Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kcal/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Elongin-C (Homo sapiens (Human)) | BDBM50463158 (CHEMBL4244103) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase MCE PC cid PC sid PDB UniChem | PDB Article PubMed | n/a | n/a | n/a | 5 | n/a | n/a | n/a | n/a | n/a |
University of Dundee Curated by ChEMBL | Assay Description Binding affinity to N-terminal His6 tagged VHL (54 to 213 residues)/ELoC (17 to 112 residues)/EloB (1 to 120 residues) (unknown origin) complex expre... | J Med Chem 61: 7387-7393 (2018) Article DOI: 10.1021/acs.jmedchem.8b00842 BindingDB Entry DOI: 10.7270/Q2639SCC | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
Elongin-C (Homo sapiens (Human)) | BDBM50463159 (CHEMBL4241500) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase MCE PC cid PC sid PDB UniChem | PDB Article PubMed | n/a | n/a | n/a | 6.70 | n/a | n/a | n/a | n/a | n/a |
University of Dundee Curated by ChEMBL | Assay Description Binding affinity to N-terminal His6 tagged VHL (54 to 213 residues)/ELoC (17 to 112 residues)/EloB (1 to 120 residues) (unknown origin) complex expre... | J Med Chem 61: 7387-7393 (2018) Article DOI: 10.1021/acs.jmedchem.8b00842 BindingDB Entry DOI: 10.7270/Q2639SCC | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
Elongin-C (Homo sapiens (Human)) | BDBM50459943 (CHEMBL4225470) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase KEGG PC cid PC sid PDB UniChem | PDB Article PubMed | n/a | n/a | n/a | 16 | n/a | n/a | n/a | n/a | n/a |
University of Dundee Curated by ChEMBL | Assay Description Binding affinity to VBC (unknown origin) at 50 uM at 20 degC by surface plasmon resonance assay | J Med Chem 61: 599-618 (2018) Article DOI: 10.1021/acs.jmedchem.7b00675 BindingDB Entry DOI: 10.7270/Q2736TJ6 | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
Elongin-C (Homo sapiens (Human)) | BDBM50459943 (CHEMBL4225470) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase KEGG PC cid PC sid PDB UniChem | PDB Article PubMed | n/a | n/a | n/a | 24 | n/a | n/a | n/a | n/a | n/a |
University of Dundee Curated by ChEMBL | Assay Description Binding affinity to VBC (unknown origin) at 50 uM at 10 degC by surface plasmon resonance assay | J Med Chem 61: 599-618 (2018) Article DOI: 10.1021/acs.jmedchem.7b00675 BindingDB Entry DOI: 10.7270/Q2736TJ6 | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
Elongin-C (Homo sapiens (Human)) | BDBM50459943 (CHEMBL4225470) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase KEGG PC cid PC sid PDB UniChem | PDB Article PubMed | n/a | n/a | n/a | 44 | n/a | n/a | n/a | n/a | n/a |
University of Dundee Curated by ChEMBL | Assay Description Binding affinity to VHL (unknown origin)/elongin C (unknown origin)/elongin B (unknown origin) by isothermal titration calorimetry-based assay | J Med Chem 61: 599-618 (2018) Article DOI: 10.1021/acs.jmedchem.7b00675 BindingDB Entry DOI: 10.7270/Q2736TJ6 | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
Elongin-C (Homo sapiens (Human)) | BDBM50459944 (CHEMBL4225537) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase MCE KEGG PC cid PC sid PDB UniChem | PDB Article PubMed | n/a | n/a | n/a | 52 | n/a | n/a | n/a | n/a | n/a |
University of Dundee Curated by ChEMBL | Assay Description Binding affinity to VBC (unknown origin) at 50 uM at 20 degC by surface plasmon resonance assay | J Med Chem 61: 599-618 (2018) Article DOI: 10.1021/acs.jmedchem.7b00675 BindingDB Entry DOI: 10.7270/Q2736TJ6 | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
Elongin-C (Homo sapiens (Human)) | BDBM50604004 (CHEMBL5205396) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 56 | n/a | n/a | n/a | n/a | n/a |
TBA | Citation and Details Article DOI: 10.1021/acs.jmedchem.1c01774 BindingDB Entry DOI: 10.7270/Q2CF9V6Z | ||||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Elongin-C (Homo sapiens (Human)) | BDBM50459880 (CHEMBL4226570) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase MCE KEGG PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 69 | n/a | n/a | n/a | n/a | n/a |
University of Dundee Curated by ChEMBL | Assay Description Binding affinity to N-terminal His6-tagged recombinant human VHL (54 to 213 residues)/elongin C (17 to 112 residues)/elongin B (1 to 104 residues) ex... | J Med Chem 61: 504-513 (2018) Article DOI: 10.1021/acs.jmedchem.6b01912 BindingDB Entry DOI: 10.7270/Q2R49TC3 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Elongin-C (Homo sapiens (Human)) | BDBM50459879 (CHEMBL4227226) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | KEGG PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 73 | n/a | n/a | n/a | n/a | n/a |
University of Dundee Curated by ChEMBL | Assay Description Binding affinity to N-terminal His6-tagged recombinant human VHL (54 to 213 residues)/elongin C (17 to 112 residues)/elongin B (1 to 104 residues) ex... | J Med Chem 61: 504-513 (2018) Article DOI: 10.1021/acs.jmedchem.6b01912 BindingDB Entry DOI: 10.7270/Q2R49TC3 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Elongin-C (Homo sapiens (Human)) | BDBM50459944 (CHEMBL4225537) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase MCE KEGG PC cid PC sid PDB UniChem | PDB Article PubMed | n/a | n/a | n/a | 80 | n/a | n/a | n/a | n/a | n/a |
University of Dundee Curated by ChEMBL | Assay Description Displacement of FAM-labeled HIF-1alpha peptide from VBC (unknown origin) by fluorescence polarization assay | J Med Chem 61: 599-618 (2018) Article DOI: 10.1021/acs.jmedchem.7b00675 BindingDB Entry DOI: 10.7270/Q2736TJ6 | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
Elongin-C (Homo sapiens (Human)) | BDBM50459944 (CHEMBL4225537) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase MCE KEGG PC cid PC sid PDB UniChem | PDB Article PubMed | n/a | n/a | n/a | 90 | n/a | n/a | n/a | n/a | n/a |
University of Dundee Curated by ChEMBL | Assay Description Binding affinity to VHL (unknown origin)/elongin C (unknown origin)/elongin B (unknown origin) by isothermal titration calorimetry-based assay | J Med Chem 61: 599-618 (2018) Article DOI: 10.1021/acs.jmedchem.7b00675 BindingDB Entry DOI: 10.7270/Q2736TJ6 | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
Elongin-C (Homo sapiens (Human)) | BDBM50459943 (CHEMBL4225470) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase KEGG PC cid PC sid PDB UniChem | PDB Article PubMed | n/a | n/a | n/a | 90 | n/a | n/a | n/a | n/a | n/a |
University of Dundee Curated by ChEMBL | Assay Description Displacement of FAM-labeled HIF-1alpha peptide from VBC (unknown origin) by fluorescence polarization assay | J Med Chem 61: 599-618 (2018) Article DOI: 10.1021/acs.jmedchem.7b00675 BindingDB Entry DOI: 10.7270/Q2736TJ6 | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
Elongin-C (Homo sapiens (Human)) | BDBM50459954 (CHEMBL4228950) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | KEGG PC cid PC sid PDB UniChem | PDB Article PubMed | n/a | n/a | n/a | 97 | n/a | n/a | n/a | n/a | n/a |
University of Dundee Curated by ChEMBL | Assay Description Binding affinity to VBC (unknown origin) at 50 uM at 20 degC by surface plasmon resonance assay | J Med Chem 61: 599-618 (2018) Article DOI: 10.1021/acs.jmedchem.7b00675 BindingDB Entry DOI: 10.7270/Q2736TJ6 | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
Elongin-C (Homo sapiens (Human)) | BDBM50459944 (CHEMBL4225537) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase MCE KEGG PC cid PC sid PDB UniChem | PDB Article PubMed | n/a | n/a | n/a | 99 | n/a | n/a | n/a | n/a | n/a |
University of Dundee Curated by ChEMBL | Assay Description Binding affinity to VBC (unknown origin) at 50 uM at 10 degC by surface plasmon resonance assay | J Med Chem 61: 599-618 (2018) Article DOI: 10.1021/acs.jmedchem.7b00675 BindingDB Entry DOI: 10.7270/Q2736TJ6 | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
Elongin-C (Homo sapiens (Human)) | BDBM50459947 (CHEMBL4225856) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | KEGG PC cid PC sid PDB UniChem | PDB Article PubMed | n/a | n/a | n/a | 105 | n/a | n/a | n/a | n/a | n/a |
University of Dundee Curated by ChEMBL | Assay Description Binding affinity to VHL (unknown origin)/elongin C (unknown origin)/elongin B (unknown origin) by isothermal titration calorimetry-based assay | J Med Chem 61: 599-618 (2018) Article DOI: 10.1021/acs.jmedchem.7b00675 BindingDB Entry DOI: 10.7270/Q2736TJ6 | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
Elongin-C (Homo sapiens (Human)) | BDBM50459876 (CHEMBL4229193) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase MCE KEGG PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 105 | n/a | n/a | n/a | n/a | n/a |
University of Dundee Curated by ChEMBL | Assay Description Binding affinity to N-terminal His6-tagged recombinant human VHL (54 to 213 residues)/elongin C (17 to 112 residues)/elongin B (1 to 104 residues) ex... | J Med Chem 61: 504-513 (2018) Article DOI: 10.1021/acs.jmedchem.6b01912 BindingDB Entry DOI: 10.7270/Q2R49TC3 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Elongin-C (Homo sapiens (Human)) | BDBM50459954 (CHEMBL4228950) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | KEGG PC cid PC sid PDB UniChem | PDB Article PubMed | n/a | n/a | n/a | 106 | n/a | n/a | n/a | n/a | n/a |
University of Dundee Curated by ChEMBL | Assay Description Binding affinity to VHL (unknown origin)/elongin C (unknown origin)/elongin B (unknown origin) by isothermal titration calorimetry-based assay | J Med Chem 61: 599-618 (2018) Article DOI: 10.1021/acs.jmedchem.7b00675 BindingDB Entry DOI: 10.7270/Q2736TJ6 | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
Elongin-C (Homo sapiens (Human)) | BDBM50099062 (CHEMBL3344081 | US10730870, Example 3 | US11512083...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase CHEMBL MCE KEGG PC cid PC sid PDB UniChem Similars | PDB Article PubMed | n/a | n/a | n/a | 107 | n/a | n/a | n/a | n/a | n/a |
University of Dundee Curated by ChEMBL | Assay Description Binding affinity to VBC (unknown origin) at 50 uM at 20 degC by surface plasmon resonance assay | J Med Chem 61: 599-618 (2018) Article DOI: 10.1021/acs.jmedchem.7b00675 BindingDB Entry DOI: 10.7270/Q2736TJ6 | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
Elongin-C (Homo sapiens (Human)) | BDBM50459881 (CHEMBL4226376) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase MCE KEGG PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 109 | n/a | n/a | n/a | n/a | n/a |
University of Dundee Curated by ChEMBL | Assay Description Binding affinity to N-terminal His6-tagged recombinant human VHL (54 to 213 residues)/elongin C (17 to 112 residues)/elongin B (1 to 104 residues) ex... | J Med Chem 61: 504-513 (2018) Article DOI: 10.1021/acs.jmedchem.6b01912 BindingDB Entry DOI: 10.7270/Q2R49TC3 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Elongin-C (Homo sapiens (Human)) | BDBM50459954 (CHEMBL4228950) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | KEGG PC cid PC sid PDB UniChem | PDB Article PubMed | n/a | n/a | n/a | 115 | n/a | n/a | n/a | n/a | n/a |
University of Dundee Curated by ChEMBL | Assay Description Binding affinity to VBC (unknown origin) at 50 uM at 10 degC by surface plasmon resonance assay | J Med Chem 61: 599-618 (2018) Article DOI: 10.1021/acs.jmedchem.7b00675 BindingDB Entry DOI: 10.7270/Q2736TJ6 | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
Elongin-C (Homo sapiens (Human)) | BDBM50459878 (CHEMBL4227834) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | KEGG PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 116 | n/a | n/a | n/a | n/a | n/a |
University of Dundee Curated by ChEMBL | Assay Description Binding affinity to N-terminal His6-tagged recombinant human VHL (54 to 213 residues)/elongin C (17 to 112 residues)/elongin B (1 to 104 residues) ex... | J Med Chem 61: 504-513 (2018) Article DOI: 10.1021/acs.jmedchem.6b01912 BindingDB Entry DOI: 10.7270/Q2R49TC3 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Elongin-C (Homo sapiens (Human)) | BDBM50099062 (CHEMBL3344081 | US10730870, Example 3 | US11512083...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase CHEMBL MCE KEGG PC cid PC sid PDB UniChem Similars | PDB Article PubMed | n/a | n/a | n/a | 123 | n/a | n/a | n/a | n/a | n/a |
University of Dundee Curated by ChEMBL | Assay Description Binding affinity to VBC (unknown origin) at 50 uM at 10 degC by surface plasmon resonance assay | J Med Chem 61: 599-618 (2018) Article DOI: 10.1021/acs.jmedchem.7b00675 BindingDB Entry DOI: 10.7270/Q2736TJ6 | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
Elongin-C (Homo sapiens (Human)) | BDBM50459949 (CHEMBL4227893) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | KEGG PC cid PC sid PDB UniChem | PDB Article PubMed | n/a | n/a | n/a | 132 | n/a | n/a | n/a | n/a | n/a |
University of Dundee Curated by ChEMBL | Assay Description Binding affinity to VHL (unknown origin)/elongin C (unknown origin)/elongin B (unknown origin) by isothermal titration calorimetry-based assay | J Med Chem 61: 599-618 (2018) Article DOI: 10.1021/acs.jmedchem.7b00675 BindingDB Entry DOI: 10.7270/Q2736TJ6 | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
Elongin-C (Homo sapiens (Human)) | BDBM50459955 (CHEMBL4228624) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | KEGG PC cid PC sid PDB UniChem | PDB Article PubMed | n/a | n/a | n/a | 138 | n/a | n/a | n/a | n/a | n/a |
University of Dundee Curated by ChEMBL | Assay Description Binding affinity to VHL (unknown origin)/elongin C (unknown origin)/elongin B (unknown origin) by isothermal titration calorimetry-based assay | J Med Chem 61: 599-618 (2018) Article DOI: 10.1021/acs.jmedchem.7b00675 BindingDB Entry DOI: 10.7270/Q2736TJ6 | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
Elongin-C (Homo sapiens (Human)) | BDBM50459877 (CHEMBL4227158) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | KEGG PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 147 | n/a | n/a | n/a | n/a | n/a |
University of Dundee Curated by ChEMBL | Assay Description Binding affinity to N-terminal His6-tagged recombinant human VHL (54 to 213 residues)/elongin C (17 to 112 residues)/elongin B (1 to 104 residues) ex... | J Med Chem 61: 504-513 (2018) Article DOI: 10.1021/acs.jmedchem.6b01912 BindingDB Entry DOI: 10.7270/Q2R49TC3 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Elongin-C (Homo sapiens (Human)) | BDBM50099062 (CHEMBL3344081 | US10730870, Example 3 | US11512083...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase CHEMBL MCE KEGG PC cid PC sid PDB UniChem Similars | PDB Article PubMed | n/a | n/a | n/a | 150 | n/a | n/a | n/a | n/a | n/a |
University of Dundee Curated by ChEMBL | Assay Description Displacement of FAM-labeled HIF-1alpha peptide from VBC (unknown origin) by fluorescence polarization assay | J Med Chem 61: 599-618 (2018) Article DOI: 10.1021/acs.jmedchem.7b00675 BindingDB Entry DOI: 10.7270/Q2736TJ6 | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
Elongin-C (Homo sapiens (Human)) | BDBM50459949 (CHEMBL4227893) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | KEGG PC cid PC sid PDB UniChem | PDB Article PubMed | n/a | n/a | n/a | 170 | n/a | n/a | n/a | n/a | n/a |
University of Dundee Curated by ChEMBL | Assay Description Displacement of FAM-labeled HIF-1alpha peptide from VBC (unknown origin) by fluorescence polarization assay | J Med Chem 61: 599-618 (2018) Article DOI: 10.1021/acs.jmedchem.7b00675 BindingDB Entry DOI: 10.7270/Q2736TJ6 | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
Elongin-C (Homo sapiens (Human)) | BDBM50459954 (CHEMBL4228950) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | KEGG PC cid PC sid PDB UniChem | PDB Article PubMed | n/a | n/a | n/a | 170 | n/a | n/a | n/a | n/a | n/a |
University of Dundee Curated by ChEMBL | Assay Description Displacement of FAM-labeled HIF-1alpha peptide from VBC (unknown origin) by fluorescence polarization assay | J Med Chem 61: 599-618 (2018) Article DOI: 10.1021/acs.jmedchem.7b00675 BindingDB Entry DOI: 10.7270/Q2736TJ6 | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
Elongin-C (Homo sapiens (Human)) | BDBM50099062 (CHEMBL3344081 | US10730870, Example 3 | US11512083...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase CHEMBL MCE KEGG PC cid PC sid PDB UniChem Similars | PDB Article PubMed | n/a | n/a | n/a | 185 | n/a | n/a | n/a | n/a | n/a |
University of Dundee Curated by ChEMBL | Assay Description Binding affinity to VHL (unknown origin)/elongin C (unknown origin)/elongin B (unknown origin) by isothermal titration calorimetry-based assay | J Med Chem 61: 599-618 (2018) Article DOI: 10.1021/acs.jmedchem.7b00675 BindingDB Entry DOI: 10.7270/Q2736TJ6 | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
Elongin-C (Homo sapiens (Human)) | BDBM50459960 (CHEMBL4225199) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | KEGG PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 200 | n/a | n/a | n/a | n/a | n/a |
University of Dundee Curated by ChEMBL | Assay Description Displacement of FAM-labeled HIF-1alpha peptide from VBC (unknown origin) by fluorescence polarization assay | J Med Chem 61: 599-618 (2018) Article DOI: 10.1021/acs.jmedchem.7b00675 BindingDB Entry DOI: 10.7270/Q2736TJ6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Elongin-C (Homo sapiens (Human)) | BDBM50459947 (CHEMBL4225856) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | KEGG PC cid PC sid PDB UniChem | PDB Article PubMed | n/a | n/a | n/a | 200 | n/a | n/a | n/a | n/a | n/a |
University of Dundee Curated by ChEMBL | Assay Description Displacement of FAM-labeled HIF-1alpha peptide from VBC (unknown origin) by fluorescence polarization assay | J Med Chem 61: 599-618 (2018) Article DOI: 10.1021/acs.jmedchem.7b00675 BindingDB Entry DOI: 10.7270/Q2736TJ6 | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
Elongin-C (Homo sapiens (Human)) | BDBM50459945 (CHEMBL4229211) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | KEGG PC cid PC sid PDB UniChem | PDB Article PubMed | n/a | n/a | n/a | 210 | n/a | n/a | n/a | n/a | n/a |
University of Dundee Curated by ChEMBL | Assay Description Binding affinity to VHL (unknown origin)/elongin C (unknown origin)/elongin B (unknown origin) by isothermal titration calorimetry-based assay | J Med Chem 61: 599-618 (2018) Article DOI: 10.1021/acs.jmedchem.7b00675 BindingDB Entry DOI: 10.7270/Q2736TJ6 | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
Elongin-C (Homo sapiens (Human)) | BDBM50459961 (CHEMBL4225714) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | KEGG PC cid PC sid PDB UniChem | PDB Article PubMed | n/a | n/a | n/a | 230 | n/a | n/a | n/a | n/a | n/a |
University of Dundee Curated by ChEMBL | Assay Description Binding affinity to VHL (unknown origin)/elongin C (unknown origin)/elongin B (unknown origin) by isothermal titration calorimetry-based assay | J Med Chem 61: 599-618 (2018) Article DOI: 10.1021/acs.jmedchem.7b00675 BindingDB Entry DOI: 10.7270/Q2736TJ6 | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
Elongin-C (Homo sapiens (Human)) | BDBM50459945 (CHEMBL4229211) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | KEGG PC cid PC sid PDB UniChem | PDB Article PubMed | n/a | n/a | n/a | 233 | n/a | n/a | n/a | n/a | n/a |
University of Dundee Curated by ChEMBL | Assay Description Binding affinity to VBC (unknown origin) at 50 uM at 20 degC by surface plasmon resonance assay | J Med Chem 61: 599-618 (2018) Article DOI: 10.1021/acs.jmedchem.7b00675 BindingDB Entry DOI: 10.7270/Q2736TJ6 | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
Elongin-C (Homo sapiens (Human)) | BDBM50459945 (CHEMBL4229211) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | KEGG PC cid PC sid PDB UniChem | PDB Article PubMed | n/a | n/a | n/a | 250 | n/a | n/a | n/a | n/a | n/a |
University of Dundee Curated by ChEMBL | Assay Description Displacement of FAM-labeled HIF-1alpha peptide from VBC (unknown origin) by fluorescence polarization assay | J Med Chem 61: 599-618 (2018) Article DOI: 10.1021/acs.jmedchem.7b00675 BindingDB Entry DOI: 10.7270/Q2736TJ6 | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
Elongin-C (Homo sapiens (Human)) | BDBM50459950 (CHEMBL4228963) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | KEGG PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 270 | n/a | n/a | n/a | n/a | n/a |
University of Dundee Curated by ChEMBL | Assay Description Displacement of FAM-labeled HIF-1alpha peptide from VBC (unknown origin) by fluorescence polarization assay | J Med Chem 61: 599-618 (2018) Article DOI: 10.1021/acs.jmedchem.7b00675 BindingDB Entry DOI: 10.7270/Q2736TJ6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Elongin-C (Homo sapiens (Human)) | BDBM50459945 (CHEMBL4229211) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | KEGG PC cid PC sid PDB UniChem | PDB Article PubMed | n/a | n/a | n/a | 271 | n/a | n/a | n/a | n/a | n/a |
University of Dundee Curated by ChEMBL | Assay Description Binding affinity to VBC (unknown origin) at 50 uM at 10 degC by surface plasmon resonance assay | J Med Chem 61: 599-618 (2018) Article DOI: 10.1021/acs.jmedchem.7b00675 BindingDB Entry DOI: 10.7270/Q2736TJ6 | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
Elongin-C (Homo sapiens (Human)) | BDBM50459955 (CHEMBL4228624) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | KEGG PC cid PC sid PDB UniChem | PDB Article PubMed | n/a | n/a | n/a | 300 | n/a | n/a | n/a | n/a | n/a |
University of Dundee Curated by ChEMBL | Assay Description Displacement of FAM-labeled HIF-1alpha peptide from VBC (unknown origin) by fluorescence polarization assay | J Med Chem 61: 599-618 (2018) Article DOI: 10.1021/acs.jmedchem.7b00675 BindingDB Entry DOI: 10.7270/Q2736TJ6 | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
Elongin-C (Homo sapiens (Human)) | BDBM50459961 (CHEMBL4225714) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | KEGG PC cid PC sid PDB UniChem | PDB Article PubMed | n/a | n/a | n/a | 320 | n/a | n/a | n/a | n/a | n/a |
University of Dundee Curated by ChEMBL | Assay Description Displacement of FAM-labeled HIF-1alpha peptide from VBC (unknown origin) by fluorescence polarization assay | J Med Chem 61: 599-618 (2018) Article DOI: 10.1021/acs.jmedchem.7b00675 BindingDB Entry DOI: 10.7270/Q2736TJ6 | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
Elongin-C (Homo sapiens (Human)) | BDBM50459948 (CHEMBL4228328 | US10730870, Example 12 | US1151208...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | KEGG PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 350 | n/a | n/a | n/a | n/a | n/a |
University of Dundee Curated by ChEMBL | Assay Description Displacement of FAM-labeled HIF-1alpha peptide from VBC (unknown origin) by fluorescence polarization assay | J Med Chem 61: 599-618 (2018) Article DOI: 10.1021/acs.jmedchem.7b00675 BindingDB Entry DOI: 10.7270/Q2736TJ6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Elongin-C (Homo sapiens (Human)) | BDBM50459953 (CHEMBL4228692) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | KEGG PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 370 | n/a | n/a | n/a | n/a | n/a |
University of Dundee Curated by ChEMBL | Assay Description Displacement of FAM-labeled HIF-1alpha peptide from VBC (unknown origin) by fluorescence polarization assay | J Med Chem 61: 599-618 (2018) Article DOI: 10.1021/acs.jmedchem.7b00675 BindingDB Entry DOI: 10.7270/Q2736TJ6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Elongin-C (Homo sapiens (Human)) | BDBM50459942 (CHEMBL4227864 | US10730870, Example 85 | US1151208...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | KEGG PC cid PC sid PDB UniChem | PDB Article PubMed | n/a | n/a | n/a | 440 | n/a | n/a | n/a | n/a | n/a |
University of Dundee Curated by ChEMBL | Assay Description Binding affinity to VBC complex (unknown origin) by ITC assay | Bioorg Med Chem 26: 2992-2995 (2018) Article DOI: 10.1016/j.bmc.2018.03.034 BindingDB Entry DOI: 10.7270/Q2HX1GB7 | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
Elongin-C (Homo sapiens (Human)) | BDBM50459959 (CHEMBL4225145) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | KEGG PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 450 | n/a | n/a | n/a | n/a | n/a |
University of Dundee Curated by ChEMBL | Assay Description Displacement of FAM-labeled HIF-1alpha peptide from VBC (unknown origin) by fluorescence polarization assay | J Med Chem 61: 599-618 (2018) Article DOI: 10.1021/acs.jmedchem.7b00675 BindingDB Entry DOI: 10.7270/Q2736TJ6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Elongin-C (Homo sapiens (Human)) | BDBM50459956 (CHEMBL4224868) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | KEGG PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 500 | n/a | n/a | n/a | n/a | n/a |
University of Dundee Curated by ChEMBL | Assay Description Displacement of FAM-labeled HIF-1alpha peptide from VBC (unknown origin) by fluorescence polarization assay | J Med Chem 61: 599-618 (2018) Article DOI: 10.1021/acs.jmedchem.7b00675 BindingDB Entry DOI: 10.7270/Q2736TJ6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Elongin-C (Homo sapiens (Human)) | BDBM50459942 (CHEMBL4227864 | US10730870, Example 85 | US1151208...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | KEGG PC cid PC sid PDB UniChem | PDB Article PubMed | n/a | n/a | n/a | 690 | n/a | n/a | n/a | n/a | n/a |
University of Dundee Curated by ChEMBL | Assay Description Binding affinity to VBC complex (unknown origin) assessed as reduction of FAM-labelled HIF1alpha peptide binding by fluorescence polarization assay | Bioorg Med Chem 26: 2992-2995 (2018) Article DOI: 10.1016/j.bmc.2018.03.034 BindingDB Entry DOI: 10.7270/Q2HX1GB7 | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
Elongin-C (Homo sapiens (Human)) | BDBM50461569 (CHEMBL4228750) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid PDB UniChem | PDB Article PubMed | n/a | n/a | n/a | 760 | n/a | n/a | n/a | n/a | n/a |
University of Dundee Curated by ChEMBL | Assay Description Binding affinity to VBC complex (unknown origin) by ITC assay | Bioorg Med Chem 26: 2992-2995 (2018) Article DOI: 10.1016/j.bmc.2018.03.034 BindingDB Entry DOI: 10.7270/Q2HX1GB7 | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
Elongin-C (Homo sapiens (Human)) | BDBM50459942 (CHEMBL4227864 | US10730870, Example 85 | US1151208...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | KEGG PC cid PC sid PDB UniChem | PDB Article PubMed | n/a | n/a | n/a | 760 | n/a | n/a | n/a | n/a | n/a |
University of Dundee Curated by ChEMBL | Assay Description Displacement of FAM-labeled HIF-1alpha peptide from VBC (unknown origin) by fluorescence polarization assay | J Med Chem 61: 599-618 (2018) Article DOI: 10.1021/acs.jmedchem.7b00675 BindingDB Entry DOI: 10.7270/Q2736TJ6 | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
Elongin-C (Homo sapiens (Human)) | BDBM50459951 (CHEMBL4229225) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | KEGG PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 770 | n/a | n/a | n/a | n/a | n/a |
University of Dundee Curated by ChEMBL | Assay Description Displacement of FAM-labeled HIF-1alpha peptide from VBC (unknown origin) by fluorescence polarization assay | J Med Chem 61: 599-618 (2018) Article DOI: 10.1021/acs.jmedchem.7b00675 BindingDB Entry DOI: 10.7270/Q2736TJ6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Elongin-C (Homo sapiens (Human)) | BDBM50461569 (CHEMBL4228750) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid PDB UniChem | PDB Article PubMed | n/a | n/a | n/a | 1.00E+3 | n/a | n/a | n/a | n/a | n/a |
University of Dundee Curated by ChEMBL | Assay Description Binding affinity to VBC complex (unknown origin) assessed as reduction of FAM-labelled HIF1alpha peptide binding by fluorescence polarization assay | Bioorg Med Chem 26: 2992-2995 (2018) Article DOI: 10.1016/j.bmc.2018.03.034 BindingDB Entry DOI: 10.7270/Q2HX1GB7 | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
Elongin-C (Homo sapiens (Human)) | BDBM50459957 (CHEMBL4229276) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | KEGG PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 1.40E+3 | n/a | n/a | n/a | n/a | n/a |
University of Dundee Curated by ChEMBL | Assay Description Displacement of FAM-labeled HIF-1alpha peptide from VBC (unknown origin) by fluorescence polarization assay | J Med Chem 61: 599-618 (2018) Article DOI: 10.1021/acs.jmedchem.7b00675 BindingDB Entry DOI: 10.7270/Q2736TJ6 | |||||||||||
More data for this Ligand-Target Pair |
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