Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kcal/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Neutral amino acid transporter B(0) (Homo sapiens (Human)) | BDBM464401 (US10793514, Compound 5) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 1.30E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Vanderbilt University US Patent | Assay Description Live-cell amino acid uptake assays using HEK293 cells were carried out in 96-well plates (CulturPlate-96, Perkin Elmer). 96-well plates were coated w... | US Patent US10793514 (2020) BindingDB Entry DOI: 10.7270/Q2TT4V1N | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neutral amino acid transporter B(0) (Homo sapiens (Human)) | BDBM464404 (US10793514, Compound 8) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 1.80E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Vanderbilt University US Patent | Assay Description Live-cell amino acid uptake assays using HEK293 cells were carried out in 96-well plates (CulturPlate-96, Perkin Elmer). 96-well plates were coated w... | US Patent US10793514 (2020) BindingDB Entry DOI: 10.7270/Q2TT4V1N | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neutral amino acid transporter B(0) (Homo sapiens (Human)) | BDBM464426 (US10793514, Compound 19) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 3.30E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Vanderbilt University US Patent | Assay Description Live-cell amino acid uptake assays using HEK293 cells were carried out in 96-well plates (CulturPlate-96, Perkin Elmer). 96-well plates were coated w... | US Patent US10793514 (2020) BindingDB Entry DOI: 10.7270/Q2TT4V1N | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neutral amino acid transporter B(0) (Homo sapiens (Human)) | BDBM50140135 (CHEMBL3753379) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | 3.70E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Vanderbilt University Medical Center Curated by ChEMBL | Assay Description Inhibition of ASCT2 (unknown origin)-mediated glutamine transport | Bioorg Med Chem Lett 26: 1044-7 (2016) Article DOI: 10.1016/j.bmcl.2015.12.031 BindingDB Entry DOI: 10.7270/Q2MC91V1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neutral amino acid transporter B(0) (Homo sapiens (Human)) | BDBM464408 (US10793514, Compound 12) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 5.10E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Vanderbilt University US Patent | Assay Description Live-cell amino acid uptake assays using HEK293 cells were carried out in 96-well plates (CulturPlate-96, Perkin Elmer). 96-well plates were coated w... | US Patent US10793514 (2020) BindingDB Entry DOI: 10.7270/Q2TT4V1N | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neutral amino acid transporter B(0) (Homo sapiens (Human)) | BDBM50140127 (CHEMBL3754498) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 7.20E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Vanderbilt University Medical Center Curated by ChEMBL | Assay Description Inhibition of ASCT2-mediated glutamine transport in human HEK293 cells using [3H]-glutamine after 15 mins by scintillation counting | Bioorg Med Chem Lett 26: 1044-7 (2016) Article DOI: 10.1016/j.bmcl.2015.12.031 BindingDB Entry DOI: 10.7270/Q2MC91V1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neutral amino acid transporter B(0) (Homo sapiens (Human)) | BDBM50140083 (CHEMBL3752210) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | 7.90E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Vanderbilt University Medical Center Curated by ChEMBL | Assay Description Inhibition of ASCT2-mediated glutamine transport in human HEK293 cells using [3H]-glutamine after 15 mins by scintillation counting | Bioorg Med Chem Lett 26: 1044-7 (2016) Article DOI: 10.1016/j.bmcl.2015.12.031 BindingDB Entry DOI: 10.7270/Q2MC91V1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neutral amino acid transporter B(0) (Homo sapiens (Human)) | BDBM50571063 (CHEMBL4867768) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 8.10E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of ASCT2 (unknown origin) | Citation and Details Article DOI: 10.1016/j.bmcl.2021.128078 BindingDB Entry DOI: 10.7270/Q29P35FB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neutral amino acid transporter B(0) (Homo sapiens (Human)) | BDBM464428 (US10793514, Compound 21) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 8.40E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Vanderbilt University US Patent | Assay Description Live-cell amino acid uptake assays using HEK293 cells were carried out in 96-well plates (CulturPlate-96, Perkin Elmer). 96-well plates were coated w... | US Patent US10793514 (2020) BindingDB Entry DOI: 10.7270/Q2TT4V1N | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neutral amino acid transporter B(0) (Homo sapiens (Human)) | BDBM464402 (US10793514, Compound 6) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 8.70E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Vanderbilt University US Patent | Assay Description Live-cell amino acid uptake assays using HEK293 cells were carried out in 96-well plates (CulturPlate-96, Perkin Elmer). 96-well plates were coated w... | US Patent US10793514 (2020) BindingDB Entry DOI: 10.7270/Q2TT4V1N | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neutral amino acid transporter B(0) (Homo sapiens (Human)) | BDBM464424 (US10793514, Compound 17) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | Purchase PC cid PC sid UniChem | US Patent | n/a | n/a | 9.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Vanderbilt University US Patent | Assay Description Live-cell amino acid uptake assays using HEK293 cells were carried out in 96-well plates (CulturPlate-96, Perkin Elmer). 96-well plates were coated w... | US Patent US10793514 (2020) BindingDB Entry DOI: 10.7270/Q2TT4V1N | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neutral amino acid transporter B(0) (Homo sapiens (Human)) | BDBM50140122 (CHEMBL3754053) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 9.60E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
China Pharmaceutical University Curated by ChEMBL | Assay Description Inhibition of ASCT2 (unknown origin) | Eur J Med Chem 163: 215-242 (2019) Article DOI: 10.1016/j.ejmech.2018.11.066 BindingDB Entry DOI: 10.7270/Q2N87F26 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neutral amino acid transporter B(0) (Homo sapiens (Human)) | BDBM50140122 (CHEMBL3754053) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 9.60E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Vanderbilt University Medical Center Curated by ChEMBL | Assay Description Inhibition of ASCT2-mediated glutamine transport in human HEK293 cells using [3H]-glutamine after 15 mins by scintillation counting | Bioorg Med Chem Lett 26: 1044-7 (2016) Article DOI: 10.1016/j.bmcl.2015.12.031 BindingDB Entry DOI: 10.7270/Q2MC91V1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neutral amino acid transporter B(0) (Homo sapiens (Human)) | BDBM464406 (US10793514, Compound 10) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 1.05E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Vanderbilt University US Patent | Assay Description Live-cell amino acid uptake assays using HEK293 cells were carried out in 96-well plates (CulturPlate-96, Perkin Elmer). 96-well plates were coated w... | US Patent US10793514 (2020) BindingDB Entry DOI: 10.7270/Q2TT4V1N | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neutral amino acid transporter B(0) (Homo sapiens (Human)) | BDBM464427 (US10793514, Compound 20) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 1.12E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Vanderbilt University US Patent | Assay Description Live-cell amino acid uptake assays using HEK293 cells were carried out in 96-well plates (CulturPlate-96, Perkin Elmer). 96-well plates were coated w... | US Patent US10793514 (2020) BindingDB Entry DOI: 10.7270/Q2TT4V1N | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neutral amino acid transporter B(0) (Homo sapiens (Human)) | BDBM50140130 (CHEMBL3752483) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.15E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Vanderbilt University Medical Center Curated by ChEMBL | Assay Description Inhibition of ASCT2-mediated glutamine transport in human HEK293 cells using [3H]-glutamine after 15 mins by scintillation counting | Bioorg Med Chem Lett 26: 1044-7 (2016) Article DOI: 10.1016/j.bmcl.2015.12.031 BindingDB Entry DOI: 10.7270/Q2MC91V1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neutral amino acid transporter B(0) (Homo sapiens (Human)) | BDBM50140133 (CHEMBL3753592) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.19E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Vanderbilt University Medical Center Curated by ChEMBL | Assay Description Inhibition of ASCT2-mediated glutamine transport in human HEK293 cells using [3H]-glutamine after 15 mins by scintillation counting | Bioorg Med Chem Lett 26: 1044-7 (2016) Article DOI: 10.1016/j.bmcl.2015.12.031 BindingDB Entry DOI: 10.7270/Q2MC91V1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neutral amino acid transporter B(0) (Homo sapiens (Human)) | BDBM464411 (US10793514, Compound 14) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 1.27E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Vanderbilt University US Patent | Assay Description Live-cell amino acid uptake assays using HEK293 cells were carried out in 96-well plates (CulturPlate-96, Perkin Elmer). 96-well plates were coated w... | US Patent US10793514 (2020) BindingDB Entry DOI: 10.7270/Q2TT4V1N | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neutral amino acid transporter B(0) (Homo sapiens (Human)) | BDBM50140082 (CHEMBL3754059) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.37E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Vanderbilt University Medical Center Curated by ChEMBL | Assay Description Inhibition of ASCT2-mediated glutamine transport in human HEK293 cells using [3H]-glutamine after 15 mins by scintillation counting | Bioorg Med Chem Lett 26: 1044-7 (2016) Article DOI: 10.1016/j.bmcl.2015.12.031 BindingDB Entry DOI: 10.7270/Q2MC91V1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neutral amino acid transporter B(0) (Homo sapiens (Human)) | BDBM464429 (US10793514, Compound 22) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 1.73E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Vanderbilt University US Patent | Assay Description Live-cell amino acid uptake assays using HEK293 cells were carried out in 96-well plates (CulturPlate-96, Perkin Elmer). 96-well plates were coated w... | US Patent US10793514 (2020) BindingDB Entry DOI: 10.7270/Q2TT4V1N | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neutral amino acid transporter B(0) (Homo sapiens (Human)) | BDBM50140084 (CHEMBL3753993) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.75E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Vanderbilt University Medical Center Curated by ChEMBL | Assay Description Inhibition of ASCT2-mediated glutamine transport in human HEK293 cells using [3H]-glutamine after 15 mins by scintillation counting | Bioorg Med Chem Lett 26: 1044-7 (2016) Article DOI: 10.1016/j.bmcl.2015.12.031 BindingDB Entry DOI: 10.7270/Q2MC91V1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neutral amino acid transporter B(0) (Homo sapiens (Human)) | BDBM50140079 (CHEMBL3753404) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.76E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Vanderbilt University Medical Center Curated by ChEMBL | Assay Description Inhibition of ASCT2-mediated glutamine transport in human HEK293 cells using [3H]-glutamine after 15 mins by scintillation counting | Bioorg Med Chem Lett 26: 1044-7 (2016) Article DOI: 10.1016/j.bmcl.2015.12.031 BindingDB Entry DOI: 10.7270/Q2MC91V1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neutral amino acid transporter B(0) (Homo sapiens (Human)) | BDBM464409 (US10793514, Compound 13) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 1.84E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Vanderbilt University US Patent | Assay Description Live-cell amino acid uptake assays using HEK293 cells were carried out in 96-well plates (CulturPlate-96, Perkin Elmer). 96-well plates were coated w... | US Patent US10793514 (2020) BindingDB Entry DOI: 10.7270/Q2TT4V1N | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neutral amino acid transporter B(0) (Homo sapiens (Human)) | BDBM464414 (US10793514, Compound 15) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 2.01E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Vanderbilt University US Patent | Assay Description Live-cell amino acid uptake assays using HEK293 cells were carried out in 96-well plates (CulturPlate-96, Perkin Elmer). 96-well plates were coated w... | US Patent US10793514 (2020) BindingDB Entry DOI: 10.7270/Q2TT4V1N | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neutral amino acid transporter B(0) (Homo sapiens (Human)) | BDBM464430 (US10793514, Compound 23) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 2.25E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Vanderbilt University US Patent | Assay Description Live-cell amino acid uptake assays using HEK293 cells were carried out in 96-well plates (CulturPlate-96, Perkin Elmer). 96-well plates were coated w... | US Patent US10793514 (2020) BindingDB Entry DOI: 10.7270/Q2TT4V1N | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neutral amino acid transporter B(0) (Homo sapiens (Human)) | BDBM464403 (US10793514, Compound 7) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 2.43E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Vanderbilt University US Patent | Assay Description Live-cell amino acid uptake assays using HEK293 cells were carried out in 96-well plates (CulturPlate-96, Perkin Elmer). 96-well plates were coated w... | US Patent US10793514 (2020) BindingDB Entry DOI: 10.7270/Q2TT4V1N | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neutral amino acid transporter B(0) (Homo sapiens (Human)) | BDBM50140123 (CHEMBL3753173) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 2.56E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Vanderbilt University Medical Center Curated by ChEMBL | Assay Description Inhibition of ASCT2-mediated glutamine transport in human HEK293 cells using [3H]-glutamine after 15 mins by scintillation counting | Bioorg Med Chem Lett 26: 1044-7 (2016) Article DOI: 10.1016/j.bmcl.2015.12.031 BindingDB Entry DOI: 10.7270/Q2MC91V1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neutral amino acid transporter B(0) (Homo sapiens (Human)) | BDBM50140132 (CHEMBL3752943) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 2.60E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Vanderbilt University Medical Center Curated by ChEMBL | Assay Description Inhibition of ASCT2-mediated glutamine transport in human HEK293 cells using [3H]-glutamine after 15 mins by scintillation counting | Bioorg Med Chem Lett 26: 1044-7 (2016) Article DOI: 10.1016/j.bmcl.2015.12.031 BindingDB Entry DOI: 10.7270/Q2MC91V1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neutral amino acid transporter B(0) (Homo sapiens (Human)) | BDBM50140136 (CHEMBL3576945) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 3.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Vanderbilt University Medical Center Curated by ChEMBL | Assay Description Inhibition of ASCT2 (unknown origin)-mediated glutamine transport | Bioorg Med Chem Lett 26: 1044-7 (2016) Article DOI: 10.1016/j.bmcl.2015.12.031 BindingDB Entry DOI: 10.7270/Q2MC91V1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neutral amino acid transporter B(0) (Homo sapiens (Human)) | BDBM50140124 (CHEMBL3754369) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 3.37E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Vanderbilt University Medical Center Curated by ChEMBL | Assay Description Inhibition of ASCT2-mediated glutamine transport in human HEK293 cells using [3H]-glutamine after 15 mins by scintillation counting | Bioorg Med Chem Lett 26: 1044-7 (2016) Article DOI: 10.1016/j.bmcl.2015.12.031 BindingDB Entry DOI: 10.7270/Q2MC91V1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neutral amino acid transporter B(0) (Homo sapiens (Human)) | BDBM50140131 (CHEMBL3752249) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 3.38E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Vanderbilt University Medical Center Curated by ChEMBL | Assay Description Inhibition of ASCT2-mediated glutamine transport in human HEK293 cells using [3H]-glutamine after 15 mins by scintillation counting | Bioorg Med Chem Lett 26: 1044-7 (2016) Article DOI: 10.1016/j.bmcl.2015.12.031 BindingDB Entry DOI: 10.7270/Q2MC91V1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neutral amino acid transporter B(0) (Homo sapiens (Human)) | BDBM464405 (US10793514, Compound 9) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 3.63E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Vanderbilt University US Patent | Assay Description Live-cell amino acid uptake assays using HEK293 cells were carried out in 96-well plates (CulturPlate-96, Perkin Elmer). 96-well plates were coated w... | US Patent US10793514 (2020) BindingDB Entry DOI: 10.7270/Q2TT4V1N | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neutral amino acid transporter B(0) (Homo sapiens (Human)) | BDBM50140126 (CHEMBL3752316) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 4.01E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Vanderbilt University Medical Center Curated by ChEMBL | Assay Description Inhibition of ASCT2-mediated glutamine transport in human HEK293 cells using [3H]-glutamine after 15 mins by scintillation counting | Bioorg Med Chem Lett 26: 1044-7 (2016) Article DOI: 10.1016/j.bmcl.2015.12.031 BindingDB Entry DOI: 10.7270/Q2MC91V1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neutral amino acid transporter B(0) (Homo sapiens (Human)) | BDBM464417 (US10793514, Compound 16) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 4.17E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Vanderbilt University US Patent | Assay Description Live-cell amino acid uptake assays using HEK293 cells were carried out in 96-well plates (CulturPlate-96, Perkin Elmer). 96-well plates were coated w... | US Patent US10793514 (2020) BindingDB Entry DOI: 10.7270/Q2TT4V1N | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neutral amino acid transporter B(0) (Homo sapiens (Human)) | BDBM50140081 (CHEMBL3752103) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 4.83E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Vanderbilt University Medical Center Curated by ChEMBL | Assay Description Inhibition of ASCT2-mediated glutamine transport in human HEK293 cells using [3H]-glutamine after 15 mins by scintillation counting | Bioorg Med Chem Lett 26: 1044-7 (2016) Article DOI: 10.1016/j.bmcl.2015.12.031 BindingDB Entry DOI: 10.7270/Q2MC91V1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neutral amino acid transporter B(0) (Homo sapiens (Human)) | BDBM50140125 (CHEMBL3753808) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 5.08E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Vanderbilt University Medical Center Curated by ChEMBL | Assay Description Inhibition of ASCT2-mediated glutamine transport in human HEK293 cells using [3H]-glutamine after 15 mins by scintillation counting | Bioorg Med Chem Lett 26: 1044-7 (2016) Article DOI: 10.1016/j.bmcl.2015.12.031 BindingDB Entry DOI: 10.7270/Q2MC91V1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neutral amino acid transporter B(0) (Homo sapiens (Human)) | BDBM50140134 (CHEMBL3753869) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 5.72E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Vanderbilt University Medical Center Curated by ChEMBL | Assay Description Inhibition of ASCT2-mediated glutamine transport in human HEK293 cells using [3H]-glutamine after 15 mins by scintillation counting | Bioorg Med Chem Lett 26: 1044-7 (2016) Article DOI: 10.1016/j.bmcl.2015.12.031 BindingDB Entry DOI: 10.7270/Q2MC91V1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neutral amino acid transporter B(0) (Homo sapiens (Human)) | BDBM50140128 (CHEMBL3752494) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 5.96E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Vanderbilt University Medical Center Curated by ChEMBL | Assay Description Inhibition of ASCT2-mediated glutamine transport in human HEK293 cells using [3H]-glutamine after 15 mins by scintillation counting | Bioorg Med Chem Lett 26: 1044-7 (2016) Article DOI: 10.1016/j.bmcl.2015.12.031 BindingDB Entry DOI: 10.7270/Q2MC91V1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neutral amino acid transporter B(0) (Homo sapiens (Human)) | BDBM464407 (US10793514, Compound 11) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 6.82E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Vanderbilt University US Patent | Assay Description Live-cell amino acid uptake assays using HEK293 cells were carried out in 96-well plates (CulturPlate-96, Perkin Elmer). 96-well plates were coated w... | US Patent US10793514 (2020) BindingDB Entry DOI: 10.7270/Q2TT4V1N | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neutral amino acid transporter B(0) (Homo sapiens (Human)) | BDBM50140080 (CHEMBL3754415) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | 6.91E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Vanderbilt University Medical Center Curated by ChEMBL | Assay Description Inhibition of ASCT2-mediated glutamine transport in human HEK293 cells using [3H]-glutamine after 15 mins by scintillation counting | Bioorg Med Chem Lett 26: 1044-7 (2016) Article DOI: 10.1016/j.bmcl.2015.12.031 BindingDB Entry DOI: 10.7270/Q2MC91V1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neutral amino acid transporter B(0) (Homo sapiens (Human)) | BDBM464425 (US10793514, Compound 18) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 8.64E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Vanderbilt University US Patent | Assay Description Live-cell amino acid uptake assays using HEK293 cells were carried out in 96-well plates (CulturPlate-96, Perkin Elmer). 96-well plates were coated w... | US Patent US10793514 (2020) BindingDB Entry DOI: 10.7270/Q2TT4V1N | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neutral amino acid transporter B(0) (Homo sapiens (Human)) | BDBM50140129 (CHEMBL3752700) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.42E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Vanderbilt University Medical Center Curated by ChEMBL | Assay Description Inhibition of ASCT2-mediated glutamine transport in human HEK293 cells using [3H]-glutamine after 15 mins by scintillation counting | Bioorg Med Chem Lett 26: 1044-7 (2016) Article DOI: 10.1016/j.bmcl.2015.12.031 BindingDB Entry DOI: 10.7270/Q2MC91V1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neutral amino acid transporter B(0) (Homo sapiens (Human)) | BDBM50088534 (CHEMBL3576929 | US10189805, Compound 5) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 3.12E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Vanderbilt University US Patent | Assay Description The glutamine uptake assays in HEK293 cells were carried out in 96 well plates (CulturPlate-96, Perkin Elmer). Cells were plated at a density of 35,0... | US Patent US10189805 (2019) BindingDB Entry DOI: 10.7270/Q2GX4DN8 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neutral amino acid transporter B(0) (Homo sapiens (Human)) | BDBM50088534 (CHEMBL3576929 | US10189805, Compound 5) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 3.12E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Vanderbilt University Medical Center Curated by ChEMBL | Assay Description Inhibition of ASCT2 (unknown origin)-mediated glutamine transport | Bioorg Med Chem Lett 26: 1044-7 (2016) Article DOI: 10.1016/j.bmcl.2015.12.031 BindingDB Entry DOI: 10.7270/Q2MC91V1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neutral amino acid transporter B(0) (Homo sapiens (Human)) | BDBM50088534 (CHEMBL3576929 | US10189805, Compound 5) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 3.12E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Vanderbilt University Institute of Imaging Science (VUIIS) Curated by ChEMBL | Assay Description Inhibition of ASCT2-mediated [3H]glutamine uptake in HEK293 cells after 15 mins by Live-cell glutamine uptake assay | Bioorg Med Chem Lett 25: 113-6 (2014) Article DOI: 10.1016/j.bmcl.2014.10.098 BindingDB Entry DOI: 10.7270/Q2CZ38X7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neutral amino acid transporter B(0) (Homo sapiens (Human)) | BDBM50088535 (CHEMBL3576928 | US10189805, Compound 4) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 4.36E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Vanderbilt University US Patent | Assay Description The glutamine uptake assays in HEK293 cells were carried out in 96 well plates (CulturPlate-96, Perkin Elmer). Cells were plated at a density of 35,0... | US Patent US10189805 (2019) BindingDB Entry DOI: 10.7270/Q2GX4DN8 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neutral amino acid transporter B(0) (Homo sapiens (Human)) | BDBM50088535 (CHEMBL3576928 | US10189805, Compound 4) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 4.36E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Vanderbilt University Institute of Imaging Science (VUIIS) Curated by ChEMBL | Assay Description Inhibition of ASCT2-mediated [3H]glutamine uptake in HEK293 cells after 15 mins by Live-cell glutamine uptake assay | Bioorg Med Chem Lett 25: 113-6 (2014) Article DOI: 10.1016/j.bmcl.2014.10.098 BindingDB Entry DOI: 10.7270/Q2CZ38X7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neutral amino acid transporter B(0) (Homo sapiens (Human)) | BDBM50088536 (CHEMBL3576927 | US10189805, Compound 3) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 6.64E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Vanderbilt University Institute of Imaging Science (VUIIS) Curated by ChEMBL | Assay Description Inhibition of ASCT2-mediated [3H]glutamine uptake in HEK293 cells after 15 mins by Live-cell glutamine uptake assay | Bioorg Med Chem Lett 25: 113-6 (2014) Article DOI: 10.1016/j.bmcl.2014.10.098 BindingDB Entry DOI: 10.7270/Q2CZ38X7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neutral amino acid transporter B(0) (Homo sapiens (Human)) | BDBM50088536 (CHEMBL3576927 | US10189805, Compound 3) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 6.64E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Vanderbilt University US Patent | Assay Description The glutamine uptake assays in HEK293 cells were carried out in 96 well plates (CulturPlate-96, Perkin Elmer). Cells were plated at a density of 35,0... | US Patent US10189805 (2019) BindingDB Entry DOI: 10.7270/Q2GX4DN8 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neutral amino acid transporter B(0) (Homo sapiens (Human)) | BDBM50088531 (CHEMBL3576943 | US10189805, Compound 19) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | US Patent | n/a | n/a | 6.77E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Vanderbilt University US Patent | Assay Description The glutamine uptake assays in HEK293 cells were carried out in 96 well plates (CulturPlate-96, Perkin Elmer). Cells were plated at a density of 35,0... | US Patent US10189805 (2019) BindingDB Entry DOI: 10.7270/Q2GX4DN8 | |||||||||||
More data for this Ligand-Target Pair |
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