Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kcal/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Peptidase (Staphylococcus aureus) | BDBM50482776 (CHEBI:70718 | Ceftaroline Fosamil | PPI-0903 | TAK...) | PDB MMDB UniProtKB/TrEMBL B.MOAD GoogleScholar AffyNet | Purchase MCE KEGG PC cid PC sid UniChem | Article PubMed | n/a | n/a | 14.6 | n/a | n/a | n/a | n/a | n/a | n/a |
Hershey Medical Center Curated by ChEMBL | Assay Description Binding affinity to against methicillin-, daptomycin-resistant, vancomycin-intermediate, beta-lactamase-positive Staphylococcus aureus 25 PBP2a by co... | Antimicrob Agents Chemother 54: 1670-7 (2010) Article DOI: 10.1128/AAC.00019-10 BindingDB Entry DOI: 10.7270/Q2B56NK6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Peptidase (Staphylococcus aureus) | BDBM50482776 (CHEBI:70718 | Ceftaroline Fosamil | PPI-0903 | TAK...) | PDB MMDB UniProtKB/TrEMBL B.MOAD GoogleScholar AffyNet | Purchase MCE KEGG PC cid PC sid UniChem | Article PubMed | n/a | n/a | 233 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Notre Dame Curated by ChEMBL | Assay Description Inhibition of methicillin-resistant Staphylococcus aureus PBP 2a | Antimicrob Agents Chemother 53: 4051-63 (2009) Article DOI: 10.1128/AAC.00084-09 BindingDB Entry DOI: 10.7270/Q2R21479 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Peptidase (Staphylococcus aureus) | BDBM50483328 (CHEMBL387640 | ME1036) | PDB MMDB UniProtKB/TrEMBL B.MOAD GoogleScholar AffyNet | Purchase PC cid PC sid UniChem | Article PubMed | n/a | n/a | 262 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Notre Dame Curated by ChEMBL | Assay Description Binding affinity to methicillin-resistant Staphylococcus aureus MF535HR PBP 2a by competitive binding assay | Antimicrob Agents Chemother 53: 4051-63 (2009) Article DOI: 10.1128/AAC.00084-09 BindingDB Entry DOI: 10.7270/Q2R21479 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Peptidase (Staphylococcus aureus) | BDBM50482776 (CHEBI:70718 | Ceftaroline Fosamil | PPI-0903 | TAK...) | PDB MMDB UniProtKB/TrEMBL B.MOAD GoogleScholar AffyNet | Purchase MCE KEGG PC cid PC sid UniChem | Article PubMed | n/a | n/a | 365 | n/a | n/a | n/a | n/a | n/a | n/a |
Hershey Medical Center Curated by ChEMBL | Assay Description Binding affinity to methicillin-, vancomycin-resistant, beta-lactamase-positive Staphylococcus aureus 510 PBP2a by competitive binding assay | Antimicrob Agents Chemother 54: 1670-7 (2010) Article DOI: 10.1128/AAC.00019-10 BindingDB Entry DOI: 10.7270/Q2B56NK6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Peptidase (Staphylococcus aureus) | BDBM50103601 (CHEBI:29007 | Ceftriaxone) | PDB MMDB UniProtKB/TrEMBL B.MOAD GoogleScholar AffyNet | KEGG PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 450 | n/a | n/a | n/a | n/a | n/a | n/a |
Hershey Medical Center Curated by ChEMBL | Assay Description Binding affinity to against methicillin-, daptomycin-resistant, vancomycin-intermediate, beta-lactamase-positive Staphylococcus aureus 25 PBP2a by co... | Antimicrob Agents Chemother 54: 1670-7 (2010) Article DOI: 10.1128/AAC.00019-10 BindingDB Entry DOI: 10.7270/Q2B56NK6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Peptidase (Staphylococcus aureus) | BDBM50482777 (CHEBI:204928 | Cefotaxime) | PDB MMDB UniProtKB/TrEMBL B.MOAD GoogleScholar AffyNet | Purchase MCE KEGG PC cid PC sid PDB UniChem | Article PubMed | n/a | n/a | 548 | n/a | n/a | n/a | n/a | n/a | n/a |
Hershey Medical Center Curated by ChEMBL | Assay Description Binding affinity to against methicillin-, daptomycin-resistant, vancomycin-intermediate, beta-lactamase-positive Staphylococcus aureus 25 PBP2a by co... | Antimicrob Agents Chemother 54: 1670-7 (2010) Article DOI: 10.1128/AAC.00019-10 BindingDB Entry DOI: 10.7270/Q2B56NK6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Peptidase (Staphylococcus aureus) | BDBM50482776 (CHEBI:70718 | Ceftaroline Fosamil | PPI-0903 | TAK...) | PDB MMDB UniProtKB/TrEMBL B.MOAD GoogleScholar AffyNet | Purchase MCE KEGG PC cid PC sid UniChem | Article PubMed | n/a | n/a | 730 | n/a | n/a | n/a | n/a | n/a | n/a |
Hershey Medical Center Curated by ChEMBL | Assay Description Binding affinity to methicillin-resistant, heteroresistant vancomycin-intermediate, beta-lactamase-negative Staphylococcus aureus 873 PBP2a by compet... | Antimicrob Agents Chemother 54: 1670-7 (2010) Article DOI: 10.1128/AAC.00019-10 BindingDB Entry DOI: 10.7270/Q2B56NK6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Peptidase (Staphylococcus aureus) | BDBM50483327 (CEFTOBIPROLE MEDOCARIL) | PDB MMDB UniProtKB/TrEMBL B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.30E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Notre Dame Curated by ChEMBL | Assay Description Inhibition of methicillin-resistant Staphylococcus aureus OC 3726 PBP 2a | Antimicrob Agents Chemother 53: 4051-63 (2009) Article DOI: 10.1128/AAC.00084-09 BindingDB Entry DOI: 10.7270/Q2R21479 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Peptidase (Staphylococcus aureus) | BDBM50482776 (CHEBI:70718 | Ceftaroline Fosamil | PPI-0903 | TAK...) | PDB MMDB UniProtKB/TrEMBL B.MOAD GoogleScholar AffyNet | Purchase MCE KEGG PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.46E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Hershey Medical Center Curated by ChEMBL | Assay Description Binding affinity to methicillin-resistant, vancomycin-intermediate, beta-lactamase-positive Staphylococcus aureus 1287 PBP2a by competitive binding a... | Antimicrob Agents Chemother 54: 1670-7 (2010) Article DOI: 10.1128/AAC.00019-10 BindingDB Entry DOI: 10.7270/Q2B56NK6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Peptidase (Staphylococcus aureus) | BDBM50482776 (CHEBI:70718 | Ceftaroline Fosamil | PPI-0903 | TAK...) | PDB MMDB UniProtKB/TrEMBL B.MOAD GoogleScholar AffyNet | Purchase MCE KEGG PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.46E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Hershey Medical Center Curated by ChEMBL | Assay Description Binding affinity to methicillin-, linezolid-resistant, vancomycin-intermediate, beta-lactamase-positive Staphylococcus aureus 2149A PBP2a by competit... | Antimicrob Agents Chemother 54: 1670-7 (2010) Article DOI: 10.1128/AAC.00019-10 BindingDB Entry DOI: 10.7270/Q2B56NK6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Peptidase (Staphylococcus aureus) | BDBM50378857 (CEFTOBIPROLE | Zeftera | Zevtera) | PDB MMDB UniProtKB/TrEMBL B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.68E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Johnson & Johnson Pharmaceutical Research and Development Curated by ChEMBL | Assay Description Inhibition of bocillin FL binding to methicillin-resistant Staphylococcus aureus OC 3726 penicillin-binding protein 2a | Antimicrob Agents Chemother 51: 2621-4 (2007) Article DOI: 10.1128/aac.00029-07 BindingDB Entry DOI: 10.7270/Q2VH5RN2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Peptidase (Staphylococcus aureus) | BDBM50103601 (CHEBI:29007 | Ceftriaxone) | PDB MMDB UniProtKB/TrEMBL B.MOAD GoogleScholar AffyNet | KEGG PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 1.80E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Hershey Medical Center Curated by ChEMBL | Assay Description Binding affinity to methicillin-, vancomycin-resistant, beta-lactamase-positive Staphylococcus aureus 510 PBP2a by competitive binding assay | Antimicrob Agents Chemother 54: 1670-7 (2010) Article DOI: 10.1128/AAC.00019-10 BindingDB Entry DOI: 10.7270/Q2B56NK6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Peptidase (Staphylococcus aureus) | BDBM50378857 (CEFTOBIPROLE | Zeftera | Zevtera) | PDB MMDB UniProtKB/TrEMBL B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.90E+3 | n/a | n/a | n/a | n/a | 7.4 | n/a |
Universit£ Catholique de Louvain Curated by ChEMBL | Assay Description Binding affinity to Staphylococcus aureus ATCC 433000 PBP2a by western blotting at pH 7.4 in presence of 100 uM Bocillin FL | Antimicrob Agents Chemother 53: 2289-97 (2009) Article DOI: 10.1128/AAC.01135-08 BindingDB Entry DOI: 10.7270/Q2NZ88MK | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Peptidase (Staphylococcus aureus) | BDBM50482777 (CHEBI:204928 | Cefotaxime) | PDB MMDB UniProtKB/TrEMBL B.MOAD GoogleScholar AffyNet | Purchase MCE KEGG PC cid PC sid PDB UniChem | Article PubMed | n/a | n/a | 2.19E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Hershey Medical Center Curated by ChEMBL | Assay Description Binding affinity to methicillin-, vancomycin-resistant, beta-lactamase-positive Staphylococcus aureus 510 PBP2a by competitive binding assay | Antimicrob Agents Chemother 54: 1670-7 (2010) Article DOI: 10.1128/AAC.00019-10 BindingDB Entry DOI: 10.7270/Q2B56NK6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Peptidase (Staphylococcus aureus) | BDBM50378857 (CEFTOBIPROLE | Zeftera | Zevtera) | PDB MMDB UniProtKB/TrEMBL B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 3.20E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
The Rockefeller University Curated by ChEMBL | Assay Description Inhibition of methicillin-resistant Staphylococcus aureus COL PBP2a by competitive assay | Antimicrob Agents Chemother 52: 2709-17 (2008) Article DOI: 10.1128/AAC.00266-08 BindingDB Entry DOI: 10.7270/Q2GH9JX8 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Peptidase (Staphylococcus aureus) | BDBM50103601 (CHEBI:29007 | Ceftriaxone) | PDB MMDB UniProtKB/TrEMBL B.MOAD GoogleScholar AffyNet | KEGG PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 3.60E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Hershey Medical Center Curated by ChEMBL | Assay Description Binding affinity to methicillin-resistant, vancomycin-intermediate, beta-lactamase-positive Staphylococcus aureus 1287 PBP2a by competitive binding a... | Antimicrob Agents Chemother 54: 1670-7 (2010) Article DOI: 10.1128/AAC.00019-10 BindingDB Entry DOI: 10.7270/Q2B56NK6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Peptidase (Staphylococcus aureus) | BDBM50482777 (CHEBI:204928 | Cefotaxime) | PDB MMDB UniProtKB/TrEMBL B.MOAD GoogleScholar AffyNet | Purchase MCE KEGG PC cid PC sid PDB UniChem | Article PubMed | n/a | n/a | 4.39E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Hershey Medical Center Curated by ChEMBL | Assay Description Binding affinity to methicillin-resistant, vancomycin-intermediate, beta-lactamase-positive Staphylococcus aureus 1287 PBP2a by competitive binding a... | Antimicrob Agents Chemother 54: 1670-7 (2010) Article DOI: 10.1128/AAC.00019-10 BindingDB Entry DOI: 10.7270/Q2B56NK6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Peptidase (Staphylococcus aureus) | BDBM50483019 (CS-023 | R-115685 | R-1558 | R-1L5685 | Ro-4908463...) | PDB MMDB UniProtKB/TrEMBL B.MOAD GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem | Article PubMed | n/a | n/a | 5.39E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Daiichi Sankyo Co., Ltd. Curated by ChEMBL | Assay Description Binding affinity to PBP2a in methicillin-resistant Staphylococcus aureus 12386-1 by [14C]benzylpenicillin labelled competitive assay | Antimicrob Agents Chemother 52: 2849-54 (2008) Article DOI: 10.1128/AAC.00413-08 BindingDB Entry DOI: 10.7270/Q24F1TK8 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Peptidase (Staphylococcus aureus) | BDBM50022787 ((+)-3,3-Dimethyl-7-oxo-6-phenylacetylamino-4-thia-...) | PDB MMDB UniProtKB/TrEMBL B.MOAD GoogleScholar AffyNet | Purchase DrugBank MCE KEGG MMDB PC cid PC sid PDB UniChem Patents Similars | Article PubMed | n/a | n/a | 5.98E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Hershey Medical Center Curated by ChEMBL | Assay Description Binding affinity to methicillin-, linezolid-resistant, vancomycin-intermediate, beta-lactamase-positive Staphylococcus aureus 2149A PBP2a by competit... | Antimicrob Agents Chemother 54: 1670-7 (2010) Article DOI: 10.1128/AAC.00019-10 BindingDB Entry DOI: 10.7270/Q2B56NK6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Peptidase (Staphylococcus aureus) | BDBM50378857 (CEFTOBIPROLE | Zeftera | Zevtera) | PDB MMDB UniProtKB/TrEMBL B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 7.40E+3 | n/a | n/a | n/a | n/a | 5.5 | n/a |
Universit£ Catholique de Louvain Curated by ChEMBL | Assay Description Binding affinity to Staphylococcus aureus ATCC 433000 PBP2a by western blotting at pH 5.5 in presence of 100 uM Bocillin FL | Antimicrob Agents Chemother 53: 2289-97 (2009) Article DOI: 10.1128/AAC.01135-08 BindingDB Entry DOI: 10.7270/Q2NZ88MK | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Peptidase (Staphylococcus aureus) | BDBM50483019 (CS-023 | R-115685 | R-1558 | R-1L5685 | Ro-4908463...) | PDB MMDB UniProtKB/TrEMBL B.MOAD GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem | Article PubMed | n/a | n/a | 9.85E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Daiichi Sankyo Co., Ltd. Curated by ChEMBL | Assay Description Binding affinity to PBP2a in methicillin-resistant Staphylococcus aureus 123-1 by [14C]benzylpenicillin labelled competitive assay | Antimicrob Agents Chemother 52: 2849-54 (2008) Article DOI: 10.1128/AAC.00413-08 BindingDB Entry DOI: 10.7270/Q24F1TK8 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Peptidase (Staphylococcus aureus) | BDBM50022787 ((+)-3,3-Dimethyl-7-oxo-6-phenylacetylamino-4-thia-...) | PDB MMDB UniProtKB/TrEMBL B.MOAD GoogleScholar AffyNet | Purchase DrugBank MCE KEGG MMDB PC cid PC sid PDB UniChem Patents Similars | Article PubMed | n/a | n/a | 1.19E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Hershey Medical Center Curated by ChEMBL | Assay Description Binding affinity to against methicillin-, daptomycin-resistant, vancomycin-intermediate, beta-lactamase-positive Staphylococcus aureus 25 PBP2a by co... | Antimicrob Agents Chemother 54: 1670-7 (2010) Article DOI: 10.1128/AAC.00019-10 BindingDB Entry DOI: 10.7270/Q2B56NK6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Peptidase (Staphylococcus aureus) | BDBM50022787 ((+)-3,3-Dimethyl-7-oxo-6-phenylacetylamino-4-thia-...) | PDB MMDB UniProtKB/TrEMBL B.MOAD GoogleScholar AffyNet | Purchase DrugBank MCE KEGG MMDB PC cid PC sid PDB UniChem Patents Similars | Article PubMed | n/a | n/a | 1.19E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Hershey Medical Center Curated by ChEMBL | Assay Description Binding affinity to methicillin-resistant, vancomycin-intermediate, beta-lactamase-positive Staphylococcus aureus 1287 PBP2a by competitive binding a... | Antimicrob Agents Chemother 54: 1670-7 (2010) Article DOI: 10.1128/AAC.00019-10 BindingDB Entry DOI: 10.7270/Q2B56NK6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Peptidase (Staphylococcus aureus) | BDBM50103601 (CHEBI:29007 | Ceftriaxone) | PDB MMDB UniProtKB/TrEMBL B.MOAD GoogleScholar AffyNet | KEGG PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | >9.01E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Johnson & Johnson Pharmaceutical Research and Development Curated by ChEMBL | Assay Description Inhibition of bocillin FL binding to methicillin-resistant Staphylococcus aureus OC 3726 penicillin-binding protein 2a | Antimicrob Agents Chemother 51: 2621-4 (2007) Article DOI: 10.1128/aac.00029-07 BindingDB Entry DOI: 10.7270/Q2VH5RN2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Peptidase (Staphylococcus aureus) | BDBM50420259 (CEFTAZIDIME) | PDB MMDB UniProtKB/TrEMBL B.MOAD GoogleScholar AffyNet | Purchase DrugBank MCE KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >9.14E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Johnson & Johnson Pharmaceutical Research and Development Curated by ChEMBL | Assay Description Inhibition of bocillin FL binding to methicillin-resistant Staphylococcus aureus OC 3726 penicillin-binding protein 2a | Antimicrob Agents Chemother 51: 2621-4 (2007) Article DOI: 10.1128/aac.00029-07 BindingDB Entry DOI: 10.7270/Q2VH5RN2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Peptidase (Staphylococcus aureus) | BDBM50129062 (CHEBI:43968 | ICI-194660 | Meropenem | Merrem | Me...) | PDB MMDB UniProtKB/TrEMBL B.MOAD GoogleScholar AffyNet | Purchase DrugBank MCE PC cid PC sid PDB UniChem Similars | Article PubMed | n/a | n/a | 1.38E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Daiichi Sankyo Co., Ltd. Curated by ChEMBL | Assay Description Binding affinity to PBP2a in methicillin-resistant Staphylococcus aureus 12386-1 by [14C]benzylpenicillin labelled competitive assay | Antimicrob Agents Chemother 52: 2849-54 (2008) Article DOI: 10.1128/AAC.00413-08 BindingDB Entry DOI: 10.7270/Q24F1TK8 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Peptidase (Staphylococcus aureus) | BDBM50022787 ((+)-3,3-Dimethyl-7-oxo-6-phenylacetylamino-4-thia-...) | PDB MMDB UniProtKB/TrEMBL B.MOAD GoogleScholar AffyNet | Purchase DrugBank MCE KEGG MMDB PC cid PC sid PDB UniChem Patents Similars | Article PubMed | n/a | n/a | 1.91E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Hershey Medical Center Curated by ChEMBL | Assay Description Binding affinity to methicillin-resistant, heteroresistant vancomycin-intermediate, beta-lactamase-negative Staphylococcus aureus 873 PBP2a by compet... | Antimicrob Agents Chemother 54: 1670-7 (2010) Article DOI: 10.1128/AAC.00019-10 BindingDB Entry DOI: 10.7270/Q2B56NK6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Peptidase (Staphylococcus aureus) | BDBM50022787 ((+)-3,3-Dimethyl-7-oxo-6-phenylacetylamino-4-thia-...) | PDB MMDB UniProtKB/TrEMBL B.MOAD GoogleScholar AffyNet | Purchase DrugBank MCE KEGG MMDB PC cid PC sid PDB UniChem Patents Similars | Article PubMed | n/a | n/a | 1.91E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Hershey Medical Center Curated by ChEMBL | Assay Description Binding affinity to methicillin-, vancomycin-resistant, beta-lactamase-positive Staphylococcus aureus 510 PBP2a by competitive binding assay | Antimicrob Agents Chemother 54: 1670-7 (2010) Article DOI: 10.1128/AAC.00019-10 BindingDB Entry DOI: 10.7270/Q2B56NK6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Peptidase (Staphylococcus aureus) | BDBM50103601 (CHEBI:29007 | Ceftriaxone) | PDB MMDB UniProtKB/TrEMBL B.MOAD GoogleScholar AffyNet | KEGG PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | >2.30E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Hershey Medical Center Curated by ChEMBL | Assay Description Binding affinity to methicillin-, linezolid-resistant, vancomycin-intermediate, beta-lactamase-positive Staphylococcus aureus 2149A PBP2a by competit... | Antimicrob Agents Chemother 54: 1670-7 (2010) Article DOI: 10.1128/AAC.00019-10 BindingDB Entry DOI: 10.7270/Q2B56NK6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Peptidase (Staphylococcus aureus) | BDBM50103601 (CHEBI:29007 | Ceftriaxone) | PDB MMDB UniProtKB/TrEMBL B.MOAD GoogleScholar AffyNet | KEGG PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | >2.30E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Hershey Medical Center Curated by ChEMBL | Assay Description Binding affinity to methicillin-resistant, heteroresistant vancomycin-intermediate, beta-lactamase-negative Staphylococcus aureus 873 PBP2a by compet... | Antimicrob Agents Chemother 54: 1670-7 (2010) Article DOI: 10.1128/AAC.00019-10 BindingDB Entry DOI: 10.7270/Q2B56NK6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Peptidase (Staphylococcus aureus) | BDBM50213266 (CHEBI:471744 | Imipenem | MK-0787) | PDB MMDB UniProtKB/TrEMBL B.MOAD GoogleScholar AffyNet | Purchase MCE KEGG PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 2.53E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Daiichi Sankyo Co., Ltd. Curated by ChEMBL | Assay Description Binding affinity to PBP2a in methicillin-resistant Staphylococcus aureus 12386-1 by [14C]benzylpenicillin labelled competitive assay | Antimicrob Agents Chemother 52: 2849-54 (2008) Article DOI: 10.1128/AAC.00413-08 BindingDB Entry DOI: 10.7270/Q24F1TK8 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Peptidase (Staphylococcus aureus) | BDBM50482777 (CHEBI:204928 | Cefotaxime) | PDB MMDB UniProtKB/TrEMBL B.MOAD GoogleScholar AffyNet | Purchase MCE KEGG PC cid PC sid PDB UniChem | Article PubMed | n/a | n/a | >2.81E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Hershey Medical Center Curated by ChEMBL | Assay Description Binding affinity to methicillin-, linezolid-resistant, vancomycin-intermediate, beta-lactamase-positive Staphylococcus aureus 2149A PBP2a by competit... | Antimicrob Agents Chemother 54: 1670-7 (2010) Article DOI: 10.1128/AAC.00019-10 BindingDB Entry DOI: 10.7270/Q2B56NK6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Peptidase (Staphylococcus aureus) | BDBM50482777 (CHEBI:204928 | Cefotaxime) | PDB MMDB UniProtKB/TrEMBL B.MOAD GoogleScholar AffyNet | Purchase MCE KEGG PC cid PC sid PDB UniChem | Article PubMed | n/a | n/a | >2.81E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Hershey Medical Center Curated by ChEMBL | Assay Description Binding affinity to methicillin-resistant, heteroresistant vancomycin-intermediate, beta-lactamase-negative Staphylococcus aureus 873 PBP2a by compet... | Antimicrob Agents Chemother 54: 1670-7 (2010) Article DOI: 10.1128/AAC.00019-10 BindingDB Entry DOI: 10.7270/Q2B56NK6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Peptidase (Staphylococcus aureus) | BDBM50129062 (CHEBI:43968 | ICI-194660 | Meropenem | Merrem | Me...) | PDB MMDB UniProtKB/TrEMBL B.MOAD GoogleScholar AffyNet | Purchase DrugBank MCE PC cid PC sid PDB UniChem Similars | Article PubMed | n/a | n/a | 3.39E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Daiichi Sankyo Co., Ltd. Curated by ChEMBL | Assay Description Binding affinity to PBP2a in methicillin-resistant Staphylococcus aureus 123-1 by [14C]benzylpenicillin labelled competitive assay | Antimicrob Agents Chemother 52: 2849-54 (2008) Article DOI: 10.1128/AAC.00413-08 BindingDB Entry DOI: 10.7270/Q24F1TK8 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Peptidase (Staphylococcus aureus) | BDBM50213266 (CHEBI:471744 | Imipenem | MK-0787) | PDB MMDB UniProtKB/TrEMBL B.MOAD GoogleScholar AffyNet | Purchase MCE KEGG PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 5.67E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Daiichi Sankyo Co., Ltd. Curated by ChEMBL | Assay Description Binding affinity to PBP2a in methicillin-resistant Staphylococcus aureus 123-1 by [14C]benzylpenicillin labelled competitive assay | Antimicrob Agents Chemother 52: 2849-54 (2008) Article DOI: 10.1128/AAC.00413-08 BindingDB Entry DOI: 10.7270/Q24F1TK8 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Peptidase (Staphylococcus aureus) | BDBM50350483 (Bactocill | OXACILLIN) | PDB MMDB UniProtKB/TrEMBL B.MOAD GoogleScholar AffyNet | Purchase DrugBank MCE KEGG PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 7.10E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
The Rockefeller University Curated by ChEMBL | Assay Description Inhibition of methicillin-resistant Staphylococcus aureus COL PBP2a by competitive assay | Antimicrob Agents Chemother 52: 2709-17 (2008) Article DOI: 10.1128/AAC.00266-08 BindingDB Entry DOI: 10.7270/Q2GH9JX8 | |||||||||||
More data for this Ligand-Target Pair |