BindingDB PrimarySearch

Found 1831 hits of ic50 data for polymerid = 5468
Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kcal/mole	IC50 nM	Kd nM	EC50/IC50 nM	k_off s^-1	k_on M^-1s^-1	pH	Temp °C
Dipeptidyl peptidase 2 (Homo sapiens (Human))	BDBM142088 (US11096924, DASH-inhibitors 2243 \| US11559537, Com...) Show SMILES C[C@H](N)C(=S)N1CCC[C@H]1B(O)O \|r\| Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem Similars	US Patent	n/a	n/a	0.200	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description This assay is described in Bachovchin et al. Nature Chemical Biology 10, 656-663 (2014). Briefly, purified enzymes are coupled to Luminex microsphere...				Citation and Details BindingDB Entry DOI: 10.7270/Q28W3J7Z
TBA					More data for this Ligand-Target Pair
Dipeptidyl peptidase 2 (Homo sapiens (Human))	BDBM50050516 (Boronic acid derivative \| CHEMBL63726 \| US11096924...) Show SMILES NCCCC[C@H](N)C(=O)N1CCC[C@H]1B(O)O Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Patents Similars	US Patent	n/a	n/a	0.200	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description This assay is described in Bachovchin et al. Nature Chemical Biology 10, 656-663 (2014). Briefly, purified enzymes are coupled to Luminex microsphere...				Citation and Details BindingDB Entry DOI: 10.7270/Q28W3J7Z
TBA					More data for this Ligand-Target Pair
Dipeptidyl peptidase 2 (Homo sapiens (Human))	BDBM50146987 ((S)-2-Amino-4-[(4-chloro-benzyl)-methyl-amino]-1-p...) Show SMILES Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	0.220	n/a	n/a	n/a	n/a	n/a	n/a
University of Antwerp Curated by ChEMBL					Assay Description Inhibition of human Dipeptidyl-peptidase II (DPP II)				J Med Chem 47: 2906-16 (2004) Article DOI: 10.1021/jm031122f BindingDB Entry DOI: 10.7270/Q2TH8M4H
University of Antwerp Curated by ChEMBL					More data for this Ligand-Target Pair
Dipeptidyl peptidase 2 (Homo sapiens (Human))	BDBM50146972 ((S)-4-(4-chlorobenzylamino)-2-amino-1-(piperidin-1...) Show SMILES Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	Purchase CHEMBL MCE PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	0.220	n/a	n/a	n/a	n/a	n/a	n/a
Laboratory of Medicinal Chemistry University of Antwerp Curated by ChEMBL					Assay Description Inhibition of DPP2				Bioorg Med Chem Lett 16: 4777-9 (2006) Article DOI: 10.1016/j.bmcl.2006.06.082 BindingDB Entry DOI: 10.7270/Q2GM86XS
					More data for this Ligand-Target Pair
Dipeptidyl peptidase 2 (Homo sapiens (Human))	BDBM50146971 (2-(S)-Amino-4-(2-chloro-benzylamino)-1-piperidin-1...) Show SMILES N[C@@H](CCNCc1ccccc1Cl)C(=O)N1CCCCC1 Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	0.230	n/a	n/a	n/a	n/a	n/a	n/a
University of Antwerp Curated by ChEMBL					Assay Description Inhibition of human Dipeptidyl-peptidase II (DPP II)				J Med Chem 47: 2906-16 (2004) Article DOI: 10.1021/jm031122f BindingDB Entry DOI: 10.7270/Q2TH8M4H
University of Antwerp Curated by ChEMBL					More data for this Ligand-Target Pair
Dipeptidyl peptidase 2 (Homo sapiens (Human))	BDBM50146973 (2-(S)-Amino-4-(2-benzyloxy-benzylamino)-1-piperidi...) Show SMILES Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	0.390	n/a	n/a	n/a	n/a	n/a	n/a
University of Antwerp Curated by ChEMBL					Assay Description Inhibition of human Dipeptidyl-peptidase II (DPP II)				J Med Chem 47: 2906-16 (2004) Article DOI: 10.1021/jm031122f BindingDB Entry DOI: 10.7270/Q2TH8M4H
University of Antwerp Curated by ChEMBL					More data for this Ligand-Target Pair
Dipeptidyl peptidase 2 (Homo sapiens (Human))	BDBM50146974 ((S)-2-Amino-4-(4-chloro-benzylamino)-1-(4-fluoro-p...) Show SMILES Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	0.390	n/a	n/a	n/a	n/a	n/a	n/a
University of Antwerp Curated by ChEMBL					Assay Description Inhibition of human Dipeptidyl-peptidase II (DPP II)				J Med Chem 47: 2906-16 (2004) Article DOI: 10.1021/jm031122f BindingDB Entry DOI: 10.7270/Q2TH8M4H
University of Antwerp Curated by ChEMBL					More data for this Ligand-Target Pair
Dipeptidyl peptidase 2 (Homo sapiens (Human))	BDBM50146952 (2-(S)-Amino-4-(4-benzyloxy-benzylamino)-1-piperidi...) Show SMILES Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	0.410	n/a	n/a	n/a	n/a	n/a	n/a
University of Antwerp Curated by ChEMBL					Assay Description Inhibition of human Dipeptidyl-peptidase II (DPP II)				J Med Chem 47: 2906-16 (2004) Article DOI: 10.1021/jm031122f BindingDB Entry DOI: 10.7270/Q2TH8M4H
University of Antwerp Curated by ChEMBL					More data for this Ligand-Target Pair
Dipeptidyl peptidase 2 (Homo sapiens (Human))	BDBM50196928 ((R)-1-((S)-2,4-diaminobutanamido)pentylboronic aci...) Show SMILES CCCC[C@H](NC(=O)[C@@H](N)CCN)B(O)O Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	0.480	n/a	n/a	n/a	n/a	n/a	n/a
Tufts University School of Medicine Curated by ChEMBL					Assay Description Inhibition of human DPP2				Bioorg Med Chem Lett 17: 507-10 (2007) Article DOI: 10.1016/j.bmcl.2006.10.012 BindingDB Entry DOI: 10.7270/Q2T43SQH
Tufts University School of Medicine Curated by ChEMBL					More data for this Ligand-Target Pair
Dipeptidyl peptidase 2 (Homo sapiens (Human))	BDBM50146972 ((S)-4-(4-chlorobenzylamino)-2-amino-1-(piperidin-1...) Show SMILES Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	Purchase CHEMBL MCE PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	0.480	n/a	n/a	n/a	n/a	n/a	n/a
University of Antwerp (UA) Curated by ChEMBL					Assay Description Inhibition of DPP2				J Med Chem 54: 5737-46 (2011) Article DOI: 10.1021/jm200383j BindingDB Entry DOI: 10.7270/Q2G73F37
University of Antwerp (UA) Curated by ChEMBL					More data for this Ligand-Target Pair
Dipeptidyl peptidase 2 (Homo sapiens (Human))	BDBM50146972 ((S)-4-(4-chlorobenzylamino)-2-amino-1-(piperidin-1...) Show SMILES Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	Purchase CHEMBL MCE PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	0.480	n/a	n/a	n/a	n/a	n/a	n/a
University of Antwerp Curated by ChEMBL					Assay Description Inhibition of human Dipeptidyl-peptidase II (DPP II)				J Med Chem 47: 2906-16 (2004) Article DOI: 10.1021/jm031122f BindingDB Entry DOI: 10.7270/Q2TH8M4H
University of Antwerp Curated by ChEMBL					More data for this Ligand-Target Pair
Dipeptidyl peptidase 2 (Homo sapiens (Human))	BDBM50171546 ((S)-2,4-Diamino-N-((R)-1-boron-dihydroxide-pentyl)...) Show SMILES CCCC[C@@H](NC(=O)[C@@H](N)CCN)B(O)O Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	0.480	n/a	n/a	n/a	n/a	n/a	n/a
ActivX Biosciences Curated by ChEMBL					Assay Description Inhibitory concentration against human dipeptidylpeptidase 7				Bioorg Med Chem Lett 15: 4256-60 (2005) Article DOI: 10.1016/j.bmcl.2005.06.076 BindingDB Entry DOI: 10.7270/Q2RR1XSW
ActivX Biosciences Curated by ChEMBL					More data for this Ligand-Target Pair
Dipeptidyl peptidase 2 (Homo sapiens (Human))	BDBM50146972 ((S)-4-(4-chlorobenzylamino)-2-amino-1-(piperidin-1...) Show SMILES Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	Purchase CHEMBL MCE PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	<0.5	n/a	n/a	n/a	n/a	n/a	n/a
University of Warwick Curated by ChEMBL					Assay Description Inhibition of DPP2 (unknown origin)				Eur J Med Chem 139: 482-491 (2017) Article DOI: 10.1016/j.ejmech.2017.08.024 BindingDB Entry DOI: 10.7270/Q25B050P
University of Warwick Curated by ChEMBL					More data for this Ligand-Target Pair
Dipeptidyl peptidase 2 (Homo sapiens (Human))	BDBM50146956 ((S)-2-Amino-4-(4-chloro-benzylamino)-1-(4-methyl-p...) Show SMILES Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	0.550	n/a	n/a	n/a	n/a	n/a	n/a
University of Antwerp Curated by ChEMBL					Assay Description Inhibition of human Dipeptidyl-peptidase II (DPP II)				J Med Chem 47: 2906-16 (2004) Article DOI: 10.1021/jm031122f BindingDB Entry DOI: 10.7270/Q2TH8M4H
University of Antwerp Curated by ChEMBL					More data for this Ligand-Target Pair
Dipeptidyl peptidase 2 (Homo sapiens (Human))	BDBM50146967 ((S)-2-Amino-4-dibenzylamino-1-piperidin-1-yl-butan...) Show SMILES Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	0.600	n/a	n/a	n/a	n/a	n/a	n/a
University of Antwerp Curated by ChEMBL					Assay Description Inhibition of human Dipeptidyl-peptidase II (DPP II)				J Med Chem 47: 2906-16 (2004) Article DOI: 10.1021/jm031122f BindingDB Entry DOI: 10.7270/Q2TH8M4H
University of Antwerp Curated by ChEMBL					More data for this Ligand-Target Pair
Dipeptidyl peptidase 2 (Homo sapiens (Human))	BDBM50191168 ((2S,4S)-4-(4-chlorobenzylamino)-2-amino-1-(piperid...) Show SMILES Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	0.620	n/a	n/a	n/a	n/a	n/a	n/a
Laboratory of Medicinal Chemistry University of Antwerp Curated by ChEMBL					Assay Description Inhibition of DPP2				Bioorg Med Chem Lett 16: 4777-9 (2006) Article DOI: 10.1016/j.bmcl.2006.06.082 BindingDB Entry DOI: 10.7270/Q2GM86XS
					More data for this Ligand-Target Pair
Dipeptidyl peptidase 2 (Homo sapiens (Human))	BDBM50146985 ((S)-2-Amino-4-(4-chloro-benzylamino)-1-(3-fluoro-p...) Show SMILES Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	0.620	n/a	n/a	n/a	n/a	n/a	n/a
University of Antwerp Curated by ChEMBL					Assay Description Inhibition of human Dipeptidyl-peptidase II (DPP II)				J Med Chem 47: 2906-16 (2004) Article DOI: 10.1021/jm031122f BindingDB Entry DOI: 10.7270/Q2TH8M4H
University of Antwerp Curated by ChEMBL					More data for this Ligand-Target Pair
Dipeptidyl peptidase 2 (Homo sapiens (Human))	BDBM50146977 (2-(S)-Amino-4-(4-methoxy-benzylamino)-1-piperidin-...) Show SMILES COc1ccc(CNCC[C@H](N)C(=O)N2CCCCC2)cc1 Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	0.660	n/a	n/a	n/a	n/a	n/a	n/a
University of Antwerp Curated by ChEMBL					Assay Description Inhibition of human Dipeptidyl-peptidase II (DPP II)				J Med Chem 47: 2906-16 (2004) Article DOI: 10.1021/jm031122f BindingDB Entry DOI: 10.7270/Q2TH8M4H
University of Antwerp Curated by ChEMBL					More data for this Ligand-Target Pair
Dipeptidyl peptidase 2 (Homo sapiens (Human))	BDBM50171555 ((S)-2,4-Diamino-1-(2-boron-dihydroxide-pyrrolidin-...) Show SMILES NCC[C@H](N)C(=O)N1CCC[C@@H]1B(O)O Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	0.720	n/a	n/a	n/a	n/a	n/a	n/a
ActivX Biosciences Curated by ChEMBL					Assay Description Inhibitory concentration against human dipeptidylpeptidase 7				Bioorg Med Chem Lett 15: 4256-60 (2005) Article DOI: 10.1016/j.bmcl.2005.06.076 BindingDB Entry DOI: 10.7270/Q2RR1XSW
ActivX Biosciences Curated by ChEMBL					More data for this Ligand-Target Pair
Dipeptidyl peptidase 2 (Homo sapiens (Human))	BDBM50146964 (2-(S)-Amino-1-piperidin-1-yl-4-[(pyridin-4-ylmethy...) Show SMILES N[C@@H](CCNCc1ccncc1)C(=O)N1CCCCC1 Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem	Article PubMed	n/a	n/a	0.75	n/a	n/a	n/a	n/a	n/a	n/a
University of Antwerp Curated by ChEMBL					Assay Description Inhibition of human Dipeptidyl-peptidase II (DPP II)				J Med Chem 47: 2906-16 (2004) Article DOI: 10.1021/jm031122f BindingDB Entry DOI: 10.7270/Q2TH8M4H
University of Antwerp Curated by ChEMBL					More data for this Ligand-Target Pair
Dipeptidyl peptidase 2 (Homo sapiens (Human))	BDBM50146957 (2-(S)-Amino-1-piperidin-1-yl-4-[(thiophen-2-ylmeth...) Show SMILES N[C@@H](CCNCc1cccs1)C(=O)N1CCCCC1 Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem	Article PubMed	n/a	n/a	0.800	n/a	n/a	n/a	n/a	n/a	n/a
University of Antwerp Curated by ChEMBL					Assay Description Inhibition of human Dipeptidyl-peptidase II (DPP II)				J Med Chem 47: 2906-16 (2004) Article DOI: 10.1021/jm031122f BindingDB Entry DOI: 10.7270/Q2TH8M4H
University of Antwerp Curated by ChEMBL					More data for this Ligand-Target Pair
Dipeptidyl peptidase 2 (Homo sapiens (Human))	BDBM50050515 (Boronic acid derivative \| CHEMBL63652 \| US11096924...) Show SMILES N[C@@H](Cc1ccccc1)C(=O)N1CCC[C@H]1B(O)O Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	US Patent	n/a	n/a	0.800	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description This assay is described in Bachovchin et al. Nature Chemical Biology 10, 656-663 (2014). Briefly, purified enzymes are coupled to Luminex microsphere...				Citation and Details BindingDB Entry DOI: 10.7270/Q28W3J7Z
TBA					More data for this Ligand-Target Pair
Dipeptidyl peptidase 2 (Homo sapiens (Human))	BDBM50196929 ((S)-2,4-diamino-1-((3aR,6aR)-hexahydrocyclopenta[b...) Show SMILES NCC[C@H](N)C(=O)N1CC[C@H]2CCC[C@@H]12 Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	0.880	n/a	n/a	n/a	n/a	n/a	n/a
Tufts University School of Medicine Curated by ChEMBL					Assay Description Inhibition of human DPP2				Bioorg Med Chem Lett 17: 507-10 (2007) Article DOI: 10.1016/j.bmcl.2006.10.012 BindingDB Entry DOI: 10.7270/Q2T43SQH
Tufts University School of Medicine Curated by ChEMBL					More data for this Ligand-Target Pair
Dipeptidyl peptidase 2 (Homo sapiens (Human))	BDBM50146954 (2-(S)-Amino-4-phenethylamino-1-piperidin-1-yl-buta...) Show SMILES N[C@@H](CCNCCc1ccccc1)C(=O)N1CCCCC1 Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem	Article PubMed	n/a	n/a	0.900	n/a	n/a	n/a	n/a	n/a	n/a
University of Antwerp Curated by ChEMBL					Assay Description Inhibition of human Dipeptidyl-peptidase II (DPP II)				J Med Chem 47: 2906-16 (2004) Article DOI: 10.1021/jm031122f BindingDB Entry DOI: 10.7270/Q2TH8M4H
University of Antwerp Curated by ChEMBL					More data for this Ligand-Target Pair
Dipeptidyl peptidase 2 (Homo sapiens (Human))	BDBM50050525 ((R)-1-((S)-2-aminopropanoyl)pyrrolidin-2-ylboronic...) Show SMILES C[C@H](N)C(=O)N1CCC[C@H]1B(O)O \|r\| Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Patents Similars	US Patent	n/a	n/a	1	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description This assay is described in Bachovchin et al. Nature Chemical Biology 10, 656-663 (2014). Briefly, purified enzymes are coupled to Luminex microsphere...				Citation and Details BindingDB Entry DOI: 10.7270/Q28W3J7Z
TBA					More data for this Ligand-Target Pair
Dipeptidyl peptidase 2 (Homo sapiens (Human))	BDBM50171648 (CHEMBL372180 \| N-alkyl Gly-boro-Pro derivative) Show SMILES Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	1	n/a	n/a	n/a	n/a	n/a	n/a
ActivX Biosciences, Inc. Curated by ChEMBL					Assay Description Inhibitory activity against human DPP7 using Ala-Pro-AMC in fluorometric assay				Bioorg Med Chem Lett 15: 4239-42 (2005) Article DOI: 10.1016/j.bmcl.2005.06.075 BindingDB Entry DOI: 10.7270/Q2CJ8D2F
ActivX Biosciences, Inc. Curated by ChEMBL					More data for this Ligand-Target Pair
Dipeptidyl peptidase 2 (Homo sapiens (Human))	BDBM50050528 (Boronic acid derivative \| CHEMBL63698 \| US11096924...) Show SMILES CC(C)C[C@H](N)C(=O)N1CCC[C@H]1B(O)O Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	US Patent	n/a	n/a	1	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description This assay is described in Bachovchin et al. Nature Chemical Biology 10, 656-663 (2014). Briefly, purified enzymes are coupled to Luminex microsphere...				Citation and Details BindingDB Entry DOI: 10.7270/Q28W3J7Z
TBA					More data for this Ligand-Target Pair
Dipeptidyl peptidase 2 (Homo sapiens (Human))	BDBM50146991 (2-(S)-Amino-4-[(naphthalen-2-ylmethyl)-amino]-1-pi...) Show SMILES Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	1.10	n/a	n/a	n/a	n/a	n/a	n/a
University of Antwerp Curated by ChEMBL					Assay Description Inhibition of human Dipeptidyl-peptidase II (DPP II)				J Med Chem 47: 2906-16 (2004) Article DOI: 10.1021/jm031122f BindingDB Entry DOI: 10.7270/Q2TH8M4H
University of Antwerp Curated by ChEMBL					More data for this Ligand-Target Pair
Dipeptidyl peptidase 2 (Homo sapiens (Human))	BDBM50146968 ((S)-2-Amino-4-(4-chloro-benzylamino)-1-(3,6-dihydr...) Show SMILES Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem	Article PubMed	n/a	n/a	1.10	n/a	n/a	n/a	n/a	n/a	n/a
University of Antwerp Curated by ChEMBL					Assay Description Inhibition of human Dipeptidyl-peptidase II (DPP II)				J Med Chem 47: 2906-16 (2004) Article DOI: 10.1021/jm031122f BindingDB Entry DOI: 10.7270/Q2TH8M4H
University of Antwerp Curated by ChEMBL					More data for this Ligand-Target Pair
Dipeptidyl peptidase 2 (Homo sapiens (Human))	BDBM50146955 (2-(S)-Amino-4-(cyclohexylmethyl-amino)-1-piperidin...) Show SMILES N[C@@H](CCNCC1CCCCC1)C(=O)N1CCCCC1 Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Patents Similars	Article PubMed	n/a	n/a	1.10	n/a	n/a	n/a	n/a	n/a	n/a
University of Antwerp Curated by ChEMBL					Assay Description Inhibition of human Dipeptidyl-peptidase II (DPP II)				J Med Chem 47: 2906-16 (2004) Article DOI: 10.1021/jm031122f BindingDB Entry DOI: 10.7270/Q2TH8M4H
University of Antwerp Curated by ChEMBL					More data for this Ligand-Target Pair
Dipeptidyl peptidase 2 (Homo sapiens (Human))	BDBM50146950 ((S)-2-Amino-4-(4-chloro-benzylamino)-1-(3-methyl-p...) Show SMILES Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	1.13	n/a	n/a	n/a	n/a	n/a	n/a
University of Antwerp Curated by ChEMBL					Assay Description Inhibition of human Dipeptidyl-peptidase II (DPP II)				J Med Chem 47: 2906-16 (2004) Article DOI: 10.1021/jm031122f BindingDB Entry DOI: 10.7270/Q2TH8M4H
University of Antwerp Curated by ChEMBL					More data for this Ligand-Target Pair
Dipeptidyl peptidase 2 (Homo sapiens (Human))	BDBM50146960 (2-(S)-Amino-4-[(naphthalen-1-ylmethyl)-amino]-1-pi...) Show SMILES Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	1.31	n/a	n/a	n/a	n/a	n/a	n/a
University of Antwerp Curated by ChEMBL					Assay Description Inhibition of human Dipeptidyl-peptidase II (DPP II)				J Med Chem 47: 2906-16 (2004) Article DOI: 10.1021/jm031122f BindingDB Entry DOI: 10.7270/Q2TH8M4H
University of Antwerp Curated by ChEMBL					More data for this Ligand-Target Pair
Dipeptidyl peptidase 2 (Homo sapiens (Human))	BDBM50146961 (2-(S)-Amino-4-(3-chloro-benzylamino)-1-piperidin-1...) Show SMILES N[C@@H](CCNCc1cccc(Cl)c1)C(=O)N1CCCCC1 Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	1.34	n/a	n/a	n/a	n/a	n/a	n/a
University of Antwerp Curated by ChEMBL					Assay Description Inhibition of human Dipeptidyl-peptidase II (DPP II)				J Med Chem 47: 2906-16 (2004) Article DOI: 10.1021/jm031122f BindingDB Entry DOI: 10.7270/Q2TH8M4H
University of Antwerp Curated by ChEMBL					More data for this Ligand-Target Pair
Dipeptidyl peptidase 2 (Homo sapiens (Human))	BDBM50050525 ((R)-1-((S)-2-aminopropanoyl)pyrrolidin-2-ylboronic...) Show SMILES C[C@H](N)C(=O)N1CCC[C@H]1B(O)O \|r\| Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Patents Similars	US Patent	n/a	n/a	1.40	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description This assay is described in Bachovchin et al. Nature Chemical Biology 10, 656-663 (2014). Briefly, purified enzymes are coupled to Luminex microsphere...				Citation and Details BindingDB Entry DOI: 10.7270/Q28W3J7Z
TBA					More data for this Ligand-Target Pair
Dipeptidyl peptidase 2 (Homo sapiens (Human))	BDBM50146988 (CHEMBL440325 \| N-((S)-3-Amino-4-oxo-4-piperidin-1-...) Show SMILES CC(=O)NCC[C@H](N)C(=O)N1CCCCC1 Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	1.5	n/a	n/a	n/a	n/a	n/a	n/a
University of Antwerp Curated by ChEMBL					Assay Description Inhibition of human Dipeptidyl-peptidase II (DPP II)				J Med Chem 47: 2906-16 (2004) Article DOI: 10.1021/jm031122f BindingDB Entry DOI: 10.7270/Q2TH8M4H
University of Antwerp Curated by ChEMBL					More data for this Ligand-Target Pair
Dipeptidyl peptidase 2 (Homo sapiens (Human))	BDBM50146978 ((S)-2-Amino-4-phenylamino-1-piperidin-1-yl-butan-1...) Show SMILES N[C@@H](CCNc1ccccc1)C(=O)N1CCCCC1 Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem	Article PubMed	n/a	n/a	1.5	n/a	n/a	n/a	n/a	n/a	n/a
University of Antwerp Curated by ChEMBL					Assay Description Inhibition of human Dipeptidyl-peptidase II (DPP II)				J Med Chem 47: 2906-16 (2004) Article DOI: 10.1021/jm031122f BindingDB Entry DOI: 10.7270/Q2TH8M4H
University of Antwerp Curated by ChEMBL					More data for this Ligand-Target Pair
Dipeptidyl peptidase 2 (Homo sapiens (Human))	BDBM50146953 (2-(S)-Amino-4-(3-methoxy-benzylamino)-1-piperidin-...) Show SMILES COc1cccc(CNCC[C@H](N)C(=O)N2CCCCC2)c1 Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	1.77	n/a	n/a	n/a	n/a	n/a	n/a
University of Antwerp Curated by ChEMBL					Assay Description Inhibition of human Dipeptidyl-peptidase II (DPP II)				J Med Chem 47: 2906-16 (2004) Article DOI: 10.1021/jm031122f BindingDB Entry DOI: 10.7270/Q2TH8M4H
University of Antwerp Curated by ChEMBL					More data for this Ligand-Target Pair
Dipeptidyl peptidase 2 (Homo sapiens (Human))	BDBM50146962 (CHEMBL101401 \| N-((S)-3-Amino-4-oxo-4-piperidin-1-...) Show SMILES N[C@@H](CCNC(N)=N)C(=O)N1CCCCC1 Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem	Article PubMed	n/a	n/a	1.80	n/a	n/a	n/a	n/a	n/a	n/a
University of Antwerp Curated by ChEMBL					Assay Description Inhibition of human Dipeptidyl-peptidase II (DPP II)				J Med Chem 47: 2906-16 (2004) Article DOI: 10.1021/jm031122f BindingDB Entry DOI: 10.7270/Q2TH8M4H
University of Antwerp Curated by ChEMBL					More data for this Ligand-Target Pair
Dipeptidyl peptidase 2 (Homo sapiens (Human))	BDBM50171649 (CHEMBL196933 \| N-alkyl Gly-boro-Pro derivative) Show SMILES OB(O)[C@@H]1CCCN1C(=O)CNC1CCCCCC1 Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	1.80	n/a	n/a	n/a	n/a	n/a	n/a
ActivX Biosciences, Inc. Curated by ChEMBL					Assay Description Inhibitory activity against human DPP7 using Ala-Pro-AMC in fluorometric assay				Bioorg Med Chem Lett 15: 4239-42 (2005) Article DOI: 10.1016/j.bmcl.2005.06.075 BindingDB Entry DOI: 10.7270/Q2CJ8D2F
ActivX Biosciences, Inc. Curated by ChEMBL					More data for this Ligand-Target Pair
Dipeptidyl peptidase 2 (Homo sapiens (Human))	BDBM50146965 (2-(S)-Amino-4-(3-phenyl-propylamino)-1-piperidin-1...) Show SMILES N[C@@H](CCNCCCc1ccccc1)C(=O)N1CCCCC1 Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem	Article PubMed	n/a	n/a	1.91	n/a	n/a	n/a	n/a	n/a	n/a
University of Antwerp Curated by ChEMBL					Assay Description Inhibition of human Dipeptidyl-peptidase II (DPP II)				J Med Chem 47: 2906-16 (2004) Article DOI: 10.1021/jm031122f BindingDB Entry DOI: 10.7270/Q2TH8M4H
University of Antwerp Curated by ChEMBL					More data for this Ligand-Target Pair
Dipeptidyl peptidase 2 (Homo sapiens (Human))	BDBM50171548 ((S)-2-(S)-Amino-1-(2-boron-dihydroxide-pyrrolidin-...) Show SMILES CCCC[C@H](N)C(=O)N1CCC[C@@H]1B(O)O Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	2	n/a	n/a	n/a	n/a	n/a	n/a
ActivX Biosciences Curated by ChEMBL					Assay Description Inhibitory concentration against human dipeptidylpeptidase 7				Bioorg Med Chem Lett 15: 4256-60 (2005) Article DOI: 10.1016/j.bmcl.2005.06.076 BindingDB Entry DOI: 10.7270/Q2RR1XSW
ActivX Biosciences Curated by ChEMBL					More data for this Ligand-Target Pair
Dipeptidyl peptidase 2 (Homo sapiens (Human))	BDBM50146975 (2-(S)-Amino-4-benzylamino-1-piperidin-1-yl-butan-1...) Show SMILES N[C@@H](CCNCc1ccccc1)C(=O)N1CCCCC1 Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	2.03	n/a	n/a	n/a	n/a	n/a	n/a
University of Antwerp Curated by ChEMBL					Assay Description Inhibition of human Dipeptidyl-peptidase II (DPP II)				J Med Chem 47: 2906-16 (2004) Article DOI: 10.1021/jm031122f BindingDB Entry DOI: 10.7270/Q2TH8M4H
University of Antwerp Curated by ChEMBL					More data for this Ligand-Target Pair
Dipeptidyl peptidase 2 (Homo sapiens (Human))	BDBM142093 (US11096924, DASH-inhibitors 1797 \| US11559537, Com...) Show SMILES Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem Similars	US Patent	n/a	n/a	2.10	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description This assay is described in Bachovchin et al. Nature Chemical Biology 10, 656-663 (2014). Briefly, purified enzymes are coupled to Luminex microsphere...				Citation and Details BindingDB Entry DOI: 10.7270/Q28W3J7Z
TBA					More data for this Ligand-Target Pair
Dipeptidyl peptidase 2 (Homo sapiens (Human))	BDBM50171645 (2-Cyclodecylamino-1-pyrrolidin-1-yl--2-borandihydr...) Show SMILES OB(O)[C@@H]1CCCN1C(=O)CNC1CCCCCCCCC1 Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	2.20	n/a	n/a	n/a	n/a	n/a	n/a
ActivX Biosciences, Inc. Curated by ChEMBL					Assay Description Inhibitory activity against human DPP7 using Ala-Pro-AMC in fluorometric assay				Bioorg Med Chem Lett 15: 4239-42 (2005) Article DOI: 10.1016/j.bmcl.2005.06.075 BindingDB Entry DOI: 10.7270/Q2CJ8D2F
ActivX Biosciences, Inc. Curated by ChEMBL					More data for this Ligand-Target Pair
Dipeptidyl peptidase 2 (Homo sapiens (Human))	BDBM50146979 ((S)-2-Amino-4-(4-chloro-benzylamino)-1-(2-methyl-p...) Show SMILES CC1CCCCN1C(=O)[C@@H](N)CCNCc1ccc(Cl)cc1 Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	2.30	n/a	n/a	n/a	n/a	n/a	n/a
University of Antwerp Curated by ChEMBL					Assay Description Inhibition of human Dipeptidyl-peptidase II (DPP II)				J Med Chem 47: 2906-16 (2004) Article DOI: 10.1021/jm031122f BindingDB Entry DOI: 10.7270/Q2TH8M4H
University of Antwerp Curated by ChEMBL					More data for this Ligand-Target Pair
Dipeptidyl peptidase 2 (Homo sapiens (Human))	BDBM50146969 (3-[((S)-3-Amino-4-oxo-4-piperidin-1-yl-butylamino)...) Show SMILES N[C@@H](CCNCc1cccc(c1)C#N)C(=O)N1CCCCC1 Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	2.70	n/a	n/a	n/a	n/a	n/a	n/a
University of Antwerp Curated by ChEMBL					Assay Description Inhibition of human Dipeptidyl-peptidase II (DPP II)				J Med Chem 47: 2906-16 (2004) Article DOI: 10.1021/jm031122f BindingDB Entry DOI: 10.7270/Q2TH8M4H
University of Antwerp Curated by ChEMBL					More data for this Ligand-Target Pair
Dipeptidyl peptidase 2 (Homo sapiens (Human))	BDBM50221977 ((2S,3S)-2-amino-3-(4'-fluoro-biphenyl-4-yl)-1-((S)...) Show SMILES Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Patents Similars	Article PubMed	n/a	n/a	2.70	n/a	n/a	n/a	n/a	n/a	n/a
Matrix Laboratories Limited Curated by ChEMBL					Assay Description Inhibition of QPP				Bioorg Med Chem 17: 1783-802 (2009) Article DOI: 10.1016/j.bmc.2009.01.061 BindingDB Entry DOI: 10.7270/Q2VD70DJ
Matrix Laboratories Limited Curated by ChEMBL					More data for this Ligand-Target Pair
Dipeptidyl peptidase 2 (Homo sapiens (Human))	BDBM50146981 (2-(S)-Amino-4-(2,4-dimethoxy-benzylamino)-1-piperi...) Show SMILES Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	2.70	n/a	n/a	n/a	n/a	n/a	n/a
University of Antwerp Curated by ChEMBL					Assay Description Inhibition of human Dipeptidyl-peptidase II (DPP II)				J Med Chem 47: 2906-16 (2004) Article DOI: 10.1021/jm031122f BindingDB Entry DOI: 10.7270/Q2TH8M4H
University of Antwerp Curated by ChEMBL					More data for this Ligand-Target Pair
Dipeptidyl peptidase 2 (Homo sapiens (Human))	BDBM50050527 (Boronic acid derivative \| CHEMBL66032 \| US11096924...) Show SMILES CC[C@H](N)C(=O)N1CCC[C@H]1B(O)O Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	US Patent	n/a	n/a	2.90	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description This assay is described in Bachovchin et al. Nature Chemical Biology 10, 656-663 (2014). Briefly, purified enzymes are coupled to Luminex microsphere...				Citation and Details BindingDB Entry DOI: 10.7270/Q28W3J7Z
TBA					More data for this Ligand-Target Pair
Dipeptidyl peptidase 2 (Homo sapiens (Human))	BDBM50191170 ((2S,4S)-4-(4-chlorobenzylamino)-2-amino-1-(piperid...) Show SMILES Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	3.40	n/a	n/a	n/a	n/a	n/a	n/a
Laboratory of Medicinal Chemistry University of Antwerp Curated by ChEMBL					Assay Description Inhibition of DPP2				Bioorg Med Chem Lett 16: 4777-9 (2006) Article DOI: 10.1016/j.bmcl.2006.06.082 BindingDB Entry DOI: 10.7270/Q2GM86XS
					More data for this Ligand-Target Pair

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