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Compile Data Set for Download or QSAR

Found 293 hits of ic50 for UniProtKB: O95835   
Target/Host
(Institution)
LigandTarget/Host
Links
Ligand
Links
Trg + Lig
Links
Ki
nM
ΔG°
kcal/mole
IC50
nM
Kd
nM
EC50/IC50
nM
koff
s-1
kon
M-1s-1
pHTemp
°C
Serine/threonine-protein kinase LATS1


(Homo sapiens (Human))
BDBM574325
PNG
(US11458138, Example 154)
Show SMILES CC1(CC1)Nc1nc(nc2cnccc12)-c1ccnc2[nH]ccc12
PDB

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TBA

Assay Description
The LATS1 biochemical HTRF assay was performed using the HTRF KinEASE-STK S1 kit (CisBio, catalogue number 62ST1PEC) according to manufacturer's ...


Citation and Details

BindingDB Entry DOI: 10.7270/Q21Z47NH
More data for this
Ligand-Target Pair
Serine/threonine-protein kinase LATS1


(Homo sapiens (Human))
BDBM574440
PNG
(US11458138, Example 320)
Show SMILES CC(C)(N)C(C)(C)Nc1nc(nc2cnccc12)-c1ccncc1
PDB

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TBA

Assay Description
The LATS1 biochemical Caliper assay was performed as following.Human LATS1 kinase domain protein was purchased from Carnabio (catalogue number 01-123...


Citation and Details

BindingDB Entry DOI: 10.7270/Q21Z47NH
More data for this
Ligand-Target Pair
Serine/threonine-protein kinase LATS1


(Homo sapiens (Human))
BDBM574429
PNG
(US11458138, Example 309)
Show SMILES CN(C)CCC(C)(C)Nc1nc(nc2cnccc12)-c1c[nH]nc1C
PDB

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TBA

Assay Description
The LATS1 biochemical Caliper assay was performed as following.Human LATS1 kinase domain protein was purchased from Carnabio (catalogue number 01-123...


Citation and Details

BindingDB Entry DOI: 10.7270/Q21Z47NH
More data for this
Ligand-Target Pair
Serine/threonine-protein kinase LATS1


(Homo sapiens (Human))
BDBM574437
PNG
(US11458138, Example 317)
Show SMILES CC(C)(CN)CNc1nc(nc2cnccc12)-c1ccncc1
PDB

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TBA

Assay Description
The LATS1 biochemical Caliper assay was performed as following.Human LATS1 kinase domain protein was purchased from Carnabio (catalogue number 01-123...


Citation and Details

BindingDB Entry DOI: 10.7270/Q21Z47NH
More data for this
Ligand-Target Pair
Serine/threonine-protein kinase LATS1


(Homo sapiens (Human))
BDBM574183
PNG
(US11458138, Example 17b)
Show SMILES C[C@H]1CCC[C@H]1Nc1nc(nc2cnccc12)-c1ccncc1 |r|
PDB

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TBA

Assay Description
The LATS1 biochemical HTRF assay was performed using the HTRF KinEASE-STK S1 kit (CisBio, catalogue number 62ST1PEC) according to manufacturer's ...


Citation and Details

BindingDB Entry DOI: 10.7270/Q21Z47NH
More data for this
Ligand-Target Pair
Serine/threonine-protein kinase LATS1


(Homo sapiens (Human))
BDBM574381
PNG
(US11458138, Example 261)
Show SMILES CC(C)(C)Nc1cc(nc2cnccc12)-c1ccncc1
PDB

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TBA

Assay Description
The LATS1 biochemical HTRF assay was performed using the HTRF KinEASE-STK S1 kit (CisBio, catalogue number 62ST1PEC) according to manufacturer's ...


Citation and Details

BindingDB Entry DOI: 10.7270/Q21Z47NH
More data for this
Ligand-Target Pair
Serine/threonine-protein kinase LATS1


(Homo sapiens (Human))
BDBM574238
PNG
(US11458138, Example 68a)
Show SMILES CC[C@H](C)Nc1nc(nc2cnccc12)-c1ccncc1 |r|
PDB

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TBA

Assay Description
The LATS1 biochemical HTRF assay was performed using the HTRF KinEASE-STK S1 kit (CisBio, catalogue number 62ST1PEC) according to manufacturer's ...


Citation and Details

BindingDB Entry DOI: 10.7270/Q21Z47NH
More data for this
Ligand-Target Pair
Serine/threonine-protein kinase LATS1


(Homo sapiens (Human))
BDBM574389
PNG
(US11458138, Example 269)
Show SMILES Cc1n[nH]cc1-c1cc(NC(C)(C)C)c2ccncc2n1
PDB

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TBA

Assay Description
The LATS1 biochemical HTRF assay was performed using the HTRF KinEASE-STK S1 kit (CisBio, catalogue number 62ST1PEC) according to manufacturer's ...


Citation and Details

BindingDB Entry DOI: 10.7270/Q21Z47NH
More data for this
Ligand-Target Pair
Serine/threonine-protein kinase LATS1


(Homo sapiens (Human))
BDBM574233
PNG
(US11458138, Example 64)
Show SMILES FC(F)(F)C1(CC1)Nc1nc(nc2cnccc12)-c1ccncc1
PDB

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TBA

Assay Description
The LATS1 biochemical HTRF assay was performed using the HTRF KinEASE-STK S1 kit (CisBio, catalogue number 62ST1PEC) according to manufacturer's ...


Citation and Details

BindingDB Entry DOI: 10.7270/Q21Z47NH
More data for this
Ligand-Target Pair
Serine/threonine-protein kinase LATS1


(Homo sapiens (Human))
BDBM574232
PNG
(US11458138, Example 63)
Show SMILES CCC(C)(C)Nc1nc(nc2cnccc12)-c1ccncc1
PDB

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TBA

Assay Description
The LATS1 biochemical HTRF assay was performed using the HTRF KinEASE-STK S1 kit (CisBio, catalogue number 62ST1PEC) according to manufacturer's ...


Citation and Details

BindingDB Entry DOI: 10.7270/Q21Z47NH
More data for this
Ligand-Target Pair
Serine/threonine-protein kinase LATS1


(Homo sapiens (Human))
BDBM574231
PNG
(US11458138, Example 62)
Show SMILES FC(F)(F)C1(CCC1)Nc1nc(nc2cnccc12)-c1ccncc1
PDB

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TBA

Assay Description
The LATS1 biochemical HTRF assay was performed using the HTRF KinEASE-STK S1 kit (CisBio, catalogue number 62ST1PEC) according to manufacturer's ...


Citation and Details

BindingDB Entry DOI: 10.7270/Q21Z47NH
More data for this
Ligand-Target Pair
Serine/threonine-protein kinase LATS1


(Homo sapiens (Human))
BDBM574270
PNG
(US11458138, Example 99)
Show SMILES CC1(CC1)Nc1nc(nc2cnccc12)-c1ccncc1
PDB

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TBA

Assay Description
The LATS1 biochemical HTRF assay was performed using the HTRF KinEASE-STK S1 kit (CisBio, catalogue number 62ST1PEC) according to manufacturer's ...


Citation and Details

BindingDB Entry DOI: 10.7270/Q21Z47NH
More data for this
Ligand-Target Pair
Serine/threonine-protein kinase LATS1


(Homo sapiens (Human))
BDBM574276
PNG
(US11458138, Example 105)
Show SMILES NCCCCCNc1nc(nc2cnccc12)-c1ccncc1
PDB

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TBA

Assay Description
The LATS1 biochemical HTRF assay was performed using the HTRF KinEASE-STK S1 kit (CisBio, catalogue number 62ST1PEC) according to manufacturer's ...


Citation and Details

BindingDB Entry DOI: 10.7270/Q21Z47NH
More data for this
Ligand-Target Pair
Serine/threonine-protein kinase LATS1


(Homo sapiens (Human))
BDBM574280
PNG
(US11458138, Example 109)
Show SMILES CN(C)CCC(C)(C)Nc1nc(nc2cnccc12)-c1ccncc1
PDB

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TBA

Assay Description
The LATS1 biochemical HTRF assay was performed using the HTRF KinEASE-STK S1 kit (CisBio, catalogue number 62ST1PEC) according to manufacturer's ...


Citation and Details

BindingDB Entry DOI: 10.7270/Q21Z47NH
More data for this
Ligand-Target Pair
Serine/threonine-protein kinase LATS1


(Homo sapiens (Human))
BDBM574282
PNG
(US11458138, Example 111)
Show SMILES FC(F)(F)c1n[nH]cc1-c1nc(NC2CCCC2)c2ccncc2n1
PDB

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TBA

Assay Description
The LATS1 biochemical HTRF assay was performed using the HTRF KinEASE-STK S1 kit (CisBio, catalogue number 62ST1PEC) according to manufacturer's ...


Citation and Details

BindingDB Entry DOI: 10.7270/Q21Z47NH
More data for this
Ligand-Target Pair
Serine/threonine-protein kinase LATS1


(Homo sapiens (Human))
BDBM574305
PNG
(US11458138, Example 134)
Show SMILES CC(C)(Nc1nc(nc2cnccc12)-c1ccncc1F)C(F)(F)F
PDB

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TBA

Assay Description
The LATS1 biochemical HTRF assay was performed using the HTRF KinEASE-STK S1 kit (CisBio, catalogue number 62ST1PEC) according to manufacturer's ...


Citation and Details

BindingDB Entry DOI: 10.7270/Q21Z47NH
More data for this
Ligand-Target Pair
Serine/threonine-protein kinase LATS1


(Homo sapiens (Human))
BDBM574326
PNG
(US11458138, Example 155)
Show SMILES CCCNc1nc(nc2cnccc12)-c1c[nH]c2ncccc12
PDB

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TBA

Assay Description
The LATS1 biochemical HTRF assay was performed using the HTRF KinEASE-STK S1 kit (CisBio, catalogue number 62ST1PEC) according to manufacturer's ...


Citation and Details

BindingDB Entry DOI: 10.7270/Q21Z47NH
More data for this
Ligand-Target Pair
Serine/threonine-protein kinase LATS1


(Homo sapiens (Human))
BDBM574369
PNG
(US11458138, Example 198)
Show SMILES CC1(CC1)Nc1nc(nc2c(Cl)nccc12)-c1ccncc1
PDB

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TBA

Assay Description
The LATS1 biochemical HTRF assay was performed using the HTRF KinEASE-STK S1 kit (CisBio, catalogue number 62ST1PEC) according to manufacturer's ...


Citation and Details

BindingDB Entry DOI: 10.7270/Q21Z47NH
More data for this
Ligand-Target Pair
Serine/threonine-protein kinase LATS1


(Homo sapiens (Human))
BDBM574370
PNG
(US11458138, Example 199)
Show SMILES Cc1nccc2c(NC3(C)CC3)nc(nc12)-c1ccncc1
PDB

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TBA

Assay Description
The LATS1 biochemical HTRF assay was performed using the HTRF KinEASE-STK S1 kit (CisBio, catalogue number 62ST1PEC) according to manufacturer's ...


Citation and Details

BindingDB Entry DOI: 10.7270/Q21Z47NH
More data for this
Ligand-Target Pair
Serine/threonine-protein kinase LATS1


(Homo sapiens (Human))
BDBM573837
PNG
(N-(2-cyclopropylpropan-2-yl)-2-(pyridin-4-yl)pyrid...)
Show SMILES CC(C)(Nc1nc(nc2cnccc12)-c1ccncc1)C1CC1
PDB

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Assay Description
The LATS1 biochemical HTRF assay was performed using the HTRF KinEASE-STK S1 kit (CisBio, catalogue number 62ST1PEC) according to manufacturer's ...


Citation and Details

BindingDB Entry DOI: 10.7270/Q21Z47NH
More data for this
Ligand-Target Pair
Serine/threonine-protein kinase LATS1


(Homo sapiens (Human))
BDBM573863
PNG
(US11458138, Example 2)
Show SMILES CCN(CC)c1nc(nc2cnccc12)-c1ccncc1
PDB

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TBA

Assay Description
The LATS1 biochemical HTRF assay was performed using the HTRF KinEASE-STK S1 kit (CisBio, catalogue number 62ST1PEC) according to manufacturer's ...


Citation and Details

BindingDB Entry DOI: 10.7270/Q21Z47NH
More data for this
Ligand-Target Pair
Serine/threonine-protein kinase LATS1


(Homo sapiens (Human))
BDBM573866
PNG
(US11458138, Example 3)
Show SMILES CCN(C(C)C)c1nc(nc2cnccc12)-c1ccncc1
PDB

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Assay Description
The LATS1 biochemical HTRF assay was performed using the HTRF KinEASE-STK S1 kit (CisBio, catalogue number 62ST1PEC) according to manufacturer's ...


Citation and Details

BindingDB Entry DOI: 10.7270/Q21Z47NH
More data for this
Ligand-Target Pair
Serine/threonine-protein kinase LATS1


(Homo sapiens (Human))
BDBM573884
PNG
(US11458138, Example 4)
Show SMILES CC(Nc1nc(nc2cnccc12)-c1ccncc1)C(F)(F)F
PDB

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Assay Description
The LATS1 biochemical HTRF assay was performed using the HTRF KinEASE-STK S1 kit (CisBio, catalogue number 62ST1PEC) according to manufacturer's ...


Citation and Details

BindingDB Entry DOI: 10.7270/Q21Z47NH
More data for this
Ligand-Target Pair
Serine/threonine-protein kinase LATS1


(Homo sapiens (Human))
BDBM573896
PNG
(US11458138, Example 6)
Show SMILES CC(C)Nc1nc(nc2cnccc12)-c1ccncc1
PDB

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Assay Description
The LATS1 biochemical HTRF assay was performed using the HTRF KinEASE-STK S1 kit (CisBio, catalogue number 62ST1PEC) according to manufacturer's ...


Citation and Details

BindingDB Entry DOI: 10.7270/Q21Z47NH
More data for this
Ligand-Target Pair
Serine/threonine-protein kinase LATS1


(Homo sapiens (Human))
BDBM574181
PNG
(US11458138, Example 17 | US11458138, Example 17a |...)
Show SMILES CC1CCCC1Nc1nc(nc2cnccc12)-c1ccncc1
PDB

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Assay Description
The LATS1 biochemical HTRF assay was performed using the HTRF KinEASE-STK S1 kit (CisBio, catalogue number 62ST1PEC) according to manufacturer's ...


Citation and Details

BindingDB Entry DOI: 10.7270/Q21Z47NH
More data for this
Ligand-Target Pair
Serine/threonine-protein kinase LATS1


(Homo sapiens (Human))
BDBM574218
PNG
(US11458138, Example 49)
Show SMILES CC(C)(O)CC(C)(C)Nc1nc(nc2cnccc12)-c1ccncc1
PDB

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Assay Description
The LATS1 biochemical HTRF assay was performed using the HTRF KinEASE-STK S1 kit (CisBio, catalogue number 62ST1PEC) according to manufacturer's ...


Citation and Details

BindingDB Entry DOI: 10.7270/Q21Z47NH
More data for this
Ligand-Target Pair
Serine/threonine-protein kinase LATS1


(Homo sapiens (Human))
BDBM574227
PNG
(US11458138, Example 58)
Show SMILES CC(C)(Nc1nc(nc2cnccc12)-c1ccncc1)C(F)(F)F
PDB

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Assay Description
The LATS1 biochemical HTRF assay was performed using the HTRF KinEASE-STK S1 kit (CisBio, catalogue number 62ST1PEC) according to manufacturer's ...


Citation and Details

BindingDB Entry DOI: 10.7270/Q21Z47NH
More data for this
Ligand-Target Pair
Serine/threonine-protein kinase LATS1


(Homo sapiens (Human))
BDBM574228
PNG
(US11458138, Example 59)
Show SMILES CC(C)(C)Nc1nc(nc2cnccc12)-c1ccncc1
PDB

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Assay Description
The LATS1 biochemical HTRF assay was performed using the HTRF KinEASE-STK S1 kit (CisBio, catalogue number 62ST1PEC) according to manufacturer's ...


Citation and Details

BindingDB Entry DOI: 10.7270/Q21Z47NH
More data for this
Ligand-Target Pair
Serine/threonine-protein kinase LATS1


(Homo sapiens (Human))
BDBM574229
PNG
(US11458138, Example 60)
Show SMILES CC1(CCC1)Nc1nc(nc2cnccc12)-c1ccncc1
PDB

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Assay Description
The LATS1 biochemical HTRF assay was performed using the HTRF KinEASE-STK S1 kit (CisBio, catalogue number 62ST1PEC) according to manufacturer's ...


Citation and Details

BindingDB Entry DOI: 10.7270/Q21Z47NH
More data for this
Ligand-Target Pair
Serine/threonine-protein kinase LATS1


(Homo sapiens (Human))
BDBM574230
PNG
(US11458138, Example 61)
Show SMILES CC(C)(CCO)Nc1nc(nc2cnccc12)-c1ccncc1
PDB

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Assay Description
The LATS1 biochemical HTRF assay was performed using the HTRF KinEASE-STK S1 kit (CisBio, catalogue number 62ST1PEC) according to manufacturer's ...


Citation and Details

BindingDB Entry DOI: 10.7270/Q21Z47NH
More data for this
Ligand-Target Pair
Serine/threonine-protein kinase LATS1


(Homo sapiens (Human))
BDBM574426
PNG
(US11458138, Example 306)
Show SMILES CN(c1cc(nc2cnccc12)-c1ccncc1)C(C)(C)C
PDB

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Assay Description
The LATS1 biochemical Caliper assay was performed as following.Human LATS1 kinase domain protein was purchased from Carnabio (catalogue number 01-123...


Citation and Details

BindingDB Entry DOI: 10.7270/Q21Z47NH
More data for this
Ligand-Target Pair
Serine/threonine-protein kinase LATS1


(Homo sapiens (Human))
BDBM574420
PNG
(US11458138, Example 300)
Show SMILES CC1(CCC1)Nc1cc(nc2cnccc12)-c1ccncc1
PDB

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Assay Description
The LATS1 biochemical Caliper assay was performed as following.Human LATS1 kinase domain protein was purchased from Carnabio (catalogue number 01-123...


Citation and Details

BindingDB Entry DOI: 10.7270/Q21Z47NH
More data for this
Ligand-Target Pair
Serine/threonine-protein kinase LATS1


(Homo sapiens (Human))
BDBM574438
PNG
(US11458138, Example 318)
Show SMILES CC(C)(CC(N)=O)Nc1nc(nc2cnccc12)-c1ccncc1
PDB

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Assay Description
The LATS1 biochemical Caliper assay was performed as following.Human LATS1 kinase domain protein was purchased from Carnabio (catalogue number 01-123...


Citation and Details

BindingDB Entry DOI: 10.7270/Q21Z47NH
More data for this
Ligand-Target Pair
Serine/threonine-protein kinase LATS1


(Homo sapiens (Human))
BDBM574427
PNG
(US11458138, Example 307)
Show SMILES CC1(CCC1)Nc1cc(nc2cnccc12)-c1ccncn1
PDB

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Assay Description
The LATS1 biochemical Caliper assay was performed as following.Human LATS1 kinase domain protein was purchased from Carnabio (catalogue number 01-123...


Citation and Details

BindingDB Entry DOI: 10.7270/Q21Z47NH
More data for this
Ligand-Target Pair
Serine/threonine-protein kinase LATS1


(Homo sapiens (Human))
BDBM574390
PNG
(US11458138, Example 270)
Show SMILES CC(C)(C)Nc1cc(nc2cnccc12)-c1ccncn1
PDB

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Assay Description
The LATS1 biochemical HTRF assay was performed using the HTRF KinEASE-STK S1 kit (CisBio, catalogue number 62ST1PEC) according to manufacturer's ...


Citation and Details

BindingDB Entry DOI: 10.7270/Q21Z47NH
More data for this
Ligand-Target Pair
Serine/threonine-protein kinase LATS1


(Homo sapiens (Human))
BDBM574237
PNG
(US11458138, Example 68 | US11458138, Example 68b)
Show SMILES CCC(C)Nc1nc(nc2cnccc12)-c1ccncc1
PDB

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Assay Description
The LATS1 biochemical HTRF assay was performed using the HTRF KinEASE-STK S1 kit (CisBio, catalogue number 62ST1PEC) according to manufacturer's ...


Citation and Details

BindingDB Entry DOI: 10.7270/Q21Z47NH
More data for this
Ligand-Target Pair
Serine/threonine-protein kinase LATS1


(Homo sapiens (Human))
BDBM574392
PNG
(US11458138, Example 272)
Show SMILES CC(C)(C)Nc1cc(nc2cnccc12)-c1ccnc2[nH]ccc12
PDB

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Assay Description
The LATS1 biochemical HTRF assay was performed using the HTRF KinEASE-STK S1 kit (CisBio, catalogue number 62ST1PEC) according to manufacturer's ...


Citation and Details

BindingDB Entry DOI: 10.7270/Q21Z47NH
More data for this
Ligand-Target Pair
Serine/threonine-protein kinase LATS1


(Homo sapiens (Human))
BDBM574407
PNG
(US11458138, Example 287)
Show SMILES CCCNc1nc(nc2cnccc12)-c1c[nH]nc1C(F)(F)F
PDB

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Assay Description
The LATS1 biochemical HTRF assay was performed using the HTRF KinEASE-STK S1 kit (CisBio, catalogue number 62ST1PEC) according to manufacturer's ...


Citation and Details

BindingDB Entry DOI: 10.7270/Q21Z47NH
More data for this
Ligand-Target Pair
Serine/threonine-protein kinase LATS1


(Homo sapiens (Human))
BDBM574391
PNG
(US11458138, Example 271)
Show SMILES CN(C)\C=C\C(=O)c1cc(NC(C)(C)C)c2ccncc2n1
PDB

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TBA

Assay Description
The LATS1 biochemical HTRF assay was performed using the HTRF KinEASE-STK S1 kit (CisBio, catalogue number 62ST1PEC) according to manufacturer's ...


Citation and Details

BindingDB Entry DOI: 10.7270/Q21Z47NH
More data for this
Ligand-Target Pair
Serine/threonine-protein kinase LATS1


(Homo sapiens (Human))
BDBM574237
PNG
(US11458138, Example 68 | US11458138, Example 68b)
Show SMILES CCC(C)Nc1nc(nc2cnccc12)-c1ccncc1
PDB

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Assay Description
The LATS1 biochemical HTRF assay was performed using the HTRF KinEASE-STK S1 kit (CisBio, catalogue number 62ST1PEC) according to manufacturer's ...


Citation and Details

BindingDB Entry DOI: 10.7270/Q21Z47NH
More data for this
Ligand-Target Pair
Serine/threonine-protein kinase LATS1


(Homo sapiens (Human))
BDBM574274
PNG
(US11458138, Example 103)
Show SMILES CC(C)CNc1nc(nc2cnccc12)-c1ccncc1
PDB

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Assay Description
The LATS1 biochemical HTRF assay was performed using the HTRF KinEASE-STK S1 kit (CisBio, catalogue number 62ST1PEC) according to manufacturer's ...


Citation and Details

BindingDB Entry DOI: 10.7270/Q21Z47NH
More data for this
Ligand-Target Pair
Serine/threonine-protein kinase LATS1


(Homo sapiens (Human))
BDBM574281
PNG
(US11458138, Example 110)
Show SMILES CC(C)(CN)Nc1nc(nc2cnccc12)-c1ccncc1
PDB

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Assay Description
The LATS1 biochemical HTRF assay was performed using the HTRF KinEASE-STK S1 kit (CisBio, catalogue number 62ST1PEC) according to manufacturer's ...


Citation and Details

BindingDB Entry DOI: 10.7270/Q21Z47NH
More data for this
Ligand-Target Pair
Serine/threonine-protein kinase LATS1


(Homo sapiens (Human))
BDBM574283
PNG
(US11458138, Example 112)
Show SMILES CC(C)(C)Nc1nc(nc2cnccc12)-c1ccnc(N)c1
PDB

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Assay Description
The LATS1 biochemical HTRF assay was performed using the HTRF KinEASE-STK S1 kit (CisBio, catalogue number 62ST1PEC) according to manufacturer's ...


Citation and Details

BindingDB Entry DOI: 10.7270/Q21Z47NH
More data for this
Ligand-Target Pair
Serine/threonine-protein kinase LATS1


(Homo sapiens (Human))
BDBM574285
PNG
(US11458138, Example 114)
Show SMILES Cc1c(-c2nc(NC(C)(C)C)c3ccncc3n2)c2cccnc2n1S(=O)(=O)c1ccc(C)cc1
PDB

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Assay Description
The LATS1 biochemical HTRF assay was performed using the HTRF KinEASE-STK S1 kit (CisBio, catalogue number 62ST1PEC) according to manufacturer's ...


Citation and Details

BindingDB Entry DOI: 10.7270/Q21Z47NH
More data for this
Ligand-Target Pair
Serine/threonine-protein kinase LATS1


(Homo sapiens (Human))
BDBM574286
PNG
(US11458138, Example 115)
Show SMILES CC(C)(C)Nc1nc(nc2cnccc12)-c1c[nH]nc1C(F)(F)F
PDB

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Assay Description
The LATS1 biochemical HTRF assay was performed using the HTRF KinEASE-STK S1 kit (CisBio, catalogue number 62ST1PEC) according to manufacturer's ...


Citation and Details

BindingDB Entry DOI: 10.7270/Q21Z47NH
More data for this
Ligand-Target Pair
Serine/threonine-protein kinase LATS1


(Homo sapiens (Human))
BDBM574304
PNG
(US11458138, Example 133)
Show SMILES Cc1n[nH]cc1-c1nc(NC2(C)CC2)c2ccncc2n1
PDB

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Assay Description
The LATS1 biochemical HTRF assay was performed using the HTRF KinEASE-STK S1 kit (CisBio, catalogue number 62ST1PEC) according to manufacturer's ...


Citation and Details

BindingDB Entry DOI: 10.7270/Q21Z47NH
More data for this
Ligand-Target Pair
Serine/threonine-protein kinase LATS1


(Homo sapiens (Human))
BDBM574306
PNG
(US11458138, Example 135)
Show SMILES Cc1n[nH]cc1-c1nc(NC(C)(C)C(F)(F)F)c2ccncc2n1
PDB

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Assay Description
The LATS1 biochemical HTRF assay was performed using the HTRF KinEASE-STK S1 kit (CisBio, catalogue number 62ST1PEC) according to manufacturer's ...


Citation and Details

BindingDB Entry DOI: 10.7270/Q21Z47NH
More data for this
Ligand-Target Pair
Serine/threonine-protein kinase LATS1


(Homo sapiens (Human))
BDBM574307
PNG
(US11458138, Example 136)
Show SMILES C[C@H](N(C)c1nc(nc2cnccc12)-c1ccncc1F)C(F)(F)F |r|
PDB

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Assay Description
The LATS1 biochemical HTRF assay was performed using the HTRF KinEASE-STK S1 kit (CisBio, catalogue number 62ST1PEC) according to manufacturer's ...


Citation and Details

BindingDB Entry DOI: 10.7270/Q21Z47NH
More data for this
Ligand-Target Pair
Serine/threonine-protein kinase LATS1


(Homo sapiens (Human))
BDBM574309
PNG
(US11458138, Example 138)
Show SMILES CC1(CC1)Nc1nc(nc2cnccc12)-c1ccnc(N)c1
PDB

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Assay Description
The LATS1 biochemical HTRF assay was performed using the HTRF KinEASE-STK S1 kit (CisBio, catalogue number 62ST1PEC) according to manufacturer's ...


Citation and Details

BindingDB Entry DOI: 10.7270/Q21Z47NH
More data for this
Ligand-Target Pair
Serine/threonine-protein kinase LATS1


(Homo sapiens (Human))
BDBM574350
PNG
(US11458138, Example 179)
Show SMILES CC1(CC1)Nc1nc(nc2cnccc12)-n1ccc2ncccc12
PDB

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Assay Description
The LATS1 biochemical HTRF assay was performed using the HTRF KinEASE-STK S1 kit (CisBio, catalogue number 62ST1PEC) according to manufacturer's ...


Citation and Details

BindingDB Entry DOI: 10.7270/Q21Z47NH
More data for this
Ligand-Target Pair
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