Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kcal/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
ATPase family AAA domain-containing protein 2B (Homo sapiens (Human)) | BDBM50539801 (CHEMBL4648912 | US11840533, Compound 70) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase MCE PC cid PC sid PDB UniChem | Article PubMed | n/a | n/a | n/a | <1 | n/a | n/a | n/a | n/a | n/a |
University of Illinois at Chicago Curated by ChEMBL | Assay Description Binding affinity to human partial length ATAD2B (Q955 to R1082 residues) expressed in bacterial expression system by BROMOscan assay | J Med Chem 63: 7186-7210 (2020) Article DOI: 10.1021/acs.jmedchem.0c00456 BindingDB Entry DOI: 10.7270/Q2PK0KPP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
ATPase family AAA domain-containing protein 2B (Homo sapiens (Human)) | BDBM50584925 (CHEMBL5079885) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid PDB UniChem | Article PubMed | n/a | n/a | n/a | 7.90 | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Binding affinity to human ATAD2B bromodomain assessed as dissociation constant by BROMOscan method | Citation and Details Article DOI: 10.1021/acs.jmedchem.1c01871 BindingDB Entry DOI: 10.7270/Q2280CH8 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
ATPase family AAA domain-containing protein 2B (Homo sapiens (Human)) | BDBM50514857 (CHEMBL4449894) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 20 | n/a | n/a | n/a | n/a | n/a |
University of Strathclyde Curated by ChEMBL | Assay Description Binding affinity to human partial length ATAD2B (Q955 to R1082 residues) expressed in bacterial expression system by BROMOscan assay | J Med Chem 63: 5212-5241 (2020) Article DOI: 10.1021/acs.jmedchem.0c00021 BindingDB Entry DOI: 10.7270/Q2RN3C7T | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
ATPase family AAA domain-containing protein 2B (Homo sapiens (Human)) | BDBM50098311 (CHEMBL3590408) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | 100 | n/a | n/a | n/a | n/a | n/a |
GlaxoSmithKline Curated by ChEMBL | Assay Description Binding affinity to ATAD2B in human HUT78 cells incubated for 45 mins by mass spectrometry based bromosphere chemoproteomic assay | J Med Chem 58: 6151-78 (2015) Article DOI: 10.1021/acs.jmedchem.5b00773 BindingDB Entry DOI: 10.7270/Q2FN17Z1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
ATPase family AAA domain-containing protein 2B (Homo sapiens (Human)) | BDBM50098305 (CHEMBL3590405) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid PDB UniChem Similars | Article PubMed | n/a | n/a | n/a | 167 | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Binding affinity to N-terminal GST tagged human ATAD2B (953-1085 residues) expressed in Escherichia coli by ITC analysis | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01178 BindingDB Entry DOI: 10.7270/Q2G44TWF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
ATPase family AAA domain-containing protein 2B (Homo sapiens (Human)) | BDBM179481 (US9675697, Cpd. No. 73) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase MCE PC cid PC sid PDB UniChem | Article PubMed | n/a | n/a | n/a | >4.00E+3 | n/a | n/a | n/a | n/a | n/a |
University of Michigan Curated by ChEMBL | Assay Description Binding affinity to human partial length ATAD2B (Q955 to R1082 residues) expressed in bacterial expression system by BROMOscan assay | J Med Chem 60: 3887-3901 (2017) Article DOI: 10.1021/acs.jmedchem.7b00193 BindingDB Entry DOI: 10.7270/Q28W3GWN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
ATPase family AAA domain-containing protein 2B (Homo sapiens (Human)) | BDBM50366670 (CHEMBL4173488) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase MCE PC cid PC sid PDB UniChem Similars | Article PubMed | n/a | n/a | n/a | >5.00E+3 | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Binding affinity to human ATAD2B (Q955 to R1082 residues) expressed in bacterial expression system by BROMOScan assay | J Med Chem 61: 6110-6120 (2018) Article DOI: 10.1021/acs.jmedchem.8b00483 BindingDB Entry DOI: 10.7270/Q26M39B1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
ATPase family AAA domain-containing protein 2B (Homo sapiens (Human)) | BDBM50547686 (CHEMBL4786330) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | KEGG PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 5.20E+3 | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Binding affinity to N-terminal GST tagged human ATAD2B (953-1085 residues) expressed in Escherichia coli by ITC analysis | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01178 BindingDB Entry DOI: 10.7270/Q2G44TWF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
ATPase family AAA domain-containing protein 2B (Homo sapiens (Human)) | BDBM50453949 (CHEMBL4208820 | US11247989, Example 87) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a | n/a |
WuXi AppTec Co., Ltd. Curated by ChEMBL | Assay Description Binding affinity to human partial length ATAD2B (Q955 to R1082 residues) expressed in bacterial expression system by BROMOscan assay | Bioorg Med Chem Lett 28: 15-23 (2018) Article DOI: 10.1016/j.bmcl.2017.11.025 BindingDB Entry DOI: 10.7270/Q2ZG6VVZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
ATPase family AAA domain-containing protein 2B (Homo sapiens (Human)) | BDBM50092310 (CHEMBL3581661 | US9675697, Cpd. No. 23) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid PDB UniChem Similars | Article PubMed | n/a | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a | n/a |
University of Michigan Curated by ChEMBL | Assay Description Binding affinity to biotinylated ATAD2B (953 to 1086 amino acid residues) (unknown origin) expressed in Rosetta2 DE3 cells by bio-layer interferometr... | J Med Chem 58: 4927-39 (2015) Article DOI: 10.1021/acs.jmedchem.5b00613 BindingDB Entry DOI: 10.7270/Q2XD13FK | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
ATPase family AAA domain-containing protein 2B (Homo sapiens (Human)) | BDBM249277 (US10017501, Compound 1020-18 | US9458145, 1020-18) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a | n/a |
Gilead Sciences, Inc. Curated by ChEMBL | Assay Description Binding affinity to human partial length ATAD2B (Q955 to R1082 residues) expressed in bacterial expression system after 1 hr by bromoscan assay | Bioorg Med Chem 27: 457-469 (2019) Article DOI: 10.1016/j.bmc.2018.11.020 BindingDB Entry DOI: 10.7270/Q2HD7ZZ6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
ATPase family AAA domain-containing protein 2B (Homo sapiens (Human)) | BDBM50560174 (GSK789) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid PDB UniChem | Article PubMed | n/a | n/a | n/a | 1.58E+4 | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Binding affinity to human partial length ATAD2B (Q955 to R1082 residues) expressed in bacterial expression system by BROMOscan assay | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c00614 BindingDB Entry DOI: 10.7270/Q27D2ZVG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
ATPase family AAA domain-containing protein 2B (Homo sapiens (Human)) | BDBM50547692 (CHEMBL4748520) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | KEGG PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 1.87E+4 | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Binding affinity to N-terminal GST tagged human ATAD2B (953-1085 residues) expressed in Escherichia coli by ITC analysis | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01178 BindingDB Entry DOI: 10.7270/Q2G44TWF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
ATPase family AAA domain-containing protein 2B (Homo sapiens (Human)) | BDBM50547691 (CHEMBL4792431) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | KEGG PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 2.81E+4 | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Binding affinity to N-terminal GST tagged human ATAD2B (953-1085 residues) expressed in Escherichia coli by ITC analysis | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01178 BindingDB Entry DOI: 10.7270/Q2G44TWF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
ATPase family AAA domain-containing protein 2B (Homo sapiens (Human)) | BDBM50547693 (CHEMBL4794843) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | KEGG PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 3.44E+4 | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Binding affinity to N-terminal GST tagged human ATAD2B (953-1085 residues) expressed in Escherichia coli by ITC analysis | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01178 BindingDB Entry DOI: 10.7270/Q2G44TWF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
ATPase family AAA domain-containing protein 2B (Homo sapiens (Human)) | BDBM50547694 (CHEMBL4748267) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | KEGG PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 3.57E+4 | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Binding affinity to N-terminal GST tagged human ATAD2B (953-1085 residues) expressed in Escherichia coli by ITC analysis | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01178 BindingDB Entry DOI: 10.7270/Q2G44TWF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
ATPase family AAA domain-containing protein 2B (Homo sapiens (Human)) | BDBM50547685 (CHEMBL4751427) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | KEGG PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 4.25E+4 | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Binding affinity to N-terminal GST tagged human ATAD2B (953-1085 residues) expressed in Escherichia coli by ITC analysis | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01178 BindingDB Entry DOI: 10.7270/Q2G44TWF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
ATPase family AAA domain-containing protein 2B (Homo sapiens (Human)) | BDBM50547687 (CHEMBL4750026) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | KEGG PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 4.80E+4 | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Binding affinity to N-terminal GST tagged human ATAD2B (953-1085 residues) expressed in Escherichia coli by ITC analysis | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01178 BindingDB Entry DOI: 10.7270/Q2G44TWF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
ATPase family AAA domain-containing protein 2B (Homo sapiens (Human)) | BDBM50547689 (CHEMBL4762063) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | KEGG PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 5.05E+4 | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Binding affinity to N-terminal GST tagged human ATAD2B (953-1085 residues) expressed in Escherichia coli by ITC analysis | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01178 BindingDB Entry DOI: 10.7270/Q2G44TWF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
ATPase family AAA domain-containing protein 2B (Homo sapiens (Human)) | BDBM50547695 (CHEMBL4762443) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | KEGG PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 2.14E+5 | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Binding affinity to N-terminal GST tagged human ATAD2B (953-1085 residues) expressed in Escherichia coli by ITC analysis | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01178 BindingDB Entry DOI: 10.7270/Q2G44TWF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
ATPase family AAA domain-containing protein 2B (Homo sapiens (Human)) | BDBM50547690 (CHEMBL4795500) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | KEGG PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 6.85E+5 | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Binding affinity to N-terminal GST tagged human ATAD2B (953-1085 residues) expressed in Escherichia coli by ITC analysis | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01178 BindingDB Entry DOI: 10.7270/Q2G44TWF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
ATPase family AAA domain-containing protein 2B (Homo sapiens (Human)) | BDBM50547688 (CHEMBL4751374) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | KEGG PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 1.16E+6 | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Binding affinity to N-terminal GST tagged human ATAD2B (953-1085 residues) expressed in Escherichia coli by ITC analysis | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01178 BindingDB Entry DOI: 10.7270/Q2G44TWF | |||||||||||
More data for this Ligand-Target Pair |