Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kcal/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
CAI-1 autoinducer sensor kinase/phosphatase CqsS (Vibrio cholerae serotype O1 (strain ATCC 39315 / E...) | BDBM50358387 (CHEMBL1922879) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 3.60E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Princeton University Curated by ChEMBL | Assay Description Antagonist activity at CqsS receptor in Vibrio cholerae MM920 assessed as inhibition of quorum sensing regulated CAI-1 induced bioluminescence after ... | Bioorg Med Chem 19: 6906-18 (2011) Article DOI: 10.1016/j.bmc.2011.09.021 BindingDB Entry DOI: 10.7270/Q27H1K1T | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
CAI-1 autoinducer sensor kinase/phosphatase CqsS (Vibrio cholerae serotype O1 (strain ATCC 39315 / E...) | BDBM50358381 (CHEMBL1922873) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 4.60E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Princeton University Curated by ChEMBL | Assay Description Antagonist activity at CqsS receptor in Vibrio cholerae MM920 assessed as inhibition of quorum sensing regulated CAI-1 induced bioluminescence after ... | Bioorg Med Chem 19: 6906-18 (2011) Article DOI: 10.1016/j.bmc.2011.09.021 BindingDB Entry DOI: 10.7270/Q27H1K1T | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
CAI-1 autoinducer sensor kinase/phosphatase CqsS (Vibrio cholerae serotype O1 (strain ATCC 39315 / E...) | BDBM50358379 (CHEMBL1922871) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 5.50E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Princeton University Curated by ChEMBL | Assay Description Antagonist activity at CqsS receptor in Vibrio cholerae MM920 assessed as inhibition of quorum sensing regulated CAI-1 induced bioluminescence after ... | Bioorg Med Chem 19: 6906-18 (2011) Article DOI: 10.1016/j.bmc.2011.09.021 BindingDB Entry DOI: 10.7270/Q27H1K1T | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
CAI-1 autoinducer sensor kinase/phosphatase CqsS (Vibrio cholerae serotype O1 (strain ATCC 39315 / E...) | BDBM50358421 (CHEMBL1922888) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 6.80E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Princeton University Curated by ChEMBL | Assay Description Antagonist activity at CqsS receptor in Vibrio cholerae MM920 assessed as inhibition of quorum sensing regulated CAI-1 induced bioluminescence after ... | Bioorg Med Chem 19: 6906-18 (2011) Article DOI: 10.1016/j.bmc.2011.09.021 BindingDB Entry DOI: 10.7270/Q27H1K1T | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
CAI-1 autoinducer sensor kinase/phosphatase CqsS (Vibrio cholerae serotype O1 (strain ATCC 39315 / E...) | BDBM50358418 (CHEMBL1922885) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 7.40E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Princeton University Curated by ChEMBL | Assay Description Antagonist activity at CqsS receptor in Vibrio cholerae MM920 assessed as inhibition of quorum sensing regulated CAI-1 induced bioluminescence after ... | Bioorg Med Chem 19: 6906-18 (2011) Article DOI: 10.1016/j.bmc.2011.09.021 BindingDB Entry DOI: 10.7270/Q27H1K1T | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
CAI-1 autoinducer sensor kinase/phosphatase CqsS (Vibrio cholerae serotype O1 (strain ATCC 39315 / E...) | BDBM50358388 (CHEMBL1922880) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 7.80E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Princeton University Curated by ChEMBL | Assay Description Antagonist activity at CqsS receptor in Vibrio cholerae MM920 assessed as inhibition of quorum sensing regulated CAI-1 induced bioluminescence after ... | Bioorg Med Chem 19: 6906-18 (2011) Article DOI: 10.1016/j.bmc.2011.09.021 BindingDB Entry DOI: 10.7270/Q27H1K1T | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
CAI-1 autoinducer sensor kinase/phosphatase CqsS (Vibrio cholerae serotype O1 (strain ATCC 39315 / E...) | BDBM50358382 (CHEMBL1922874) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.14E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Princeton University Curated by ChEMBL | Assay Description Antagonist activity at CqsS receptor in Vibrio cholerae MM920 assessed as inhibition of quorum sensing regulated CAI-1 induced bioluminescence after ... | Bioorg Med Chem 19: 6906-18 (2011) Article DOI: 10.1016/j.bmc.2011.09.021 BindingDB Entry DOI: 10.7270/Q27H1K1T | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
CAI-1 autoinducer sensor kinase/phosphatase CqsS (Vibrio cholerae serotype O1 (strain ATCC 39315 / E...) | BDBM50358428 (CHEMBL1922895) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.36E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Princeton University Curated by ChEMBL | Assay Description Antagonist activity at CqsS receptor in Vibrio cholerae MM920 assessed as inhibition of quorum sensing regulated CAI-1 induced bioluminescence after ... | Bioorg Med Chem 19: 6906-18 (2011) Article DOI: 10.1016/j.bmc.2011.09.021 BindingDB Entry DOI: 10.7270/Q27H1K1T | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
CAI-1 autoinducer sensor kinase/phosphatase CqsS (Vibrio cholerae serotype O1 (strain ATCC 39315 / E...) | BDBM50358420 (CHEMBL1922887) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.37E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Princeton University Curated by ChEMBL | Assay Description Antagonist activity at CqsS receptor in Vibrio cholerae MM920 assessed as inhibition of quorum sensing regulated CAI-1 induced bioluminescence after ... | Bioorg Med Chem 19: 6906-18 (2011) Article DOI: 10.1016/j.bmc.2011.09.021 BindingDB Entry DOI: 10.7270/Q27H1K1T | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
CAI-1 autoinducer sensor kinase/phosphatase CqsS (Vibrio cholerae serotype O1 (strain ATCC 39315 / E...) | BDBM50358386 (CHEMBL1922878) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.72E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Princeton University Curated by ChEMBL | Assay Description Antagonist activity at CqsS receptor in Vibrio cholerae MM920 assessed as inhibition of quorum sensing regulated CAI-1 induced bioluminescence after ... | Bioorg Med Chem 19: 6906-18 (2011) Article DOI: 10.1016/j.bmc.2011.09.021 BindingDB Entry DOI: 10.7270/Q27H1K1T | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
CAI-1 autoinducer sensor kinase/phosphatase CqsS (Vibrio cholerae serotype O1 (strain ATCC 39315 / E...) | BDBM50358389 (CHEMBL1922881) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.74E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Princeton University Curated by ChEMBL | Assay Description Antagonist activity at CqsS receptor in Vibrio cholerae MM920 assessed as inhibition of quorum sensing regulated CAI-1 induced bioluminescence after ... | Bioorg Med Chem 19: 6906-18 (2011) Article DOI: 10.1016/j.bmc.2011.09.021 BindingDB Entry DOI: 10.7270/Q27H1K1T | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
CAI-1 autoinducer sensor kinase/phosphatase CqsS (Vibrio cholerae serotype O1 (strain ATCC 39315 / E...) | BDBM50358419 (CHEMBL1922886) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.78E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Princeton University Curated by ChEMBL | Assay Description Antagonist activity at CqsS receptor in Vibrio cholerae MM920 assessed as inhibition of quorum sensing regulated CAI-1 induced bioluminescence after ... | Bioorg Med Chem 19: 6906-18 (2011) Article DOI: 10.1016/j.bmc.2011.09.021 BindingDB Entry DOI: 10.7270/Q27H1K1T | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
CAI-1 autoinducer sensor kinase/phosphatase CqsS (Vibrio cholerae serotype O1 (strain ATCC 39315 / E...) | BDBM50358427 (CHEMBL1922894) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.85E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Princeton University Curated by ChEMBL | Assay Description Antagonist activity at CqsS receptor in Vibrio cholerae MM920 assessed as inhibition of quorum sensing regulated CAI-1 induced bioluminescence after ... | Bioorg Med Chem 19: 6906-18 (2011) Article DOI: 10.1016/j.bmc.2011.09.021 BindingDB Entry DOI: 10.7270/Q27H1K1T | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
CAI-1 autoinducer sensor kinase/phosphatase CqsS (Vibrio cholerae serotype O1 (strain ATCC 39315 / E...) | BDBM50358426 (CHEMBL1922893) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >5.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Princeton University Curated by ChEMBL | Assay Description Antagonist activity at CqsS receptor in Vibrio cholerae MM920 assessed as inhibition of quorum sensing regulated CAI-1 induced bioluminescence after ... | Bioorg Med Chem 19: 6906-18 (2011) Article DOI: 10.1016/j.bmc.2011.09.021 BindingDB Entry DOI: 10.7270/Q27H1K1T | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
CAI-1 autoinducer sensor kinase/phosphatase CqsS (Vibrio cholerae serotype O1 (strain ATCC 39315 / E...) | BDBM50358425 (CHEMBL1922892) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >5.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Princeton University Curated by ChEMBL | Assay Description Antagonist activity at CqsS receptor in Vibrio cholerae MM920 assessed as inhibition of quorum sensing regulated CAI-1 induced bioluminescence after ... | Bioorg Med Chem 19: 6906-18 (2011) Article DOI: 10.1016/j.bmc.2011.09.021 BindingDB Entry DOI: 10.7270/Q27H1K1T | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
CAI-1 autoinducer sensor kinase/phosphatase CqsS (Vibrio cholerae serotype O1 (strain ATCC 39315 / E...) | BDBM50358424 (CHEMBL1922891) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >5.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Princeton University Curated by ChEMBL | Assay Description Antagonist activity at CqsS receptor in Vibrio cholerae MM920 assessed as inhibition of quorum sensing regulated CAI-1 induced bioluminescence after ... | Bioorg Med Chem 19: 6906-18 (2011) Article DOI: 10.1016/j.bmc.2011.09.021 BindingDB Entry DOI: 10.7270/Q27H1K1T | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
CAI-1 autoinducer sensor kinase/phosphatase CqsS (Vibrio cholerae serotype O1 (strain ATCC 39315 / E...) | BDBM50358423 (CHEMBL1922890) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >5.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Princeton University Curated by ChEMBL | Assay Description Antagonist activity at CqsS receptor in Vibrio cholerae MM920 assessed as inhibition of quorum sensing regulated CAI-1 induced bioluminescence after ... | Bioorg Med Chem 19: 6906-18 (2011) Article DOI: 10.1016/j.bmc.2011.09.021 BindingDB Entry DOI: 10.7270/Q27H1K1T | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
CAI-1 autoinducer sensor kinase/phosphatase CqsS (Vibrio cholerae serotype O1 (strain ATCC 39315 / E...) | BDBM50358422 (CHEMBL1922889) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | >5.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Princeton University Curated by ChEMBL | Assay Description Antagonist activity at CqsS receptor in Vibrio cholerae MM920 assessed as inhibition of quorum sensing regulated CAI-1 induced bioluminescence after ... | Bioorg Med Chem 19: 6906-18 (2011) Article DOI: 10.1016/j.bmc.2011.09.021 BindingDB Entry DOI: 10.7270/Q27H1K1T | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
CAI-1 autoinducer sensor kinase/phosphatase CqsS (Vibrio cholerae serotype O1 (strain ATCC 39315 / E...) | BDBM50358417 (CHEMBL1922884) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >5.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Princeton University Curated by ChEMBL | Assay Description Antagonist activity at CqsS receptor in Vibrio cholerae MM920 assessed as inhibition of quorum sensing regulated CAI-1 induced bioluminescence after ... | Bioorg Med Chem 19: 6906-18 (2011) Article DOI: 10.1016/j.bmc.2011.09.021 BindingDB Entry DOI: 10.7270/Q27H1K1T | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
CAI-1 autoinducer sensor kinase/phosphatase CqsS (Vibrio cholerae serotype O1 (strain ATCC 39315 / E...) | BDBM50358391 (CHEMBL1922883) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >5.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Princeton University Curated by ChEMBL | Assay Description Antagonist activity at CqsS receptor in Vibrio cholerae MM920 assessed as inhibition of quorum sensing regulated CAI-1 induced bioluminescence after ... | Bioorg Med Chem 19: 6906-18 (2011) Article DOI: 10.1016/j.bmc.2011.09.021 BindingDB Entry DOI: 10.7270/Q27H1K1T | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
CAI-1 autoinducer sensor kinase/phosphatase CqsS (Vibrio cholerae serotype O1 (strain ATCC 39315 / E...) | BDBM50358390 (CHEMBL1922882) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >5.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Princeton University Curated by ChEMBL | Assay Description Antagonist activity at CqsS receptor in Vibrio cholerae MM920 assessed as inhibition of quorum sensing regulated CAI-1 induced bioluminescence after ... | Bioorg Med Chem 19: 6906-18 (2011) Article DOI: 10.1016/j.bmc.2011.09.021 BindingDB Entry DOI: 10.7270/Q27H1K1T | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
CAI-1 autoinducer sensor kinase/phosphatase CqsS (Vibrio cholerae serotype O1 (strain ATCC 39315 / E...) | BDBM50358385 (CHEMBL1922877) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >5.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Princeton University Curated by ChEMBL | Assay Description Antagonist activity at CqsS receptor in Vibrio cholerae MM920 assessed as inhibition of quorum sensing regulated CAI-1 induced bioluminescence after ... | Bioorg Med Chem 19: 6906-18 (2011) Article DOI: 10.1016/j.bmc.2011.09.021 BindingDB Entry DOI: 10.7270/Q27H1K1T | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
CAI-1 autoinducer sensor kinase/phosphatase CqsS (Vibrio cholerae serotype O1 (strain ATCC 39315 / E...) | BDBM50358384 (CHEMBL1922876) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >5.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Princeton University Curated by ChEMBL | Assay Description Antagonist activity at CqsS receptor in Vibrio cholerae MM920 assessed as inhibition of quorum sensing regulated CAI-1 induced bioluminescence after ... | Bioorg Med Chem 19: 6906-18 (2011) Article DOI: 10.1016/j.bmc.2011.09.021 BindingDB Entry DOI: 10.7270/Q27H1K1T | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
CAI-1 autoinducer sensor kinase/phosphatase CqsS (Vibrio cholerae serotype O1 (strain ATCC 39315 / E...) | BDBM50358383 (CHEMBL1922875) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >5.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Princeton University Curated by ChEMBL | Assay Description Antagonist activity at CqsS receptor in Vibrio cholerae MM920 assessed as inhibition of quorum sensing regulated CAI-1 induced bioluminescence after ... | Bioorg Med Chem 19: 6906-18 (2011) Article DOI: 10.1016/j.bmc.2011.09.021 BindingDB Entry DOI: 10.7270/Q27H1K1T | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
CAI-1 autoinducer sensor kinase/phosphatase CqsS (Vibrio cholerae serotype O1 (strain ATCC 39315 / E...) | BDBM50358429 (CHEMBL1922896) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | >5.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Princeton University Curated by ChEMBL | Assay Description Antagonist activity at CqsS receptor in Vibrio cholerae MM920 assessed as inhibition of quorum sensing regulated CAI-1 induced bioluminescence after ... | Bioorg Med Chem 19: 6906-18 (2011) Article DOI: 10.1016/j.bmc.2011.09.021 BindingDB Entry DOI: 10.7270/Q27H1K1T | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
CAI-1 autoinducer sensor kinase/phosphatase CqsS (Vibrio cholerae serotype O1 (strain ATCC 39315 / E...) | BDBM50358380 (CHEMBL1922872) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >5.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Princeton University Curated by ChEMBL | Assay Description Antagonist activity at CqsS receptor in Vibrio cholerae MM920 assessed as inhibition of quorum sensing regulated CAI-1 induced bioluminescence after ... | Bioorg Med Chem 19: 6906-18 (2011) Article DOI: 10.1016/j.bmc.2011.09.021 BindingDB Entry DOI: 10.7270/Q27H1K1T | |||||||||||
More data for this Ligand-Target Pair |