Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Platelet-activating factor receptor (Homo sapiens (Human)) | BDBM50018316 (2-Butyl-3',4'-dimethoxy-biphenyl-4-carboxylic acid...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | n/a | n/a | 4 | n/a | n/a | n/a | n/a | n/a | n/a |
Roche Research Center Curated by ChEMBL | Assay Description Inhibition of platelet activating factor receptor binding activity in dog platelets using [3H]-PAF as radioligand. | J Med Chem 32: 1814-20 (1989) BindingDB Entry DOI: 10.7270/Q2SQ8ZCJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet-activating factor receptor (Homo sapiens (Human)) | BDBM50018341 (2-Ethyl-3',4'-dimethoxy-biphenyl-4-carboxylic acid...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | n/a | n/a | 4 | n/a | n/a | n/a | n/a | n/a | n/a |
Roche Research Center Curated by ChEMBL | Assay Description Inhibition of platelet activating factor receptor binding activity in dog platelets using [3H]-PAF as radioligand. | J Med Chem 32: 1814-20 (1989) BindingDB Entry DOI: 10.7270/Q2SQ8ZCJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet-activating factor receptor (Homo sapiens (Human)) | BDBM50018315 (2-Ethynyl-3',4'-dimethoxy-biphenyl-4-carboxylic ac...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | n/a | n/a | 5 | n/a | n/a | n/a | n/a | n/a | n/a |
Roche Research Center Curated by ChEMBL | Assay Description Inhibition of platelet activating factor receptor binding activity in dog platelets using [3H]-PAF as radioligand. | J Med Chem 32: 1814-20 (1989) BindingDB Entry DOI: 10.7270/Q2SQ8ZCJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet-activating factor receptor (Homo sapiens (Human)) | BDBM50018325 (CHEMBL53584 | [1,1';2',1'']Terphenyl-4'-carboxylic...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | n/a | n/a | 5 | n/a | n/a | n/a | n/a | n/a | n/a |
Roche Research Center Curated by ChEMBL | Assay Description Inhibition of platelet activating factor receptor binding activity in dog platelets using [3H]-PAF as radioligand. | J Med Chem 32: 1814-20 (1989) BindingDB Entry DOI: 10.7270/Q2SQ8ZCJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet-activating factor receptor (Homo sapiens (Human)) | BDBM50018321 (3',4'-Dimethoxy-biphenyl-4-carboxylic acid (1-meth...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | n/a | n/a | 15 | n/a | n/a | n/a | n/a | n/a | n/a |
Roche Research Center Curated by ChEMBL | Assay Description Inhibition of platelet activating factor receptor binding activity in dog platelets using [3H]-PAF as radioligand. | J Med Chem 32: 1814-20 (1989) BindingDB Entry DOI: 10.7270/Q2SQ8ZCJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet-activating factor receptor (Homo sapiens (Human)) | BDBM50018338 (2-Butyl-3',4'-dimethoxy-biphenyl-4-carboxylic acid...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 18 | n/a | n/a | n/a | n/a | n/a | n/a |
Roche Research Center Curated by ChEMBL | Assay Description Inhibition of platelet activating factor receptor binding activity in dog platelets using [3H]-PAF as radioligand. | J Med Chem 32: 1814-20 (1989) BindingDB Entry DOI: 10.7270/Q2SQ8ZCJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet-activating factor receptor (Homo sapiens (Human)) | BDBM50018337 (3'-Methoxy-biphenyl-4-carboxylic acid (1-methyl-4-...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 20 | n/a | n/a | n/a | n/a | n/a | n/a |
Roche Research Center Curated by ChEMBL | Assay Description Inhibition of platelet activating factor receptor binding activity in dog platelets using [3H]-PAF as radioligand. | J Med Chem 32: 1814-20 (1989) BindingDB Entry DOI: 10.7270/Q2SQ8ZCJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet-activating factor receptor (Homo sapiens (Human)) | BDBM50018320 (3',4'-Dimethoxy-2-propyl-biphenyl-4-carboxylic aci...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | n/a | n/a | 50 | n/a | n/a | n/a | n/a | n/a | n/a |
Roche Research Center Curated by ChEMBL | Assay Description Inhibition of platelet activating factor receptor binding activity in dog platelets using [3H]-PAF as radioligand. | J Med Chem 32: 1814-20 (1989) BindingDB Entry DOI: 10.7270/Q2SQ8ZCJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet-activating factor receptor (Homo sapiens (Human)) | BDBM50018324 (CHEMBL299760 | [1,1';2',1'']Terphenyl-4'-carboxyli...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 50 | n/a | n/a | n/a | n/a | n/a | n/a |
Roche Research Center Curated by ChEMBL | Assay Description Inhibition of platelet activating factor receptor binding activity in dog platelets using [3H]-PAF as radioligand. | J Med Chem 32: 1814-20 (1989) BindingDB Entry DOI: 10.7270/Q2SQ8ZCJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet-activating factor receptor (Homo sapiens (Human)) | BDBM50018329 (3',4'-Dimethoxy-biphenyl-4-carbothioic acid (1-met...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 60 | n/a | n/a | n/a | n/a | n/a | n/a |
Roche Research Center Curated by ChEMBL | Assay Description Inhibition of platelet activating factor receptor binding activity in dog platelets using [3H]-PAF as radioligand. | J Med Chem 32: 1814-20 (1989) BindingDB Entry DOI: 10.7270/Q2SQ8ZCJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet-activating factor receptor (Homo sapiens (Human)) | BDBM50018326 (2-Allyl-3',4'-dimethoxy-biphenyl-4-carboxylic acid...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | n/a | n/a | 80 | n/a | n/a | n/a | n/a | n/a | n/a |
Roche Research Center Curated by ChEMBL | Assay Description Inhibition of platelet activating factor receptor binding activity in dog platelets using [3H]-PAF as radioligand. | J Med Chem 32: 1814-20 (1989) BindingDB Entry DOI: 10.7270/Q2SQ8ZCJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet-activating factor receptor (Homo sapiens (Human)) | BDBM50018322 (4,4''-Dimethoxy-[1,1';2',1'']terphenyl-4'-carboxyl...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 125 | n/a | n/a | n/a | n/a | n/a | n/a |
Roche Research Center Curated by ChEMBL | Assay Description Inhibition of platelet activating factor receptor binding activity in dog platelets using [3H]-PAF as radioligand. | J Med Chem 32: 1814-20 (1989) BindingDB Entry DOI: 10.7270/Q2SQ8ZCJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet-activating factor receptor (Homo sapiens (Human)) | BDBM50018336 (3',4'-Dimethoxy-biphenyl-4-carbothioic acid (4-pyr...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 140 | n/a | n/a | n/a | n/a | n/a | n/a |
Roche Research Center Curated by ChEMBL | Assay Description Inhibition of platelet activating factor receptor binding activity in dog platelets using [3H]-PAF as radioligand. | J Med Chem 32: 1814-20 (1989) BindingDB Entry DOI: 10.7270/Q2SQ8ZCJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet-activating factor receptor (Homo sapiens (Human)) | BDBM50018327 (2-Bromo-3',4'-dimethoxy-biphenyl-4-carboxylic acid...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 180 | n/a | n/a | n/a | n/a | n/a | n/a |
Roche Research Center Curated by ChEMBL | Assay Description Inhibition of platelet activating factor receptor binding activity in dog platelets using [3H]-PAF as radioligand. | J Med Chem 32: 1814-20 (1989) BindingDB Entry DOI: 10.7270/Q2SQ8ZCJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet-activating factor receptor (Homo sapiens (Human)) | BDBM50018323 (3,3''-Dimethoxy-[1,1';2',1'']terphenyl-4'-carboxyl...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 200 | n/a | n/a | n/a | n/a | n/a | n/a |
Roche Research Center Curated by ChEMBL | Assay Description Inhibition of platelet activating factor receptor binding activity in dog platelets using [3H]-PAF as radioligand. | J Med Chem 32: 1814-20 (1989) BindingDB Entry DOI: 10.7270/Q2SQ8ZCJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet-activating factor receptor (Homo sapiens (Human)) | BDBM50018319 (3',4'-Dimethoxy-2-nitro-biphenyl-4-carboxylic acid...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 200 | n/a | n/a | n/a | n/a | n/a | n/a |
Roche Research Center Curated by ChEMBL | Assay Description Inhibition of platelet activating factor receptor binding activity in dog platelets using [3H]-PAF as radioligand. | J Med Chem 32: 1814-20 (1989) BindingDB Entry DOI: 10.7270/Q2SQ8ZCJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet-activating factor receptor (Homo sapiens (Human)) | BDBM50018328 (3',4'-Dimethyl-biphenyl-4-carboxylic acid (4-pyrid...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | n/a | n/a | 200 | n/a | n/a | n/a | n/a | n/a | n/a |
Roche Research Center Curated by ChEMBL | Assay Description Inhibition of platelet activating factor receptor binding activity in dog platelets using [3H]-PAF as radioligand. | J Med Chem 32: 1814-20 (1989) BindingDB Entry DOI: 10.7270/Q2SQ8ZCJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet-activating factor receptor (Homo sapiens (Human)) | BDBM50018331 (3',4'-Dimethoxy-2-nitro-biphenyl-4-carboxylic acid...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 200 | n/a | n/a | n/a | n/a | n/a | n/a |
Roche Research Center Curated by ChEMBL | Assay Description Inhibition of platelet activating factor receptor binding activity in dog platelets using [3H]-PAF as radioligand. | J Med Chem 32: 1814-20 (1989) BindingDB Entry DOI: 10.7270/Q2SQ8ZCJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet-activating factor receptor (Homo sapiens (Human)) | BDBM50018330 (2-Bromo-3',4'-dimethoxy-biphenyl-4-carboxylic acid...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 220 | n/a | n/a | n/a | n/a | n/a | n/a |
Roche Research Center Curated by ChEMBL | Assay Description Inhibition of platelet activating factor receptor binding activity in dog platelets using [3H]-PAF as radioligand. | J Med Chem 32: 1814-20 (1989) BindingDB Entry DOI: 10.7270/Q2SQ8ZCJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet-activating factor receptor (Homo sapiens (Human)) | BDBM50018318 (3'-Methoxy-biphenyl-4-carboxylic acid (4-pyridin-3...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 280 | n/a | n/a | n/a | n/a | n/a | n/a |
Roche Research Center Curated by ChEMBL | Assay Description Inhibition of platelet activating factor receptor binding activity in dog platelets using [3H]-PAF as radioligand. | J Med Chem 32: 1814-20 (1989) BindingDB Entry DOI: 10.7270/Q2SQ8ZCJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet-activating factor receptor (Homo sapiens (Human)) | BDBM50018333 (2,3',4'-Trimethoxy-biphenyl-4-carboxylic acid (4-p...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 300 | n/a | n/a | n/a | n/a | n/a | n/a |
Roche Research Center Curated by ChEMBL | Assay Description Inhibition of platelet activating factor receptor binding activity in dog platelets using [3H]-PAF as radioligand. | J Med Chem 32: 1814-20 (1989) BindingDB Entry DOI: 10.7270/Q2SQ8ZCJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet-activating factor receptor (Homo sapiens (Human)) | BDBM50018317 (3'-Hydroxy-biphenyl-4-carboxylic acid (4-pyridin-3...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | n/a | n/a | 300 | n/a | n/a | n/a | n/a | n/a | n/a |
Roche Research Center Curated by ChEMBL | Assay Description Inhibition of platelet activating factor receptor binding activity in dog platelets using [3H]-PAF as radioligand. | J Med Chem 32: 1814-20 (1989) BindingDB Entry DOI: 10.7270/Q2SQ8ZCJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet-activating factor receptor (Homo sapiens (Human)) | BDBM50018332 (3',4'-Dimethoxy-biphenyl-4-carboxylic acid (4-pyri...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 400 | n/a | n/a | n/a | n/a | n/a | n/a |
Roche Research Center Curated by ChEMBL | Assay Description Inhibition of platelet activating factor receptor binding activity in dog platelets using [3H]-PAF as radioligand. | J Med Chem 32: 1814-20 (1989) BindingDB Entry DOI: 10.7270/Q2SQ8ZCJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet-activating factor receptor (Homo sapiens (Human)) | BDBM50018334 (3'-Methyl-biphenyl-4-carboxylic acid (4-pyridin-3-...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 500 | n/a | n/a | n/a | n/a | n/a | n/a |
Roche Research Center Curated by ChEMBL | Assay Description Inhibition of platelet activating factor receptor binding activity in dog platelets using [3H]-PAF as radioligand. | J Med Chem 32: 1814-20 (1989) BindingDB Entry DOI: 10.7270/Q2SQ8ZCJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet-activating factor receptor (Homo sapiens (Human)) | BDBM50018335 (Biphenyl-4-carboxylic acid (4-pyridin-3-yl-butyl)-...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 630 | n/a | n/a | n/a | n/a | n/a | n/a |
Roche Research Center Curated by ChEMBL | Assay Description Inhibition of platelet activating factor receptor binding activity in dog platelets using [3H]-PAF as radioligand. | J Med Chem 32: 1814-20 (1989) BindingDB Entry DOI: 10.7270/Q2SQ8ZCJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet-activating factor receptor (Homo sapiens (Human)) | BDBM50018339 (3'-(Cyclohepta-1,3,5-trienyloxy)-biphenyl-4-carbox...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | PubMed | n/a | n/a | 700 | n/a | n/a | n/a | n/a | n/a | n/a |
Roche Research Center Curated by ChEMBL | Assay Description Inhibition of platelet-activating factor receptor binding activity in dog platelets using [3H]-PAF as radioligand. | J Med Chem 32: 1814-20 (1989) BindingDB Entry DOI: 10.7270/Q2SQ8ZCJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet-activating factor receptor (Homo sapiens (Human)) | BDBM50018340 (2,3'-Difluoro-biphenyl-4-carboxylic acid (4-pyridi...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 2.10E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Roche Research Center Curated by ChEMBL | Assay Description Inhibition of platelet activating factor receptor binding activity in dog platelets using [3H]-PAF as radioligand. | J Med Chem 32: 1814-20 (1989) BindingDB Entry DOI: 10.7270/Q2SQ8ZCJ | |||||||||||
More data for this Ligand-Target Pair |