Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Prolyl 4-hydroxylase subunit alpha-1 (Rattus norvegicus) | BDBM26106 (CHEMBL90852 | N-oxalyl glycine, 1a | NOG | Oxalylg...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase CHEMBL MCE MMDB PC cid PC sid PDB UniChem Patents Similars | PubMed | 540 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
ICI Pharmaceuticals Curated by ChEMBL | Assay Description Compound was evaluated for the inhibition of prolyl 4-hydroxylase | J Med Chem 35: 2652-8 (1992) BindingDB Entry DOI: 10.7270/Q28P5ZF9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Prolyl 4-hydroxylase subunit alpha-1 (Rattus norvegicus) | BDBM26114 (CHEMBL88972 | pyridine carboxylate, 6b | pyridine-...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid PDB UniChem Patents | PubMed | 800 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
ICI Pharmaceuticals Curated by ChEMBL | Assay Description Inhibitory activity against prolyl 4-hydroxylase | J Med Chem 35: 2652-8 (1992) BindingDB Entry DOI: 10.7270/Q28P5ZF9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Prolyl 4-hydroxylase subunit alpha-1 (Rattus norvegicus) | BDBM26106 (CHEMBL90852 | N-oxalyl glycine, 1a | NOG | Oxalylg...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase CHEMBL MCE MMDB PC cid PC sid PDB UniChem Patents Similars | PubMed | n/a | n/a | 2.89E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
ICI Pharmaceuticals Curated by ChEMBL | Assay Description Compound was evaluated for the inhibition of prolyl 4-hydroxylase | J Med Chem 35: 2652-8 (1992) BindingDB Entry DOI: 10.7270/Q28P5ZF9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Prolyl 4-hydroxylase subunit alpha-1 (Rattus norvegicus) | BDBM26114 (CHEMBL88972 | pyridine carboxylate, 6b | pyridine-...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid PDB UniChem Patents | PubMed | n/a | n/a | 5.18E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
ICI Pharmaceuticals Curated by ChEMBL | Assay Description Compound was evaluated for the inhibition of prolyl 4-hydroxylase | J Med Chem 35: 2652-8 (1992) BindingDB Entry DOI: 10.7270/Q28P5ZF9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Prolyl 4-hydroxylase subunit alpha-1 (Rattus norvegicus) | BDBM50000866 (2-(Oxalyl-amino)-propionic acid (0.25H2O) | CHEMBL...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | n/a | n/a | 3.82E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
ICI Pharmaceuticals Curated by ChEMBL | Assay Description Compound was evaluated for the inhibition of prolyl 4-hydroxylase | J Med Chem 35: 2652-8 (1992) BindingDB Entry DOI: 10.7270/Q28P5ZF9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Prolyl 4-hydroxylase subunit alpha-1 (Rattus norvegicus) | BDBM50000865 (2-(Oxalyl-amino)-propionic acid | CHEMBL314979) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid PDB UniChem Patents Similars | PubMed | n/a | n/a | 9.07E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
ICI Pharmaceuticals Curated by ChEMBL | Assay Description Compound was evaluated for the inhibition of prolyl 4-hydroxylase | J Med Chem 35: 2652-8 (1992) BindingDB Entry DOI: 10.7270/Q28P5ZF9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Prolyl 4-hydroxylase subunit alpha-1 (Rattus norvegicus) | BDBM50000864 (CHEMBL314175 | N-(2-Methanesulfonylamino-2-oxo-eth...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | PubMed | n/a | n/a | 4.14E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
ICI Pharmaceuticals Curated by ChEMBL | Assay Description Compound was evaluated for the inhibition of prolyl 4-hydroxylase | J Med Chem 35: 2652-8 (1992) BindingDB Entry DOI: 10.7270/Q28P5ZF9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Prolyl 4-hydroxylase subunit alpha-1 (Rattus norvegicus) | BDBM50000863 (2-(Oxalyl-amino)-propionic acid | CHEMBL88472) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid PDB UniChem Patents Similars | PubMed | n/a | n/a | 6.21E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
ICI Pharmaceuticals Curated by ChEMBL | Assay Description Compound was evaluated for the inhibition of prolyl 4-hydroxylase at 50 ug/mL | J Med Chem 35: 2652-8 (1992) BindingDB Entry DOI: 10.7270/Q28P5ZF9 | |||||||||||
More data for this Ligand-Target Pair |