Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kcal/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Histone-lysine N-methyltransferase Su(var)3-9 (Drosophila melanogaster) | BDBM50315537 (CHEMBL1089316 | chaetocin) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 600 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Inhibition of recombinant Drosophila melanogaster SUV39 by radioactive filter-binding assay | Eur J Med Chem 56: 179-194 (2012) Article DOI: 10.1016/j.ejmech.2012.08.010 BindingDB Entry DOI: 10.7270/Q2TQ62NX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histone-lysine N-methyltransferase Su(var)3-9 (Drosophila melanogaster) | BDBM50315537 (CHEMBL1089316 | chaetocin) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 600 | n/a | n/a | n/a | n/a | n/a | n/a |
Ludwig-Maximillians University of Munich Curated by ChEMBL | Assay Description Inhibition of Drosophila melanogaster SU(VAR)3-9 | Nat Chem Biol 1: 143-5 (2005) Article DOI: 10.1038/nchembio721 BindingDB Entry DOI: 10.7270/Q2PK0JZV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histone-lysine N-methyltransferase Su(var)3-9 (Drosophila melanogaster) | BDBM50315537 (CHEMBL1089316 | chaetocin) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 600 | n/a | n/a | n/a | n/a | n/a | n/a |
Imperial College London Curated by ChEMBL | Assay Description Inhibition of Drosophila melanogaster Histone-lysine N-methyltransferase Su(var)3-9 | J Med Chem 56: 8616-25 (2013) Article DOI: 10.1021/jm401063r BindingDB Entry DOI: 10.7270/Q2NS0WDK | |||||||||||
More data for this Ligand-Target Pair |