Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kcal/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Polynucleotide kinase (Enterobacteria phage T4) | BDBM50356642 (CHEMBL1917196) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Kyoto Prefectural University Curated by ChEMBL | Assay Description Inhibition of T4 polynucleotide kinase using 5'-hydroxyl termini of DNA and [gamma-32ATP] after 30 mins by liquid scintillation counting | Bioorg Med Chem 19: 5803-12 (2011) Article DOI: 10.1016/j.bmc.2011.08.023 BindingDB Entry DOI: 10.7270/Q2DZ0989 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Polynucleotide kinase (Enterobacteria phage T4) | BDBM50356643 (CHEMBL1917198) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Kyoto Prefectural University Curated by ChEMBL | Assay Description Inhibition of T4 polynucleotide kinase using 5'-hydroxyl termini of DNA and [gamma-32ATP] after 30 mins by liquid scintillation counting | Bioorg Med Chem 19: 5803-12 (2011) Article DOI: 10.1016/j.bmc.2011.08.023 BindingDB Entry DOI: 10.7270/Q2DZ0989 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Polynucleotide kinase (Enterobacteria phage T4) | BDBM50448689 (CHEMBL3127730) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >2.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Kobe Gakuin University Curated by ChEMBL | Assay Description Inhibition of T4 bacteriophage polynucleotide kinase assessed as inhibition of incorporation of dTTP into poly(dA)/oligo(dT)18 after 60 mins | Bioorg Med Chem 22: 1070-6 (2014) Article DOI: 10.1016/j.bmc.2013.12.038 BindingDB Entry DOI: 10.7270/Q22V2HMW | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Polynucleotide kinase (Enterobacteria phage T4) | BDBM50448688 (Pecilocin | Variotin) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | Purchase MCE KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >2.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Kobe Gakuin University Curated by ChEMBL | Assay Description Inhibition of T4 bacteriophage polynucleotide kinase assessed as inhibition of incorporation of dTTP into poly(dA)/oligo(dT)18 after 60 mins | Bioorg Med Chem 22: 1070-6 (2014) Article DOI: 10.1016/j.bmc.2013.12.038 BindingDB Entry DOI: 10.7270/Q22V2HMW | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Polynucleotide kinase (Enterobacteria phage T4) | BDBM50379292 (CHEMBL2011646) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >2.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Science University of Tokyo Curated by ChEMBL | Assay Description Inhibition of T4 arnN8l pseT 1 polynucleotide kinase assessed as inhibition of Salmon sperm DNA phosphorylation using [gamma32P]ATP by liquid scintil... | J Nat Prod 75: 135-41 (2012) Article DOI: 10.1021/np200523b BindingDB Entry DOI: 10.7270/Q2T154NG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Polynucleotide kinase (Enterobacteria phage T4) | BDBM50379294 (CHEMBL2011647) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >2.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Science University of Tokyo Curated by ChEMBL | Assay Description Inhibition of T4 arnN8l pseT 1 polynucleotide kinase assessed as inhibition of Salmon sperm DNA phosphorylation using [gamma32P]ATP by liquid scintil... | J Nat Prod 75: 135-41 (2012) Article DOI: 10.1021/np200523b BindingDB Entry DOI: 10.7270/Q2T154NG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Polynucleotide kinase (Enterobacteria phage T4) | BDBM50448690 (CHEMBL3127728) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | >2.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Kobe Gakuin University Curated by ChEMBL | Assay Description Inhibition of T4 bacteriophage polynucleotide kinase assessed as inhibition of incorporation of dTTP into poly(dA)/oligo(dT)18 after 60 mins | Bioorg Med Chem 22: 1070-6 (2014) Article DOI: 10.1016/j.bmc.2013.12.038 BindingDB Entry DOI: 10.7270/Q22V2HMW | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Polynucleotide kinase (Enterobacteria phage T4) | BDBM50448691 (CHEMBL3127729) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | >2.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Kobe Gakuin University Curated by ChEMBL | Assay Description Inhibition of T4 bacteriophage polynucleotide kinase assessed as inhibition of incorporation of dTTP into poly(dA)/oligo(dT)18 after 60 mins | Bioorg Med Chem 22: 1070-6 (2014) Article DOI: 10.1016/j.bmc.2013.12.038 BindingDB Entry DOI: 10.7270/Q22V2HMW | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Polynucleotide kinase (Enterobacteria phage T4) | BDBM50379293 (CHEMBL2011648) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >2.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Science University of Tokyo Curated by ChEMBL | Assay Description Inhibition of T4 arnN8l pseT 1 polynucleotide kinase assessed as inhibition of Salmon sperm DNA phosphorylation using [gamma32P]ATP by liquid scintil... | J Nat Prod 75: 135-41 (2012) Article DOI: 10.1021/np200523b BindingDB Entry DOI: 10.7270/Q2T154NG | |||||||||||
More data for this Ligand-Target Pair |