Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kcal/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Proteasome subunit alpha type-6 (Homo sapiens (Human)) | BDBM588478 ((R)-N-(2,5-dichlorobenzoyl)-3- methylmercaptopropi...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | UniChem | US Patent | n/a | n/a | 4.86 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description The proteasome used in the present invention is human erythrocyte 20S proteasome, and the enzyme, fluorescent substrate and test buffer are all purch... | Citation and Details BindingDB Entry DOI: 10.7270/Q27P937G | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Proteasome subunit alpha type-6 (Homo sapiens (Human)) | BDBM50516758 (CHEMBL4444471 | US11542283, Compound V-9A) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | KEGG PC cid PC sid UniChem | US Patent | n/a | n/a | 5.69 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description The proteasome used in the present invention is human erythrocyte 20S proteasome, and the enzyme, fluorescent substrate and test buffer are all purch... | Citation and Details BindingDB Entry DOI: 10.7270/Q27P937G | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Proteasome subunit alpha type-6 (Homo sapiens (Human)) | BDBM588482 ((R)-N-(2,5-dichlorobenzoyl)-3- methylmercaptopropi...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | UniChem | US Patent | n/a | n/a | 6.60 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description The proteasome used in the present invention is human erythrocyte 20S proteasome, and the enzyme, fluorescent substrate and test buffer are all purch... | Citation and Details BindingDB Entry DOI: 10.7270/Q27P937G | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Proteasome subunit alpha type-6 (Homo sapiens (Human)) | BDBM50462603 (CHEMBL4248209 | US11542283, Compound V-8A) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 7.02 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description The proteasome used in the present invention is human erythrocyte 20S proteasome, and the enzyme, fluorescent substrate and test buffer are all purch... | Citation and Details BindingDB Entry DOI: 10.7270/Q27P937G | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Proteasome subunit alpha type-6 (Homo sapiens (Human)) | BDBM50462621 (CHEMBL1813256 | MLN-9708 | US11542283, Compound ML...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase PC cid PC sid UniChem | US Patent | n/a | n/a | 7.47 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description The proteasome used in the present invention is human erythrocyte 20S proteasome, and the enzyme, fluorescent substrate and test buffer are all purch... | Citation and Details BindingDB Entry DOI: 10.7270/Q27P937G | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Proteasome subunit alpha type-6 (Homo sapiens (Human)) | BDBM50462625 (CHEMBL4243375 | US11542283, Compound IV-8) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 7.52 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description The proteasome used in the present invention is human erythrocyte 20S proteasome, and the enzyme, fluorescent substrate and test buffer are all purch... | Citation and Details BindingDB Entry DOI: 10.7270/Q27P937G | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Proteasome subunit alpha type-6 (Homo sapiens (Human)) | BDBM588480 ((S)-N-(2,5-dichlorobenzoyl)-3- methoxypropionamido...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | UniChem | US Patent | n/a | n/a | 8.20 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description The proteasome used in the present invention is human erythrocyte 20S proteasome, and the enzyme, fluorescent substrate and test buffer are all purch... | Citation and Details BindingDB Entry DOI: 10.7270/Q27P937G | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Proteasome subunit alpha type-6 (Homo sapiens (Human)) | BDBM50069989 ((R)-3-methyl-1-((S)-3-phenyl-2-(pyrazine-2-carboxa...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL DrugBank MCE MMDB PC cid PC sid PDB UniChem Patents Similars | DrugBank PDB US Patent | n/a | n/a | 9.92 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description The proteasome used in the present invention is human erythrocyte 20S proteasome, and the enzyme, fluorescent substrate and test buffer are all purch... | Citation and Details BindingDB Entry DOI: 10.7270/Q27P937G | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) |