Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kcal/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Bombesin receptor subtype-3 (Mus musculus) | BDBM50533323 (CHEMBL4435571) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 0.800 | n/a | n/a | n/a | n/a |
Daiichi Sankyo Co., Ltd Curated by ChEMBL | Assay Description Agonist activity at mouse BRS3 expressed in CHOK1 cells measured after 1 hrs by IP-One HTRF assay | Bioorg Med Chem Lett 26: 4205-10 (2016) Article DOI: 10.1016/j.bmcl.2016.07.056 BindingDB Entry DOI: 10.7270/Q2CF9TMX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bombesin receptor subtype-3 (Mus musculus) | BDBM50533323 (CHEMBL4435571) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 0.800 | n/a | n/a | n/a | n/a |
Daiichi Sankyo Co., Ltd Curated by ChEMBL | Assay Description Agonist activity at mouse BRS3 expressed in CHOK1 cells measured after 1 hrs by IP-One HTRF assay | Bioorg Med Chem Lett 26: 4205-10 (2016) Article DOI: 10.1016/j.bmcl.2016.07.056 BindingDB Entry DOI: 10.7270/Q2CF9TMX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bombesin receptor subtype-3 (Mus musculus) | BDBM50447496 (CHEMBL3115400) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 1 | n/a | n/a | n/a | n/a |
Daiichi Sankyo Co., Ltd Curated by ChEMBL | Assay Description Agonist activity at mouse BRS-3 expressed in CHOK1 cells after 1 hr by HTRF assay | Bioorg Med Chem Lett 24: 750-5 (2014) Article DOI: 10.1016/j.bmcl.2013.12.106 BindingDB Entry DOI: 10.7270/Q2J967WH | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bombesin receptor subtype-3 (Mus musculus) | BDBM50447496 (CHEMBL3115400) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 1 | n/a | n/a | n/a | n/a |
Daiichi Sankyo Co., Ltd Curated by ChEMBL | Assay Description Agonist activity at mouse BRS3 expressed in CHO-K1 cells by IP-One HTRF assay | Bioorg Med Chem 23: 89-104 (2014) Article DOI: 10.1016/j.bmc.2014.11.018 BindingDB Entry DOI: 10.7270/Q2VT1TPX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bombesin receptor subtype-3 (Mus musculus) | BDBM50533320 (CHEMBL4580739) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 2 | n/a | n/a | n/a | n/a |
Daiichi Sankyo Co., Ltd Curated by ChEMBL | Assay Description Agonist activity at mouse BRS3 expressed in CHOK1 cells measured after 1 hrs by IP-One HTRF assay | Bioorg Med Chem Lett 26: 4205-10 (2016) Article DOI: 10.1016/j.bmcl.2016.07.056 BindingDB Entry DOI: 10.7270/Q2CF9TMX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bombesin receptor subtype-3 (Mus musculus) | BDBM50533320 (CHEMBL4580739) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 2 | n/a | n/a | n/a | n/a |
Daiichi Sankyo Co., Ltd Curated by ChEMBL | Assay Description Agonist activity at mouse BRS3 expressed in CHOK1 cells measured after 1 hrs by IP-One HTRF assay | Bioorg Med Chem Lett 26: 4205-10 (2016) Article DOI: 10.1016/j.bmcl.2016.07.056 BindingDB Entry DOI: 10.7270/Q2CF9TMX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bombesin receptor subtype-3 (Mus musculus) | BDBM50447497 (CHEMBL3115399) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 2.70 | n/a | n/a | n/a | n/a |
Daiichi Sankyo Co., Ltd Curated by ChEMBL | Assay Description Agonist activity at mouse BRS3 expressed in CHO-K1 cells by IP-One HTRF assay | Bioorg Med Chem 23: 89-104 (2014) Article DOI: 10.1016/j.bmc.2014.11.018 BindingDB Entry DOI: 10.7270/Q2VT1TPX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bombesin receptor subtype-3 (Mus musculus) | BDBM50447497 (CHEMBL3115399) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 2.70 | n/a | n/a | n/a | n/a |
Daiichi Sankyo Co., Ltd Curated by ChEMBL | Assay Description Agonist activity at mouse BRS-3 expressed in CHOK1 cells after 1 hr by HTRF assay | Bioorg Med Chem Lett 24: 750-5 (2014) Article DOI: 10.1016/j.bmcl.2013.12.106 BindingDB Entry DOI: 10.7270/Q2J967WH | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bombesin receptor subtype-3 (Mus musculus) | BDBM50447477 (CHEMBL3115388) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 2.70 | n/a | n/a | n/a | n/a |
Daiichi Sankyo Co., Ltd Curated by ChEMBL | Assay Description Agonist activity at mouse BRS3 expressed in CHO-K1 cells by IP-One HTRF assay | Bioorg Med Chem 23: 89-104 (2014) Article DOI: 10.1016/j.bmc.2014.11.018 BindingDB Entry DOI: 10.7270/Q2VT1TPX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bombesin receptor subtype-3 (Mus musculus) | BDBM50447477 (CHEMBL3115388) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 2.70 | n/a | n/a | n/a | n/a |
Daiichi Sankyo Co., Ltd Curated by ChEMBL | Assay Description Agonist activity at mouse BRS-3 expressed in CHOK1 cells after 1 hr by HTRF assay | Bioorg Med Chem Lett 24: 750-5 (2014) Article DOI: 10.1016/j.bmcl.2013.12.106 BindingDB Entry DOI: 10.7270/Q2J967WH | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bombesin receptor subtype-3 (Mus musculus) | BDBM50447492 (CHEMBL3115373) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 2.80 | n/a | n/a | n/a | n/a |
Daiichi Sankyo Co., Ltd Curated by ChEMBL | Assay Description Agonist activity at mouse BRS3 expressed in CHO-K1 cells by IP-One HTRF assay | Bioorg Med Chem 23: 89-104 (2014) Article DOI: 10.1016/j.bmc.2014.11.018 BindingDB Entry DOI: 10.7270/Q2VT1TPX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bombesin receptor subtype-3 (Mus musculus) | BDBM50314969 (2-(4-(2-(4-(2,2-dimethylbutyl)-1H-imidazol-2-yl)et...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | 2.80 | n/a | n/a | n/a | n/a |
Merck Research Laboratories Curated by ChEMBL | Assay Description Agonist activity at mouse BRS-3 expressed in HEK293 cells coexpressing AEQ over 10 mins by aequorin bioluminescence assay | Bioorg Med Chem Lett 20: 2074-7 (2010) Article DOI: 10.1016/j.bmcl.2010.02.076 BindingDB Entry DOI: 10.7270/Q2XW4JX6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bombesin receptor subtype-3 (Mus musculus) | BDBM50447492 (CHEMBL3115373) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 2.80 | n/a | n/a | n/a | n/a |
Daiichi Sankyo Co., Ltd Curated by ChEMBL | Assay Description Agonist activity at mouse BRS-3 expressed in CHOK1 cells after 1 hr by HTRF assay | Bioorg Med Chem Lett 24: 750-5 (2014) Article DOI: 10.1016/j.bmcl.2013.12.106 BindingDB Entry DOI: 10.7270/Q2J967WH | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bombesin receptor subtype-3 (Mus musculus) | BDBM50316914 (5-((4'-(2-(4-(2,2-dimethylbutyl)-1H-imidazol-2-yl)...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | 2.90 | n/a | n/a | n/a | n/a |
AMRI Curated by ChEMBL | Assay Description Agonist activity at mouse BRS3 | Bioorg Med Chem Lett 20: 2912-5 (2010) Article DOI: 10.1016/j.bmcl.2010.03.028 BindingDB Entry DOI: 10.7270/Q2416X7S | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bombesin receptor subtype-3 (Mus musculus) | BDBM50533327 (CHEMBL4461212) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 3 | n/a | n/a | n/a | n/a |
Daiichi Sankyo Co., Ltd Curated by ChEMBL | Assay Description Agonist activity at mouse BRS3 expressed in CHOK1 cells measured after 1 hrs by IP-One HTRF assay | Bioorg Med Chem Lett 26: 4205-10 (2016) Article DOI: 10.1016/j.bmcl.2016.07.056 BindingDB Entry DOI: 10.7270/Q2CF9TMX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bombesin receptor subtype-3 (Mus musculus) | BDBM50533327 (CHEMBL4461212) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 3 | n/a | n/a | n/a | n/a |
Daiichi Sankyo Co., Ltd Curated by ChEMBL | Assay Description Agonist activity at mouse BRS3 expressed in CHOK1 cells measured after 1 hrs by IP-One HTRF assay | Bioorg Med Chem Lett 26: 4205-10 (2016) Article DOI: 10.1016/j.bmcl.2016.07.056 BindingDB Entry DOI: 10.7270/Q2CF9TMX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bombesin receptor subtype-3 (Mus musculus) | BDBM50314977 (5-(4-(2-(4-(2,2-dimethylbutyl)-1H-imidazol-2-yl)et...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 3.10 | n/a | n/a | n/a | n/a |
Merck Research Laboratories Curated by ChEMBL | Assay Description Agonist activity at mouse BRS-3 expressed in HEK293 cells coexpressing AEQ over 10 mins by aequorin bioluminescence assay | Bioorg Med Chem Lett 20: 2074-7 (2010) Article DOI: 10.1016/j.bmcl.2010.02.076 BindingDB Entry DOI: 10.7270/Q2XW4JX6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bombesin receptor subtype-3 (Mus musculus) | BDBM50447479 (CHEMBL3115386) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 3.40 | n/a | n/a | n/a | n/a |
Daiichi Sankyo Co., Ltd Curated by ChEMBL | Assay Description Agonist activity at mouse BRS3 expressed in CHO-K1 cells by IP-One HTRF assay | Bioorg Med Chem 23: 89-104 (2014) Article DOI: 10.1016/j.bmc.2014.11.018 BindingDB Entry DOI: 10.7270/Q2VT1TPX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bombesin receptor subtype-3 (Mus musculus) | BDBM50447479 (CHEMBL3115386) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 3.40 | n/a | n/a | n/a | n/a |
Daiichi Sankyo Co., Ltd Curated by ChEMBL | Assay Description Agonist activity at mouse BRS-3 expressed in CHOK1 cells after 1 hr by HTRF assay | Bioorg Med Chem Lett 24: 750-5 (2014) Article DOI: 10.1016/j.bmcl.2013.12.106 BindingDB Entry DOI: 10.7270/Q2J967WH | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bombesin receptor subtype-3 (Mus musculus) | BDBM50447499 (CHEMBL3115397) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 3.5 | n/a | n/a | n/a | n/a |
Daiichi Sankyo Co., Ltd Curated by ChEMBL | Assay Description Agonist activity at mouse BRS-3 expressed in CHOK1 cells after 1 hr by HTRF assay | Bioorg Med Chem Lett 24: 750-5 (2014) Article DOI: 10.1016/j.bmcl.2013.12.106 BindingDB Entry DOI: 10.7270/Q2J967WH | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bombesin receptor subtype-3 (Mus musculus) | BDBM50447475 (CHEMBL3115390) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 3.5 | n/a | n/a | n/a | n/a |
Daiichi Sankyo Co., Ltd Curated by ChEMBL | Assay Description Agonist activity at mouse BRS3 expressed in CHO-K1 cells by IP-One HTRF assay | Bioorg Med Chem 23: 89-104 (2014) Article DOI: 10.1016/j.bmc.2014.11.018 BindingDB Entry DOI: 10.7270/Q2VT1TPX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bombesin receptor subtype-3 (Mus musculus) | BDBM50447475 (CHEMBL3115390) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 3.5 | n/a | n/a | n/a | n/a |
Daiichi Sankyo Co., Ltd Curated by ChEMBL | Assay Description Agonist activity at mouse BRS-3 expressed in CHOK1 cells after 1 hr by HTRF assay | Bioorg Med Chem Lett 24: 750-5 (2014) Article DOI: 10.1016/j.bmcl.2013.12.106 BindingDB Entry DOI: 10.7270/Q2J967WH | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bombesin receptor subtype-3 (Mus musculus) | BDBM50041425 (CHEMBL3356412) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 3.70 | n/a | n/a | n/a | n/a |
Daiichi Sankyo Co., Ltd Curated by ChEMBL | Assay Description Agonist activity at mouse BRS3 expressed in CHO-K1 cells by IP-One HTRF assay | Bioorg Med Chem 23: 89-104 (2014) Article DOI: 10.1016/j.bmc.2014.11.018 BindingDB Entry DOI: 10.7270/Q2VT1TPX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bombesin receptor subtype-3 (Mus musculus) | BDBM50314974 (6-(4-(2-(4-(2,2-dimethylbutyl)-1H-imidazol-2-yl)et...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 3.90 | n/a | n/a | n/a | n/a |
Merck Research Laboratories Curated by ChEMBL | Assay Description Agonist activity at mouse BRS-3 expressed in HEK293 cells coexpressing AEQ over 10 mins by aequorin bioluminescence assay | Bioorg Med Chem Lett 20: 2074-7 (2010) Article DOI: 10.1016/j.bmcl.2010.02.076 BindingDB Entry DOI: 10.7270/Q2XW4JX6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bombesin receptor subtype-3 (Mus musculus) | BDBM50533331 (CHEMBL4448589) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 4 | n/a | n/a | n/a | n/a |
Daiichi Sankyo Co., Ltd Curated by ChEMBL | Assay Description Agonist activity at mouse BRS3 expressed in CHOK1 cells measured after 1 hrs by IP-One HTRF assay | Bioorg Med Chem Lett 26: 4205-10 (2016) Article DOI: 10.1016/j.bmcl.2016.07.056 BindingDB Entry DOI: 10.7270/Q2CF9TMX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bombesin receptor subtype-3 (Mus musculus) | BDBM50533331 (CHEMBL4448589) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 4 | n/a | n/a | n/a | n/a |
Daiichi Sankyo Co., Ltd Curated by ChEMBL | Assay Description Agonist activity at mouse BRS3 expressed in CHOK1 cells measured after 1 hrs by IP-One HTRF assay | Bioorg Med Chem Lett 26: 4205-10 (2016) Article DOI: 10.1016/j.bmcl.2016.07.056 BindingDB Entry DOI: 10.7270/Q2CF9TMX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bombesin receptor subtype-3 (Mus musculus) | BDBM50314970 (3-(4-(2-(4-(2,2-dimethylbutyl)-1H-imidazol-2-yl)et...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 4.30 | n/a | n/a | n/a | n/a |
Merck Research Laboratories Curated by ChEMBL | Assay Description Agonist activity at mouse BRS-3 expressed in HEK293 cells coexpressing AEQ over 10 mins by aequorin bioluminescence assay | Bioorg Med Chem Lett 20: 2074-7 (2010) Article DOI: 10.1016/j.bmcl.2010.02.076 BindingDB Entry DOI: 10.7270/Q2XW4JX6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bombesin receptor subtype-3 (Mus musculus) | BDBM50316912 (5-((4'-(2-(4-(2,2-dimethylbutyl)-1H-imidazol-2-yl)...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 4.60 | n/a | n/a | n/a | n/a |
AMRI Curated by ChEMBL | Assay Description Agonist activity at mouse BRS3 | Bioorg Med Chem Lett 20: 2912-5 (2010) Article DOI: 10.1016/j.bmcl.2010.03.028 BindingDB Entry DOI: 10.7270/Q2416X7S | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bombesin receptor subtype-3 (Mus musculus) | BDBM50314965 (4'-(2-(4-(cyclohexylmethyl)-1H-imidazol-2-yl)ethyl...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | 4.70 | n/a | n/a | n/a | n/a |
Merck Research Laboratories Curated by ChEMBL | Assay Description Agonist activity at mouse BRS-3 expressed in HEK293 cells coexpressing AEQ over 10 mins by aequorin bioluminescence assay | Bioorg Med Chem Lett 20: 2074-7 (2010) Article DOI: 10.1016/j.bmcl.2010.02.076 BindingDB Entry DOI: 10.7270/Q2XW4JX6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bombesin receptor subtype-3 (Mus musculus) | BDBM50533326 (CHEMBL4593256) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 5 | n/a | n/a | n/a | n/a |
Daiichi Sankyo Co., Ltd Curated by ChEMBL | Assay Description Agonist activity at mouse BRS3 expressed in CHOK1 cells measured after 1 hrs by IP-One HTRF assay | Bioorg Med Chem Lett 26: 4205-10 (2016) Article DOI: 10.1016/j.bmcl.2016.07.056 BindingDB Entry DOI: 10.7270/Q2CF9TMX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bombesin receptor subtype-3 (Mus musculus) | BDBM50533326 (CHEMBL4593256) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 5 | n/a | n/a | n/a | n/a |
Daiichi Sankyo Co., Ltd Curated by ChEMBL | Assay Description Agonist activity at mouse BRS3 expressed in CHOK1 cells measured after 1 hrs by IP-One HTRF assay | Bioorg Med Chem Lett 26: 4205-10 (2016) Article DOI: 10.1016/j.bmcl.2016.07.056 BindingDB Entry DOI: 10.7270/Q2CF9TMX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bombesin receptor subtype-3 (Mus musculus) | BDBM50041423 (CHEMBL3356410) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 5.40 | n/a | n/a | n/a | n/a |
Daiichi Sankyo Co., Ltd Curated by ChEMBL | Assay Description Agonist activity at mouse BRS3 expressed in CHO-K1 cells by IP-One HTRF assay | Bioorg Med Chem 23: 89-104 (2014) Article DOI: 10.1016/j.bmc.2014.11.018 BindingDB Entry DOI: 10.7270/Q2VT1TPX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bombesin receptor subtype-3 (Mus musculus) | BDBM50041424 (CHEMBL3356411) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 5.60 | n/a | n/a | n/a | n/a |
Daiichi Sankyo Co., Ltd Curated by ChEMBL | Assay Description Agonist activity at mouse BRS3 expressed in CHO-K1 cells by IP-One HTRF assay | Bioorg Med Chem 23: 89-104 (2014) Article DOI: 10.1016/j.bmc.2014.11.018 BindingDB Entry DOI: 10.7270/Q2VT1TPX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bombesin receptor subtype-3 (Mus musculus) | BDBM50313743 (4'-(2-(5-(cycloheptylmethyl)-1H-imidazol-2-yl)ethy...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 5.70 | n/a | n/a | n/a | n/a |
Merck Research Laboratories Curated by ChEMBL | Assay Description Agonistic activity at mouse BRS3 expressed in HEK293AEO cells by aequorin bioluminescence assay | Bioorg Med Chem Lett 20: 1913-7 (2010) Article DOI: 10.1016/j.bmcl.2010.01.154 BindingDB Entry DOI: 10.7270/Q2M045KD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bombesin receptor subtype-3 (Mus musculus) | BDBM50316911 (5-((4'-(2-(4-(2,2-dimethylbutyl)-1H-imidazol-2-yl)...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 5.80 | n/a | n/a | n/a | n/a |
AMRI Curated by ChEMBL | Assay Description Agonist activity at mouse BRS3 | Bioorg Med Chem Lett 20: 2912-5 (2010) Article DOI: 10.1016/j.bmcl.2010.03.028 BindingDB Entry DOI: 10.7270/Q2416X7S | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bombesin receptor subtype-3 (Mus musculus) | BDBM50313748 (4'-(2-(5-(3,3-dimethylbutyl)-1H-imidazol-2-yl)ethy...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 6.20 | n/a | n/a | n/a | n/a |
Merck Research Laboratories Curated by ChEMBL | Assay Description Agonistic activity at mouse BRS3 expressed in HEK293AEO cells by aequorin bioluminescence assay | Bioorg Med Chem Lett 20: 1913-7 (2010) Article DOI: 10.1016/j.bmcl.2010.01.154 BindingDB Entry DOI: 10.7270/Q2M045KD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bombesin receptor subtype-3 (Mus musculus) | BDBM50313749 (4'-(2-(5-neopentyl-1H-imidazol-2-yl)ethyl)biphenyl...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | 6.30 | n/a | n/a | n/a | n/a |
Merck Research Laboratories Curated by ChEMBL | Assay Description Agonistic activity at mouse BRS3 expressed in HEK293AEO cells by aequorin bioluminescence assay | Bioorg Med Chem Lett 20: 1913-7 (2010) Article DOI: 10.1016/j.bmcl.2010.01.154 BindingDB Entry DOI: 10.7270/Q2M045KD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bombesin receptor subtype-3 (Mus musculus) | BDBM50314979 (4-(4-(2-(4-(2,2-dimethylbutyl)-1H-imidazol-2-yl)et...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents | Article PubMed | n/a | n/a | n/a | n/a | 6.90 | n/a | n/a | n/a | n/a |
Merck Research Laboratories Curated by ChEMBL | Assay Description Agonist activity at mouse BRS-3 expressed in HEK293 cells coexpressing AEQ over 10 mins by aequorin bioluminescence assay | Bioorg Med Chem Lett 20: 2074-7 (2010) Article DOI: 10.1016/j.bmcl.2010.02.076 BindingDB Entry DOI: 10.7270/Q2XW4JX6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bombesin receptor subtype-3 (Mus musculus) | BDBM50533333 (CHEMBL4464287) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 7 | n/a | n/a | n/a | n/a |
Daiichi Sankyo Co., Ltd Curated by ChEMBL | Assay Description Agonist activity at mouse BRS3 expressed in CHOK1 cells measured after 1 hrs by IP-One HTRF assay | Bioorg Med Chem Lett 26: 4205-10 (2016) Article DOI: 10.1016/j.bmcl.2016.07.056 BindingDB Entry DOI: 10.7270/Q2CF9TMX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bombesin receptor subtype-3 (Mus musculus) | BDBM50533333 (CHEMBL4464287) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 7 | n/a | n/a | n/a | n/a |
Daiichi Sankyo Co., Ltd Curated by ChEMBL | Assay Description Agonist activity at mouse BRS3 expressed in CHOK1 cells measured after 1 hrs by IP-One HTRF assay | Bioorg Med Chem Lett 26: 4205-10 (2016) Article DOI: 10.1016/j.bmcl.2016.07.056 BindingDB Entry DOI: 10.7270/Q2CF9TMX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bombesin receptor subtype-3 (Mus musculus) | BDBM50313740 (4'-(2-(5-(cyclobutylmethyl)-1H-imidazol-2-yl)ethyl...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 7.10 | n/a | n/a | n/a | n/a |
Merck Research Laboratories Curated by ChEMBL | Assay Description Agonistic activity at mouse BRS3 expressed in HEK293AEO cells by aequorin bioluminescence assay | Bioorg Med Chem Lett 20: 1913-7 (2010) Article DOI: 10.1016/j.bmcl.2010.01.154 BindingDB Entry DOI: 10.7270/Q2M045KD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bombesin receptor subtype-3 (Mus musculus) | BDBM50313742 (4'-(2-(5-(cyclohexylmethyl)-1H-imidazol-2-yl)ethyl...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 7.30 | n/a | n/a | n/a | n/a |
Merck Research Laboratories Curated by ChEMBL | Assay Description Agonistic activity at mouse BRS3 expressed in HEK293AEO cells by aequorin bioluminescence assay | Bioorg Med Chem Lett 20: 1913-7 (2010) Article DOI: 10.1016/j.bmcl.2010.01.154 BindingDB Entry DOI: 10.7270/Q2M045KD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bombesin receptor subtype-3 (Mus musculus) | BDBM50313741 (4'-(2-(5-(cyclopentylmethyl)-1H-imidazol-2-yl)ethy...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | 7.90 | n/a | n/a | n/a | n/a |
Merck Research Laboratories Curated by ChEMBL | Assay Description Agonistic activity at mouse BRS3 expressed in HEK293AEO cells by aequorin bioluminescence assay | Bioorg Med Chem Lett 20: 1913-7 (2010) Article DOI: 10.1016/j.bmcl.2010.01.154 BindingDB Entry DOI: 10.7270/Q2M045KD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bombesin receptor subtype-3 (Mus musculus) | BDBM50313736 (4'-(2-(5-(3-fluorobenzyl)-1H-imidazol-2-yl)ethyl)b...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 7.90 | n/a | n/a | n/a | n/a |
Merck Research Laboratories Curated by ChEMBL | Assay Description Agonistic activity at mouse BRS3 expressed in HEK293AEO cells by aequorin bioluminescence assay | Bioorg Med Chem Lett 20: 1913-7 (2010) Article DOI: 10.1016/j.bmcl.2010.01.154 BindingDB Entry DOI: 10.7270/Q2M045KD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bombesin receptor subtype-3 (Mus musculus) | BDBM50313738 (4'-(2-(5-(2,3-difluorobenzyl)-1H-imidazol-2-yl)eth...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 8 | n/a | n/a | n/a | n/a |
Merck Research Laboratories Curated by ChEMBL | Assay Description Agonistic activity at mouse BRS3 expressed in HEK293AEO cells by aequorin bioluminescence assay | Bioorg Med Chem Lett 20: 1913-7 (2010) Article DOI: 10.1016/j.bmcl.2010.01.154 BindingDB Entry DOI: 10.7270/Q2M045KD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bombesin receptor subtype-3 (Mus musculus) | BDBM50041426 (CHEMBL3356413) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 8.10 | n/a | n/a | n/a | n/a |
Daiichi Sankyo Co., Ltd Curated by ChEMBL | Assay Description Agonist activity at mouse BRS3 expressed in CHO-K1 cells by IP-One HTRF assay | Bioorg Med Chem 23: 89-104 (2014) Article DOI: 10.1016/j.bmc.2014.11.018 BindingDB Entry DOI: 10.7270/Q2VT1TPX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bombesin receptor subtype-3 (Mus musculus) | BDBM50447498 (CHEMBL3115398) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 8.70 | n/a | n/a | n/a | n/a |
Daiichi Sankyo Co., Ltd Curated by ChEMBL | Assay Description Agonist activity at mouse BRS-3 expressed in CHOK1 cells after 1 hr by HTRF assay | Bioorg Med Chem Lett 24: 750-5 (2014) Article DOI: 10.1016/j.bmcl.2013.12.106 BindingDB Entry DOI: 10.7270/Q2J967WH | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bombesin receptor subtype-3 (Mus musculus) | BDBM50447484 (CHEMBL3115381) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 8.70 | n/a | n/a | n/a | n/a |
Daiichi Sankyo Co., Ltd Curated by ChEMBL | Assay Description Agonist activity at mouse BRS-3 expressed in CHOK1 cells after 1 hr by HTRF assay | Bioorg Med Chem Lett 24: 750-5 (2014) Article DOI: 10.1016/j.bmcl.2013.12.106 BindingDB Entry DOI: 10.7270/Q2J967WH | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bombesin receptor subtype-3 (Mus musculus) | BDBM50314981 (1-(4-(2-(4-(2,2-dimethylbutyl)-1H-imidazol-2-yl)et...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | 9 | n/a | n/a | n/a | n/a |
Merck Research Laboratories Curated by ChEMBL | Assay Description Agonist activity at mouse BRS-3 expressed in HEK293 cells coexpressing AEQ over 10 mins by aequorin bioluminescence assay | Bioorg Med Chem Lett 20: 2074-7 (2010) Article DOI: 10.1016/j.bmcl.2010.02.076 BindingDB Entry DOI: 10.7270/Q2XW4JX6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bombesin receptor subtype-3 (Mus musculus) | BDBM50313729 (4'-(2-(5-(2-methylbenzyl)-1H-imidazol-2-yl)ethyl)b...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 9.30 | n/a | n/a | n/a | n/a |
Merck Research Laboratories Curated by ChEMBL | Assay Description Agonistic activity at mouse BRS3 expressed in HEK293AEO cells by aequorin bioluminescence assay | Bioorg Med Chem Lett 20: 1913-7 (2010) Article DOI: 10.1016/j.bmcl.2010.01.154 BindingDB Entry DOI: 10.7270/Q2M045KD | |||||||||||
More data for this Ligand-Target Pair |
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