Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kcal/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
RCG37580 (Rattus norvegicus) | BDBM50030788 (CHEMBL3342358) | KEGG UniProtKB/TrEMBL GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 0.400 | n/a | n/a | n/a | n/a |
Novartis Institutes for BioMedical Research Curated by ChEMBL | Assay Description Agonist activity at rat GPR39 by IP1 assay | ACS Med Chem Lett 5: 1114-8 (2014) Article DOI: 10.1021/ml500240d BindingDB Entry DOI: 10.7270/Q2MC91MW | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
RCG37580 (Rattus norvegicus) | BDBM50030788 (CHEMBL3342358) | KEGG UniProtKB/TrEMBL GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 0.400 | n/a | n/a | n/a | n/a |
Novartis Institutes for BioMedical Research Curated by ChEMBL | Assay Description Agonist activity at rat GPR39 expressed in HEK293 cells by IP1 assay | ACS Med Chem Lett 5: 1114-8 (2014) Article DOI: 10.1021/ml500240d BindingDB Entry DOI: 10.7270/Q2MC91MW | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
RCG37580 (Rattus norvegicus) | BDBM50030774 (CHEMBL3342379) | KEGG UniProtKB/TrEMBL GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 0.600 | n/a | n/a | n/a | n/a |
Novartis Institutes for BioMedical Research Curated by ChEMBL | Assay Description Agonist activity at rat GPR39 expressed in HEK293 cells by IP1 assay | ACS Med Chem Lett 5: 1114-8 (2014) Article DOI: 10.1021/ml500240d BindingDB Entry DOI: 10.7270/Q2MC91MW | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
RCG37580 (Rattus norvegicus) | BDBM50030789 (CHEMBL3341764) | KEGG UniProtKB/TrEMBL GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 1 | n/a | n/a | n/a | n/a |
Novartis Institutes for BioMedical Research Curated by ChEMBL | Assay Description Agonist activity at rat GPR39 by IP1 assay | ACS Med Chem Lett 5: 1114-8 (2014) Article DOI: 10.1021/ml500240d BindingDB Entry DOI: 10.7270/Q2MC91MW | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
RCG37580 (Rattus norvegicus) | BDBM50030776 (CHEMBL3342377) | KEGG UniProtKB/TrEMBL GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 2 | n/a | n/a | n/a | n/a |
Novartis Institutes for BioMedical Research Curated by ChEMBL | Assay Description Agonist activity at rat GPR39 expressed in HEK293 cells by IP1 assay | ACS Med Chem Lett 5: 1114-8 (2014) Article DOI: 10.1021/ml500240d BindingDB Entry DOI: 10.7270/Q2MC91MW | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
RCG37580 (Rattus norvegicus) | BDBM50030777 (CHEMBL3342376) | KEGG UniProtKB/TrEMBL GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 3 | n/a | n/a | n/a | n/a |
Novartis Institutes for BioMedical Research Curated by ChEMBL | Assay Description Agonist activity at rat GPR39 expressed in HEK293 cells by IP1 assay | ACS Med Chem Lett 5: 1114-8 (2014) Article DOI: 10.1021/ml500240d BindingDB Entry DOI: 10.7270/Q2MC91MW | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
RCG37580 (Rattus norvegicus) | BDBM50030790 (CHEMBL3342357) | KEGG UniProtKB/TrEMBL GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 12 | n/a | n/a | n/a | n/a |
Novartis Institutes for BioMedical Research Curated by ChEMBL | Assay Description Agonist activity at rat GPR39 by IP1 assay | ACS Med Chem Lett 5: 1114-8 (2014) Article DOI: 10.1021/ml500240d BindingDB Entry DOI: 10.7270/Q2MC91MW | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
RCG37580 (Rattus norvegicus) | BDBM16 (Zn2+ | zinc(2+) ion) | KEGG UniProtKB/TrEMBL GoogleScholar AffyNet | Purchase MCE KEGG MMDB PC cid PC sid PDB UniChem | Article PubMed | n/a | n/a | n/a | n/a | 4.04E+3 | n/a | n/a | n/a | n/a |
Novartis Institutes for BioMedical Research Curated by ChEMBL | Assay Description Agonist activity at rat GPR39 expressed in HEK293 cells by IP1 assay | ACS Med Chem Lett 5: 1114-8 (2014) Article DOI: 10.1021/ml500240d BindingDB Entry DOI: 10.7270/Q2MC91MW | |||||||||||
More data for this Ligand-Target Pair |