Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kcal/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Elongation factor 1-alpha 2 (Homo sapiens (Human)) | BDBM50347602 (CHEMBL1802815) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 2.43 | n/a | n/a | n/a | n/a | n/a |
University of California Davis Curated by ChEMBL | Assay Description Binding affinity to eEF1A2 expressed in human MDA-MB-231 cells using 1 uM biotinylated compound immobilized on streptavidin sensor chip by surface pl... | J Med Chem 54: 4339-49 (2011) Article DOI: 10.1021/jm101440r BindingDB Entry DOI: 10.7270/Q24M94X7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Elongation factor 1-alpha 2 (Homo sapiens (Human)) | BDBM50347603 (CHEMBL1802973) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 4.54 | n/a | n/a | n/a | n/a | n/a |
University of California Davis Curated by ChEMBL | Assay Description Binding affinity to eEF1A2 expressed in human MDA-MB-231 cells using 1 uM biotinylated compound immobilized on streptavidin sensor chip by surface pl... | J Med Chem 54: 4339-49 (2011) Article DOI: 10.1021/jm101440r BindingDB Entry DOI: 10.7270/Q24M94X7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Elongation factor 1-alpha 2 (Homo sapiens (Human)) | BDBM50347601 (CHEMBL1802814) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 4.89 | n/a | n/a | n/a | n/a | n/a |
University of California Davis Curated by ChEMBL | Assay Description Binding affinity to eEF1A2 expressed in human MDA-MB-231 cells using 1 uM biotinylated compound immobilized on streptavidin sensor chip by surface pl... | J Med Chem 54: 4339-49 (2011) Article DOI: 10.1021/jm101440r BindingDB Entry DOI: 10.7270/Q24M94X7 | |||||||||||
More data for this Ligand-Target Pair |