Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Platelet-activating factor receptor (Cavia porcellus) | BDBM50000714 (3-[4-(2-Chloro-phenyl)-9-methyl-6H-1-thia-5,7,8,9a...) | MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Patents Similars | PubMed | 98 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Abbott Laboratories Curated by ChEMBL | Assay Description In vitro intrinsic binding affinity at platelet activating factor receptor using rabbit platelet membranes | J Med Chem 35: 2055-61 (1992) BindingDB Entry DOI: 10.7270/Q2NZ86K9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet-activating factor receptor (Cavia porcellus) | BDBM50000717 (2-{7-[4-(4-Fluoro-phenyl)-1-methyl-butyl]-5-methox...) | MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 142 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Abbott Laboratories Curated by ChEMBL | Assay Description In vitro intrinsic binding affinity at platelet activating factor receptor using rabbit platelet membranes | J Med Chem 35: 2055-61 (1992) BindingDB Entry DOI: 10.7270/Q2NZ86K9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet-activating factor receptor (Cavia porcellus) | BDBM50000701 (2-{7-[4-(4-Fluoro-phenyl)-1-methyl-butyl]-10,10-di...) | MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 157 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Abbott Laboratories Curated by ChEMBL | Assay Description In vitro intrinsic binding affinity at platelet activating factor receptor using rabbit platelet membranes | J Med Chem 35: 2055-61 (1992) BindingDB Entry DOI: 10.7270/Q2NZ86K9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet-activating factor receptor (Cavia porcellus) | BDBM50000707 (2-{7-[4-(4-Fluoro-phenyl)-1-methyl-butyl]-10,10-di...) | MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 167 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Abbott Laboratories Curated by ChEMBL | Assay Description In vitro intrinsic binding affinity at platelet activating factor receptor using rabbit platelet membranes | J Med Chem 35: 2055-61 (1992) BindingDB Entry DOI: 10.7270/Q2NZ86K9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet-activating factor receptor (Cavia porcellus) | BDBM50000722 (2-{7-[4-(4-Fluoro-phenyl)-1-methyl-butyl]-5-hydrox...) | MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 331 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Abbott Laboratories Curated by ChEMBL | Assay Description In vitro intrinsic binding affinity at platelet activating factor receptor using rabbit platelet membranes | J Med Chem 35: 2055-61 (1992) BindingDB Entry DOI: 10.7270/Q2NZ86K9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet-activating factor receptor (Cavia porcellus) | BDBM50000720 (2-{7-[4-(4-Fluoro-phenyl)-1-methyl-butyl]-10,10-di...) | MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 345 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Abbott Laboratories Curated by ChEMBL | Assay Description In vitro intrinsic binding affinity at platelet activating factor receptor using rabbit platelet membranes | J Med Chem 35: 2055-61 (1992) BindingDB Entry DOI: 10.7270/Q2NZ86K9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet-activating factor receptor (Cavia porcellus) | BDBM50000719 (CHEMBL62812 | {7-[4-(4-Fluoro-phenyl)-1-methyl-but...) | MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 390 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Abbott Laboratories Curated by ChEMBL | Assay Description In vitro intrinsic binding affinity at platelet activating factor receptor using rabbit platelet membranes | J Med Chem 35: 2055-61 (1992) BindingDB Entry DOI: 10.7270/Q2NZ86K9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet-activating factor receptor (Cavia porcellus) | BDBM50000708 (4-{7-[4-(4-Fluoro-phenyl)-1-methyl-butyl]-5-hydrox...) | MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 656 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Abbott Laboratories Curated by ChEMBL | Assay Description In vitro intrinsic binding affinity at platelet activating factor receptor using rabbit platelet membranes | J Med Chem 35: 2055-61 (1992) BindingDB Entry DOI: 10.7270/Q2NZ86K9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet-activating factor receptor (Cavia porcellus) | BDBM50000700 (4-{7-[4-(4-Fluoro-phenyl)-1-methyl-butyl]-5-methox...) | MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 690 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Abbott Laboratories Curated by ChEMBL | Assay Description In vitro intrinsic binding affinity at platelet activating factor receptor using rabbit platelet membranes | J Med Chem 35: 2055-61 (1992) BindingDB Entry DOI: 10.7270/Q2NZ86K9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet-activating factor receptor (Cavia porcellus) | BDBM50000716 (CHEMBL61680 | {7-[4-(4-Fluoro-phenyl)-1-methyl-but...) | MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 925 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Abbott Laboratories Curated by ChEMBL | Assay Description In vitro intrinsic binding affinity at platelet activating factor receptor using rabbit platelet membranes | J Med Chem 35: 2055-61 (1992) BindingDB Entry DOI: 10.7270/Q2NZ86K9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet-activating factor receptor (Cavia porcellus) | BDBM50000718 (2-{7-[4-(4-Fluoro-phenyl)-1-methyl-butyl]-5-methox...) | MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 945 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Abbott Laboratories Curated by ChEMBL | Assay Description In vitro intrinsic binding affinity at platelet activating factor receptor using rabbit platelet membranes | J Med Chem 35: 2055-61 (1992) BindingDB Entry DOI: 10.7270/Q2NZ86K9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet-activating factor receptor (Cavia porcellus) | BDBM50000705 (2-({7-[4-(4-Fluoro-phenyl)-1-methyl-butyl]-5-hydro...) | MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 1.58E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Abbott Laboratories Curated by ChEMBL | Assay Description In vitro intrinsic binding affinity at platelet activating factor receptor using rabbit platelet membranes | J Med Chem 35: 2055-61 (1992) BindingDB Entry DOI: 10.7270/Q2NZ86K9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet-activating factor receptor (Cavia porcellus) | BDBM50000712 (7-[4-(4-Fluoro-phenyl)-1-methyl-butyl]-10,10-dimet...) | MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 3.25E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Abbott Laboratories Curated by ChEMBL | Assay Description In vitro intrinsic binding affinity at platelet activating factor receptor using rabbit platelet membranes | J Med Chem 35: 2055-61 (1992) BindingDB Entry DOI: 10.7270/Q2NZ86K9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet-activating factor receptor (Cavia porcellus) | BDBM50000711 (2-{7-[4-(4-Fluoro-phenyl)-1-methyl-butyl]-5-hydrox...) | MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | PubMed | 3.30E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Abbott Laboratories Curated by ChEMBL | Assay Description In vitro intrinsic binding affinity at platelet activating factor receptor using rabbit platelet membranes | J Med Chem 35: 2055-61 (1992) BindingDB Entry DOI: 10.7270/Q2NZ86K9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet-activating factor receptor (Cavia porcellus) | BDBM50000715 (2-[7-(1,2-Dimethyl-heptyl)-5-hydroxy-10,10-dimethy...) | MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 3.68E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Abbott Laboratories Curated by ChEMBL | Assay Description In vitro intrinsic binding affinity at platelet activating factor receptor using rabbit platelet membranes | J Med Chem 35: 2055-61 (1992) BindingDB Entry DOI: 10.7270/Q2NZ86K9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet-activating factor receptor (Cavia porcellus) | BDBM50000702 (7-[4-(4-Fluoro-phenyl)-1-methyl-butyl]-5-methoxy-1...) | MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 4.21E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Abbott Laboratories Curated by ChEMBL | Assay Description In vitro intrinsic binding affinity at platelet activating factor receptor using rabbit platelet membranes | J Med Chem 35: 2055-61 (1992) BindingDB Entry DOI: 10.7270/Q2NZ86K9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet-activating factor receptor (Cavia porcellus) | BDBM50000710 (3-{7-[4-(4-Fluoro-phenyl)-1-methyl-butyl]-5-methox...) | MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 4.40E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Abbott Laboratories Curated by ChEMBL | Assay Description In vitro intrinsic binding affinity at platelet activating factor receptor using rabbit platelet membranes | J Med Chem 35: 2055-61 (1992) BindingDB Entry DOI: 10.7270/Q2NZ86K9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet-activating factor receptor (Cavia porcellus) | BDBM50000699 (3-{7-[4-(4-Fluoro-phenyl)-1-methyl-butyl]-5-methox...) | MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 5.50E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Abbott Laboratories Curated by ChEMBL | Assay Description In vitro intrinsic binding affinity at platelet activating factor receptor using rabbit platelet membranes | J Med Chem 35: 2055-61 (1992) BindingDB Entry DOI: 10.7270/Q2NZ86K9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet-activating factor receptor (Cavia porcellus) | BDBM50000709 (5-{7-[4-(4-Fluoro-phenyl)-1-methyl-butyl]-5-methox...) | MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 5.50E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Abbott Laboratories Curated by ChEMBL | Assay Description In vitro intrinsic binding affinity at platelet activating factor receptor using rabbit platelet membranes | J Med Chem 35: 2055-61 (1992) BindingDB Entry DOI: 10.7270/Q2NZ86K9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet-activating factor receptor (Cavia porcellus) | BDBM50000724 (2-(5-Hydroxy-7-isopropyl-10,10-dimethyl-1,2,4,10-t...) | MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 9.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Abbott Laboratories Curated by ChEMBL | Assay Description In vitro intrinsic binding affinity at platelet activating factor receptor using rabbit platelet membranes | J Med Chem 35: 2055-61 (1992) BindingDB Entry DOI: 10.7270/Q2NZ86K9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet-activating factor receptor (Cavia porcellus) | BDBM50000725 (7-[4-(4-Fluoro-phenyl)-1-methyl-butyl]-10,10-dimet...) | MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | 1.18E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Abbott Laboratories Curated by ChEMBL | Assay Description In vitro intrinsic binding affinity at platelet activating factor receptor using rabbit platelet membranes | J Med Chem 35: 2055-61 (1992) BindingDB Entry DOI: 10.7270/Q2NZ86K9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet-activating factor receptor (Cavia porcellus) | BDBM50000721 (2-{7-[4-(4-Fluoro-phenyl)-1-methyl-butyl]-5-hydrox...) | MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 1.58E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Abbott Laboratories Curated by ChEMBL | Assay Description In vitro intrinsic binding affinity at platelet activating factor receptor using rabbit platelet membranes | J Med Chem 35: 2055-61 (1992) BindingDB Entry DOI: 10.7270/Q2NZ86K9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet-activating factor receptor (Cavia porcellus) | BDBM50000703 (7-[4-(4-Fluoro-phenyl)-1-methyl-butyl]-5-methoxy-1...) | MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 1.69E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Abbott Laboratories Curated by ChEMBL | Assay Description In vitro intrinsic binding affinity at platelet activating factor receptor using rabbit platelet membranes | J Med Chem 35: 2055-61 (1992) BindingDB Entry DOI: 10.7270/Q2NZ86K9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet-activating factor receptor (Cavia porcellus) | BDBM50000723 (1-{7-[4-(4-Fluoro-phenyl)-1-methyl-butyl]-5-hydrox...) | MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 2.05E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Abbott Laboratories Curated by ChEMBL | Assay Description In vitro intrinsic binding affinity at platelet activating factor receptor using rabbit platelet membranes | J Med Chem 35: 2055-61 (1992) BindingDB Entry DOI: 10.7270/Q2NZ86K9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet-activating factor receptor (Cavia porcellus) | BDBM50000726 (4-{7-[4-(4-Fluoro-phenyl)-1-methyl-butyl]-5-hydrox...) | MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 2.07E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Abbott Laboratories Curated by ChEMBL | Assay Description In vitro intrinsic binding affinity at platelet activating factor receptor using rabbit platelet membranes | J Med Chem 35: 2055-61 (1992) BindingDB Entry DOI: 10.7270/Q2NZ86K9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet-activating factor receptor (Cavia porcellus) | BDBM50000713 (2-[5-{4-[4-(4-Fluoro-phenyl)-1-methyl-butyl]-2,6-d...) | MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 2.35E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Abbott Laboratories Curated by ChEMBL | Assay Description In vitro intrinsic binding affinity at platelet activating factor receptor using rabbit platelet membranes | J Med Chem 35: 2055-61 (1992) BindingDB Entry DOI: 10.7270/Q2NZ86K9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet-activating factor receptor (Cavia porcellus) | BDBM50000706 (6-{7-[4-(4-Fluoro-phenyl)-1-methyl-butyl]-5-methox...) | MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 2.50E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Abbott Laboratories Curated by ChEMBL | Assay Description In vitro intrinsic binding affinity at platelet activating factor receptor using rabbit platelet membranes | J Med Chem 35: 2055-61 (1992) BindingDB Entry DOI: 10.7270/Q2NZ86K9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet-activating factor receptor (Cavia porcellus) | BDBM50000704 (7-[4-(4-Fluoro-phenyl)-1-methyl-butyl]-1,4,4-trime...) | MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | PubMed | 4.38E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Abbott Laboratories Curated by ChEMBL | Assay Description In vitro intrinsic binding affinity at platelet activating factor receptor using rabbit platelet membranes | J Med Chem 35: 2055-61 (1992) BindingDB Entry DOI: 10.7270/Q2NZ86K9 | |||||||||||
More data for this Ligand-Target Pair |