BindingDB PrimarySearch

Found 40 hits of ic50 for UniProtKB: P00516
Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kcal/mole	IC50 nM	Kd nM	EC50/IC50 nM	k_off s^-1	k_on M^-1s^-1	pH	Temp °C
cGMP-dependent protein kinase 1 (Bos taurus (bovine))	BDBM2579 ((2S,3R,4R,6R)-3-methoxy-2-methyl-4-(methylamino)-2...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet	Purchase CHEMBL MCE KEGG MMDB PC cid PC sid PDB UniChem Patents Similars	Article	n/a	n/a	18	n/a	n/a	n/a	n/a	n/a	n/a
Tumor Biology Center					Assay Description The activity of cGPK, activated by cGMP, is measured by its ability to transfer phosphate from [gamma-32P]ATP to histone.				Bioorg Med Chem Lett 5: 55-60 (1995) Article DOI: 10.1016/0960-894X(94)00458-R BindingDB Entry DOI: 10.7270/Q2CF9N8C
Tumor Biology Center					More data for this Ligand-Target Pair
cGMP-dependent protein kinase 1 (Bos taurus (bovine))	BDBM2579 ((2S,3R,4R,6R)-3-methoxy-2-methyl-4-(methylamino)-2...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet	Purchase CHEMBL MCE KEGG MMDB PC cid PC sid PDB UniChem Patents Similars	Article	n/a	n/a	18	n/a	n/a	n/a	n/a	n/a	n/a
TBA Curated by ChEMBL					Assay Description In vitro for inhibitory activity against cGMP-dependent protein kinase from bovine lung (G-kinase)				Bioorg Med Chem Lett 3: 1959-1964 (1993) Article DOI: 10.1016/S0960-894X(01)80995-1 BindingDB Entry DOI: 10.7270/Q2QC03DJ
TBA Curated by ChEMBL					More data for this Ligand-Target Pair
cGMP-dependent protein kinase 1 (Bos taurus (bovine))	BDBM3040 (23-(3-aminopropyl)-3-methyl-3,13,23-triazahexacycl...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet	PC cid PC sid UniChem Similars	Article	n/a	n/a	220	n/a	n/a	n/a	n/a	n/a	n/a
Tumor Biology Center					Assay Description The activity of cGPK, activated by cGMP, is measured by its ability to transfer phosphate from [gamma-32P]ATP to histone.				Bioorg Med Chem Lett 5: 55-60 (1995) Article DOI: 10.1016/0960-894X(94)00458-R BindingDB Entry DOI: 10.7270/Q2CF9N8C
Tumor Biology Center					More data for this Ligand-Target Pair
cGMP-dependent protein kinase 1 (Bos taurus (bovine))	BDBM50280868 (12-(2,3-dihydroxypropyl)-6,7,12,13-tetrahydro-5H-i...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article	n/a	n/a	280	n/a	n/a	n/a	n/a	n/a	n/a
TBA Curated by ChEMBL					Assay Description In vitro for inhibitory activity against cGMP-dependent protein kinase from bovine lung (G-kinase)				Bioorg Med Chem Lett 3: 1959-1964 (1993) Article DOI: 10.1016/S0960-894X(01)80995-1 BindingDB Entry DOI: 10.7270/Q2QC03DJ
TBA Curated by ChEMBL					More data for this Ligand-Target Pair
cGMP-dependent protein kinase 1 (Bos taurus (bovine))	BDBM50280877 (2-(5-oxo-6,7,12,13-tetrahydro-5H-indolo[2,3-a]pyrr...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Patents Similars	Article	n/a	n/a	320	n/a	n/a	n/a	n/a	n/a	n/a
TBA Curated by ChEMBL					Assay Description In vitro for inhibitory activity against cGMP-dependent protein kinase from bovine lung (G-kinase)				Bioorg Med Chem Lett 3: 1959-1964 (1993) Article DOI: 10.1016/S0960-894X(01)80995-1 BindingDB Entry DOI: 10.7270/Q2QC03DJ
TBA Curated by ChEMBL					More data for this Ligand-Target Pair
cGMP-dependent protein kinase 1 (Bos taurus (bovine))	BDBM10840 (4-(5-bromo-1H-indol-3-yl)pyrimidin-2-amine \| Merid...) Show SMILES Nc1nccc(n1)-c1c[nH]c2ccc(Br)cc12 Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet	Purchase MCE PC cid PC sid UniChem Patents Similars	Article PubMed	n/a	n/a	400	n/a	n/a	n/a	n/a	n/a	30
CNRS					Assay Description Kinase activities were assayed in buffers containing substrate, enzyme, and inhibitor at 30°C in the presence of 15 uM ATP/[gamma-32P] ATP. 32P ...				Bioorg Med Chem Lett 14: 1703-7 (2004) Article DOI: 10.1016/j.bmcl.2004.01.050 BindingDB Entry DOI: 10.7270/Q2BZ648W
CNRS					More data for this Ligand-Target Pair
cGMP-dependent protein kinase 1 (Bos taurus (bovine))	BDBM50280876 (12-methyl-6,7,12,13-tetrahydro-5H-indolo[2,3-a]pyr...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Patents Similars	Article	n/a	n/a	400	n/a	n/a	n/a	n/a	n/a	n/a
TBA Curated by ChEMBL					Assay Description In vitro for inhibitory activity against cGMP-dependent protein kinase from bovine lung (G-kinase)				Bioorg Med Chem Lett 3: 1959-1964 (1993) Article DOI: 10.1016/S0960-894X(01)80995-1 BindingDB Entry DOI: 10.7270/Q2QC03DJ
TBA Curated by ChEMBL					More data for this Ligand-Target Pair
cGMP-dependent protein kinase 1 (Bos taurus (bovine))	BDBM3036 (23-[3-(dimethylamino)propyl]-3,13,23-triazahexacyc...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet	PC cid PC sid UniChem Patents Similars	Article	n/a	n/a	420	n/a	n/a	n/a	n/a	n/a	n/a
Tumor Biology Center					Assay Description The activity of cGPK, activated by cGMP, is measured by its ability to transfer phosphate from [gamma-32P]ATP to histone.				Bioorg Med Chem Lett 5: 55-60 (1995) Article DOI: 10.1016/0960-894X(94)00458-R BindingDB Entry DOI: 10.7270/Q2CF9N8C
Tumor Biology Center					More data for this Ligand-Target Pair
cGMP-dependent protein kinase 1 (Bos taurus (bovine))	BDBM10842 (3-(2-aminopyrimidin-4-yl)-7-bromo-1H-indol-4-ol \| ...) Show SMILES Nc1nccc(n1)-c1c[nH]c2c(Br)ccc(O)c12 Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet	PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	600	n/a	n/a	n/a	n/a	n/a	30
CNRS					Assay Description Kinase activities were assayed in buffers containing substrate, enzyme, and inhibitor at 30°C in the presence of 15 uM ATP/[gamma-32P] ATP. 32P ...				Bioorg Med Chem Lett 14: 1703-7 (2004) Article DOI: 10.1016/j.bmcl.2004.01.050 BindingDB Entry DOI: 10.7270/Q2BZ648W
CNRS					More data for this Ligand-Target Pair
cGMP-dependent protein kinase 1 (Bos taurus (bovine))	BDBM10843 (4-(5,6-dibromo-1H-indol-3-yl)pyrimidin-2-amine \| M...) Show SMILES Nc1nccc(n1)-c1c[nH]c2cc(Br)c(Br)cc12 Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet	PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	600	n/a	n/a	n/a	n/a	n/a	30
CNRS					Assay Description Kinase activities were assayed in buffers containing substrate, enzyme, and inhibitor at 30°C in the presence of 15 uM ATP/[gamma-32P] ATP. 32P ...				Bioorg Med Chem Lett 14: 1703-7 (2004) Article DOI: 10.1016/j.bmcl.2004.01.050 BindingDB Entry DOI: 10.7270/Q2BZ648W
CNRS					More data for this Ligand-Target Pair
cGMP-dependent protein kinase 1 (Bos taurus (bovine))	BDBM2581 (3,13,23-triazahexacyclo[14.7.0.0^{2,10}.0^{4,9}.0^...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet	Purchase CHEMBL DrugBank MCE PC cid PC sid PDB UniChem Patents Similars	Article	n/a	n/a	650	n/a	n/a	n/a	n/a	n/a	n/a
TBA Curated by ChEMBL					Assay Description In vitro for inhibitory activity against cGMP-dependent protein kinase from bovine lung (G-kinase)				Bioorg Med Chem Lett 3: 1959-1964 (1993) Article DOI: 10.1016/S0960-894X(01)80995-1 BindingDB Entry DOI: 10.7270/Q2QC03DJ
TBA Curated by ChEMBL					More data for this Ligand-Target Pair
cGMP-dependent protein kinase 1 (Bos taurus (bovine))	BDBM50280879 (12,13-diethyl-6,7,12,13-tetrahydro-5H-indolo[2,3-a...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Patents Similars	Article	n/a	n/a	700	n/a	n/a	n/a	n/a	n/a	n/a
TBA Curated by ChEMBL					Assay Description In vitro for inhibitory activity against cGMP-dependent protein kinase from bovine lung (G-kinase)				Bioorg Med Chem Lett 3: 1959-1964 (1993) Article DOI: 10.1016/S0960-894X(01)80995-1 BindingDB Entry DOI: 10.7270/Q2QC03DJ
TBA Curated by ChEMBL					More data for this Ligand-Target Pair
cGMP-dependent protein kinase 1 (Bos taurus (bovine))	BDBM50280870 (12-(2,2-difluoroethyl)-13-methyl-6,7,12,13-tetrahy...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article	n/a	n/a	710	n/a	n/a	n/a	n/a	n/a	n/a
TBA Curated by ChEMBL					Assay Description In vitro for inhibitory activity against cGMP-dependent protein kinase from bovine lung (G-kinase)				Bioorg Med Chem Lett 3: 1959-1964 (1993) Article DOI: 10.1016/S0960-894X(01)80995-1 BindingDB Entry DOI: 10.7270/Q2QC03DJ
TBA Curated by ChEMBL					More data for this Ligand-Target Pair
cGMP-dependent protein kinase 1 (Bos taurus (bovine))	BDBM10841 (4-(6-bromo-1H-indol-3-yl)pyrimidin-2-amine \| Merid...) Show SMILES Nc1nccc(n1)-c1c[nH]c2cc(Br)ccc12 Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet	Purchase PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	800	n/a	n/a	n/a	n/a	n/a	30
CNRS					Assay Description Kinase activities were assayed in buffers containing substrate, enzyme, and inhibitor at 30°C in the presence of 15 uM ATP/[gamma-32P] ATP. 32P ...				Bioorg Med Chem Lett 14: 1703-7 (2004) Article DOI: 10.1016/j.bmcl.2004.01.050 BindingDB Entry DOI: 10.7270/Q2BZ648W
CNRS					More data for this Ligand-Target Pair
cGMP-dependent protein kinase 1 (Bos taurus (bovine))	BDBM3039 (23-[3-(dimethylamino)propyl]-3-methyl-3,13,23-tria...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet	PC cid PC sid UniChem Similars	Article	n/a	n/a	870	n/a	n/a	n/a	n/a	n/a	n/a
Tumor Biology Center					Assay Description The activity of cGPK, activated by cGMP, is measured by its ability to transfer phosphate from [gamma-32P]ATP to histone.				Bioorg Med Chem Lett 5: 55-60 (1995) Article DOI: 10.1016/0960-894X(94)00458-R BindingDB Entry DOI: 10.7270/Q2CF9N8C
Tumor Biology Center					More data for this Ligand-Target Pair
cGMP-dependent protein kinase 1 (Bos taurus (bovine))	BDBM3047 (4-{19-methoxy-23-methyl-12,14-dioxo-3,13,23-triaza...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet	PC cid PC sid UniChem Similars	Article	n/a	n/a	1.00E+3	n/a	n/a	n/a	n/a	n/a	n/a
Tumor Biology Center					Assay Description The activity of cGPK, activated by cGMP, is measured by its ability to transfer phosphate from [gamma-32P]ATP to histone.				Bioorg Med Chem Lett 5: 55-60 (1995) Article DOI: 10.1016/0960-894X(94)00458-R BindingDB Entry DOI: 10.7270/Q2CF9N8C
Tumor Biology Center					More data for this Ligand-Target Pair
cGMP-dependent protein kinase 1 (Bos taurus (bovine))	BDBM50284317 (3-(9-methoxy-13-methyl-5,7-dioxo-6,7,12,13-tetrahy...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article	n/a	n/a	1.00E+3	n/a	n/a	n/a	n/a	n/a	n/a
Tumor Biology Center					Assay Description Tested for inhibition of cGMP-dependent protein kinase from bovine lung				Bioorg Med Chem Lett 5: 55-60 (1995) Article DOI: 10.1016/0960-894X(94)00458-R BindingDB Entry DOI: 10.7270/Q2CF9N8C
Tumor Biology Center					More data for this Ligand-Target Pair
cGMP-dependent protein kinase 1 (Bos taurus (bovine))	BDBM10839 (3-(2-aminopyrimidin-4-yl)-6-bromo-1H-indol-4-ol \| ...) Show SMILES Nc1nccc(n1)-c1c[nH]c2cc(Br)cc(O)c12 Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet	PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	1.00E+3	n/a	n/a	n/a	n/a	n/a	30
CNRS					Assay Description Kinase activities were assayed in buffers containing substrate, enzyme, and inhibitor at 30°C in the presence of 15 uM ATP/[gamma-32P] ATP. 32P ...				Bioorg Med Chem Lett 14: 1703-7 (2004) Article DOI: 10.1016/j.bmcl.2004.01.050 BindingDB Entry DOI: 10.7270/Q2BZ648W
CNRS					More data for this Ligand-Target Pair
cGMP-dependent protein kinase 1 (Bos taurus (bovine))	BDBM50280873 (2-(13-ethyl-5-oxo-6,7,12,13-tetrahydro-5H-indolo[2...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article	n/a	n/a	1.30E+3	n/a	n/a	n/a	n/a	n/a	n/a
TBA Curated by ChEMBL					Assay Description In vitro for inhibitory activity against cGMP-dependent protein kinase from bovine lung (G-kinase)				Bioorg Med Chem Lett 3: 1959-1964 (1993) Article DOI: 10.1016/S0960-894X(01)80995-1 BindingDB Entry DOI: 10.7270/Q2QC03DJ
TBA Curated by ChEMBL					More data for this Ligand-Target Pair
cGMP-dependent protein kinase 1 (Bos taurus (bovine))	BDBM3034 (3-{7,19-dimethoxy-23-methyl-14-oxo-3,13,23-triazah...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet	Purchase PC cid PC sid UniChem Similars	Article	n/a	n/a	2.00E+3	n/a	n/a	n/a	n/a	n/a	n/a
Tumor Biology Center					Assay Description The activity of cGPK, activated by cGMP, is measured by its ability to transfer phosphate from [gamma-32P]ATP to histone.				Bioorg Med Chem Lett 5: 55-60 (1995) Article DOI: 10.1016/0960-894X(94)00458-R BindingDB Entry DOI: 10.7270/Q2CF9N8C
Tumor Biology Center					More data for this Ligand-Target Pair
cGMP-dependent protein kinase 1 (Bos taurus (bovine))	BDBM3048 (23-[3-(dimethylamino)-2-hydroxypropyl]-3-methyl-3,...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet	PC cid PC sid UniChem Similars	Article	n/a	n/a	2.10E+3	n/a	n/a	n/a	n/a	n/a	n/a
Tumor Biology Center					Assay Description The activity of cGPK, activated by cGMP, is measured by its ability to transfer phosphate from [gamma-32P]ATP to histone.				Bioorg Med Chem Lett 5: 55-60 (1995) Article DOI: 10.1016/0960-894X(94)00458-R BindingDB Entry DOI: 10.7270/Q2CF9N8C
Tumor Biology Center					More data for this Ligand-Target Pair
cGMP-dependent protein kinase 1 (Bos taurus (bovine))	BDBM3045 (3-{19-methoxy-23-methyl-12,14-dioxo-3,13,23-triaza...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet	PC cid PC sid UniChem Similars	Article	n/a	n/a	>3.00E+3	n/a	n/a	n/a	n/a	n/a	n/a
Tumor Biology Center					Assay Description The activity of cGPK, activated by cGMP, is measured by its ability to transfer phosphate from [gamma-32P]ATP to histone.				Bioorg Med Chem Lett 5: 55-60 (1995) Article DOI: 10.1016/0960-894X(94)00458-R BindingDB Entry DOI: 10.7270/Q2CF9N8C
Tumor Biology Center					More data for this Ligand-Target Pair
cGMP-dependent protein kinase 1 (Bos taurus (bovine))	BDBM3044 (3-{7-methoxy-23-methyl-12,14-dioxo-3,13,23-triazah...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet	PC cid PC sid UniChem Patents Similars	Article	n/a	n/a	>3.00E+3	n/a	n/a	n/a	n/a	n/a	n/a
Tumor Biology Center					Assay Description Tested for inhibition of cGMP-dependent protein kinase from bovine lung				Bioorg Med Chem Lett 5: 55-60 (1995) Article DOI: 10.1016/0960-894X(94)00458-R BindingDB Entry DOI: 10.7270/Q2CF9N8C
Tumor Biology Center					More data for this Ligand-Target Pair
cGMP-dependent protein kinase 1 (Bos taurus (bovine))	BDBM50284318 (13-(3-dimethylamino-2-hydroxypropyl)-3-methoxy-12-...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Patents Similars	Article	n/a	n/a	4.80E+3	n/a	n/a	n/a	n/a	n/a	n/a
Tumor Biology Center					Assay Description Tested for inhibition of cGMP-dependent protein kinase from bovine lung				Bioorg Med Chem Lett 5: 55-60 (1995) Article DOI: 10.1016/0960-894X(94)00458-R BindingDB Entry DOI: 10.7270/Q2CF9N8C
Tumor Biology Center					More data for this Ligand-Target Pair
cGMP-dependent protein kinase 1 (Bos taurus (bovine))	BDBM3049 (23-[3-(dimethylamino)-2-hydroxypropyl]-7-methoxy-3...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet	PC cid PC sid UniChem Similars	Article	n/a	n/a	4.80E+3	n/a	n/a	n/a	n/a	n/a	n/a
Tumor Biology Center					Assay Description The activity of cGPK, activated by cGMP, is measured by its ability to transfer phosphate from [gamma-32P]ATP to histone.				Bioorg Med Chem Lett 5: 55-60 (1995) Article DOI: 10.1016/0960-894X(94)00458-R BindingDB Entry DOI: 10.7270/Q2CF9N8C
Tumor Biology Center					More data for this Ligand-Target Pair
cGMP-dependent protein kinase 1 (Bos taurus (bovine))	BDBM50280869 (13-methyl-12-propyl-6,7,12,13-tetrahydro-5H-indolo...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article	n/a	n/a	5.10E+3	n/a	n/a	n/a	n/a	n/a	n/a
TBA Curated by ChEMBL					Assay Description In vitro for inhibitory activity against cGMP-dependent protein kinase from bovine lung (G-kinase)				Bioorg Med Chem Lett 3: 1959-1964 (1993) Article DOI: 10.1016/S0960-894X(01)80995-1 BindingDB Entry DOI: 10.7270/Q2QC03DJ
TBA Curated by ChEMBL					More data for this Ligand-Target Pair
cGMP-dependent protein kinase 1 (Bos taurus (bovine))	BDBM50280878 (12,13-dimethyl-6,7,12,13-tetrahydro-5H-indolo[2,3-...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article	n/a	n/a	5.50E+3	n/a	n/a	n/a	n/a	n/a	n/a
TBA Curated by ChEMBL					Assay Description In vitro for inhibitory activity against cGMP-dependent protein kinase from bovine lung (G-kinase)				Bioorg Med Chem Lett 3: 1959-1964 (1993) Article DOI: 10.1016/S0960-894X(01)80995-1 BindingDB Entry DOI: 10.7270/Q2QC03DJ
TBA Curated by ChEMBL					More data for this Ligand-Target Pair
cGMP-dependent protein kinase 1 (Bos taurus (bovine))	BDBM3033 (3-{23-methyl-14-oxo-3,13,23-triazahexacyclo[14.7.0...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet	Purchase CHEMBL MCE PC cid PC sid PDB UniChem Patents Similars	Article	n/a	n/a	6.20E+3	n/a	n/a	n/a	n/a	n/a	n/a
Tumor Biology Center					Assay Description The activity of cGPK, activated by cGMP, is measured by its ability to transfer phosphate from [gamma-32P]ATP to histone.				Bioorg Med Chem Lett 5: 55-60 (1995) Article DOI: 10.1016/0960-894X(94)00458-R BindingDB Entry DOI: 10.7270/Q2CF9N8C
Tumor Biology Center					More data for this Ligand-Target Pair
cGMP-dependent protein kinase 1 (Bos taurus (bovine))	BDBM3033 (3-{23-methyl-14-oxo-3,13,23-triazahexacyclo[14.7.0...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet	Purchase CHEMBL MCE PC cid PC sid PDB UniChem Patents Similars	Article	n/a	n/a	6.20E+3	n/a	n/a	n/a	n/a	n/a	n/a
TBA Curated by ChEMBL					Assay Description In vitro for inhibitory activity against cGMP-dependent protein kinase from bovine lung (G-kinase)				Bioorg Med Chem Lett 3: 1959-1964 (1993) Article DOI: 10.1016/S0960-894X(01)80995-1 BindingDB Entry DOI: 10.7270/Q2QC03DJ
TBA Curated by ChEMBL					More data for this Ligand-Target Pair
cGMP-dependent protein kinase 1 (Bos taurus (bovine))	BDBM3043 (3-{23-methyl-12,14-dioxo-3,13,23-triazahexacyclo[1...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet	Purchase PC cid PC sid UniChem Similars	Article	n/a	n/a	7.20E+3	n/a	n/a	n/a	n/a	n/a	n/a
Tumor Biology Center					Assay Description The activity of cGPK, activated by cGMP, is measured by its ability to transfer phosphate from [gamma-32P]ATP to histone.				Bioorg Med Chem Lett 5: 55-60 (1995) Article DOI: 10.1016/0960-894X(94)00458-R BindingDB Entry DOI: 10.7270/Q2CF9N8C
Tumor Biology Center					More data for this Ligand-Target Pair
cGMP-dependent protein kinase 1 (Bos taurus (bovine))	BDBM3041 (23-[3-(dimethylamino)-2-hydroxypropyl]-3-methyl-3,...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet	PC cid PC sid UniChem Patents Similars	Article	n/a	n/a	9.40E+3	n/a	n/a	n/a	n/a	n/a	n/a
Tumor Biology Center					Assay Description The activity of cGPK, activated by cGMP, is measured by its ability to transfer phosphate from [gamma-32P]ATP to histone.				Bioorg Med Chem Lett 5: 55-60 (1995) Article DOI: 10.1016/0960-894X(94)00458-R BindingDB Entry DOI: 10.7270/Q2CF9N8C
Tumor Biology Center					More data for this Ligand-Target Pair
cGMP-dependent protein kinase 1 (Bos taurus (bovine))	BDBM50280874 (3-(5-oxo-6,7,12,13-tetrahydro-5H-indolo[2,3-a]pyrr...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Patents Similars	Article	n/a	n/a	2.10E+4	n/a	n/a	n/a	n/a	n/a	n/a
TBA Curated by ChEMBL					Assay Description In vitro for inhibitory activity against cGMP-dependent protein kinase from bovine lung (G-kinase)				Bioorg Med Chem Lett 3: 1959-1964 (1993) Article DOI: 10.1016/S0960-894X(01)80995-1 BindingDB Entry DOI: 10.7270/Q2QC03DJ
TBA Curated by ChEMBL					More data for this Ligand-Target Pair
cGMP-dependent protein kinase 1 (Bos taurus (bovine))	BDBM50284316 (12-(3-dimethylamino-2-hydroxypropyl)-9-methoxy-13-...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article	n/a	n/a	2.30E+4	n/a	n/a	n/a	n/a	n/a	n/a
Tumor Biology Center					Assay Description Tested for inhibition of cGMP-dependent protein kinase from bovine lung				Bioorg Med Chem Lett 5: 55-60 (1995) Article DOI: 10.1016/0960-894X(94)00458-R BindingDB Entry DOI: 10.7270/Q2CF9N8C
Tumor Biology Center					More data for this Ligand-Target Pair
cGMP-dependent protein kinase 1 (Bos taurus (bovine))	BDBM3042 (23-[3-(dimethylamino)-2-hydroxypropyl]-7-methoxy-3...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet	PC cid PC sid UniChem Similars	Article	n/a	n/a	2.30E+4	n/a	n/a	n/a	n/a	n/a	n/a
Tumor Biology Center					Assay Description The activity of cGPK, activated by cGMP, is measured by its ability to transfer phosphate from [gamma-32P]ATP to histone.				Bioorg Med Chem Lett 5: 55-60 (1995) Article DOI: 10.1016/0960-894X(94)00458-R BindingDB Entry DOI: 10.7270/Q2CF9N8C
Tumor Biology Center					More data for this Ligand-Target Pair
cGMP-dependent protein kinase 1 (Bos taurus (bovine))	BDBM50280867 (2-(6,13-dimethyl-5-oxo-6,7,12,13-tetrahydro-5H-ind...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article	n/a	n/a	>3.00E+4	n/a	n/a	n/a	n/a	n/a	n/a
TBA Curated by ChEMBL					Assay Description In vitro for inhibitory activity against cGMP-dependent protein kinase from bovine lung (G-kinase)				Bioorg Med Chem Lett 3: 1959-1964 (1993) Article DOI: 10.1016/S0960-894X(01)80995-1 BindingDB Entry DOI: 10.7270/Q2QC03DJ
TBA Curated by ChEMBL					More data for this Ligand-Target Pair
cGMP-dependent protein kinase 1 (Bos taurus (bovine))	BDBM10838 (3-(2-aminopyrimidin-4-yl)-1H-indol-4-ol \| Meridian...) Show SMILES Nc1nccc(n1)-c1c[nH]c2cccc(O)c12 Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet	PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	2.00E+5	n/a	n/a	n/a	n/a	n/a	30
CNRS					Assay Description Kinase activities were assayed in buffers containing substrate, enzyme, and inhibitor at 30°C in the presence of 15 uM ATP/[gamma-32P] ATP. 32P ...				Bioorg Med Chem Lett 14: 1703-7 (2004) Article DOI: 10.1016/j.bmcl.2004.01.050 BindingDB Entry DOI: 10.7270/Q2BZ648W
CNRS					More data for this Ligand-Target Pair
cGMP-dependent protein kinase 1 (Bos taurus (bovine))	BDBM10844 (4-(1H-indol-3-yl)pyrimidin-2-amine \| Meridianin G) Show SMILES Nc1nccc(n1)-c1c[nH]c2ccccc12 Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet	Purchase MCE PC cid PC sid PDB UniChem Patents Similars	Article PubMed	n/a	n/a	4.00E+5	n/a	n/a	n/a	n/a	n/a	30
CNRS					Assay Description Kinase activities were assayed in buffers containing substrate, enzyme, and inhibitor at 30°C in the presence of 15 uM ATP/[gamma-32P] ATP. 32P ...				Bioorg Med Chem Lett 14: 1703-7 (2004) Article DOI: 10.1016/j.bmcl.2004.01.050 BindingDB Entry DOI: 10.7270/Q2BZ648W
CNRS					More data for this Ligand-Target Pair
cGMP-dependent protein kinase 1 (Bos taurus (bovine))	BDBM10845 (4-(5-bromo-1H-indol-2-yl)pyrimidin-2-amine \| isome...) Show SMILES Nc1nccc(n1)-c1cc2cc(Br)ccc2[nH]1 Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet	PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	>1.00E+6	n/a	n/a	n/a	n/a	n/a	30
CNRS					Assay Description Kinase activities were assayed in buffers containing substrate, enzyme, and inhibitor at 30°C in the presence of 15 uM ATP/[gamma-32P] ATP. 32P ...				Bioorg Med Chem Lett 14: 1703-7 (2004) Article DOI: 10.1016/j.bmcl.2004.01.050 BindingDB Entry DOI: 10.7270/Q2BZ648W
CNRS					More data for this Ligand-Target Pair
cGMP-dependent protein kinase 1 (Bos taurus (bovine))	BDBM10846 (4-(1H-indol-2-yl)pyrimidin-2-amine \| isomeridianin...) Show SMILES Nc1nccc(n1)-c1cc2ccccc2[nH]1 Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet	PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	1.00E+6	n/a	n/a	n/a	n/a	n/a	30
CNRS					Assay Description Kinase activities were assayed in buffers containing substrate, enzyme, and inhibitor at 30°C in the presence of 15 uM ATP/[gamma-32P] ATP. 32P ...				Bioorg Med Chem Lett 14: 1703-7 (2004) Article DOI: 10.1016/j.bmcl.2004.01.050 BindingDB Entry DOI: 10.7270/Q2BZ648W
CNRS					More data for this Ligand-Target Pair
cGMP-dependent protein kinase 1 (Bos taurus (bovine))	BDBM7533 ((2R)-2-[[6-(benzylamino)-9-isopropyl-purin-2-yl]am...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet	Purchase CHEMBL MCE MMDB PC cid PC sid PDB UniChem Patents Similars	Article PubMed	n/a	n/a	>1.00E+6	n/a	n/a	n/a	n/a	n/a	30
CNRS					Assay Description Kinase activities were assayed in buffers containing substrate, enzyme, and inhibitor at 30°C in the presence of 15 uM ATP/[gamma-32P] ATP. 32P ...				Bioorg Med Chem Lett 14: 1703-7 (2004) Article DOI: 10.1016/j.bmcl.2004.01.050 BindingDB Entry DOI: 10.7270/Q2BZ648W
CNRS					More data for this Ligand-Target Pair