Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kcal/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Endothelial lipase (Mus musculus (Mouse)) | BDBM50443626 (CHEMBL3092451) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | 4 | n/a | n/a | n/a | n/a | n/a | n/a |
Therachem Research Medilab (India) Pvt. Ltd. Curated by ChEMBL | Assay Description Inhibition of mouse endothelial lipase using PLAi as substrate measured for 30 mins by cell-based fluorescence assay | ACS Med Chem Lett 4: 1016-7 (2013) Article DOI: 10.1021/ml400361q BindingDB Entry DOI: 10.7270/Q22J6DBG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Endothelial lipase (Mus musculus (Mouse)) | BDBM199225 (US9216998, 8) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 4 | n/a | n/a | n/a | n/a | 7.2 | n/a |
Janssen Pharmaceutica NV US Patent | Assay Description To assay for cell surface lipase activity, cells expressing human endothelial lipase (EL) or LPL were plated in CellBIND® 384-well plates (Corning, L... | US Patent US9216998 (2015) BindingDB Entry DOI: 10.7270/Q22N513F | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Endothelial lipase (Mus musculus (Mouse)) | BDBM50443627 (CHEMBL3092450 | US9216998, 5) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | US Patent | n/a | n/a | 17 | n/a | n/a | n/a | n/a | 7.2 | n/a |
Janssen Pharmaceutica NV US Patent | Assay Description To assay for cell surface lipase activity, cells expressing human endothelial lipase (EL) or LPL were plated in CellBIND® 384-well plates (Corning, L... | US Patent US9216998 (2015) BindingDB Entry DOI: 10.7270/Q22N513F | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Endothelial lipase (Mus musculus (Mouse)) | BDBM50443627 (CHEMBL3092450 | US9216998, 5) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | 17 | n/a | n/a | n/a | n/a | n/a | n/a |
Therachem Research Medilab (India) Pvt. Ltd. Curated by ChEMBL | Assay Description Inhibition of mouse endothelial lipase using PLAi as substrate measured for 30 mins by cell-based fluorescence assay | ACS Med Chem Lett 4: 1016-7 (2013) Article DOI: 10.1021/ml400361q BindingDB Entry DOI: 10.7270/Q22J6DBG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Endothelial lipase (Mus musculus (Mouse)) | BDBM199219 (US9216998, 7 | US9216998, Reference Compound 2) | UniProtKB/SwissProt GoogleScholar AffyNet | Purchase PC cid PC sid UniChem | US Patent | n/a | n/a | 26 | n/a | n/a | n/a | n/a | 7.2 | n/a |
Janssen Pharmaceutica NV US Patent | Assay Description To assay for cell surface lipase activity, cells expressing human endothelial lipase (EL) or LPL were plated in CellBIND® 384-well plates (Corning, L... | US Patent US9216998 (2015) BindingDB Entry DOI: 10.7270/Q22N513F | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Endothelial lipase (Mus musculus (Mouse)) | BDBM50443625 (CHEMBL3092448 | US9216998, 25) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | US Patent | n/a | n/a | 31 | n/a | n/a | n/a | n/a | 7.2 | n/a |
Janssen Pharmaceutica NV US Patent | Assay Description To assay for cell surface lipase activity, cells expressing human endothelial lipase (EL) or LPL were plated in CellBIND® 384-well plates (Corning, L... | US Patent US9216998 (2015) BindingDB Entry DOI: 10.7270/Q22N513F | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Endothelial lipase (Mus musculus (Mouse)) | BDBM50443625 (CHEMBL3092448 | US9216998, 25) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | 31 | n/a | n/a | n/a | n/a | n/a | n/a |
Therachem Research Medilab (India) Pvt. Ltd. Curated by ChEMBL | Assay Description Inhibition of mouse endothelial lipase using PLAi as substrate measured for 30 mins by cell-based fluorescence assay | ACS Med Chem Lett 4: 1016-7 (2013) Article DOI: 10.1021/ml400361q BindingDB Entry DOI: 10.7270/Q22J6DBG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Endothelial lipase (Mus musculus (Mouse)) | BDBM50443625 (CHEMBL3092448 | US9216998, 25) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | 31 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Calabria Curated by ChEMBL | Assay Description Inhibition of endothelial lipase in mouse cells after 30 mins by fluorescence assay | Eur J Med Chem 151: 121-144 (2018) Article DOI: 10.1016/j.ejmech.2018.03.061 BindingDB Entry DOI: 10.7270/Q2HM5C4Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Endothelial lipase (Mus musculus (Mouse)) | BDBM199205 (US9216998, 9) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 36 | n/a | n/a | n/a | n/a | 7.2 | n/a |
Janssen Pharmaceutica NV US Patent | Assay Description To assay for cell surface lipase activity, cells expressing human endothelial lipase (EL) or LPL were plated in CellBIND® 384-well plates (Corning, L... | US Patent US9216998 (2015) BindingDB Entry DOI: 10.7270/Q22N513F | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Endothelial lipase (Mus musculus (Mouse)) | BDBM199219 (US9216998, 7 | US9216998, Reference Compound 2) | UniProtKB/SwissProt GoogleScholar AffyNet | Purchase PC cid PC sid UniChem | US Patent | n/a | n/a | 48 | n/a | n/a | n/a | n/a | 7.2 | n/a |
Janssen Pharmaceutica NV US Patent | Assay Description To assay for cell surface lipase activity, cells expressing human endothelial lipase (EL) or LPL were plated in CellBIND® 384-well plates (Corning, L... | US Patent US9216998 (2015) BindingDB Entry DOI: 10.7270/Q22N513F | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Endothelial lipase (Mus musculus (Mouse)) | BDBM199226 (US9216998, 10) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 75 | n/a | n/a | n/a | n/a | 7.2 | n/a |
Janssen Pharmaceutica NV US Patent | Assay Description To assay for cell surface lipase activity, cells expressing human endothelial lipase (EL) or LPL were plated in CellBIND® 384-well plates (Corning, L... | US Patent US9216998 (2015) BindingDB Entry DOI: 10.7270/Q22N513F | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Endothelial lipase (Mus musculus (Mouse)) | BDBM199207 (US9216998, 19) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 87 | n/a | n/a | n/a | n/a | 7.2 | n/a |
Janssen Pharmaceutica NV US Patent | Assay Description To assay for cell surface lipase activity, cells expressing human endothelial lipase (EL) or LPL were plated in CellBIND® 384-well plates (Corning, L... | US Patent US9216998 (2015) BindingDB Entry DOI: 10.7270/Q22N513F | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Endothelial lipase (Mus musculus (Mouse)) | BDBM50522804 (CHEMBL4437751) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 94 | n/a | n/a | n/a | n/a | n/a | n/a |
Bristol-Myers Squibb Curated by ChEMBL | Assay Description Inhibition of mouse endothelial lipase expressed in HEK293F cells using D31-POPC-HDL as substrate incubated for 2 hrs in presence of mouse plasma by ... | Bioorg Med Chem Lett 29: 1918-1921 (2019) Article DOI: 10.1016/j.bmcl.2019.05.048 BindingDB Entry DOI: 10.7270/Q2JH3QMN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Endothelial lipase (Mus musculus (Mouse)) | BDBM199221 (US9216998, 3) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 96 | n/a | n/a | n/a | n/a | 7.2 | n/a |
Janssen Pharmaceutica NV US Patent | Assay Description To assay for cell surface lipase activity, cells expressing human endothelial lipase (EL) or LPL were plated in CellBIND® 384-well plates (Corning, L... | US Patent US9216998 (2015) BindingDB Entry DOI: 10.7270/Q22N513F | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Endothelial lipase (Mus musculus (Mouse)) | BDBM50458640 (CHEMBL4203934) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 100 | n/a | n/a | n/a | n/a | n/a | n/a |
Bristol-Myers Squibb Curated by ChEMBL | Assay Description Inhibition of recombinant mouse endothelial lipase expressed in HEK293F cells using HDL as substrate pretreated for 10 mins followed by substrate add... | ACS Med Chem Lett 9: 673-678 (2018) Article DOI: 10.1021/acsmedchemlett.8b00138 BindingDB Entry DOI: 10.7270/Q2JS9T2R | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Endothelial lipase (Mus musculus (Mouse)) | BDBM50522808 (CHEMBL4520847) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 100 | n/a | n/a | n/a | n/a | n/a | n/a |
Bristol-Myers Squibb Curated by ChEMBL | Assay Description Inhibition of mouse endothelial lipase expressed in HEK293F cells using D31-POPC-HDL as substrate incubated for 2 hrs in presence of mouse plasma by ... | Bioorg Med Chem Lett 29: 1918-1921 (2019) Article DOI: 10.1016/j.bmcl.2019.05.048 BindingDB Entry DOI: 10.7270/Q2JH3QMN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Endothelial lipase (Mus musculus (Mouse)) | BDBM199229 (US9216998, 27) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 108 | n/a | n/a | n/a | n/a | 7.2 | n/a |
Janssen Pharmaceutica NV US Patent | Assay Description To assay for cell surface lipase activity, cells expressing human endothelial lipase (EL) or LPL were plated in CellBIND® 384-well plates (Corning, L... | US Patent US9216998 (2015) BindingDB Entry DOI: 10.7270/Q22N513F | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Endothelial lipase (Mus musculus (Mouse)) | BDBM50522805 (CHEMBL4514272) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 120 | n/a | n/a | n/a | n/a | n/a | n/a |
Bristol-Myers Squibb Curated by ChEMBL | Assay Description Inhibition of mouse endothelial lipase expressed in HEK293F cells using D31-POPC-HDL as substrate incubated for 2 hrs in presence of mouse plasma by ... | Bioorg Med Chem Lett 29: 1918-1921 (2019) Article DOI: 10.1016/j.bmcl.2019.05.048 BindingDB Entry DOI: 10.7270/Q2JH3QMN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Endothelial lipase (Mus musculus (Mouse)) | BDBM199209 (US9216998, 13) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 124 | n/a | n/a | n/a | n/a | 7.2 | n/a |
Janssen Pharmaceutica NV US Patent | Assay Description To assay for cell surface lipase activity, cells expressing human endothelial lipase (EL) or LPL were plated in CellBIND® 384-well plates (Corning, L... | US Patent US9216998 (2015) BindingDB Entry DOI: 10.7270/Q22N513F | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Endothelial lipase (Mus musculus (Mouse)) | BDBM199208 (US9216998, 12) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 131 | n/a | n/a | n/a | n/a | 7.2 | n/a |
Janssen Pharmaceutica NV US Patent | Assay Description To assay for cell surface lipase activity, cells expressing human endothelial lipase (EL) or LPL were plated in CellBIND® 384-well plates (Corning, L... | US Patent US9216998 (2015) BindingDB Entry DOI: 10.7270/Q22N513F | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Endothelial lipase (Mus musculus (Mouse)) | BDBM199223 (US9216998, 6) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 136 | n/a | n/a | n/a | n/a | 7.2 | n/a |
Janssen Pharmaceutica NV US Patent | Assay Description To assay for cell surface lipase activity, cells expressing human endothelial lipase (EL) or LPL were plated in CellBIND® 384-well plates (Corning, L... | US Patent US9216998 (2015) BindingDB Entry DOI: 10.7270/Q22N513F | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Endothelial lipase (Mus musculus (Mouse)) | BDBM199216 (US9216998, 22) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 142 | n/a | n/a | n/a | n/a | 7.2 | n/a |
Janssen Pharmaceutica NV US Patent | Assay Description To assay for cell surface lipase activity, cells expressing human endothelial lipase (EL) or LPL were plated in CellBIND® 384-well plates (Corning, L... | US Patent US9216998 (2015) BindingDB Entry DOI: 10.7270/Q22N513F | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Endothelial lipase (Mus musculus (Mouse)) | BDBM199210 (US9216998, 14) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 162 | n/a | n/a | n/a | n/a | 7.2 | n/a |
Janssen Pharmaceutica NV US Patent | Assay Description To assay for cell surface lipase activity, cells expressing human endothelial lipase (EL) or LPL were plated in CellBIND® 384-well plates (Corning, L... | US Patent US9216998 (2015) BindingDB Entry DOI: 10.7270/Q22N513F | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Endothelial lipase (Mus musculus (Mouse)) | BDBM151238 (US8987314, B34) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 190 | n/a | n/a | n/a | n/a | n/a | n/a |
Bristol-Myers Squibb Curated by ChEMBL | Assay Description Inhibition of mouse endothelial lipase expressed in HEK293F cells using D31-POPC-HDL as substrate incubated for 2 hrs in presence of mouse plasma by ... | Bioorg Med Chem Lett 29: 1918-1921 (2019) Article DOI: 10.1016/j.bmcl.2019.05.048 BindingDB Entry DOI: 10.7270/Q2JH3QMN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Endothelial lipase (Mus musculus (Mouse)) | BDBM199220 (US9216998, 1) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 195 | n/a | n/a | n/a | n/a | 7.2 | n/a |
Janssen Pharmaceutica NV US Patent | Assay Description To assay for cell surface lipase activity, cells expressing human endothelial lipase (EL) or LPL were plated in CellBIND® 384-well plates (Corning, L... | US Patent US9216998 (2015) BindingDB Entry DOI: 10.7270/Q22N513F | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Endothelial lipase (Mus musculus (Mouse)) | BDBM50506505 (CHEMBL4460376) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 200 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Inhibition of endothelial lipase in hepatic lipase knock-out mouse plasma | J Med Chem 63: 1660-1670 (2020) Article DOI: 10.1021/acs.jmedchem.9b01831 BindingDB Entry DOI: 10.7270/Q28G8PZS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Endothelial lipase (Mus musculus (Mouse)) | BDBM50506504 (CHEMBL4460663) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 200 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Inhibition of endothelial lipase in hepatic lipase knock-out mouse plasma | J Med Chem 63: 1660-1670 (2020) Article DOI: 10.1021/acs.jmedchem.9b01831 BindingDB Entry DOI: 10.7270/Q28G8PZS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Endothelial lipase (Mus musculus (Mouse)) | BDBM151212 (US8987314, B3) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 200 | n/a | n/a | n/a | n/a | n/a | n/a |
Bristol-Myers Squibb Curated by ChEMBL | Assay Description Inhibition of mouse endothelial lipase expressed in HEK293F cells using D31-POPC-HDL as substrate incubated for 2 hrs in presence of mouse plasma by ... | Bioorg Med Chem Lett 29: 1918-1921 (2019) Article DOI: 10.1016/j.bmcl.2019.05.048 BindingDB Entry DOI: 10.7270/Q2JH3QMN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Endothelial lipase (Mus musculus (Mouse)) | BDBM50506498 (CHEMBL4581886) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 200 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Inhibition of endothelial lipase in hepatic lipase knock-out mouse plasma | J Med Chem 63: 1660-1670 (2020) Article DOI: 10.1021/acs.jmedchem.9b01831 BindingDB Entry DOI: 10.7270/Q28G8PZS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Endothelial lipase (Mus musculus (Mouse)) | BDBM50506506 (CHEMBL4465833) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 200 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Inhibition of endothelial lipase in hepatic lipase knock-out mouse plasma | J Med Chem 63: 1660-1670 (2020) Article DOI: 10.1021/acs.jmedchem.9b01831 BindingDB Entry DOI: 10.7270/Q28G8PZS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Endothelial lipase (Mus musculus (Mouse)) | BDBM199222 (US9216998, 4) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 205 | n/a | n/a | n/a | n/a | 7.2 | n/a |
Janssen Pharmaceutica NV US Patent | Assay Description To assay for cell surface lipase activity, cells expressing human endothelial lipase (EL) or LPL were plated in CellBIND® 384-well plates (Corning, L... | US Patent US9216998 (2015) BindingDB Entry DOI: 10.7270/Q22N513F | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Endothelial lipase (Mus musculus (Mouse)) | BDBM199215 (US9216998, 21) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 237 | n/a | n/a | n/a | n/a | 7.2 | n/a |
Janssen Pharmaceutica NV US Patent | Assay Description To assay for cell surface lipase activity, cells expressing human endothelial lipase (EL) or LPL were plated in CellBIND® 384-well plates (Corning, L... | US Patent US9216998 (2015) BindingDB Entry DOI: 10.7270/Q22N513F | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Endothelial lipase (Mus musculus (Mouse)) | BDBM319015 (N-[(cyclopropyl- carbamoyl) methyl]-2-[6-(6- fluor...) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 290 | n/a | n/a | n/a | n/a | n/a | n/a |
Bristol-Myers Squibb Curated by ChEMBL | Assay Description Inhibition of mouse endothelial lipase expressed in HEK293F cells using D31-POPC-HDL as substrate incubated for 2 hrs in presence of mouse plasma by ... | Bioorg Med Chem Lett 29: 1918-1921 (2019) Article DOI: 10.1016/j.bmcl.2019.05.048 BindingDB Entry DOI: 10.7270/Q2JH3QMN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Endothelial lipase (Mus musculus (Mouse)) | BDBM50522805 (CHEMBL4514272) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 310 | n/a | n/a | n/a | n/a | n/a | n/a |
Bristol-Myers Squibb Curated by ChEMBL | Assay Description Inhibition of endothelial lipase in hepatic lipase knock-out mouse plasma using D31-POPC-HDL as substrate incubated for 2 hrs by LC/MS analysis | Bioorg Med Chem Lett 29: 1918-1921 (2019) Article DOI: 10.1016/j.bmcl.2019.05.048 BindingDB Entry DOI: 10.7270/Q2JH3QMN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Endothelial lipase (Mus musculus (Mouse)) | BDBM151303 (US8987314, B101) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 320 | n/a | n/a | n/a | n/a | n/a | n/a |
Bristol-Myers Squibb Curated by ChEMBL | Assay Description Inhibition of mouse endothelial lipase expressed in HEK293F cells using D31-POPC-HDL as substrate incubated for 2 hrs in presence of mouse plasma by ... | Bioorg Med Chem Lett 29: 1918-1921 (2019) Article DOI: 10.1016/j.bmcl.2019.05.048 BindingDB Entry DOI: 10.7270/Q2JH3QMN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Endothelial lipase (Mus musculus (Mouse)) | BDBM199218 (US9216998, 24) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 340 | n/a | n/a | n/a | n/a | 7.2 | n/a |
Janssen Pharmaceutica NV US Patent | Assay Description To assay for cell surface lipase activity, cells expressing human endothelial lipase (EL) or LPL were plated in CellBIND® 384-well plates (Corning, L... | US Patent US9216998 (2015) BindingDB Entry DOI: 10.7270/Q22N513F | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Endothelial lipase (Mus musculus (Mouse)) | BDBM199217 (US9216998, 23) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 346 | n/a | n/a | n/a | n/a | 7.2 | n/a |
Janssen Pharmaceutica NV US Patent | Assay Description To assay for cell surface lipase activity, cells expressing human endothelial lipase (EL) or LPL were plated in CellBIND® 384-well plates (Corning, L... | US Patent US9216998 (2015) BindingDB Entry DOI: 10.7270/Q22N513F | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Endothelial lipase (Mus musculus (Mouse)) | BDBM50433475 (CHEMBL2381067) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | 470 | n/a | n/a | n/a | n/a | n/a | n/a |
Janssen Research and Development, LLC Curated by ChEMBL | Assay Description Inhibition of mouse EL expressed in HEK293 cells using PED-A1 as substrate by spectrophotometry | Bioorg Med Chem Lett 23: 2595-7 (2013) Article DOI: 10.1016/j.bmcl.2013.02.113 BindingDB Entry DOI: 10.7270/Q24T6KQV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Endothelial lipase (Mus musculus (Mouse)) | BDBM199214 (US9216998, 20) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 479 | n/a | n/a | n/a | n/a | 7.2 | n/a |
Janssen Pharmaceutica NV US Patent | Assay Description To assay for cell surface lipase activity, cells expressing human endothelial lipase (EL) or LPL were plated in CellBIND® 384-well plates (Corning, L... | US Patent US9216998 (2015) BindingDB Entry DOI: 10.7270/Q22N513F | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Endothelial lipase (Mus musculus (Mouse)) | BDBM319014 (N-[(cyclopropyl- carbamoyl) methyl]-2-[6-(6- fluor...) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 600 | n/a | n/a | n/a | n/a | n/a | n/a |
Bristol-Myers Squibb Curated by ChEMBL | Assay Description Inhibition of mouse endothelial lipase expressed in HEK293F cells using D31-POPC-HDL as substrate incubated for 2 hrs in presence of mouse plasma by ... | Bioorg Med Chem Lett 29: 1918-1921 (2019) Article DOI: 10.1016/j.bmcl.2019.05.048 BindingDB Entry DOI: 10.7270/Q2JH3QMN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Endothelial lipase (Mus musculus (Mouse)) | BDBM199228 (US9216998, 26) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 618 | n/a | n/a | n/a | n/a | 7.2 | n/a |
Janssen Pharmaceutica NV US Patent | Assay Description To assay for cell surface lipase activity, cells expressing human endothelial lipase (EL) or LPL were plated in CellBIND® 384-well plates (Corning, L... | US Patent US9216998 (2015) BindingDB Entry DOI: 10.7270/Q22N513F | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Endothelial lipase (Mus musculus (Mouse)) | BDBM199206 (US9216998, 15) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 677 | n/a | n/a | n/a | n/a | 7.2 | n/a |
Janssen Pharmaceutica NV US Patent | Assay Description To assay for cell surface lipase activity, cells expressing human endothelial lipase (EL) or LPL were plated in CellBIND® 384-well plates (Corning, L... | US Patent US9216998 (2015) BindingDB Entry DOI: 10.7270/Q22N513F | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Endothelial lipase (Mus musculus (Mouse)) | BDBM50433472 (CHEMBL2381069) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | 680 | n/a | n/a | n/a | n/a | n/a | n/a |
Janssen Research and Development, LLC Curated by ChEMBL | Assay Description Inhibition of mouse EL expressed in HEK293 cells using PED-A1 as substrate by spectrophotometry | Bioorg Med Chem Lett 23: 2595-7 (2013) Article DOI: 10.1016/j.bmcl.2013.02.113 BindingDB Entry DOI: 10.7270/Q24T6KQV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Endothelial lipase (Mus musculus (Mouse)) | BDBM199211 (US9216998, 16) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 1.00E+3 | n/a | n/a | n/a | n/a | 7.2 | n/a |
Janssen Pharmaceutica NV US Patent | Assay Description To assay for cell surface lipase activity, cells expressing human endothelial lipase (EL) or LPL were plated in CellBIND® 384-well plates (Corning, L... | US Patent US9216998 (2015) BindingDB Entry DOI: 10.7270/Q22N513F | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Endothelial lipase (Mus musculus (Mouse)) | BDBM199227 (US9216998, 11) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 1.20E+3 | n/a | n/a | n/a | n/a | 7.2 | n/a |
Janssen Pharmaceutica NV US Patent | Assay Description To assay for cell surface lipase activity, cells expressing human endothelial lipase (EL) or LPL were plated in CellBIND® 384-well plates (Corning, L... | US Patent US9216998 (2015) BindingDB Entry DOI: 10.7270/Q22N513F | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Endothelial lipase (Mus musculus (Mouse)) | BDBM199213 (US9216998, 18) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 1.89E+3 | n/a | n/a | n/a | n/a | 7.2 | n/a |
Janssen Pharmaceutica NV US Patent | Assay Description To assay for cell surface lipase activity, cells expressing human endothelial lipase (EL) or LPL were plated in CellBIND® 384-well plates (Corning, L... | US Patent US9216998 (2015) BindingDB Entry DOI: 10.7270/Q22N513F | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Endothelial lipase (Mus musculus (Mouse)) | BDBM199212 (US9216998, 17) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 3.62E+3 | n/a | n/a | n/a | n/a | 7.2 | n/a |
Janssen Pharmaceutica NV US Patent | Assay Description To assay for cell surface lipase activity, cells expressing human endothelial lipase (EL) or LPL were plated in CellBIND® 384-well plates (Corning, L... | US Patent US9216998 (2015) BindingDB Entry DOI: 10.7270/Q22N513F | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Endothelial lipase (Mus musculus (Mouse)) | BDBM50522805 (CHEMBL4514272) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 2.60E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Bristol-Myers Squibb Curated by ChEMBL | Assay Description Inhibition of hepatic lipase in endothelial lipase knock-out mouse plasma using D31-POPC-HDL as substrate incubated for 2 hrs by LC/MS analysis | Bioorg Med Chem Lett 29: 1918-1921 (2019) Article DOI: 10.1016/j.bmcl.2019.05.048 BindingDB Entry DOI: 10.7270/Q2JH3QMN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Endothelial lipase (Mus musculus (Mouse)) | BDBM50433474 (CHEMBL2381068) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | >3.30E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Janssen Research and Development, LLC Curated by ChEMBL | Assay Description Inhibition of mouse EL expressed in HEK293 cells using PED-A1 as substrate by spectrophotometry | Bioorg Med Chem Lett 23: 2595-7 (2013) Article DOI: 10.1016/j.bmcl.2013.02.113 BindingDB Entry DOI: 10.7270/Q24T6KQV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Endothelial lipase (Mus musculus (Mouse)) | BDBM50443624 (CHEMBL3092449 | US9216998, 28) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | US Patent | n/a | n/a | 3.33E+4 | n/a | n/a | n/a | n/a | 7.2 | n/a |
Janssen Pharmaceutica NV US Patent | Assay Description To assay for cell surface lipase activity, cells expressing human endothelial lipase (EL) or LPL were plated in CellBIND® 384-well plates (Corning, L... | US Patent US9216998 (2015) BindingDB Entry DOI: 10.7270/Q22N513F | |||||||||||
More data for this Ligand-Target Pair |
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