc.2015.04.066 BindingDB Entry DOI: 10.7270/Q2Z321DW
Universit£ de Haute Alsace Curated by ChEMBL					More data for this Ligand-Target Pair

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