Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kcal/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Taste receptor type 2 member 14 (Homo sapiens (Human)) | BDBM50044849 (CHEMBL3311308) | UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | <1.00E+4 | n/a | n/a | n/a | n/a |
GlaxoSmithKline Curated by ChEMBL | Assay Description Agonist activity at human TAS2R14 expressed in U2OS cells by Ga16gust44 Clone 7A FLIPR/summary (Abse5) assay | Bioorg Med Chem Lett 24: 3100-3 (2014) Article DOI: 10.1016/j.bmcl.2014.05.012 BindingDB Entry DOI: 10.7270/Q2CC1292 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Taste receptor type 2 member 14 (Homo sapiens (Human)) | BDBM211262 (US9247759, 10-10) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 4.00E+4 | n/a | n/a | n/a | n/a |
Firmenich SA Curated by ChEMBL | Assay Description Agonist activity at TAS2R14 (unknown origin) by stably expressed cell-based assay | J Med Chem 63: 4957-4977 (2020) Article DOI: 10.1021/acs.jmedchem.0c00388 BindingDB Entry DOI: 10.7270/Q2VH5S56 | |||||||||||
More data for this Ligand-Target Pair |