Compile Data Set for Download or QSAR

Found 87 hits of ic50 data for polymerid = 5523,9360   

Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kcal/mole	IC50 nM	Kd nM	EC50/IC50 nM	koff s-1	kon M-1s-1	pH	Temp °C
Urokinase plasminogen activator surface receptor (Homo sapiens (Human))	BDBM50120747 (CHEMBL412236 | cyclic uPA-derived peptide) Show SMILES CC(C)C[C@H]1NC(=O)[C@H](CCC(O)=O)NC(=O)[C@@H](CC(N)=O)NC(=O)[C@@H](N)CSSC[C@H](NC(=O)[C@H]2CCCN2C(=O)[C@@H](NC(=O)[C@@H](CCC(N)=O)NC(=O)[C@H](Cc2cnc[nH]2)NC1=O)C(C)C)C(=O)N[C@@H](CC(N)=O)C(O)=O Show InChI InChI=1S/C46H71N15O16S2/c1-20(2)12-26-40(70)57-27(13-22-16-51-19-52-22)41(71)53-24(7-9-32(48)62)39(69)60-36(21(3)4)45(75)61-11-5-6-31(61)44(74)59-30(43(73)58-29(46(76)77)15-34(50)64)18-79-78-17-23(47)37(67)55-28(14-33(49)63)42(72)54-25(38(68)56-26)8-10-35(65)66/h16,19-21,23-31,36H,5-15,17-18,47H2,1-4H3,(H2,48,62)(H2,49,63)(H2,50,64)(H,51,52)(H,53,71)(H,54,72)(H,55,67)(H,56,68)(H,57,70)(H,58,73)(H,59,74)(H,60,69)(H,65,66)(H,76,77)/t23-,24+,25-,26+,27-,28+,29-,30-,31+,36-/m0/s1	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	PubMed	n/a	n/a	40	n/a	n/a	n/a	n/a	n/a	n/a
Technische Universität München Curated by ChEMBL					Assay Description Inhibitory activity of the compound against human Urokinase plasminogen activator receptor (uPAR) was determined				J Med Chem 45: 4984-94 (2002) BindingDB Entry DOI: 10.7270/Q2P84B7C
					More data for this Ligand-Target Pair
Urokinase plasminogen activator surface receptor (Homo sapiens (Human))	BDBM50120746 (CHEMBL405302 | cyclic uPA-derived peptide) Show SMILES CC(C)[C@@H]1NC(=O)[C@@H](CCC(N)=O)NC(=O)[C@H](Cc2cnc[nH]2)NC(=O)[C@@H](Cc2cccc3ccccc23)NC(=O)[C@H](CCC(O)=O)NC(=O)[C@@H](CC(N)=O)NC(=O)[C@@H](N)CSSC[C@H](NC(=O)[C@H]2CCCN2C1=O)C(=O)N[C@@H](CC(N)=O)C(O)=O Show InChI InChI=1S/C53H71N15O16S2/c1-25(2)43-52(82)68-16-6-11-38(68)51(81)66-37(50(80)65-36(53(83)84)20-41(57)71)23-86-85-22-30(54)44(74)62-35(19-40(56)70)49(79)61-32(13-15-42(72)73)45(75)63-33(17-27-9-5-8-26-7-3-4-10-29(26)27)47(77)64-34(18-28-21-58-24-59-28)48(78)60-31(46(76)67-43)12-14-39(55)69/h3-5,7-10,21,24-25,30-38,43H,6,11-20,22-23,54H2,1-2H3,(H2,55,69)(H2,56,70)(H2,57,71)(H,58,59)(H,60,78)(H,61,79)(H,62,74)(H,63,75)(H,64,77)(H,65,80)(H,66,81)(H,67,76)(H,72,73)(H,83,84)/t30-,31+,32-,33+,34-,35+,36-,37-,38+,43-/m0/s1	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	PubMed	n/a	n/a	50	n/a	n/a	n/a	n/a	n/a	n/a
Technische Universität München Curated by ChEMBL					Assay Description Inhibitory activity of the compound against human Urokinase plasminogen activator receptor (uPAR) was determined				J Med Chem 45: 4984-94 (2002) BindingDB Entry DOI: 10.7270/Q2P84B7C
					More data for this Ligand-Target Pair
Urokinase plasminogen activator surface receptor (Homo sapiens (Human))	BDBM50120740 (CHEMBL405999 | cyclic uPA-derived peptide) Show SMILES CCCC[C@@H]1NC(=O)[C@@H](CC(N)=O)NC(=O)[C@@H](N)CSSC[C@H](NC(=O)[C@H]2CCCN2C(=O)[C@@H](NC(=O)[C@@H](CCC(N)=O)NC(=O)[C@H](Cc2cnc[nH]2)NC(=O)[C@@H](CC(C)C)NC1=O)C(C)C)C(=O)N[C@@H](CC(N)=O)C(O)=O Show InChI InChI=1S/C47H75N15O14S2/c1-6-7-9-26-39(67)57-28(14-22(2)3)41(69)58-29(15-24-18-52-21-53-24)42(70)55-27(11-12-34(49)63)40(68)61-37(23(4)5)46(74)62-13-8-10-33(62)45(73)60-32(44(72)59-31(47(75)76)17-36(51)65)20-78-77-19-25(48)38(66)56-30(16-35(50)64)43(71)54-26/h18,21-23,25-33,37H,6-17,19-20,48H2,1-5H3,(H2,49,63)(H2,50,64)(H2,51,65)(H,52,53)(H,54,71)(H,55,70)(H,56,66)(H,57,67)(H,58,69)(H,59,72)(H,60,73)(H,61,68)(H,75,76)/t25-,26-,27+,28+,29-,30+,31-,32-,33+,37-/m0/s1	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	PubMed	n/a	n/a	60	n/a	n/a	n/a	n/a	n/a	n/a
Technische Universität München Curated by ChEMBL					Assay Description Inhibitory activity of the compound against human Urokinase plasminogen activator receptor (uPAR) was determined				J Med Chem 45: 4984-94 (2002) BindingDB Entry DOI: 10.7270/Q2P84B7C
					More data for this Ligand-Target Pair
Urokinase plasminogen activator surface receptor (Homo sapiens (Human))	BDBM50120745 (CHEMBL263158 | cyclic uPA-derived peptide) Show SMILES CC(C)[C@@H]1NC(=O)[C@@H](CCC(N)=O)NC(=O)[C@H](Cc2cnc[nH]2)NC(=O)[C@@H](Cc2ccc3ccccc3c2)NC(=O)[C@H](CCC(O)=O)NC(=O)[C@@H](CC(N)=O)NC(=O)[C@@H](N)CSSC[C@H](NC(=O)[C@H]2CCCN2C1=O)C(=O)N[C@@H](CC(N)=O)C(O)=O Show InChI InChI=1S/C53H71N15O16S2/c1-25(2)43-52(82)68-15-5-8-38(68)51(81)66-37(50(80)65-36(53(83)84)20-41(57)71)23-86-85-22-30(54)44(74)62-35(19-40(56)70)49(79)61-32(12-14-42(72)73)45(75)63-33(17-26-9-10-27-6-3-4-7-28(27)16-26)47(77)64-34(18-29-21-58-24-59-29)48(78)60-31(46(76)67-43)11-13-39(55)69/h3-4,6-7,9-10,16,21,24-25,30-38,43H,5,8,11-15,17-20,22-23,54H2,1-2H3,(H2,55,69)(H2,56,70)(H2,57,71)(H,58,59)(H,60,78)(H,61,79)(H,62,74)(H,63,75)(H,64,77)(H,65,80)(H,66,81)(H,67,76)(H,72,73)(H,83,84)/t30-,31+,32-,33+,34-,35+,36-,37-,38+,43-/m0/s1	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	PubMed	n/a	n/a	80	n/a	n/a	n/a	n/a	n/a	n/a
Technische Universität München Curated by ChEMBL					Assay Description Inhibitory activity of the compound against human Urokinase plasminogen activator receptor (uPAR) was determined				J Med Chem 45: 4984-94 (2002) BindingDB Entry DOI: 10.7270/Q2P84B7C
					More data for this Ligand-Target Pair
Urokinase plasminogen activator surface receptor (Homo sapiens (Human))	BDBM50120743 (CHEMBL385968 | cyclic uPA-derived peptide) Show SMILES CC(C)C[C@H]1NC(=O)[C@H](CCC(O)=O)NC(=O)[C@@H](CC(N)=O)NC(=O)[C@H](CO)NC(=O)CNC(=O)[C@@H](N)CSSC[C@@H](NC(=O)[C@@H](CC(N)=O)NC(=O)[C@H](CO)NC(=O)[C@H]2CCCN2C(=O)[C@@H](NC(=O)[C@@H](CCC(N)=O)NC(=O)[C@H](Cc2cnc[nH]2)NC1=O)C(C)C)C(O)=O Show InChI InChI=1S/C54H84N18O21S2/c1-23(2)12-29-46(84)66-30(13-25-16-59-22-61-25)47(85)63-27(7-9-37(56)75)45(83)71-42(24(3)4)53(91)72-11-5-6-36(72)52(90)69-34(19-74)51(89)68-32(15-39(58)77)49(87)70-35(54(92)93)21-95-94-20-26(55)43(81)60-17-40(78)62-33(18-73)50(88)67-31(14-38(57)76)48(86)64-28(44(82)65-29)8-10-41(79)80/h16,22-24,26-36,42,73-74H,5-15,17-21,55H2,1-4H3,(H2,56,75)(H2,57,76)(H2,58,77)(H,59,61)(H,60,81)(H,62,78)(H,63,85)(H,64,86)(H,65,82)(H,66,84)(H,67,88)(H,68,89)(H,69,90)(H,70,87)(H,71,83)(H,79,80)(H,92,93)/t26-,27+,28-,29+,30-,31+,32+,33-,34-,35+,36+,42-/m0/s1	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	PubMed	n/a	n/a	200	n/a	n/a	n/a	n/a	n/a	n/a
Technische Universität München Curated by ChEMBL					Assay Description Inhibitory activity of the compound against human Urokinase plasminogen activator receptor (uPAR) was determined				J Med Chem 45: 4984-94 (2002) BindingDB Entry DOI: 10.7270/Q2P84B7C
					More data for this Ligand-Target Pair
Urokinase plasminogen activator surface receptor (Homo sapiens (Human))	BDBM50549787 (CHEMBL4791246) Show SMILES O=C(N1CCOCC1)c1cc(nc2c(cccc12)-c1cccs1)-c1ccccc1 Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	500	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Binding affinity to recombinant soluble form urokinase-type plasminogen activator receptor (unknown origin) expressed in S2 cells assessed as inhibit...				Citation and Details Article DOI: 10.1021/acsmedchemlett.0c00422 BindingDB Entry DOI: 10.7270/Q21C21G5
					More data for this Ligand-Target Pair
Urokinase plasminogen activator surface receptor (Homo sapiens (Human))	BDBM50549794 (CHEMBL4753144) Show SMILES Fc1cccc(c1)-c1cc(C(=O)N2CCOCC2)c2cccc(-c3cccs3)c2n1 Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	500	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Binding affinity to recombinant soluble form urokinase-type plasminogen activator receptor (unknown origin) expressed in S2 cells assessed as inhibit...				Citation and Details Article DOI: 10.1021/acsmedchemlett.0c00422 BindingDB Entry DOI: 10.7270/Q21C21G5
					More data for this Ligand-Target Pair
Urokinase plasminogen activator surface receptor (Homo sapiens (Human))	BDBM50120749 (CHEMBL412223 | cyclic uPA-derived peptide) Show SMILES CC(C)C[C@H]1NC(=O)[C@H](CCC(O)=O)NC(=O)[C@@H](CC(N)=O)NC(=O)[C@H](CO)NC(=O)CNC(=O)[C@H](N)CSSC[C@@H](NC(=O)[C@@H](CC(N)=O)NC(=O)[C@H](CO)NC(=O)[C@H]2CCCN2C(=O)[C@@H](NC(=O)[C@@H](CCC(N)=O)NC(=O)[C@H](Cc2cnc[nH]2)NC1=O)C(C)C)C(O)=O Show InChI InChI=1S/C54H84N18O21S2/c1-23(2)12-29-46(84)66-30(13-25-16-59-22-61-25)47(85)63-27(7-9-37(56)75)45(83)71-42(24(3)4)53(91)72-11-5-6-36(72)52(90)69-34(19-74)51(89)68-32(15-39(58)77)49(87)70-35(54(92)93)21-95-94-20-26(55)43(81)60-17-40(78)62-33(18-73)50(88)67-31(14-38(57)76)48(86)64-28(44(82)65-29)8-10-41(79)80/h16,22-24,26-36,42,73-74H,5-15,17-21,55H2,1-4H3,(H2,56,75)(H2,57,76)(H2,58,77)(H,59,61)(H,60,81)(H,62,78)(H,63,85)(H,64,86)(H,65,82)(H,66,84)(H,67,88)(H,68,89)(H,69,90)(H,70,87)(H,71,83)(H,79,80)(H,92,93)/t26-,27-,28+,29-,30+,31-,32-,33+,34+,35-,36-,42+/m1/s1	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	PubMed	n/a	n/a	700	n/a	n/a	n/a	n/a	n/a	n/a
Technische Universität München Curated by ChEMBL					Assay Description Inhibitory activity of the compound against human Urokinase plasminogen activator receptor (uPAR) was determined				J Med Chem 45: 4984-94 (2002) BindingDB Entry DOI: 10.7270/Q2P84B7C
					More data for this Ligand-Target Pair
Urokinase plasminogen activator surface receptor (Homo sapiens (Human))	BDBM50120742 (CHEMBL264653 | cyclic uPA-derived peptide) Show SMILES CC(C)C[C@H]1NC(=O)[C@H](CCC(O)=O)NC(=O)[C@@H](CC(N)=O)NC(=O)[C@H](N)CSSC[C@@H](NC(=O)[C@H]2CCCN2C(=O)[C@@H](NC(=O)[C@@H](CCC(N)=O)NC(=O)[C@H](Cc2cnc[nH]2)NC1=O)C(C)C)C(=O)N[C@@H](CC(N)=O)C(O)=O Show InChI InChI=1S/C46H71N15O16S2/c1-20(2)12-26-40(70)57-27(13-22-16-51-19-52-22)41(71)53-24(7-9-32(48)62)39(69)60-36(21(3)4)45(75)61-11-5-6-31(61)44(74)59-30(43(73)58-29(46(76)77)15-34(50)64)18-79-78-17-23(47)37(67)55-28(14-33(49)63)42(72)54-25(38(68)56-26)8-10-35(65)66/h16,19-21,23-31,36H,5-15,17-18,47H2,1-4H3,(H2,48,62)(H2,49,63)(H2,50,64)(H,51,52)(H,53,71)(H,54,72)(H,55,67)(H,56,68)(H,57,70)(H,58,73)(H,59,74)(H,60,69)(H,65,66)(H,76,77)/t23-,24-,25+,26-,27+,28-,29+,30-,31-,36+/m1/s1	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	PubMed	n/a	n/a	900	n/a	n/a	n/a	n/a	n/a	n/a
Technische Universität München Curated by ChEMBL					Assay Description Inhibitory activity of the compound against human Urokinase plasminogen activator receptor (uPAR) was determined				J Med Chem 45: 4984-94 (2002) BindingDB Entry DOI: 10.7270/Q2P84B7C
					More data for this Ligand-Target Pair
Urokinase plasminogen activator surface receptor (Homo sapiens (Human))	BDBM50549789 (CHEMBL4752534) Show SMILES COc1ccc(cc1)-c1cc(C(=O)N2CCOCC2)c2cccc(-c3cccs3)c2n1 Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	2.20E+3	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Binding affinity to recombinant soluble form urokinase-type plasminogen activator receptor (unknown origin) expressed in S2 cells assessed as inhibit...				Citation and Details Article DOI: 10.1021/acsmedchemlett.0c00422 BindingDB Entry DOI: 10.7270/Q21C21G5
					More data for this Ligand-Target Pair
Urokinase plasminogen activator surface receptor (Homo sapiens (Human))	BDBM50549790 (CHEMBL4748577) Show SMILES COc1cccc(c1)-c1cc(C(=O)N2CCOCC2)c2cccc(-c3cccs3)c2n1 Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	2.20E+3	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Binding affinity to recombinant soluble form urokinase-type plasminogen activator receptor (unknown origin) expressed in S2 cells assessed as inhibit...				Citation and Details Article DOI: 10.1021/acsmedchemlett.0c00422 BindingDB Entry DOI: 10.7270/Q21C21G5
					More data for this Ligand-Target Pair
Urokinase plasminogen activator surface receptor (Homo sapiens (Human))	BDBM50549787 (CHEMBL4791246) Show SMILES O=C(N1CCOCC1)c1cc(nc2c(cccc12)-c1cccs1)-c1ccccc1 Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	4.90E+3	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Inhibition of AE147-FAM peptide binding to recombinant soluble form urokinase-type plasminogen activator receptor (unknown origin) expressed in S2 ce...				Citation and Details Article DOI: 10.1021/acsmedchemlett.0c00422 BindingDB Entry DOI: 10.7270/Q21C21G5
					More data for this Ligand-Target Pair
Urokinase plasminogen activator surface receptor (Homo sapiens (Human))	BDBM50401180 (CHEMBL2206354) Show SMILES CC1CC(C)CN(C1)c1cc(Nc2cccc(c2)C(O)=O)c2C(=O)c3ccccc3-c3onc1c23 Show InChI InChI=1S/C28H25N3O4/c1-15-10-16(2)14-31(13-15)22-12-21(29-18-7-5-6-17(11-18)28(33)34)23-24-25(22)30-35-27(24)20-9-4-3-8-19(20)26(23)32/h3-9,11-12,15-16,29H,10,13-14H2,1-2H3,(H,33,34)	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	Purchase CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	5.00E+3	n/a	n/a	n/a	n/a	n/a	n/a
Indiana University Curated by ChEMBL					Assay Description Inhibition of urokinase receptor binding to uPA amino terminal fragment by ELISA				Bioorg Med Chem 20: 4760-73 (2012) Article DOI: 10.1016/j.bmc.2012.06.002 BindingDB Entry DOI: 10.7270/Q24F1RXX
					More data for this Ligand-Target Pair
Urokinase plasminogen activator surface receptor (Homo sapiens (Human))	BDBM50549788 (CHEMBL4748144) Show SMILES O=C(N1CCOCC1)c1cc(nc2c(cccc12)-c1cncs1)-c1ccccc1 Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	5.80E+3	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Inhibition of AE147-FAM peptide binding to recombinant soluble form urokinase-type plasminogen activator receptor (unknown origin) expressed in S2 ce...				Citation and Details Article DOI: 10.1021/acsmedchemlett.0c00422 BindingDB Entry DOI: 10.7270/Q21C21G5
					More data for this Ligand-Target Pair
Urokinase plasminogen activator surface receptor (Homo sapiens (Human))	BDBM50549801 (CHEMBL4742729) Show SMILES O=C(N1CCOCC1)c1cc(nc2c(CCc3ccccc3)cccc12)-c1ccccc1 Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	6.20E+3	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Inhibition of AE147-FAM peptide binding to recombinant soluble form urokinase-type plasminogen activator receptor (unknown origin) expressed in S2 ce...				Citation and Details Article DOI: 10.1021/acsmedchemlett.0c00422 BindingDB Entry DOI: 10.7270/Q21C21G5
					More data for this Ligand-Target Pair
Urokinase plasminogen activator surface receptor (Homo sapiens (Human))	BDBM50401189 (CHEMBL2205795) Show SMILES CC1CCCN(C1)c1cc(Nc2cccc(c2)C(O)=O)c2C(=O)c3ccccc3-c3onc1c23 Show InChI InChI=1S/C27H23N3O4/c1-15-6-5-11-30(14-15)21-13-20(28-17-8-4-7-16(12-17)27(32)33)22-23-24(21)29-34-26(23)19-10-3-2-9-18(19)25(22)31/h2-4,7-10,12-13,15,28H,5-6,11,14H2,1H3,(H,32,33)	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	Purchase CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	7.00E+3	n/a	n/a	n/a	n/a	n/a	n/a
Indiana University Curated by ChEMBL					Assay Description Inhibition of urokinase receptor binding to uPA amino terminal fragment by ELISA				Bioorg Med Chem 20: 4760-73 (2012) Article DOI: 10.1016/j.bmc.2012.06.002 BindingDB Entry DOI: 10.7270/Q24F1RXX
					More data for this Ligand-Target Pair
Urokinase plasminogen activator surface receptor (Homo sapiens (Human))	BDBM50549794 (CHEMBL4753144) Show SMILES Fc1cccc(c1)-c1cc(C(=O)N2CCOCC2)c2cccc(-c3cccs3)c2n1 Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	7.50E+3	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Inhibition of AE147-FAM peptide binding to recombinant soluble form urokinase-type plasminogen activator receptor (unknown origin) expressed in S2 ce...				Citation and Details Article DOI: 10.1021/acsmedchemlett.0c00422 BindingDB Entry DOI: 10.7270/Q21C21G5
					More data for this Ligand-Target Pair
Urokinase plasminogen activator surface receptor (Homo sapiens (Human))	BDBM50549796 (CHEMBL4740414) Show SMILES O=C(N1CCOCC1)c1cc(nc2c(cccc12)C#Cc1ccccc1)-c1ccccc1 Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	8.50E+3	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Inhibition of AE147-FAM peptide binding to recombinant soluble form urokinase-type plasminogen activator receptor (unknown origin) expressed in S2 ce...				Citation and Details Article DOI: 10.1021/acsmedchemlett.0c00422 BindingDB Entry DOI: 10.7270/Q21C21G5
					More data for this Ligand-Target Pair
Urokinase plasminogen activator surface receptor (Homo sapiens (Human))	BDBM50549793 (CHEMBL4760716) Show SMILES O=C(N1CCOCC1)c1cc(nc2c(cccc12)-c1cccs1)-c1cccnc1 Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	8.50E+3	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Binding affinity to recombinant soluble form urokinase-type plasminogen activator receptor (unknown origin) expressed in S2 cells assessed as inhibit...				Citation and Details Article DOI: 10.1021/acsmedchemlett.0c00422 BindingDB Entry DOI: 10.7270/Q21C21G5
					More data for this Ligand-Target Pair
Urokinase plasminogen activator surface receptor (Homo sapiens (Human))	BDBM50549787 (CHEMBL4791246) Show SMILES O=C(N1CCOCC1)c1cc(nc2c(cccc12)-c1cccs1)-c1ccccc1 Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	8.60E+3	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Binding affinity to recombinant soluble form urokinase-type plasminogen activator receptor (unknown origin) expressed in S2 cells assessed as inhibit...				Citation and Details Article DOI: 10.1021/acsmedchemlett.0c00422 BindingDB Entry DOI: 10.7270/Q21C21G5
					More data for this Ligand-Target Pair
Urokinase plasminogen activator surface receptor (Homo sapiens (Human))	BDBM50549792 (CHEMBL4790155) Show SMILES O=C(N1CCOCC1)c1cc(nc2c(cncc12)-c1cccs1)-c1ccccc1 Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	9.30E+3	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Inhibition of AE147-FAM peptide binding to recombinant soluble form urokinase-type plasminogen activator receptor (unknown origin) expressed in S2 ce...				Citation and Details Article DOI: 10.1021/acsmedchemlett.0c00422 BindingDB Entry DOI: 10.7270/Q21C21G5
					More data for this Ligand-Target Pair
Urokinase plasminogen activator surface receptor (Homo sapiens (Human))	BDBM50549800 (CHEMBL4748584) Show SMILES C1CC(CCN1)n1ccc(n1)-c1cc(nc2c(cccc12)-c1cccs1)-c1ccccc1 Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	9.50E+3	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Inhibition of AE147-FAM peptide binding to recombinant soluble form urokinase-type plasminogen activator receptor (unknown origin) expressed in S2 ce...				Citation and Details Article DOI: 10.1021/acsmedchemlett.0c00422 BindingDB Entry DOI: 10.7270/Q21C21G5
					More data for this Ligand-Target Pair
Urokinase plasminogen activator surface receptor (Homo sapiens (Human))	BDBM50549797 (CHEMBL4757892) Show SMILES O=C(N1CCOCC1)c1cc(nc2c(cccc12)-c1ccccc1)-c1ccccc1 Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	9.80E+3	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Inhibition of AE147-FAM peptide binding to recombinant soluble form urokinase-type plasminogen activator receptor (unknown origin) expressed in S2 ce...				Citation and Details Article DOI: 10.1021/acsmedchemlett.0c00422 BindingDB Entry DOI: 10.7270/Q21C21G5
					More data for this Ligand-Target Pair
Urokinase plasminogen activator surface receptor (Homo sapiens (Human))	BDBM50401178 (CHEMBL2206358) Show SMILES CC1CC(C)CN(C1)c1cc(Nc2ccccc2C(O)=O)c2C(=O)c3ccccc3-c3onc1c23 Show InChI InChI=1S/C28H25N3O4/c1-15-11-16(2)14-31(13-15)22-12-21(29-20-10-6-5-9-19(20)28(33)34)23-24-25(22)30-35-27(24)18-8-4-3-7-17(18)26(23)32/h3-10,12,15-16,29H,11,13-14H2,1-2H3,(H,33,34)	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	Purchase CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	1.00E+4	n/a	n/a	n/a	n/a	n/a	n/a
Indiana University Curated by ChEMBL					Assay Description Inhibition of urokinase receptor binding to uPA amino terminal fragment by ELISA				Bioorg Med Chem 20: 4760-73 (2012) Article DOI: 10.1016/j.bmc.2012.06.002 BindingDB Entry DOI: 10.7270/Q24F1RXX
					More data for this Ligand-Target Pair
Urokinase plasminogen activator surface receptor (Homo sapiens (Human))	BDBM50401187 (CHEMBL2205797) Show SMILES CC1CCCCN1c1cc(Nc2cccc(c2)C(O)=O)c2C(=O)c3ccccc3-c3onc1c23 Show InChI InChI=1S/C27H23N3O4/c1-15-7-4-5-12-30(15)21-14-20(28-17-9-6-8-16(13-17)27(32)33)22-23-24(21)29-34-26(23)19-11-3-2-10-18(19)25(22)31/h2-3,6,8-11,13-15,28H,4-5,7,12H2,1H3,(H,32,33)	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	Purchase CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	1.00E+4	n/a	n/a	n/a	n/a	n/a	n/a
Indiana University Curated by ChEMBL					Assay Description Inhibition of urokinase receptor binding to uPA amino terminal fragment by ELISA				Bioorg Med Chem 20: 4760-73 (2012) Article DOI: 10.1016/j.bmc.2012.06.002 BindingDB Entry DOI: 10.7270/Q24F1RXX
					More data for this Ligand-Target Pair
Urokinase plasminogen activator surface receptor (Homo sapiens (Human))	BDBM50549792 (CHEMBL4790155) Show SMILES O=C(N1CCOCC1)c1cc(nc2c(cncc12)-c1cccs1)-c1ccccc1 Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	1.04E+4	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Binding affinity to recombinant soluble form urokinase-type plasminogen activator receptor (unknown origin) expressed in S2 cells assessed as inhibit...				Citation and Details Article DOI: 10.1021/acsmedchemlett.0c00422 BindingDB Entry DOI: 10.7270/Q21C21G5
					More data for this Ligand-Target Pair
Urokinase plasminogen activator surface receptor (Homo sapiens (Human))	BDBM50401188 (CHEMBL2205796) Show SMILES CC1CCCN(C1)c1cc(=Cc2ccc(cc2)C(O)=O)c2c(O)c3ccccc3c3onc1c23 |w:10.11| Show InChI InChI=1S/C28H24N2O4/c1-16-5-4-12-30(15-16)22-14-19(13-17-8-10-18(11-9-17)28(32)33)23-24-25(22)29-34-27(24)21-7-3-2-6-20(21)26(23)31/h2-3,6-11,13-14,16,31H,4-5,12,15H2,1H3,(H,32,33)	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	1.10E+4	n/a	n/a	n/a	n/a	n/a	n/a
Indiana University Curated by ChEMBL					Assay Description Inhibition of urokinase receptor binding to uPA amino terminal fragment by ELISA				Bioorg Med Chem 20: 4760-73 (2012) Article DOI: 10.1016/j.bmc.2012.06.002 BindingDB Entry DOI: 10.7270/Q24F1RXX
					More data for this Ligand-Target Pair
Urokinase plasminogen activator surface receptor (Homo sapiens (Human))	BDBM50549790 (CHEMBL4748577) Show SMILES COc1cccc(c1)-c1cc(C(=O)N2CCOCC2)c2cccc(-c3cccs3)c2n1 Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	1.20E+4	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Inhibition of AE147-FAM peptide binding to recombinant soluble form urokinase-type plasminogen activator receptor (unknown origin) expressed in S2 ce...				Citation and Details Article DOI: 10.1021/acsmedchemlett.0c00422 BindingDB Entry DOI: 10.7270/Q21C21G5
					More data for this Ligand-Target Pair
Urokinase plasminogen activator surface receptor (Homo sapiens (Human))	BDBM50549789 (CHEMBL4752534) Show SMILES COc1ccc(cc1)-c1cc(C(=O)N2CCOCC2)c2cccc(-c3cccs3)c2n1 Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	1.23E+4	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Inhibition of AE147-FAM peptide binding to recombinant soluble form urokinase-type plasminogen activator receptor (unknown origin) expressed in S2 ce...				Citation and Details Article DOI: 10.1021/acsmedchemlett.0c00422 BindingDB Entry DOI: 10.7270/Q21C21G5
					More data for this Ligand-Target Pair
Urokinase plasminogen activator surface receptor (Homo sapiens (Human))	BDBM50549799 (CHEMBL4740458) Show SMILES O=C(N1CCNCC1)c1cc(nc2c(cccc12)-c1cccs1)-c1ccccc1 Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	1.31E+4	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Inhibition of AE147-FAM peptide binding to recombinant soluble form urokinase-type plasminogen activator receptor (unknown origin) expressed in S2 ce...				Citation and Details Article DOI: 10.1021/acsmedchemlett.0c00422 BindingDB Entry DOI: 10.7270/Q21C21G5
					More data for this Ligand-Target Pair
Urokinase plasminogen activator surface receptor (Homo sapiens (Human))	BDBM50549791 (CHEMBL4755034) Show SMILES Clc1cccc(c1)N1CCN(CC1)C(=O)c1cc(nc2c(cccc12)-c1cccs1)-c1ccccc1 Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	1.34E+4	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Binding affinity to recombinant soluble form urokinase-type plasminogen activator receptor (unknown origin) expressed in S2 cells assessed as inhibit...				Citation and Details Article DOI: 10.1021/acsmedchemlett.0c00422 BindingDB Entry DOI: 10.7270/Q21C21G5
					More data for this Ligand-Target Pair
Urokinase plasminogen activator surface receptor (Homo sapiens (Human))	BDBM50549797 (CHEMBL4757892) Show SMILES O=C(N1CCOCC1)c1cc(nc2c(cccc12)-c1ccccc1)-c1ccccc1 Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	1.39E+4	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Binding affinity to recombinant soluble form urokinase-type plasminogen activator receptor (unknown origin) expressed in S2 cells assessed as inhibit...				Citation and Details Article DOI: 10.1021/acsmedchemlett.0c00422 BindingDB Entry DOI: 10.7270/Q21C21G5
					More data for this Ligand-Target Pair
Urokinase plasminogen activator surface receptor (Homo sapiens (Human))	BDBM222392 (IPR-2260 (45)) Show SMILES COC(=O)c1cccc(c1)-c1ccc(cc1)N1C(C(C(=O)c2ccc(Cl)cc2)=C(O)C1=O)c1cccc(F)c1 |t:30| Show InChI InChI=1S/C31H21ClFNO5/c1-39-31(38)22-6-2-4-20(16-22)18-10-14-25(15-11-18)34-27(21-5-3-7-24(33)17-21)26(29(36)30(34)37)28(35)19-8-12-23(32)13-9-19/h2-17,27,36H,1H3	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	400	n/a	1.57E+4	n/a	n/a	n/a	n/a	n/a	n/a
Indiana University School of Medicine					Assay Description Polarized fluorescence intensities were measured using an EnVision Multilabel plate reader (PerkinElmer) with excitation and emission wavelengths of ...				Biochemistry 56: 1768-1784 (2017) Article DOI: 10.1021/acs.biochem.6b01039 BindingDB Entry DOI: 10.7270/Q2NS0SQC
					More data for this Ligand-Target Pair
Urokinase plasminogen activator surface receptor (Homo sapiens (Human))	BDBM222351 (IPR-1201 (4)) Show SMILES Cc1ccc(cc1Br)N1C(C(C(=O)c2ccc(Cl)c(C)c2)=C(O)C1=O)c1cccc(F)c1 |t:22| Show InChI InChI=1S/C25H18BrClFNO3/c1-13-6-8-18(12-19(13)26)29-22(15-4-3-5-17(28)11-15)21(24(31)25(29)32)23(30)16-7-9-20(27)14(2)10-16/h3-12,22,31H,1-2H3	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	1.00E+3	n/a	1.63E+4	n/a	n/a	n/a	n/a	n/a	n/a
Indiana University School of Medicine					Assay Description Polarized fluorescence intensities were measured using an EnVision Multilabel plate reader (PerkinElmer) with excitation and emission wavelengths of ...				Biochemistry 56: 1768-1784 (2017) Article DOI: 10.1021/acs.biochem.6b01039 BindingDB Entry DOI: 10.7270/Q2NS0SQC
					More data for this Ligand-Target Pair
Urokinase plasminogen activator surface receptor (Homo sapiens (Human))	BDBM50401186 (CHEMBL2206348) Show SMILES CC1CC(C)CN(C1)c1cc(NCCC(O)=O)c2C(=O)c3ccccc3-c3onc1c23 Show InChI InChI=1S/C24H25N3O4/c1-13-9-14(2)12-27(11-13)18-10-17(25-8-7-19(28)29)20-21-22(18)26-31-24(21)16-6-4-3-5-15(16)23(20)30/h3-6,10,13-14,25H,7-9,11-12H2,1-2H3,(H,28,29)	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	Purchase CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	1.80E+4	n/a	n/a	n/a	n/a	n/a	n/a
Indiana University Curated by ChEMBL					Assay Description Inhibition of urokinase receptor binding to uPA amino terminal fragment by ELISA				Bioorg Med Chem 20: 4760-73 (2012) Article DOI: 10.1016/j.bmc.2012.06.002 BindingDB Entry DOI: 10.7270/Q24F1RXX
					More data for this Ligand-Target Pair
Urokinase plasminogen activator surface receptor (Homo sapiens (Human))	BDBM222350 (IPR-1110 (1)) Show SMILES Cc1ccc(cc1Br)N1C(C(C(=O)c2ccc(Cl)cc2)=C(O)C1=O)c1cccc(F)c1 |t:21| Show InChI InChI=1S/C24H16BrClFNO3/c1-13-5-10-18(12-19(13)25)28-21(15-3-2-4-17(27)11-15)20(23(30)24(28)31)22(29)14-6-8-16(26)9-7-14/h2-12,21,30H,1H3	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	Purchase PC cid PC sid UniChem	Article PubMed	700	n/a	1.84E+4	n/a	n/a	n/a	n/a	n/a	n/a
Indiana University School of Medicine					Assay Description Polarized fluorescence intensities were measured using an EnVision Multilabel plate reader (PerkinElmer) with excitation and emission wavelengths of ...				Biochemistry 56: 1768-1784 (2017) Article DOI: 10.1021/acs.biochem.6b01039 BindingDB Entry DOI: 10.7270/Q2NS0SQC
					More data for this Ligand-Target Pair
Urokinase plasminogen activator surface receptor (Homo sapiens (Human))	BDBM222370 (IPR-1174 (23)) Show SMILES CCCCCCOc1cc(ccc1C)N1C(C(C(=O)c2ccc(Cl)cc2)=C(O)C1=O)c1cccc(F)c1 |t:27| Show InChI InChI=1S/C30H29ClFNO4/c1-3-4-5-6-16-37-25-18-24(15-10-19(25)2)33-27(21-8-7-9-23(32)17-21)26(29(35)30(33)36)28(34)20-11-13-22(31)14-12-20/h7-15,17-18,27,35H,3-6,16H2,1-2H3	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	1.20E+3	n/a	1.84E+4	n/a	n/a	n/a	n/a	n/a	n/a
Indiana University School of Medicine					Assay Description Polarized fluorescence intensities were measured using an EnVision Multilabel plate reader (PerkinElmer) with excitation and emission wavelengths of ...				Biochemistry 56: 1768-1784 (2017) Article DOI: 10.1021/acs.biochem.6b01039 BindingDB Entry DOI: 10.7270/Q2NS0SQC
					More data for this Ligand-Target Pair
Urokinase plasminogen activator surface receptor (Homo sapiens (Human))	BDBM50401181 (CHEMBL2206353) Show SMILES CC1CCCN(C1)c1cc(NCCCC(O)=O)c2C(=O)c3ccccc3-c3onc1c23 Show InChI InChI=1S/C24H25N3O4/c1-14-6-5-11-27(13-14)18-12-17(25-10-4-9-19(28)29)20-21-22(18)26-31-24(21)16-8-3-2-7-15(16)23(20)30/h2-3,7-8,12,14,25H,4-6,9-11,13H2,1H3,(H,28,29)	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	Purchase CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	2.00E+4	n/a	n/a	n/a	n/a	n/a	n/a
Indiana University Curated by ChEMBL					Assay Description Inhibition of urokinase receptor binding to uPA amino terminal fragment by ELISA				Bioorg Med Chem 20: 4760-73 (2012) Article DOI: 10.1016/j.bmc.2012.06.002 BindingDB Entry DOI: 10.7270/Q24F1RXX
					More data for this Ligand-Target Pair
Urokinase plasminogen activator surface receptor (Homo sapiens (Human))	BDBM222354 (IPR-1178 (7)) Show SMILES Cc1ccc(cc1Br)N1C(C(C(=O)c2ccc(Cl)cc2)=C(O)C1=O)c1cccc(Cl)c1 |t:21| Show InChI InChI=1S/C24H16BrCl2NO3/c1-13-5-10-18(12-19(13)25)28-21(15-3-2-4-17(27)11-15)20(23(30)24(28)31)22(29)14-6-8-16(26)9-7-14/h2-12,21,30H,1H3	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	1.10E+3	n/a	2.02E+4	n/a	n/a	n/a	n/a	n/a	n/a
Indiana University School of Medicine					Assay Description Polarized fluorescence intensities were measured using an EnVision Multilabel plate reader (PerkinElmer) with excitation and emission wavelengths of ...				Biochemistry 56: 1768-1784 (2017) Article DOI: 10.1021/acs.biochem.6b01039 BindingDB Entry DOI: 10.7270/Q2NS0SQC
					More data for this Ligand-Target Pair
Urokinase plasminogen activator surface receptor (Homo sapiens (Human))	BDBM222375 (IPR-1190 (28)) Show SMILES COc1cc(ccc1F)C1N(C(=O)C(O)=C1C(=O)c1ccc(Cl)cc1)c1ccc(C)c(Br)c1 |c:15| Show InChI InChI=1S/C25H18BrClFNO4/c1-13-3-9-17(12-18(13)26)29-22(15-6-10-19(28)20(11-15)33-2)21(24(31)25(29)32)23(30)14-4-7-16(27)8-5-14/h3-12,22,31H,1-2H3	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	2.60E+3	n/a	2.10E+4	n/a	n/a	n/a	n/a	n/a	n/a
Indiana University School of Medicine					Assay Description Polarized fluorescence intensities were measured using an EnVision Multilabel plate reader (PerkinElmer) with excitation and emission wavelengths of ...				Biochemistry 56: 1768-1784 (2017) Article DOI: 10.1021/acs.biochem.6b01039 BindingDB Entry DOI: 10.7270/Q2NS0SQC
					More data for this Ligand-Target Pair
Urokinase plasminogen activator surface receptor (Homo sapiens (Human))	BDBM50401190 (CHEMBL2205794) Show SMILES OC(=O)c1ccccc1Nc1cc(N2CCCC2)c2noc3-c4ccccc4C(=O)c1c23 Show InChI InChI=1S/C25H19N3O4/c29-23-14-7-1-2-8-15(14)24-21-20(23)18(26-17-10-4-3-9-16(17)25(30)31)13-19(22(21)27-32-24)28-11-5-6-12-28/h1-4,7-10,13,26H,5-6,11-12H2,(H,30,31)	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	Purchase CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	2.10E+4	n/a	n/a	n/a	n/a	n/a	n/a
Indiana University Curated by ChEMBL					Assay Description Inhibition of urokinase receptor binding to uPA amino terminal fragment by ELISA				Bioorg Med Chem 20: 4760-73 (2012) Article DOI: 10.1016/j.bmc.2012.06.002 BindingDB Entry DOI: 10.7270/Q24F1RXX
					More data for this Ligand-Target Pair
Urokinase plasminogen activator surface receptor (Homo sapiens (Human))	BDBM222393 (IPR-1609 (46)) Show SMILES OC1=C(C(N(CCc2ccc(Cl)c(Cl)c2)C1=O)c1cccc(F)c1)C(=O)c1cccc(Cl)c1 |t:1| Show InChI InChI=1S/C25H17Cl3FNO3/c26-17-5-1-4-16(12-17)23(31)21-22(15-3-2-6-18(29)13-15)30(25(33)24(21)32)10-9-14-7-8-19(27)20(28)11-14/h1-8,11-13,22,32H,9-10H2	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	600	n/a	2.16E+4	n/a	n/a	n/a	n/a	n/a	n/a
Indiana University School of Medicine					Assay Description Polarized fluorescence intensities were measured using an EnVision Multilabel plate reader (PerkinElmer) with excitation and emission wavelengths of ...				Biochemistry 56: 1768-1784 (2017) Article DOI: 10.1021/acs.biochem.6b01039 BindingDB Entry DOI: 10.7270/Q2NS0SQC
					More data for this Ligand-Target Pair
Urokinase plasminogen activator surface receptor (Homo sapiens (Human))	BDBM50549793 (CHEMBL4760716) Show SMILES O=C(N1CCOCC1)c1cc(nc2c(cccc12)-c1cccs1)-c1cccnc1 Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	2.27E+4	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Inhibition of AE147-FAM peptide binding to recombinant soluble form urokinase-type plasminogen activator receptor (unknown origin) expressed in S2 ce...				Citation and Details Article DOI: 10.1021/acsmedchemlett.0c00422 BindingDB Entry DOI: 10.7270/Q21C21G5
					More data for this Ligand-Target Pair
Urokinase plasminogen activator surface receptor (Homo sapiens (Human))	BDBM222360 (IPR-1171 (13)) Show SMILES Cc1ccc(cc1I)N1C(C(C(=O)c2ccc(Cl)cc2)=C(O)C1=O)c1cccc(F)c1 |t:21| Show InChI InChI=1S/C24H16ClFINO3/c1-13-5-10-18(12-19(13)27)28-21(15-3-2-4-17(26)11-15)20(23(30)24(28)31)22(29)14-6-8-16(25)9-7-14/h2-12,21,30H,1H3	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	1.30E+3	n/a	2.30E+4	n/a	n/a	n/a	n/a	n/a	n/a
Indiana University School of Medicine					Assay Description Polarized fluorescence intensities were measured using an EnVision Multilabel plate reader (PerkinElmer) with excitation and emission wavelengths of ...				Biochemistry 56: 1768-1784 (2017) Article DOI: 10.1021/acs.biochem.6b01039 BindingDB Entry DOI: 10.7270/Q2NS0SQC
					More data for this Ligand-Target Pair
Urokinase plasminogen activator surface receptor (Homo sapiens (Human))	BDBM222386 (IPR-1168 (39)) Show SMILES OC1=C(C(N(CCc2ccc(Cl)c(Cl)c2)C1=O)c1cccc(F)c1)C(=O)c1ccc(Cl)cc1 |t:1| Show InChI InChI=1S/C25H17Cl3FNO3/c26-17-7-5-15(6-8-17)23(31)21-22(16-2-1-3-18(29)13-16)30(25(33)24(21)32)11-10-14-4-9-19(27)20(28)12-14/h1-9,12-13,22,32H,10-11H2	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	900	n/a	2.31E+4	n/a	n/a	n/a	n/a	n/a	n/a
Indiana University School of Medicine					Assay Description Polarized fluorescence intensities were measured using an EnVision Multilabel plate reader (PerkinElmer) with excitation and emission wavelengths of ...				Biochemistry 56: 1768-1784 (2017) Article DOI: 10.1021/acs.biochem.6b01039 BindingDB Entry DOI: 10.7270/Q2NS0SQC
					More data for this Ligand-Target Pair
Urokinase plasminogen activator surface receptor (Homo sapiens (Human))	BDBM222391 (IPR-1607 (44)) Show SMILES OC1=C(C(N(C1=O)c1ccc(cc1)-c1ccccc1)c1cccc(F)c1)C(=O)c1ccc(Cl)cc1 |t:1| Show InChI InChI=1S/C29H19ClFNO3/c30-22-13-9-20(10-14-22)27(33)25-26(21-7-4-8-23(31)17-21)32(29(35)28(25)34)24-15-11-19(12-16-24)18-5-2-1-3-6-18/h1-17,26,34H	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	800	n/a	2.40E+4	n/a	n/a	n/a	n/a	n/a	n/a
Indiana University School of Medicine					Assay Description Polarized fluorescence intensities were measured using an EnVision Multilabel plate reader (PerkinElmer) with excitation and emission wavelengths of ...				Biochemistry 56: 1768-1784 (2017) Article DOI: 10.1021/acs.biochem.6b01039 BindingDB Entry DOI: 10.7270/Q2NS0SQC
					More data for this Ligand-Target Pair
Urokinase plasminogen activator surface receptor (Homo sapiens (Human))	BDBM50401184 (CHEMBL2206350) Show SMILES CC1CCCN(C1)c1cc(NCCC(O)=O)c2C(=O)c3ccccc3-c3onc1c23 Show InChI InChI=1S/C23H23N3O4/c1-13-5-4-10-26(12-13)17-11-16(24-9-8-18(27)28)19-20-21(17)25-30-23(20)15-7-3-2-6-14(15)22(19)29/h2-3,6-7,11,13,24H,4-5,8-10,12H2,1H3,(H,27,28)	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	Purchase CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	2.40E+4	n/a	n/a	n/a	n/a	n/a	n/a
Indiana University Curated by ChEMBL					Assay Description Inhibition of urokinase receptor binding to uPA amino terminal fragment by ELISA				Bioorg Med Chem 20: 4760-73 (2012) Article DOI: 10.1016/j.bmc.2012.06.002 BindingDB Entry DOI: 10.7270/Q24F1RXX
					More data for this Ligand-Target Pair
Urokinase plasminogen activator surface receptor (Homo sapiens (Human))	BDBM50549795 (CHEMBL4748990) Show SMILES O=C(N1CCOCC1)c1cc(nc2c(cccc12)N1C(=O)c2ccccc2C1=O)-c1ccccc1 Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	2.50E+4	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description Inhibition of AE147-FAM peptide binding to recombinant soluble form urokinase-type plasminogen activator receptor (unknown origin) expressed in S2 ce...				Citation and Details Article DOI: 10.1021/acsmedchemlett.0c00422 BindingDB Entry DOI: 10.7270/Q21C21G5
					More data for this Ligand-Target Pair
Urokinase plasminogen activator surface receptor (Homo sapiens (Human))	BDBM222355 (IPR-1187 (8)) Show SMILES CCc1cccc(c1)C1N(C(=O)C(O)=C1C(=O)c1ccc(Cl)cc1)c1ccc(C)c(Br)c1 |c:14| Show InChI InChI=1S/C26H21BrClNO3/c1-3-16-5-4-6-18(13-16)23-22(24(30)17-8-10-19(28)11-9-17)25(31)26(32)29(23)20-12-7-15(2)21(27)14-20/h4-14,23,31H,3H2,1-2H3	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	2.50E+3	n/a	2.64E+4	n/a	n/a	n/a	n/a	n/a	n/a
Indiana University School of Medicine					Assay Description Polarized fluorescence intensities were measured using an EnVision Multilabel plate reader (PerkinElmer) with excitation and emission wavelengths of ...				Biochemistry 56: 1768-1784 (2017) Article DOI: 10.1021/acs.biochem.6b01039 BindingDB Entry DOI: 10.7270/Q2NS0SQC
					More data for this Ligand-Target Pair
Urokinase plasminogen activator surface receptor (Homo sapiens (Human))	BDBM222352 (IPR-1200 (5)) Show SMILES Cc1ccc(cc1Br)N1C(C(C(=O)c2ccc(cc2)C(C)(C)C)=C(O)C1=O)c1cccc(F)c1 |t:24| Show InChI InChI=1S/C28H25BrFNO3/c1-16-8-13-21(15-22(16)29)31-24(18-6-5-7-20(30)14-18)23(26(33)27(31)34)25(32)17-9-11-19(12-10-17)28(2,3)4/h5-15,24,33H,1-4H3	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	2.70E+3	n/a	2.74E+4	n/a	n/a	n/a	n/a	n/a	n/a
Indiana University School of Medicine					Assay Description Polarized fluorescence intensities were measured using an EnVision Multilabel plate reader (PerkinElmer) with excitation and emission wavelengths of ...				Biochemistry 56: 1768-1784 (2017) Article DOI: 10.1021/acs.biochem.6b01039 BindingDB Entry DOI: 10.7270/Q2NS0SQC
					More data for this Ligand-Target Pair

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