Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Cytosol aminopeptidase [33-68,L62W] (Sus scrofa (Pig)) | BDBM234297 (Met-ψ[P(O)(OH)CH2]-Ala (5)) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | 3.64E+3 | -31.0 | n/a | n/a | n/a | n/a | n/a | 8.4 | 25 |
Academy of Sciences of the Czech Republic | Assay Description LAP was assayed in 75 mM triethanolamine hydrochloride buffer (pH = 8.4, containing 5 mM MgCl2) at 25°C. The substrate (L-leucine-p-nitroanilide) was... | J Enzyme Inhib Med Chem 26: 155-61 (2011) Article DOI: 10.3109/14756366.2010.482047 BindingDB Entry DOI: 10.7270/Q22N515B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cytosol aminopeptidase [33-68,L62W] (Sus scrofa (Pig)) | BDBM234295 (Met-PH (2)) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid PDB UniChem | Article PubMed | 2.20E+4 | -26.6 | n/a | n/a | n/a | n/a | n/a | 8.4 | 25 |
Academy of Sciences of the Czech Republic | Assay Description LAP was assayed in 75 mM triethanolamine hydrochloride buffer (pH = 8.4, containing 5 mM MgCl2) at 25°C. The substrate (L-leucine-p-nitroanilide) was... | J Enzyme Inhib Med Chem 26: 155-61 (2011) Article DOI: 10.3109/14756366.2010.482047 BindingDB Entry DOI: 10.7270/Q22N515B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cytosol aminopeptidase [33-68,L62W] (Sus scrofa (Pig)) | BDBM234294 (Met-P (1)) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid PDB UniChem | Article PubMed | 2.26E+4 | -26.5 | n/a | n/a | n/a | n/a | n/a | 8.4 | 25 |
Academy of Sciences of the Czech Republic | Assay Description LAP was assayed in 75 mM triethanolamine hydrochloride buffer (pH = 8.4, containing 5 mM MgCl2) at 25°C. The substrate (L-leucine-p-nitroanilide) was... | J Enzyme Inhib Med Chem 26: 155-61 (2011) Article DOI: 10.3109/14756366.2010.482047 BindingDB Entry DOI: 10.7270/Q22N515B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cytosol aminopeptidase [33-68,L62W] (Sus scrofa (Pig)) | BDBM50316030 (1-aminopentylphosphonic acid | CHEMBL1089899 | Nle...) | UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid PDB UniChem Patents Similars | Article PubMed | 5.80E+4 | -24.2 | n/a | n/a | n/a | n/a | n/a | 8.4 | 25 |
Academy of Sciences of the Czech Republic | Assay Description LAP was assayed in 75 mM triethanolamine hydrochloride buffer (pH = 8.4, containing 5 mM MgCl2) at 25°C. The substrate (L-leucine-p-nitroanilide) was... | J Enzyme Inhib Med Chem 26: 155-61 (2011) Article DOI: 10.3109/14756366.2010.482047 BindingDB Entry DOI: 10.7270/Q22N515B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cytosol aminopeptidase [33-68,L62W] (Sus scrofa (Pig)) | BDBM234296 (Nle-PH (4)) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | 7.39E+4 | -23.6 | n/a | n/a | n/a | n/a | n/a | 8.4 | 25 |
Academy of Sciences of the Czech Republic | Assay Description LAP was assayed in 75 mM triethanolamine hydrochloride buffer (pH = 8.4, containing 5 mM MgCl2) at 25°C. The substrate (L-leucine-p-nitroanilide) was... | J Enzyme Inhib Med Chem 26: 155-61 (2011) Article DOI: 10.3109/14756366.2010.482047 BindingDB Entry DOI: 10.7270/Q22N515B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cytosol aminopeptidase [33-68,L62W] (Sus scrofa (Pig)) | BDBM234299 (Nle-ψ[P(O)(OH)O]-L-AlaOMe (7)) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | 2.19E+5 | -20.9 | n/a | n/a | n/a | n/a | n/a | 8.4 | 25 |
Academy of Sciences of the Czech Republic | Assay Description LAP was assayed in 75 mM triethanolamine hydrochloride buffer (pH = 8.4, containing 5 mM MgCl2) at 25°C. The substrate (L-leucine-p-nitroanilide) was... | J Enzyme Inhib Med Chem 26: 155-61 (2011) Article DOI: 10.3109/14756366.2010.482047 BindingDB Entry DOI: 10.7270/Q22N515B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cytosol aminopeptidase [33-68,L62W] (Sus scrofa (Pig)) | BDBM234298 (Nle-ψ[P(O)(OH)O]-L-Ala (6)) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | 2.69E+5 | -20.4 | n/a | n/a | n/a | n/a | n/a | 8.4 | 25 |
Academy of Sciences of the Czech Republic | Assay Description LAP was assayed in 75 mM triethanolamine hydrochloride buffer (pH = 8.4, containing 5 mM MgCl2) at 25°C. The substrate (L-leucine-p-nitroanilide) was... | J Enzyme Inhib Med Chem 26: 155-61 (2011) Article DOI: 10.3109/14756366.2010.482047 BindingDB Entry DOI: 10.7270/Q22N515B | |||||||||||
More data for this Ligand-Target Pair |