Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Melanocortin receptor 5 (Mus musculus (Mouse)) | BDBM50027084 (Melatonan) | UniProtKB/SwissProt GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 0.190 | n/a | n/a | n/a | n/a |
University of Cergy-Pontoise Curated by ChEMBL | Assay Description Activity at mouse MC5R expressed in HEK293 cells assessed as cAMP accumulation by CRE/beta-galactosidase reporter gene assay | J Med Chem 57: 9424-34 (2014) Article DOI: 10.1021/jm501027w BindingDB Entry DOI: 10.7270/Q21G0NVT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 5 (Mus musculus (Mouse)) | BDBM50031469 (CHEMBL3358552) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 0.0700 | n/a | n/a | n/a | n/a |
University of Cergy-Pontoise Curated by ChEMBL | Assay Description Activity at mouse MC5R expressed in HEK293 cells assessed as cAMP accumulation by CRE/beta-galactosidase reporter gene assay | J Med Chem 57: 9424-34 (2014) Article DOI: 10.1021/jm501027w BindingDB Entry DOI: 10.7270/Q21G0NVT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 5 (Mus musculus (Mouse)) | BDBM50031470 (CHEMBL3358551) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 0.150 | n/a | n/a | n/a | n/a |
University of Cergy-Pontoise Curated by ChEMBL | Assay Description Activity at mouse MC5R expressed in HEK293 cells assessed as cAMP accumulation by CRE/beta-galactosidase reporter gene assay | J Med Chem 57: 9424-34 (2014) Article DOI: 10.1021/jm501027w BindingDB Entry DOI: 10.7270/Q21G0NVT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 5 (Mus musculus (Mouse)) | BDBM50031471 (CHEMBL3358550) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 0.150 | n/a | n/a | n/a | n/a |
University of Cergy-Pontoise Curated by ChEMBL | Assay Description Activity at mouse MC5R expressed in HEK293 cells assessed as cAMP accumulation by CRE/beta-galactosidase reporter gene assay | J Med Chem 57: 9424-34 (2014) Article DOI: 10.1021/jm501027w BindingDB Entry DOI: 10.7270/Q21G0NVT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 5 (Mus musculus (Mouse)) | BDBM50031473 (CHEMBL3358549) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | 0.0450 | n/a | n/a | n/a | n/a |
University of Cergy-Pontoise Curated by ChEMBL | Assay Description Activity at mouse MC5R expressed in HEK293 cells assessed as cAMP accumulation by CRE/beta-galactosidase reporter gene assay | J Med Chem 57: 9424-34 (2014) Article DOI: 10.1021/jm501027w BindingDB Entry DOI: 10.7270/Q21G0NVT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 5 (Mus musculus (Mouse)) | BDBM50031476 (CHEMBL3358548) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 1.90 | n/a | n/a | n/a | n/a |
University of Cergy-Pontoise Curated by ChEMBL | Assay Description Activity at mouse MC5R expressed in HEK293 cells assessed as cAMP accumulation by CRE/beta-galactosidase reporter gene assay | J Med Chem 57: 9424-34 (2014) Article DOI: 10.1021/jm501027w BindingDB Entry DOI: 10.7270/Q21G0NVT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 5 (Mus musculus (Mouse)) | BDBM50031477 (CHEMBL3358547) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 1.80 | n/a | n/a | n/a | n/a |
University of Cergy-Pontoise Curated by ChEMBL | Assay Description Activity at mouse MC5R expressed in HEK293 cells assessed as cAMP accumulation by CRE/beta-galactosidase reporter gene assay | J Med Chem 57: 9424-34 (2014) Article DOI: 10.1021/jm501027w BindingDB Entry DOI: 10.7270/Q21G0NVT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 5 (Mus musculus (Mouse)) | BDBM50031478 (CHEMBL3358546) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 0.130 | n/a | n/a | n/a | n/a |
University of Cergy-Pontoise Curated by ChEMBL | Assay Description Activity at mouse MC5R expressed in HEK293 cells assessed as cAMP accumulation by CRE/beta-galactosidase reporter gene assay | J Med Chem 57: 9424-34 (2014) Article DOI: 10.1021/jm501027w BindingDB Entry DOI: 10.7270/Q21G0NVT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 5 (Mus musculus (Mouse)) | BDBM50031479 (CHEMBL3358545) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 0.0420 | n/a | n/a | n/a | n/a |
University of Cergy-Pontoise Curated by ChEMBL | Assay Description Activity at mouse MC5R expressed in HEK293 cells assessed as cAMP accumulation by CRE/beta-galactosidase reporter gene assay | J Med Chem 57: 9424-34 (2014) Article DOI: 10.1021/jm501027w BindingDB Entry DOI: 10.7270/Q21G0NVT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 5 (Mus musculus (Mouse)) | BDBM50031486 (CHEMBL3358544) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 0.340 | n/a | n/a | n/a | n/a |
University of Cergy-Pontoise Curated by ChEMBL | Assay Description Activity at mouse MC5R expressed in HEK293 cells assessed as cAMP accumulation by CRE/beta-galactosidase reporter gene assay | J Med Chem 57: 9424-34 (2014) Article DOI: 10.1021/jm501027w BindingDB Entry DOI: 10.7270/Q21G0NVT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 5 (Mus musculus (Mouse)) | BDBM50031487 (CHEMBL3358543) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 1.90 | n/a | n/a | n/a | n/a |
University of Cergy-Pontoise Curated by ChEMBL | Assay Description Activity at mouse MC5R expressed in HEK293 cells assessed as cAMP accumulation by CRE/beta-galactosidase reporter gene assay | J Med Chem 57: 9424-34 (2014) Article DOI: 10.1021/jm501027w BindingDB Entry DOI: 10.7270/Q21G0NVT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 5 (Mus musculus (Mouse)) | BDBM50031488 (CHEMBL3358541) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 0.0510 | n/a | n/a | n/a | n/a |
University of Cergy-Pontoise Curated by ChEMBL | Assay Description Activity at mouse MC5R expressed in HEK293 cells assessed as cAMP accumulation by CRE/beta-galactosidase reporter gene assay | J Med Chem 57: 9424-34 (2014) Article DOI: 10.1021/jm501027w BindingDB Entry DOI: 10.7270/Q21G0NVT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 5 (Mus musculus (Mouse)) | BDBM50031489 (CHEMBL3352878) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 0.230 | n/a | n/a | n/a | n/a |
University of Cergy-Pontoise Curated by ChEMBL | Assay Description Activity at mouse MC5R expressed in HEK293 cells assessed as cAMP accumulation by CRE/beta-galactosidase reporter gene assay | J Med Chem 57: 9424-34 (2014) Article DOI: 10.1021/jm501027w BindingDB Entry DOI: 10.7270/Q21G0NVT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 5 (Mus musculus (Mouse)) | BDBM50031490 (CHEMBL3358540) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 0.130 | n/a | n/a | n/a | n/a |
University of Cergy-Pontoise Curated by ChEMBL | Assay Description Activity at mouse MC5R expressed in HEK293 cells assessed as cAMP accumulation by CRE/beta-galactosidase reporter gene assay | J Med Chem 57: 9424-34 (2014) Article DOI: 10.1021/jm501027w BindingDB Entry DOI: 10.7270/Q21G0NVT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 5 (Mus musculus (Mouse)) | BDBM50031492 (CHEMBL3358539) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 0.0860 | n/a | n/a | n/a | n/a |
University of Cergy-Pontoise Curated by ChEMBL | Assay Description Activity at mouse MC5R expressed in HEK293 cells assessed as cAMP accumulation by CRE/beta-galactosidase reporter gene assay | J Med Chem 57: 9424-34 (2014) Article DOI: 10.1021/jm501027w BindingDB Entry DOI: 10.7270/Q21G0NVT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 5 (Mus musculus (Mouse)) | BDBM50031493 (CHEMBL3358538) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 5 | n/a | n/a | n/a | n/a |
University of Cergy-Pontoise Curated by ChEMBL | Assay Description Activity at mouse MC5R expressed in HEK293 cells assessed as cAMP accumulation by CRE/beta-galactosidase reporter gene assay | J Med Chem 57: 9424-34 (2014) Article DOI: 10.1021/jm501027w BindingDB Entry DOI: 10.7270/Q21G0NVT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 5 (Mus musculus (Mouse)) | BDBM50031494 (CHEMBL3358537) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 1.90 | n/a | n/a | n/a | n/a |
University of Cergy-Pontoise Curated by ChEMBL | Assay Description Activity at mouse MC5R expressed in HEK293 cells assessed as cAMP accumulation by CRE/beta-galactosidase reporter gene assay | J Med Chem 57: 9424-34 (2014) Article DOI: 10.1021/jm501027w BindingDB Entry DOI: 10.7270/Q21G0NVT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 5 (Mus musculus (Mouse)) | BDBM50031495 (CHEMBL3358536) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 0.180 | n/a | n/a | n/a | n/a |
University of Cergy-Pontoise Curated by ChEMBL | Assay Description Activity at mouse MC5R expressed in HEK293 cells assessed as cAMP accumulation by CRE/beta-galactosidase reporter gene assay | J Med Chem 57: 9424-34 (2014) Article DOI: 10.1021/jm501027w BindingDB Entry DOI: 10.7270/Q21G0NVT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 5 (Mus musculus (Mouse)) | BDBM50031496 (CHEMBL3358535) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 0.130 | n/a | n/a | n/a | n/a |
University of Cergy-Pontoise Curated by ChEMBL | Assay Description Activity at mouse MC5R expressed in HEK293 cells assessed as cAMP accumulation by CRE/beta-galactosidase reporter gene assay | J Med Chem 57: 9424-34 (2014) Article DOI: 10.1021/jm501027w BindingDB Entry DOI: 10.7270/Q21G0NVT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 5 (Mus musculus (Mouse)) | BDBM50031497 (CHEMBL3358534) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 5.30 | n/a | n/a | n/a | n/a |
University of Cergy-Pontoise Curated by ChEMBL | Assay Description Activity at mouse MC5R expressed in HEK293 cells assessed as cAMP accumulation by CRE/beta-galactosidase reporter gene assay | J Med Chem 57: 9424-34 (2014) Article DOI: 10.1021/jm501027w BindingDB Entry DOI: 10.7270/Q21G0NVT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 5 (Mus musculus (Mouse)) | BDBM50031498 (CHEMBL3358533) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 3.20 | n/a | n/a | n/a | n/a |
University of Cergy-Pontoise Curated by ChEMBL | Assay Description Activity at mouse MC5R expressed in HEK293 cells assessed as cAMP accumulation by CRE/beta-galactosidase reporter gene assay | J Med Chem 57: 9424-34 (2014) Article DOI: 10.1021/jm501027w BindingDB Entry DOI: 10.7270/Q21G0NVT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 4 (Mus musculus) | BDBM50027084 (Melatonan) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 0.0600 | n/a | n/a | n/a | n/a |
University of Cergy-Pontoise Curated by ChEMBL | Assay Description Activity at mouse MC4R expressed in HEK293 cells assessed as cAMP accumulation by CRE/beta-galactosidase reporter gene assay | J Med Chem 57: 9424-34 (2014) Article DOI: 10.1021/jm501027w BindingDB Entry DOI: 10.7270/Q21G0NVT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 4 (Mus musculus) | BDBM50031469 (CHEMBL3358552) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 0.0670 | n/a | n/a | n/a | n/a |
University of Cergy-Pontoise Curated by ChEMBL | Assay Description Activity at mouse MC4R expressed in HEK293 cells assessed as cAMP accumulation by CRE/beta-galactosidase reporter gene assay | J Med Chem 57: 9424-34 (2014) Article DOI: 10.1021/jm501027w BindingDB Entry DOI: 10.7270/Q21G0NVT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 4 (Mus musculus) | BDBM50031470 (CHEMBL3358551) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 0.140 | n/a | n/a | n/a | n/a |
University of Cergy-Pontoise Curated by ChEMBL | Assay Description Activity at mouse MC4R expressed in HEK293 cells assessed as cAMP accumulation by CRE/beta-galactosidase reporter gene assay | J Med Chem 57: 9424-34 (2014) Article DOI: 10.1021/jm501027w BindingDB Entry DOI: 10.7270/Q21G0NVT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 4 (Mus musculus) | BDBM50031471 (CHEMBL3358550) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 0.140 | n/a | n/a | n/a | n/a |
University of Cergy-Pontoise Curated by ChEMBL | Assay Description Activity at mouse MC4R expressed in HEK293 cells assessed as cAMP accumulation by CRE/beta-galactosidase reporter gene assay | J Med Chem 57: 9424-34 (2014) Article DOI: 10.1021/jm501027w BindingDB Entry DOI: 10.7270/Q21G0NVT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 4 (Mus musculus) | BDBM50031473 (CHEMBL3358549) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | 0.0480 | n/a | n/a | n/a | n/a |
University of Cergy-Pontoise Curated by ChEMBL | Assay Description Activity at mouse MC4R expressed in HEK293 cells assessed as cAMP accumulation by CRE/beta-galactosidase reporter gene assay | J Med Chem 57: 9424-34 (2014) Article DOI: 10.1021/jm501027w BindingDB Entry DOI: 10.7270/Q21G0NVT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 4 (Mus musculus) | BDBM50031476 (CHEMBL3358548) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 0.850 | n/a | n/a | n/a | n/a |
University of Cergy-Pontoise Curated by ChEMBL | Assay Description Activity at mouse MC4R expressed in HEK293 cells assessed as cAMP accumulation by CRE/beta-galactosidase reporter gene assay | J Med Chem 57: 9424-34 (2014) Article DOI: 10.1021/jm501027w BindingDB Entry DOI: 10.7270/Q21G0NVT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 4 (Mus musculus) | BDBM50031477 (CHEMBL3358547) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 0.580 | n/a | n/a | n/a | n/a |
University of Cergy-Pontoise Curated by ChEMBL | Assay Description Activity at mouse MC4R expressed in HEK293 cells assessed as cAMP accumulation by CRE/beta-galactosidase reporter gene assay | J Med Chem 57: 9424-34 (2014) Article DOI: 10.1021/jm501027w BindingDB Entry DOI: 10.7270/Q21G0NVT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 4 (Mus musculus) | BDBM50031478 (CHEMBL3358546) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 0.140 | n/a | n/a | n/a | n/a |
University of Cergy-Pontoise Curated by ChEMBL | Assay Description Activity at mouse MC4R expressed in HEK293 cells assessed as cAMP accumulation by CRE/beta-galactosidase reporter gene assay | J Med Chem 57: 9424-34 (2014) Article DOI: 10.1021/jm501027w BindingDB Entry DOI: 10.7270/Q21G0NVT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 4 (Mus musculus) | BDBM50031479 (CHEMBL3358545) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 0.0510 | n/a | n/a | n/a | n/a |
University of Cergy-Pontoise Curated by ChEMBL | Assay Description Activity at mouse MC4R expressed in HEK293 cells assessed as cAMP accumulation by CRE/beta-galactosidase reporter gene assay | J Med Chem 57: 9424-34 (2014) Article DOI: 10.1021/jm501027w BindingDB Entry DOI: 10.7270/Q21G0NVT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 4 (Mus musculus) | BDBM50031486 (CHEMBL3358544) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 0.220 | n/a | n/a | n/a | n/a |
University of Cergy-Pontoise Curated by ChEMBL | Assay Description Activity at mouse MC4R expressed in HEK293 cells assessed as cAMP accumulation by CRE/beta-galactosidase reporter gene assay | J Med Chem 57: 9424-34 (2014) Article DOI: 10.1021/jm501027w BindingDB Entry DOI: 10.7270/Q21G0NVT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 4 (Mus musculus) | BDBM50031487 (CHEMBL3358543) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 1.60 | n/a | n/a | n/a | n/a |
University of Cergy-Pontoise Curated by ChEMBL | Assay Description Activity at mouse MC4R expressed in HEK293 cells assessed as cAMP accumulation by CRE/beta-galactosidase reporter gene assay | J Med Chem 57: 9424-34 (2014) Article DOI: 10.1021/jm501027w BindingDB Entry DOI: 10.7270/Q21G0NVT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 4 (Mus musculus) | BDBM50031499 (CHEMBL3358542) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 0.310 | n/a | n/a | n/a | n/a |
University of Cergy-Pontoise Curated by ChEMBL | Assay Description Activity at mouse MC4R expressed in HEK293 cells assessed as cAMP accumulation by CRE/beta-galactosidase reporter gene assay | J Med Chem 57: 9424-34 (2014) Article DOI: 10.1021/jm501027w BindingDB Entry DOI: 10.7270/Q21G0NVT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 4 (Mus musculus) | BDBM50031500 (CHEMBL2372859) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 0.210 | n/a | n/a | n/a | n/a |
University of Cergy-Pontoise Curated by ChEMBL | Assay Description Activity at mouse MC4R expressed in HEK293 cells assessed as cAMP accumulation by CRE/beta-galactosidase reporter gene assay | J Med Chem 57: 9424-34 (2014) Article DOI: 10.1021/jm501027w BindingDB Entry DOI: 10.7270/Q21G0NVT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 4 (Mus musculus) | BDBM50017181 (CHEMBL441738) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL DrugBank MCE PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 0.200 | n/a | n/a | n/a | n/a |
University of Cergy-Pontoise Curated by ChEMBL | Assay Description Activity at mouse MC4R expressed in HEK293 cells assessed as cAMP accumulation by CRE/beta-galactosidase reporter gene assay | J Med Chem 57: 9424-34 (2014) Article DOI: 10.1021/jm501027w BindingDB Entry DOI: 10.7270/Q21G0NVT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 4 (Mus musculus) | BDBM50031488 (CHEMBL3358541) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 0.0580 | n/a | n/a | n/a | n/a |
University of Cergy-Pontoise Curated by ChEMBL | Assay Description Activity at mouse MC4R expressed in HEK293 cells assessed as cAMP accumulation by CRE/beta-galactosidase reporter gene assay | J Med Chem 57: 9424-34 (2014) Article DOI: 10.1021/jm501027w BindingDB Entry DOI: 10.7270/Q21G0NVT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 4 (Mus musculus) | BDBM50031489 (CHEMBL3352878) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 0.290 | n/a | n/a | n/a | n/a |
University of Cergy-Pontoise Curated by ChEMBL | Assay Description Activity at mouse MC4R expressed in HEK293 cells assessed as cAMP accumulation by CRE/beta-galactosidase reporter gene assay | J Med Chem 57: 9424-34 (2014) Article DOI: 10.1021/jm501027w BindingDB Entry DOI: 10.7270/Q21G0NVT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 4 (Mus musculus) | BDBM50031490 (CHEMBL3358540) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 0.140 | n/a | n/a | n/a | n/a |
University of Cergy-Pontoise Curated by ChEMBL | Assay Description Activity at mouse MC4R expressed in HEK293 cells assessed as cAMP accumulation by CRE/beta-galactosidase reporter gene assay | J Med Chem 57: 9424-34 (2014) Article DOI: 10.1021/jm501027w BindingDB Entry DOI: 10.7270/Q21G0NVT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 4 (Mus musculus) | BDBM50031492 (CHEMBL3358539) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 0.0980 | n/a | n/a | n/a | n/a |
University of Cergy-Pontoise Curated by ChEMBL | Assay Description Activity at mouse MC4R expressed in HEK293 cells assessed as cAMP accumulation by CRE/beta-galactosidase reporter gene assay | J Med Chem 57: 9424-34 (2014) Article DOI: 10.1021/jm501027w BindingDB Entry DOI: 10.7270/Q21G0NVT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 4 (Mus musculus) | BDBM50031493 (CHEMBL3358538) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 2.20 | n/a | n/a | n/a | n/a |
University of Cergy-Pontoise Curated by ChEMBL | Assay Description Activity at mouse MC4R expressed in HEK293 cells assessed as cAMP accumulation by CRE/beta-galactosidase reporter gene assay | J Med Chem 57: 9424-34 (2014) Article DOI: 10.1021/jm501027w BindingDB Entry DOI: 10.7270/Q21G0NVT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 4 (Mus musculus) | BDBM50031494 (CHEMBL3358537) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 0.810 | n/a | n/a | n/a | n/a |
University of Cergy-Pontoise Curated by ChEMBL | Assay Description Activity at mouse MC4R expressed in HEK293 cells assessed as cAMP accumulation by CRE/beta-galactosidase reporter gene assay | J Med Chem 57: 9424-34 (2014) Article DOI: 10.1021/jm501027w BindingDB Entry DOI: 10.7270/Q21G0NVT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 4 (Mus musculus) | BDBM50031495 (CHEMBL3358536) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 0.190 | n/a | n/a | n/a | n/a |
University of Cergy-Pontoise Curated by ChEMBL | Assay Description Activity at mouse MC4R expressed in HEK293 cells assessed as cAMP accumulation by CRE/beta-galactosidase reporter gene assay | J Med Chem 57: 9424-34 (2014) Article DOI: 10.1021/jm501027w BindingDB Entry DOI: 10.7270/Q21G0NVT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 4 (Mus musculus) | BDBM50031496 (CHEMBL3358535) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 0.130 | n/a | n/a | n/a | n/a |
University of Cergy-Pontoise Curated by ChEMBL | Assay Description Activity at mouse MC4R expressed in HEK293 cells assessed as cAMP accumulation by CRE/beta-galactosidase reporter gene assay | J Med Chem 57: 9424-34 (2014) Article DOI: 10.1021/jm501027w BindingDB Entry DOI: 10.7270/Q21G0NVT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 4 (Mus musculus) | BDBM50031497 (CHEMBL3358534) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 2.20 | n/a | n/a | n/a | n/a |
University of Cergy-Pontoise Curated by ChEMBL | Assay Description Activity at mouse MC4R expressed in HEK293 cells assessed as cAMP accumulation by CRE/beta-galactosidase reporter gene assay | J Med Chem 57: 9424-34 (2014) Article DOI: 10.1021/jm501027w BindingDB Entry DOI: 10.7270/Q21G0NVT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 4 (Mus musculus) | BDBM50031498 (CHEMBL3358533) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 1.5 | n/a | n/a | n/a | n/a |
University of Cergy-Pontoise Curated by ChEMBL | Assay Description Activity at mouse MC4R expressed in HEK293 cells assessed as cAMP accumulation by CRE/beta-galactosidase reporter gene assay | J Med Chem 57: 9424-34 (2014) Article DOI: 10.1021/jm501027w BindingDB Entry DOI: 10.7270/Q21G0NVT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 3 (Mus musculus) | BDBM50027084 (Melatonan) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 0.180 | n/a | n/a | n/a | n/a |
University of Cergy-Pontoise Curated by ChEMBL | Assay Description Activity at mouse MC3R expressed in HEK293 cells assessed as cAMP accumulation by CRE/beta-galactosidase reporter gene assay | J Med Chem 57: 9424-34 (2014) Article DOI: 10.1021/jm501027w BindingDB Entry DOI: 10.7270/Q21G0NVT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 3 (Mus musculus) | BDBM50031489 (CHEMBL3352878) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 2.30 | n/a | n/a | n/a | n/a |
University of Cergy-Pontoise Curated by ChEMBL | Assay Description Activity at mouse MC3R expressed in HEK293 cells assessed as cAMP accumulation by CRE/beta-galactosidase reporter gene assay | J Med Chem 57: 9424-34 (2014) Article DOI: 10.1021/jm501027w BindingDB Entry DOI: 10.7270/Q21G0NVT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 3 (Mus musculus) | BDBM50031490 (CHEMBL3358540) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 1.30 | n/a | n/a | n/a | n/a |
University of Cergy-Pontoise Curated by ChEMBL | Assay Description Activity at mouse MC3R expressed in HEK293 cells assessed as cAMP accumulation by CRE/beta-galactosidase reporter gene assay | J Med Chem 57: 9424-34 (2014) Article DOI: 10.1021/jm501027w BindingDB Entry DOI: 10.7270/Q21G0NVT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 3 (Mus musculus) | BDBM50031492 (CHEMBL3358539) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 0.860 | n/a | n/a | n/a | n/a |
University of Cergy-Pontoise Curated by ChEMBL | Assay Description Activity at mouse MC3R expressed in HEK293 cells assessed as cAMP accumulation by CRE/beta-galactosidase reporter gene assay | J Med Chem 57: 9424-34 (2014) Article DOI: 10.1021/jm501027w BindingDB Entry DOI: 10.7270/Q21G0NVT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanocortin receptor 3 (Mus musculus) | BDBM50031493 (CHEMBL3358538) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 3.70 | n/a | n/a | n/a | n/a |
University of Cergy-Pontoise Curated by ChEMBL | Assay Description Activity at mouse MC3R expressed in HEK293 cells assessed as cAMP accumulation by CRE/beta-galactosidase reporter gene assay | J Med Chem 57: 9424-34 (2014) Article DOI: 10.1021/jm501027w BindingDB Entry DOI: 10.7270/Q21G0NVT | |||||||||||
More data for this Ligand-Target Pair |
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