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Compile Data Set for Download or QSAR

Found 1067 hits of ic50 for UniProtKB: O14744   
Target/Host
(Institution)
LigandTarget/Host
Links
Ligand
Links
Trg + Lig
Links
Ki
nM
ΔG°
kcal/mole
IC50
nM
Kd
nM
EC50/IC50
nM
koff
s-1
kon
M-1s-1
pHTemp
°C
Protein arginine N-methyltransferase 5


(Homo sapiens (Human))
BDBM364153
PNG
(US9856252, 45)
PDB

UniProtKB/SwissProt

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n/an/a 83n/an/an/an/an/an/a



Bristol-Myers Squibb Company





J Med Chem 49: 2440-55 (2006)

More data for this
Ligand-Target Pair
Protein arginine N-methyltransferase 5


(Homo sapiens (Human))
BDBM337050
PNG
(US9745291, Compound 96 | US9765068, Compound 96)
Show SMILES CN1CCC(C1)n1ncc2cc(OCC(=O)NCC(O)CN3CCc4ccccc4C3)ccc12
PDB

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US Patent
n/an/a<100n/an/an/an/an/an/a



Epizyme, Inc.

US Patent




US Patent US9765068 (2017)


BindingDB Entry DOI: 10.7270/Q2959KN3
More data for this
Ligand-Target Pair
Protein arginine N-methyltransferase 5


(Homo sapiens (Human))
BDBM337052
PNG
(US9745291, Compound 98 | US9765068, Compound 98)
Show SMILES COc1ccc2cccc(OCC(=O)NC[C@@H](O)CN3CCc4ccccc4C3)c2n1 |r|
PDB

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n/an/a<100n/an/an/an/an/an/a



Epizyme, Inc.

US Patent




US Patent US9765068 (2017)


BindingDB Entry DOI: 10.7270/Q2959KN3
More data for this
Ligand-Target Pair
Protein arginine N-methyltransferase 5


(Homo sapiens (Human))
BDBM337053
PNG
(US9745291, Compound 99 | US9765068, Compound 99)
Show SMILES CN1CCc2c(C1)cccc2OCC(=O)NCC(O)CN1CCc2ccccc2C1
PDB

UniProtKB/SwissProt

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n/an/a<100n/an/an/an/an/an/a



Epizyme, Inc.

US Patent




US Patent US9765068 (2017)


BindingDB Entry DOI: 10.7270/Q2959KN3
More data for this
Ligand-Target Pair
Protein arginine N-methyltransferase 5


(Homo sapiens (Human))
BDBM337054
PNG
(US9745291, Compound 100 | US9765068, Compound 100)
Show SMILES OC(CNC(=O)COc1cccc2OCCOc12)CN1CCc2ccccc2C1
PDB

UniProtKB/SwissProt

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n/an/a<100n/an/an/an/an/an/a



Epizyme, Inc.

US Patent




US Patent US9765068 (2017)


BindingDB Entry DOI: 10.7270/Q2959KN3
More data for this
Ligand-Target Pair
Protein arginine N-methyltransferase 5


(Homo sapiens (Human))
BDBM337055
PNG
(US9745291, Compound 101 | US9765068, Compound 101)
Show SMILES CC(=O)N1CCc2c(C1)cccc2OCC(=O)NCC(O)CN1CCc2ccccc2C1
PDB

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n/an/a<100n/an/an/an/an/an/a



Epizyme, Inc.

US Patent




US Patent US9765068 (2017)


BindingDB Entry DOI: 10.7270/Q2959KN3
More data for this
Ligand-Target Pair
Protein arginine N-methyltransferase 5


(Homo sapiens (Human))
BDBM337056
PNG
(US9745291, Compound 102 | US9765068, Compound 102)
Show SMILES CS(=O)(=O)N1CCc2c(C1)cccc2OCC(=O)NCC(O)CN1CCc2ccccc2C1
PDB

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n/an/a<100n/an/an/an/an/an/a



Epizyme, Inc.

US Patent




US Patent US9765068 (2017)


BindingDB Entry DOI: 10.7270/Q2959KN3
More data for this
Ligand-Target Pair
Protein arginine N-methyltransferase 5


(Homo sapiens (Human))
BDBM337057
PNG
(US9745291, Compound 103 | US9765068, Compound 103)
Show SMILES OC(CNC(=O)COc1ccccc1C1CCNCC1)CN1CCc2ccccc2C1
PDB

UniProtKB/SwissProt

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n/an/a<100n/an/an/an/an/an/a



Epizyme, Inc.

US Patent




US Patent US9765068 (2017)


BindingDB Entry DOI: 10.7270/Q2959KN3
More data for this
Ligand-Target Pair
Protein arginine N-methyltransferase 5


(Homo sapiens (Human))
BDBM337059
PNG
(US9745291, Compound 105 | US9765068, Compound 105)
Show SMILES CN(C)c1ccc2cccc(OCC(=O)NC[C@@H](O)CN3CCc4ccccc4C3)c2n1 |r|
PDB

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n/an/a<100n/an/an/an/an/an/a



Epizyme, Inc.

US Patent




US Patent US9765068 (2017)


BindingDB Entry DOI: 10.7270/Q2959KN3
More data for this
Ligand-Target Pair
Protein arginine N-methyltransferase 5


(Homo sapiens (Human))
BDBM337061
PNG
(US9745291, Compound 107 | US9765068, Compound 107)
Show SMILES OC(CNC(=O)COc1ccccc1S(=O)(=O)N1CCNCC1)CN1CCc2ccccc2C1
PDB

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n/an/a<100n/an/an/an/an/an/a



Epizyme, Inc.

US Patent




US Patent US9765068 (2017)


BindingDB Entry DOI: 10.7270/Q2959KN3
More data for this
Ligand-Target Pair
Protein arginine N-methyltransferase 5


(Homo sapiens (Human))
BDBM337062
PNG
(US9745291, Compound 108 | US9765068, Compound 108)
Show SMILES CN1CCN(CC1)S(=O)(=O)c1ccccc1OCC(=O)NCC(O)CN1CCc2ccccc2C1
PDB

UniProtKB/SwissProt

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n/an/a<100n/an/an/an/an/an/a



Epizyme, Inc.

US Patent




US Patent US9765068 (2017)


BindingDB Entry DOI: 10.7270/Q2959KN3
More data for this
Ligand-Target Pair
Protein arginine N-methyltransferase 5


(Homo sapiens (Human))
BDBM337063
PNG
(US9745291, Compound 109 | US9765068, Compound 109)
Show SMILES CN(C)S(=O)(=O)c1ccccc1OCC(=O)NCC(O)CN1CCc2ccccc2C1
PDB

UniProtKB/SwissProt

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n/an/a<100n/an/an/an/an/an/a



Epizyme, Inc.

US Patent




US Patent US9765068 (2017)


BindingDB Entry DOI: 10.7270/Q2959KN3
More data for this
Ligand-Target Pair
Protein arginine N-methyltransferase 5


(Homo sapiens (Human))
BDBM337064
PNG
(US9745291, Compound 110 | US9765068, Compound 110)
Show SMILES OC(CNC(=O)COc1ccccc1S(=O)(=O)N1CCCC1)CN1CCc2ccccc2C1
PDB

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n/an/a<100n/an/an/an/an/an/a



Epizyme, Inc.

US Patent




US Patent US9765068 (2017)


BindingDB Entry DOI: 10.7270/Q2959KN3
More data for this
Ligand-Target Pair
Protein arginine N-methyltransferase 5


(Homo sapiens (Human))
BDBM337065
PNG
(US9745291, Compound 111 | US9765068, Compound 111)
Show SMILES OC(CNC(=O)COc1ccccc1S(=O)(=O)N1CCC(O)C1)CN1CCc2ccccc2C1
PDB

UniProtKB/SwissProt

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n/an/a<100n/an/an/an/an/an/a



Epizyme, Inc.

US Patent




US Patent US9765068 (2017)


BindingDB Entry DOI: 10.7270/Q2959KN3
More data for this
Ligand-Target Pair
PRMT5/MEP50 Enzyme


(Homo sapiens (Human))
BDBM343957
PNG
(1-(3,4-dihydroisoquinolin-2(1H)-yl)-3-((4-(1-(tetr...)
Show SMILES OC(CNc1cc(ccn1)-c1ccc2ncn(C3CCOCC3)c2c1)CN1CCc2ccccc2C1
PDB

UniProtKB/SwissProt

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n/an/a<100n/an/an/an/an/an/a



Epizyme, Inc.

US Patent




US Patent US9777008 (2017)


BindingDB Entry DOI: 10.7270/Q26975QQ
More data for this
Ligand-Target Pair
PRMT5/MEP50 Enzyme


(Homo sapiens (Human))
BDBM343958
PNG
(US9777008, Compound 252)
Show SMILES CN1CCC(CC1)n1cnc2ccc(cc12)-c1ccnc(NCC(O)CN2CCc3ccccc3C2)c1
PDB

UniProtKB/SwissProt

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n/an/a<100n/an/an/an/an/an/a



Epizyme, Inc.

US Patent




US Patent US9777008 (2017)


BindingDB Entry DOI: 10.7270/Q26975QQ
More data for this
Ligand-Target Pair
PRMT5/MEP50 Enzyme


(Homo sapiens (Human))
BDBM343959
PNG
(US9777008, Compound 253)
Show SMILES OC(COc1cccc(c1)-c1ncc2ccn(C3CCNCC3)c2n1)CN1CCc2ccccc2C1
PDB

UniProtKB/SwissProt

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n/an/a<100n/an/an/an/an/an/a



Epizyme, Inc.

US Patent




US Patent US9777008 (2017)


BindingDB Entry DOI: 10.7270/Q26975QQ
More data for this
Ligand-Target Pair
PRMT5/MEP50 Enzyme


(Homo sapiens (Human))
BDBM343960
PNG
(US9777008, Compound 254)
Show SMILES OC(CNc1cc(ccn1)-c1ncc2ccn(C3CNC3)c2n1)CN1CCc2ccccc2C1
PDB

UniProtKB/SwissProt

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n/an/a<100n/an/an/an/an/an/a



Epizyme, Inc.

US Patent




US Patent US9777008 (2017)


BindingDB Entry DOI: 10.7270/Q26975QQ
More data for this
Ligand-Target Pair
PRMT5/MEP50 Enzyme


(Homo sapiens (Human))
BDBM343961
PNG
(US9777008, Compound 255)
Show SMILES OC(CNc1cc(ccn1)-c1ncc2ccn(C3CCNCC3)c2n1)CN1CCc2ccccc2C1
PDB

UniProtKB/SwissProt

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n/an/a<100n/an/an/an/an/an/a



Epizyme, Inc.

US Patent




US Patent US9777008 (2017)


BindingDB Entry DOI: 10.7270/Q26975QQ
More data for this
Ligand-Target Pair
PRMT5/MEP50 Enzyme


(Homo sapiens (Human))
BDBM343962
PNG
(US9777008, Compound 256)
Show SMILES CC(=O)N1CCC(CC1)n1ccc2cnc(nc12)-c1ccnc(NCC(O)CN2CCc3ccccc3C2)c1
PDB

UniProtKB/SwissProt

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n/an/a<100n/an/an/an/an/an/a



Epizyme, Inc.

US Patent




US Patent US9777008 (2017)


BindingDB Entry DOI: 10.7270/Q26975QQ
More data for this
Ligand-Target Pair
PRMT5/MEP50 Enzyme


(Homo sapiens (Human))
BDBM343963
PNG
((R)-1-(3,4-dihydroisoquinolin-2(1H)-yl)-3-(3-(quin...)
Show SMILES O[C@@H](COc1cccc(c1)-c1cccc2cccnc12)CN1CCc2ccccc2C1 |r|
PDB

UniProtKB/SwissProt

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n/an/a<100n/an/an/an/an/an/a



Epizyme, Inc.

US Patent




US Patent US9777008 (2017)


BindingDB Entry DOI: 10.7270/Q26975QQ
More data for this
Ligand-Target Pair
PRMT5/MEP50 Enzyme


(Homo sapiens (Human))
BDBM343967
PNG
(US9777008, Compound 261)
Show SMILES Cn1cc2ccc(nc2n1)-c1cccc(NCC(O)CN2CCc3ccccc3C2)c1
PDB

UniProtKB/SwissProt

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n/an/a<100n/an/an/an/an/an/a



Epizyme, Inc.

US Patent




US Patent US9777008 (2017)


BindingDB Entry DOI: 10.7270/Q26975QQ
More data for this
Ligand-Target Pair
PRMT5/MEP50 Enzyme


(Homo sapiens (Human))
BDBM343971
PNG
(US9777008, Compound 265)
Show SMILES OC(CNc1cc(ccn1)-c1ccc2ncn(C3COC3)c2c1)CN1CCc2ccccc2C1
PDB

UniProtKB/SwissProt

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n/an/a<100n/an/an/an/an/an/a



Epizyme, Inc.

US Patent




US Patent US9777008 (2017)


BindingDB Entry DOI: 10.7270/Q26975QQ
More data for this
Ligand-Target Pair
PRMT5/MEP50 Enzyme


(Homo sapiens (Human))
BDBM343972
PNG
(1-(3,4-dihydroisoquinolin-2(1H)-yl)-3-(3-(3-methyl...)
Show SMILES Cc1ncc2ccc(cn12)-c1cccc(OCC(O)CN2CCc3ccccc3C2)c1
PDB

UniProtKB/SwissProt

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n/an/a<100n/an/an/an/an/an/a



Epizyme, Inc.

US Patent




US Patent US9777008 (2017)


BindingDB Entry DOI: 10.7270/Q26975QQ
More data for this
Ligand-Target Pair
PRMT5/MEP50 Enzyme


(Homo sapiens (Human))
BDBM343975
PNG
(US9777008, Compound 269)
Show SMILES OC(COc1cccc(c1)-c1ccc2ncn(C3COC3)c2c1)CN1CCc2ccccc2C1
PDB

UniProtKB/SwissProt

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n/an/a<100n/an/an/an/an/an/a



Epizyme, Inc.

US Patent




US Patent US9777008 (2017)


BindingDB Entry DOI: 10.7270/Q26975QQ
More data for this
Ligand-Target Pair
PRMT5/MEP50 Enzyme


(Homo sapiens (Human))
BDBM343979
PNG
(N-(3-(3,4-dihydroisoquinolin-2(1H)-yl)-2-hydroxypr...)
Show SMILES CC(=O)N(CC(O)CN1CCc2ccccc2C1)c1cccc(c1)-c1ccc2ncn(C)c2c1
PDB

UniProtKB/SwissProt

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n/an/a<100n/an/an/an/an/an/a



Epizyme, Inc.

US Patent




US Patent US9777008 (2017)


BindingDB Entry DOI: 10.7270/Q26975QQ
More data for this
Ligand-Target Pair
PRMT5/MEP50 Enzyme


(Homo sapiens (Human))
BDBM343981
PNG
(US9777008, Compound 275)
Show SMILES Cn1cnc2ccc(cc12)-c1ccnc(NC[C@H](O)CN2CCc3ccccc3C2)c1 |r|
PDB

UniProtKB/SwissProt

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n/an/a<100n/an/an/an/an/an/a



Epizyme, Inc.

US Patent




US Patent US9777008 (2017)


BindingDB Entry DOI: 10.7270/Q26975QQ
More data for this
Ligand-Target Pair
3D
3D Structure (crystal)
Protein arginine N-methyltransferase 5


(Homo sapiens (Human))
BDBM336958
PNG
(US9745291, Compound 4 | US9765068, Compound 4)
Show SMILES OC(CNC(=O)COc1cccc2N(Cc3ccccc3)CCCc12)CN1CCc2ccccc2C1
PDB

UniProtKB/SwissProt

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n/an/a<100n/an/an/an/an/an/a



Epizyme, Inc.

US Patent




US Patent US9765068 (2017)


BindingDB Entry DOI: 10.7270/Q2959KN3
More data for this
Ligand-Target Pair
Protein arginine N-methyltransferase 5


(Homo sapiens (Human))
BDBM336960
PNG
(US9745291, Compound 6 | US9765068, Compound 6)
Show SMILES OC(CNC(=O)COc1cccc2cccnc12)CN1CCc2ccccc2C1
PDB

UniProtKB/SwissProt

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n/an/a<100n/an/an/an/an/an/a



Epizyme, Inc.

US Patent




US Patent US9765068 (2017)


BindingDB Entry DOI: 10.7270/Q2959KN3
More data for this
Ligand-Target Pair
3D
3D Structure (crystal)
Protein arginine N-methyltransferase 5


(Homo sapiens (Human))
BDBM336973
PNG
(US9745291, Compound 19 | US9765068, Compound 19)
Show SMILES CC(Oc1ccccc1)C(=O)NCC(O)CN1CCc2ccccc2C1
PDB

UniProtKB/SwissProt

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n/an/a<100n/an/an/an/an/an/a



Epizyme, Inc.

US Patent




US Patent US9765068 (2017)


BindingDB Entry DOI: 10.7270/Q2959KN3
More data for this
Ligand-Target Pair
Protein arginine N-methyltransferase 5


(Homo sapiens (Human))
BDBM336974
PNG
(US9745291, Compound 20 | US9765068, Compound 20)
Show SMILES COc1cccc(OCC(=O)NCC(O)CN2CCc3ccccc3C2)c1
PDB

UniProtKB/SwissProt

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n/an/a<100n/an/an/an/an/an/a



Epizyme, Inc.

US Patent




US Patent US9765068 (2017)


BindingDB Entry DOI: 10.7270/Q2959KN3
More data for this
Ligand-Target Pair
Protein arginine N-methyltransferase 5


(Homo sapiens (Human))
BDBM336976
PNG
(US9745291, Compound 22 | US9765068, Compound 22)
Show SMILES COc1ccccc1OCC(=O)NCC(O)CN1CCc2ccccc2C1
PDB

UniProtKB/SwissProt

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n/an/a<100n/an/an/an/an/an/a



Epizyme, Inc.

US Patent




US Patent US9765068 (2017)


BindingDB Entry DOI: 10.7270/Q2959KN3
More data for this
Ligand-Target Pair
Protein arginine N-methyltransferase 5


(Homo sapiens (Human))
BDBM336977
PNG
(US9745291, Compound 23 | US9765068, Compound 23)
Show SMILES Cn1ncc2ccc(OCC(=O)NCC(O)CN3CCc4ccccc4C3)cc12
PDB

UniProtKB/SwissProt

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n/an/a<100n/an/an/an/an/an/a



Epizyme, Inc.

US Patent




US Patent US9765068 (2017)


BindingDB Entry DOI: 10.7270/Q2959KN3
More data for this
Ligand-Target Pair
Protein arginine N-methyltransferase 5


(Homo sapiens (Human))
BDBM336980
PNG
(US9745291, Compound 26 | US9765068, Compound 26)
Show SMILES Cc1cccc(OCC(=O)NCC(O)CN2CCc3ccccc3C2)c1
PDB

UniProtKB/SwissProt

antibodypedia
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US Patent
n/an/a<100n/an/an/an/an/an/a



Epizyme, Inc.

US Patent




US Patent US9765068 (2017)


BindingDB Entry DOI: 10.7270/Q2959KN3
More data for this
Ligand-Target Pair
Protein arginine N-methyltransferase 5


(Homo sapiens (Human))
BDBM336981
PNG
(US9745291, Compound 27 | US9765068, Compound 27)
Show SMILES CN(C)c1cccc(OCC(=O)NCC(O)CN2CCc3ccccc3C2)c1
PDB

UniProtKB/SwissProt

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US Patent
n/an/a<100n/an/an/an/an/an/a



Epizyme, Inc.

US Patent




US Patent US9765068 (2017)


BindingDB Entry DOI: 10.7270/Q2959KN3
More data for this
Ligand-Target Pair
Protein arginine N-methyltransferase 5


(Homo sapiens (Human))
BDBM336982
PNG
(US9745291, Compound 28 | US9765068, Compound 28)
Show SMILES CS(=O)(=O)Nc1cccc(OCC(=O)NCC(O)CN2CCc3ccccc3C2)c1
PDB

UniProtKB/SwissProt

antibodypedia
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PC sid
UniChem
US Patent
n/an/a<100n/an/an/an/an/an/a



Epizyme, Inc.

US Patent




US Patent US9765068 (2017)


BindingDB Entry DOI: 10.7270/Q2959KN3
More data for this
Ligand-Target Pair
Protein arginine N-methyltransferase 5


(Homo sapiens (Human))
BDBM336991
PNG
(US9745291, Compound 37 | US9765068, Compound 37)
Show SMILES CS(=O)(=O)c1ccccc1OCC(=O)NCC(O)CN1CCc2ccccc2C1
PDB

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Epizyme, Inc.

US Patent




US Patent US9765068 (2017)


BindingDB Entry DOI: 10.7270/Q2959KN3
More data for this
Ligand-Target Pair
Protein arginine N-methyltransferase 5


(Homo sapiens (Human))
BDBM336992
PNG
(US9745291, Compound 38 | US9765068, Compound 38)
Show SMILES CN(C)c1ccccc1OCC(=O)NCC(O)CN1CCc2ccccc2C1
PDB

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Epizyme, Inc.

US Patent




US Patent US9765068 (2017)


BindingDB Entry DOI: 10.7270/Q2959KN3
More data for this
Ligand-Target Pair
Protein arginine N-methyltransferase 5


(Homo sapiens (Human))
BDBM336993
PNG
(US9745291, Compound 39 | US9765068, Compound 39)
Show SMILES CC(Oc1cccc2cccnc12)C(=O)NCC(O)CN1CCc2ccccc2C1
PDB

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Epizyme, Inc.

US Patent




US Patent US9765068 (2017)


BindingDB Entry DOI: 10.7270/Q2959KN3
More data for this
Ligand-Target Pair
Protein arginine N-methyltransferase 5


(Homo sapiens (Human))
BDBM336994
PNG
(US9745291, Compound 40 | US9765068, Compound 40)
Show SMILES OC(CNC(=O)COc1ccccc1C1CCCCC1)CN1CCc2ccccc2C1
PDB

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Epizyme, Inc.

US Patent




US Patent US9765068 (2017)


BindingDB Entry DOI: 10.7270/Q2959KN3
More data for this
Ligand-Target Pair
Protein arginine N-methyltransferase 5


(Homo sapiens (Human))
BDBM336997
PNG
(US9745291, Compound 43 | US9765068, Compound 43)
Show SMILES CC(C)(Oc1cccc2cccnc12)C(=O)NCC(O)CN1CCc2ccccc2C1
PDB

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Epizyme, Inc.

US Patent




US Patent US9765068 (2017)


BindingDB Entry DOI: 10.7270/Q2959KN3
More data for this
Ligand-Target Pair
Protein arginine N-methyltransferase 5


(Homo sapiens (Human))
BDBM336999
PNG
(US9745291, Compound 269 | US9745291, Compound 45 |...)
Show SMILES O[C@H](CNC(=O)COc1cccc2cccnc12)CN1CCc2ccccc2C1 |r|
PDB

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Epizyme, Inc.

US Patent




US Patent US9765068 (2017)


BindingDB Entry DOI: 10.7270/Q2959KN3
More data for this
Ligand-Target Pair
3D
3D Structure (crystal)
Protein arginine N-methyltransferase 5


(Homo sapiens (Human))
BDBM337001
PNG
(US9745291, Compound 47 | US9765068, Compound 47)
Show SMILES CS(=O)(=O)c1cccc(OCC(=O)NCC(O)CN2CCc3ccccc3C2)c1
PDB

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Epizyme, Inc.

US Patent




US Patent US9765068 (2017)


BindingDB Entry DOI: 10.7270/Q2959KN3
More data for this
Ligand-Target Pair
Protein arginine N-methyltransferase 5


(Homo sapiens (Human))
BDBM337002
PNG
(US9745291, Compound 48 | US9765068, Compound 48)
Show SMILES OC(CNC(=O)COc1cccc2ccc(nc12)N1CCOCC1)CN1CCc2ccccc2C1
PDB

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Epizyme, Inc.

US Patent




US Patent US9765068 (2017)


BindingDB Entry DOI: 10.7270/Q2959KN3
More data for this
Ligand-Target Pair
Protein arginine N-methyltransferase 5


(Homo sapiens (Human))
BDBM337003
PNG
(US9745291, Compound 49 | US9765068, Compound 49)
Show SMILES OC(CNC(=O)COc1ccccc1N1CCOCC1)CN1CCc2ccccc2C1
PDB

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Epizyme, Inc.

US Patent




US Patent US9765068 (2017)


BindingDB Entry DOI: 10.7270/Q2959KN3
More data for this
Ligand-Target Pair
Protein arginine N-methyltransferase 5


(Homo sapiens (Human))
BDBM337004
PNG
(US9745291, Compound 50 | US9765068, Compound 50)
Show SMILES OC(CNC(=O)COc1ccccc1-c1cc[nH]n1)CN1CCc2ccccc2C1
PDB

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Epizyme, Inc.

US Patent




US Patent US9765068 (2017)


BindingDB Entry DOI: 10.7270/Q2959KN3
More data for this
Ligand-Target Pair
Protein arginine N-methyltransferase 5


(Homo sapiens (Human))
BDBM337007
PNG
(US9745291, Compound 53 | US9765068, Compound 53)
Show SMILES CS(=O)(=O)Nc1ccccc1OCC(=O)NCC(O)CN1CCc2ccccc2C1
PDB

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Epizyme, Inc.

US Patent




US Patent US9765068 (2017)


BindingDB Entry DOI: 10.7270/Q2959KN3
More data for this
Ligand-Target Pair
Protein arginine N-methyltransferase 5


(Homo sapiens (Human))
BDBM337018
PNG
(US9745291, Compound 64 | US9765068, Compound 64)
Show SMILES OC(CNC(=O)COc1cccc2CCCCc12)CN1CCc2ccccc2C1
PDB

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Epizyme, Inc.

US Patent




US Patent US9765068 (2017)


BindingDB Entry DOI: 10.7270/Q2959KN3
More data for this
Ligand-Target Pair
Protein arginine N-methyltransferase 5


(Homo sapiens (Human))
BDBM337019
PNG
(US9745291, Compound 65 | US9765068, Compound 65)
Show SMILES NS(=O)(=O)c1ccccc1OCC(=O)NCC(O)CN1CCc2ccccc2C1
PDB

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Epizyme, Inc.

US Patent




US Patent US9765068 (2017)


BindingDB Entry DOI: 10.7270/Q2959KN3
More data for this
Ligand-Target Pair
Protein arginine N-methyltransferase 5


(Homo sapiens (Human))
BDBM337020
PNG
(US9745291, Compound 66 | US9765068, Compound 66)
Show SMILES OC(CNC(=O)COc1cccc2ccccc12)CN1CCc2ccccc2C1
PDB

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Epizyme, Inc.

US Patent




US Patent US9765068 (2017)


BindingDB Entry DOI: 10.7270/Q2959KN3
More data for this
Ligand-Target Pair
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