Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kcal/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Thiol:disulfide interchange protein DsbA (Escherichia coli (strain K12)) | BDBM50062483 (CHEMBL3397433) | PDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | 2.20E+3 | n/a | n/a | n/a | n/a | n/a |
University of Queensland Curated by ChEMBL | Assay Description Binding affinity to oxidized Escherichia coli DsbA by isothermal titration calorimetry assay | J Med Chem 58: 577-87 (2015) Article DOI: 10.1021/jm500955s BindingDB Entry DOI: 10.7270/Q2BP04GJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Thiol:disulfide interchange protein DsbA (Escherichia coli (strain K12)) | BDBM50062385 (CHEMBL3397424) | PDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | 2.70E+3 | n/a | n/a | n/a | n/a | n/a |
University of Queensland Curated by ChEMBL | Assay Description Binding affinity to oxidized Escherichia coli DsbA by isothermal titration calorimetry assay | J Med Chem 58: 577-87 (2015) Article DOI: 10.1021/jm500955s BindingDB Entry DOI: 10.7270/Q2BP04GJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Thiol:disulfide interchange protein DsbA (Escherichia coli (strain K12)) | BDBM50062386 (CHEMBL3397425) | PDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | 2.80E+3 | n/a | n/a | n/a | n/a | n/a |
University of Queensland Curated by ChEMBL | Assay Description Binding affinity to oxidized Escherichia coli DsbA by isothermal titration calorimetry assay | J Med Chem 58: 577-87 (2015) Article DOI: 10.1021/jm500955s BindingDB Entry DOI: 10.7270/Q2BP04GJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Thiol:disulfide interchange protein DsbA (Escherichia coli (strain K12)) | BDBM50062490 (CHEMBL3397418) | PDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | 2.90E+3 | n/a | n/a | n/a | n/a | n/a |
University of Queensland Curated by ChEMBL | Assay Description Binding affinity to oxidized Escherichia coli DsbA by isothermal titration calorimetry assay | J Med Chem 58: 577-87 (2015) Article DOI: 10.1021/jm500955s BindingDB Entry DOI: 10.7270/Q2BP04GJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Thiol:disulfide interchange protein DsbA (Escherichia coli (strain K12)) | BDBM50062484 (CHEMBL3397434) | PDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | 3.00E+3 | n/a | n/a | n/a | n/a | n/a |
University of Queensland Curated by ChEMBL | Assay Description Binding affinity to oxidized Escherichia coli DsbA by isothermal titration calorimetry assay | J Med Chem 58: 577-87 (2015) Article DOI: 10.1021/jm500955s BindingDB Entry DOI: 10.7270/Q2BP04GJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Thiol:disulfide interchange protein DsbA (Escherichia coli (strain K12)) | BDBM50062448 (CHEMBL3397430) | PDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | 3.10E+3 | n/a | n/a | n/a | n/a | n/a |
University of Queensland Curated by ChEMBL | Assay Description Binding affinity to oxidized Escherichia coli DsbA by isothermal titration calorimetry assay | J Med Chem 58: 577-87 (2015) Article DOI: 10.1021/jm500955s BindingDB Entry DOI: 10.7270/Q2BP04GJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Thiol:disulfide interchange protein DsbA (Escherichia coli (strain K12)) | BDBM50062487 (CHEMBL3397415) | PDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | 4.00E+3 | n/a | n/a | n/a | n/a | n/a |
University of Queensland Curated by ChEMBL | Assay Description Binding affinity to oxidized Escherichia coli DsbA by isothermal titration calorimetry assay | J Med Chem 58: 577-87 (2015) Article DOI: 10.1021/jm500955s BindingDB Entry DOI: 10.7270/Q2BP04GJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Thiol:disulfide interchange protein DsbA (Escherichia coli (strain K12)) | BDBM50062481 (CHEMBL3397431) | PDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | 4.40E+3 | n/a | n/a | n/a | n/a | n/a |
University of Queensland Curated by ChEMBL | Assay Description Binding affinity to oxidized Escherichia coli DsbA by isothermal titration calorimetry assay | J Med Chem 58: 577-87 (2015) Article DOI: 10.1021/jm500955s BindingDB Entry DOI: 10.7270/Q2BP04GJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Thiol:disulfide interchange protein DsbA (Escherichia coli (strain K12)) | BDBM50062388 (CHEMBL3397426) | PDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | 5.50E+3 | n/a | n/a | n/a | n/a | n/a |
University of Queensland Curated by ChEMBL | Assay Description Binding affinity to oxidized Escherichia coli DsbA by isothermal titration calorimetry assay | J Med Chem 58: 577-87 (2015) Article DOI: 10.1021/jm500955s BindingDB Entry DOI: 10.7270/Q2BP04GJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Thiol:disulfide interchange protein DsbA (Escherichia coli (strain K12)) | BDBM50062485 (CHEMBL3397435) | PDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | 5.70E+3 | n/a | n/a | n/a | n/a | n/a |
University of Queensland Curated by ChEMBL | Assay Description Binding affinity to oxidized Escherichia coli DsbA by isothermal titration calorimetry assay | J Med Chem 58: 577-87 (2015) Article DOI: 10.1021/jm500955s BindingDB Entry DOI: 10.7270/Q2BP04GJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Thiol:disulfide interchange protein DsbA (Escherichia coli (strain K12)) | BDBM50062389 (CHEMBL3397427) | PDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | 5.80E+3 | n/a | n/a | n/a | n/a | n/a |
University of Queensland Curated by ChEMBL | Assay Description Binding affinity to oxidized Escherichia coli DsbA by isothermal titration calorimetry assay | J Med Chem 58: 577-87 (2015) Article DOI: 10.1021/jm500955s BindingDB Entry DOI: 10.7270/Q2BP04GJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Thiol:disulfide interchange protein DsbA (Escherichia coli (strain K12)) | BDBM50062488 (CHEMBL3397416) | PDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | 5.90E+3 | n/a | n/a | n/a | n/a | n/a |
University of Queensland Curated by ChEMBL | Assay Description Binding affinity to oxidized Escherichia coli DsbA by isothermal titration calorimetry assay | J Med Chem 58: 577-87 (2015) Article DOI: 10.1021/jm500955s BindingDB Entry DOI: 10.7270/Q2BP04GJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Thiol:disulfide interchange protein DsbA (Escherichia coli (strain K12)) | BDBM50062486 (CHEMBL3397436) | PDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | 8.30E+3 | n/a | n/a | n/a | n/a | n/a |
University of Queensland Curated by ChEMBL | Assay Description Binding affinity to oxidized Escherichia coli DsbA by isothermal titration calorimetry assay | J Med Chem 58: 577-87 (2015) Article DOI: 10.1021/jm500955s BindingDB Entry DOI: 10.7270/Q2BP04GJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Thiol:disulfide interchange protein DsbA (Escherichia coli (strain K12)) | BDBM50062493 (CHEMBL3397421) | PDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | 9.70E+3 | n/a | n/a | n/a | n/a | n/a |
University of Queensland Curated by ChEMBL | Assay Description Binding affinity to oxidized Escherichia coli DsbA by isothermal titration calorimetry assay | J Med Chem 58: 577-87 (2015) Article DOI: 10.1021/jm500955s BindingDB Entry DOI: 10.7270/Q2BP04GJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Thiol:disulfide interchange protein DsbA (Escherichia coli (strain K12)) | BDBM50062482 (CHEMBL3397432) | PDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | 1.07E+4 | n/a | n/a | n/a | n/a | n/a |
University of Queensland Curated by ChEMBL | Assay Description Binding affinity to oxidized Escherichia coli DsbA by isothermal titration calorimetry assay | J Med Chem 58: 577-87 (2015) Article DOI: 10.1021/jm500955s BindingDB Entry DOI: 10.7270/Q2BP04GJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Thiol:disulfide interchange protein DsbA (Escherichia coli (strain K12)) | BDBM50062390 (CHEMBL3397428) | PDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | 1.13E+4 | n/a | n/a | n/a | n/a | n/a |
University of Queensland Curated by ChEMBL | Assay Description Binding affinity to oxidized Escherichia coli DsbA by isothermal titration calorimetry assay | J Med Chem 58: 577-87 (2015) Article DOI: 10.1021/jm500955s BindingDB Entry DOI: 10.7270/Q2BP04GJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Thiol:disulfide interchange protein DsbA (Escherichia coli (strain K12)) | BDBM50062363 (CHEMBL3397422) | PDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | 1.20E+4 | n/a | n/a | n/a | n/a | n/a |
University of Queensland Curated by ChEMBL | Assay Description Binding affinity to oxidized Escherichia coli DsbA by isothermal titration calorimetry assay | J Med Chem 58: 577-87 (2015) Article DOI: 10.1021/jm500955s BindingDB Entry DOI: 10.7270/Q2BP04GJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Thiol:disulfide interchange protein DsbA (Escherichia coli (strain K12)) | BDBM50062489 (CHEMBL3397417) | PDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | 1.31E+4 | n/a | n/a | n/a | n/a | n/a |
University of Queensland Curated by ChEMBL | Assay Description Binding affinity to oxidized Escherichia coli DsbA by isothermal titration calorimetry assay | J Med Chem 58: 577-87 (2015) Article DOI: 10.1021/jm500955s BindingDB Entry DOI: 10.7270/Q2BP04GJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Thiol:disulfide interchange protein DsbA (Escherichia coli (strain K12)) | BDBM50062364 (CHEMBL3397423) | PDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | 1.31E+4 | n/a | n/a | n/a | n/a | n/a |
University of Queensland Curated by ChEMBL | Assay Description Binding affinity to oxidized Escherichia coli DsbA by isothermal titration calorimetry assay | J Med Chem 58: 577-87 (2015) Article DOI: 10.1021/jm500955s BindingDB Entry DOI: 10.7270/Q2BP04GJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Thiol:disulfide interchange protein DsbA (Escherichia coli (strain K12)) | BDBM50062492 (CHEMBL3397420) | PDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | 1.49E+4 | n/a | n/a | n/a | n/a | n/a |
University of Queensland Curated by ChEMBL | Assay Description Binding affinity to oxidized Escherichia coli DsbA by isothermal titration calorimetry assay | J Med Chem 58: 577-87 (2015) Article DOI: 10.1021/jm500955s BindingDB Entry DOI: 10.7270/Q2BP04GJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Thiol:disulfide interchange protein DsbA (Escherichia coli (strain K12)) | BDBM50062491 (CHEMBL3397419) | PDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | 1.80E+4 | n/a | n/a | n/a | n/a | n/a |
University of Queensland Curated by ChEMBL | Assay Description Binding affinity to oxidized Escherichia coli DsbA by isothermal titration calorimetry assay | J Med Chem 58: 577-87 (2015) Article DOI: 10.1021/jm500955s BindingDB Entry DOI: 10.7270/Q2BP04GJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Thiol:disulfide interchange protein DsbA (Escherichia coli (strain K12)) | BDBM50539928 (CHEMBL4635874) | PDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid PDB UniChem | PDB Article PubMed | n/a | n/a | n/a | 6.20E+4 | n/a | n/a | n/a | n/a | n/a |
Monash University (Parkville Campus) Curated by ChEMBL | Assay Description Binding affinity to uniformly labeled 15N oxidized Escherichia coli DsbA by 1H-15N HSQC NMR spectroscopy | J Med Chem 63: 6863-6875 (2020) Article DOI: 10.1021/acs.jmedchem.0c00111 BindingDB Entry DOI: 10.7270/Q2X3520R | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
Thiol:disulfide interchange protein DsbA (Escherichia coli (strain K12)) | BDBM50539930 (CHEMBL4640751) | PDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid PDB UniChem | PDB Article PubMed | n/a | n/a | n/a | 2.30E+5 | n/a | n/a | n/a | n/a | n/a |
Monash University (Parkville Campus) Curated by ChEMBL | Assay Description Binding affinity to uniformly labeled 15N oxidized Escherichia coli DsbA by 1H-15N HSQC NMR spectroscopy | J Med Chem 63: 6863-6875 (2020) Article DOI: 10.1021/acs.jmedchem.0c00111 BindingDB Entry DOI: 10.7270/Q2X3520R | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
Thiol:disulfide interchange protein DsbA (Escherichia coli (strain K12)) | BDBM50576685 (CHEMBL4871128) | PDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid PDB UniChem | PDB Article PubMed | n/a | n/a | n/a | 2.74E+5 | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Binding affinity to 15N-labelled Escherichia coli DsbA measured by 1H-15N HSQC NMR spectroscopy | Citation and Details Article DOI: 10.1016/j.bmc.2021.116315 BindingDB Entry DOI: 10.7270/Q2765K51 | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
Thiol:disulfide interchange protein DsbA (Escherichia coli (strain K12)) | BDBM50539926 (CHEMBL4648660) | PDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid PDB UniChem | PDB Article PubMed | n/a | n/a | n/a | 2.90E+5 | n/a | n/a | n/a | n/a | n/a |
Monash University (Parkville Campus) Curated by ChEMBL | Assay Description Binding affinity to uniformly labeled 15N oxidized Escherichia coli DsbA by 1H-15N HSQC NMR spectroscopy | J Med Chem 63: 6863-6875 (2020) Article DOI: 10.1021/acs.jmedchem.0c00111 BindingDB Entry DOI: 10.7270/Q2X3520R | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
Thiol:disulfide interchange protein DsbA (Escherichia coli (strain K12)) | BDBM50539927 (CHEMBL4641779) | PDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid PDB UniChem | PDB Article PubMed | n/a | n/a | n/a | 3.65E+5 | n/a | n/a | n/a | n/a | n/a |
Monash University (Parkville Campus) Curated by ChEMBL | Assay Description Binding affinity to uniformly labeled 15N oxidized Escherichia coli DsbA by 1H-15N HSQC NMR spectroscopy | J Med Chem 63: 6863-6875 (2020) Article DOI: 10.1021/acs.jmedchem.0c00111 BindingDB Entry DOI: 10.7270/Q2X3520R | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
Thiol:disulfide interchange protein DsbA (Escherichia coli (strain K12)) | BDBM50576683 (CHEMBL4854940) | PDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 4.03E+5 | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Binding affinity to 15N-labelled Escherichia coli DsbA measured by 1H-15N HSQC NMR spectroscopy | Citation and Details Article DOI: 10.1016/j.bmc.2021.116315 BindingDB Entry DOI: 10.7270/Q2765K51 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Thiol:disulfide interchange protein DsbA (Escherichia coli (strain K12)) | BDBM50539929 (CHEMBL4638876) | PDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 4.30E+5 | n/a | n/a | n/a | n/a | n/a |
Monash University (Parkville Campus) Curated by ChEMBL | Assay Description Binding affinity to uniformly labeled 15N oxidized Escherichia coli DsbA by 1H-15N HSQC NMR spectroscopy | J Med Chem 63: 6863-6875 (2020) Article DOI: 10.1021/acs.jmedchem.0c00111 BindingDB Entry DOI: 10.7270/Q2X3520R | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Thiol:disulfide interchange protein DsbA (Escherichia coli (strain K12)) | BDBM50576682 (CHEMBL4855609) | PDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 4.60E+5 | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Binding affinity to 15N-labelled Escherichia coli DsbA measured by 1H-15N HSQC NMR spectroscopy | Citation and Details Article DOI: 10.1016/j.bmc.2021.116315 BindingDB Entry DOI: 10.7270/Q2765K51 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Thiol:disulfide interchange protein DsbA (Escherichia coli (strain K12)) | BDBM50539925 (CHEMBL4633160) | PDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid PDB UniChem | PDB Article PubMed | n/a | n/a | n/a | 4.80E+5 | n/a | n/a | n/a | n/a | n/a |
Monash University (Parkville Campus) Curated by ChEMBL | Assay Description Binding affinity to uniformly labeled 15N oxidized Escherichia coli DsbA by 1H-15N HSQC NMR spectroscopy | J Med Chem 63: 6863-6875 (2020) Article DOI: 10.1021/acs.jmedchem.0c00111 BindingDB Entry DOI: 10.7270/Q2X3520R | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
Thiol:disulfide interchange protein DsbA (Escherichia coli (strain K12)) | BDBM50539924 (CHEMBL4634926) | PDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | KEGG PC cid PC sid PDB UniChem | PDB Article PubMed | n/a | n/a | n/a | 4.90E+5 | n/a | n/a | n/a | n/a | n/a |
Monash University (Parkville Campus) Curated by ChEMBL | Assay Description Binding affinity to uniformly labeled 15N oxidized Escherichia coli DsbA by 1H-15N HSQC NMR spectroscopy | J Med Chem 63: 6863-6875 (2020) Article DOI: 10.1021/acs.jmedchem.0c00111 BindingDB Entry DOI: 10.7270/Q2X3520R | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
Thiol:disulfide interchange protein DsbA (Escherichia coli (strain K12)) | BDBM50576684 (CHEMBL4848780) | PDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid PDB UniChem | PDB Article PubMed | n/a | n/a | n/a | 5.31E+5 | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Binding affinity to 15N-labelled Escherichia coli DsbA measured by 1H-15N HSQC NMR spectroscopy | Citation and Details Article DOI: 10.1016/j.bmc.2021.116315 BindingDB Entry DOI: 10.7270/Q2765K51 | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
Thiol:disulfide interchange protein DsbA (Escherichia coli (strain K12)) | BDBM50576679 (CHEMBL4851994) | PDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 8.20E+5 | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Binding affinity to 15N-labelled Escherichia coli DsbA measured by 1H-15N HSQC NMR spectroscopy | Citation and Details Article DOI: 10.1016/j.bmc.2021.116315 BindingDB Entry DOI: 10.7270/Q2765K51 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Thiol:disulfide interchange protein DsbA (Escherichia coli (strain K12)) | BDBM50576676 (CHEMBL4868312) | PDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 8.30E+5 | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Binding affinity to 15N-labelled Escherichia coli DsbA measured by 1H-15N HSQC NMR spectroscopy | Citation and Details Article DOI: 10.1016/j.bmc.2021.116315 BindingDB Entry DOI: 10.7270/Q2765K51 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Thiol:disulfide interchange protein DsbA (Escherichia coli (strain K12)) | BDBM50576686 (CHEMBL4875684) | PDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid PDB UniChem | PDB Article PubMed | n/a | n/a | n/a | 9.78E+5 | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Binding affinity to 15N-labelled Escherichia coli DsbA measured by 1H-15N HSQC NMR spectroscopy | Citation and Details Article DOI: 10.1016/j.bmc.2021.116315 BindingDB Entry DOI: 10.7270/Q2765K51 | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
Thiol:disulfide interchange protein DsbA (Escherichia coli (strain K12)) | BDBM50539932 (CHEMBL4641638) | PDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | >1.00E+6 | n/a | n/a | n/a | n/a | n/a |
Monash University (Parkville Campus) Curated by ChEMBL | Assay Description Binding affinity to uniformly labeled 15N oxidized Escherichia coli DsbA by 1H-15N HSQC NMR spectroscopy | J Med Chem 63: 6863-6875 (2020) Article DOI: 10.1021/acs.jmedchem.0c00111 BindingDB Entry DOI: 10.7270/Q2X3520R | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Thiol:disulfide interchange protein DsbA (Escherichia coli (strain K12)) | BDBM50576681 (CHEMBL4846499) | PDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | >1.00E+6 | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Binding affinity to 15N-labelled Escherichia coli DsbA measured by 1H-15N HSQC NMR spectroscopy | Citation and Details Article DOI: 10.1016/j.bmc.2021.116315 BindingDB Entry DOI: 10.7270/Q2765K51 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Thiol:disulfide interchange protein DsbA (Escherichia coli (strain K12)) | BDBM50576677 (CHEMBL4877192) | PDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid PDB UniChem | PDB Article PubMed | n/a | n/a | n/a | 1.10E+6 | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Binding affinity to 15N-labelled Escherichia coli DsbA measured by 1H-15N HSQC NMR spectroscopy | Citation and Details Article DOI: 10.1016/j.bmc.2021.116315 BindingDB Entry DOI: 10.7270/Q2765K51 | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
Thiol:disulfide interchange protein DsbA (Escherichia coli (strain K12)) | BDBM50539931 (CHEMBL4646259) | PDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 1.10E+6 | n/a | n/a | n/a | n/a | n/a |
Monash University (Parkville Campus) Curated by ChEMBL | Assay Description Binding affinity to uniformly labeled 15N oxidized Escherichia coli DsbA by 1H-15N HSQC NMR spectroscopy | J Med Chem 63: 6863-6875 (2020) Article DOI: 10.1021/acs.jmedchem.0c00111 BindingDB Entry DOI: 10.7270/Q2X3520R | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Thiol:disulfide interchange protein DsbA (Escherichia coli (strain K12)) | BDBM50576680 (CHEMBL4860222) | PDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid PDB UniChem | PDB Article PubMed | n/a | n/a | n/a | 1.14E+6 | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Binding affinity to 15N-labelled Escherichia coli DsbA measured by 1H-15N HSQC NMR spectroscopy | Citation and Details Article DOI: 10.1016/j.bmc.2021.116315 BindingDB Entry DOI: 10.7270/Q2765K51 | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
Thiol:disulfide interchange protein DsbA (Escherichia coli (strain K12)) | BDBM50576678 (CHEMBL4852788) | PDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 2.30E+6 | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Binding affinity to 15N-labelled Escherichia coli DsbA measured by 1H-15N HSQC NMR spectroscopy | Citation and Details Article DOI: 10.1016/j.bmc.2021.116315 BindingDB Entry DOI: 10.7270/Q2765K51 | |||||||||||
More data for this Ligand-Target Pair |