Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Proteinase-activated receptor 1 (Homo sapiens (Human)) | BDBM50173419 ((3R,3aS,4S,4aR,8aS,9aR)-3-Methyl-4-{(E)-2-[5-(3-tr...) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 2.70 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Schering-Plough Research Institute Curated by ChEMBL | Assay Description Inhibitory constant aganist Protease-activated receptor 1 | J Med Chem 48: 5884-7 (2005) Article DOI: 10.1021/jm0502236 BindingDB Entry DOI: 10.7270/Q2V69J5Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Proteinase-activated receptor 1 (Homo sapiens (Human)) | BDBM50173417 ((3R,3aS,4S,4aR,8aS,9aR)-4-(2-(6-ethylpyridin-2-yl)...) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 12 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Schering-Plough Research Institute Curated by ChEMBL | Assay Description Inhibitory constant aganist Protease-activated receptor 1 | J Med Chem 48: 5884-7 (2005) Article DOI: 10.1021/jm0502236 BindingDB Entry DOI: 10.7270/Q2V69J5Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Proteinase-activated receptor 1 (Homo sapiens (Human)) | BDBM50173437 ((3R,3aS,4S,4aR,8aS,9aR)-4-{(E)-2-[5-(3-Chloro-phen...) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 10 | n/a | n/a | n/a | n/a | n/a | n/a |
Schering-Plough Research Institute Curated by ChEMBL | Assay Description In vitro inhibitory concentration aganist human protease activated receptor 1 using [3H]-haTRAP as radioligand | J Med Chem 48: 5884-7 (2005) Article DOI: 10.1021/jm0502236 BindingDB Entry DOI: 10.7270/Q2V69J5Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Proteinase-activated receptor 1 (Homo sapiens (Human)) | BDBM50173419 ((3R,3aS,4S,4aR,8aS,9aR)-3-Methyl-4-{(E)-2-[5-(3-tr...) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 11 | n/a | n/a | n/a | n/a | n/a | n/a |
Schering-Plough Research Institute Curated by ChEMBL | Assay Description In vitro inhibitory concentration aganist human protease activated receptor 1 using [3H]-haTRAP as radioligand | J Med Chem 48: 5884-7 (2005) Article DOI: 10.1021/jm0502236 BindingDB Entry DOI: 10.7270/Q2V69J5Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Proteinase-activated receptor 1 (Homo sapiens (Human)) | BDBM50173433 ((3R,3aS,4S,4aR,8aS,9aR)-4-{(E)-2-[5-(2-Methoxy-phe...) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 11 | n/a | n/a | n/a | n/a | n/a | n/a |
Schering-Plough Research Institute Curated by ChEMBL | Assay Description In vitro inhibitory concentration aganist human protease activated receptor 1 using [3H]-haTRAP as radioligand | J Med Chem 48: 5884-7 (2005) Article DOI: 10.1021/jm0502236 BindingDB Entry DOI: 10.7270/Q2V69J5Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Proteinase-activated receptor 1 (Homo sapiens (Human)) | BDBM50173419 ((3R,3aS,4S,4aR,8aS,9aR)-3-Methyl-4-{(E)-2-[5-(3-tr...) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 11 | n/a | n/a | n/a | n/a | n/a | n/a |
Schering-Plough Research Institute Curated by ChEMBL | Assay Description In vitro inhibitory concentration aganist human protease activated receptor 1 using [3H]-haTRAP as radioligand | J Med Chem 48: 5884-7 (2005) Article DOI: 10.1021/jm0502236 BindingDB Entry DOI: 10.7270/Q2V69J5Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Proteinase-activated receptor 1 (Homo sapiens (Human)) | BDBM50173409 ((3R,3aS,4S,4aR,8aS,9aR)-3-Methyl-4-[(E)-2-(5-m-tol...) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 13 | n/a | n/a | n/a | n/a | n/a | n/a |
Schering-Plough Research Institute Curated by ChEMBL | Assay Description In vitro inhibitory concentration aganist human protease activated receptor 1 using [3H]-haTRAP as radioligand | J Med Chem 48: 5884-7 (2005) Article DOI: 10.1021/jm0502236 BindingDB Entry DOI: 10.7270/Q2V69J5Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Proteinase-activated receptor 1 (Homo sapiens (Human)) | BDBM50173410 ((3R,3aS,4S,4aR,8aS,9aR)-3-Methyl-4-[(E)-2-(5-o-tol...) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 14 | n/a | n/a | n/a | n/a | n/a | n/a |
Schering-Plough Research Institute Curated by ChEMBL | Assay Description In vitro inhibitory concentration aganist human protease activated receptor 1 using [3H]-haTRAP as radioligand | J Med Chem 48: 5884-7 (2005) Article DOI: 10.1021/jm0502236 BindingDB Entry DOI: 10.7270/Q2V69J5Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Proteinase-activated receptor 1 (Homo sapiens (Human)) | BDBM50173418 ((3R,3aS,4S,4aR,8aS,9aR)-4-{(E)-2-[5-(3-Isopropyl-p...) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 19 | n/a | n/a | n/a | n/a | n/a | n/a |
Schering-Plough Research Institute Curated by ChEMBL | Assay Description In vitro inhibitory concentration aganist human protease activated receptor 1 using [3H]-haTRAP as radioligand | J Med Chem 48: 5884-7 (2005) Article DOI: 10.1021/jm0502236 BindingDB Entry DOI: 10.7270/Q2V69J5Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Proteinase-activated receptor 1 (Homo sapiens (Human)) | BDBM50173451 ((3R,3aS,4S,4aR,8aS,9aR)-4-[(E)-2-(5-Benzyloxy-pyri...) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 19 | n/a | n/a | n/a | n/a | n/a | n/a |
Schering-Plough Research Institute Curated by ChEMBL | Assay Description In vitro inhibitory concentration aganist human protease activated receptor 1 using [3H]-haTRAP as radioligand | J Med Chem 48: 5884-7 (2005) Article DOI: 10.1021/jm0502236 BindingDB Entry DOI: 10.7270/Q2V69J5Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Proteinase-activated receptor 1 (Homo sapiens (Human)) | BDBM50173417 ((3R,3aS,4S,4aR,8aS,9aR)-4-(2-(6-ethylpyridin-2-yl)...) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 20 | n/a | n/a | n/a | n/a | n/a | n/a |
Schering-Plough Research Institute Curated by ChEMBL | Assay Description In vitro inhibitory concentration aganist human protease activated receptor 1 using [3H]-haTRAP as radioligand | J Med Chem 48: 5884-7 (2005) Article DOI: 10.1021/jm0502236 BindingDB Entry DOI: 10.7270/Q2V69J5Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Proteinase-activated receptor 1 (Homo sapiens (Human)) | BDBM50173438 ((3R,3aS,4S,4aR,8aS,9aR)-4-{(E)-2-[5-(2-Fluoro-phen...) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 22 | n/a | n/a | n/a | n/a | n/a | n/a |
Schering-Plough Research Institute Curated by ChEMBL | Assay Description In vitro inhibitory concentration aganist human protease activated receptor 1 using [3H]-haTRAP as radioligand | J Med Chem 48: 5884-7 (2005) Article DOI: 10.1021/jm0502236 BindingDB Entry DOI: 10.7270/Q2V69J5Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Proteinase-activated receptor 1 (Homo sapiens (Human)) | BDBM50173436 (3-{6-[(E)-2-((3R,3aS,4S,4aR,8aS,9aR)-3-Methyl-1-ox...) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 25 | n/a | n/a | n/a | n/a | n/a | n/a |
Schering-Plough Research Institute Curated by ChEMBL | Assay Description In vitro inhibitory concentration aganist human protease activated receptor 1 using [3H]-haTRAP as radioligand | J Med Chem 48: 5884-7 (2005) Article DOI: 10.1021/jm0502236 BindingDB Entry DOI: 10.7270/Q2V69J5Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Proteinase-activated receptor 1 (Homo sapiens (Human)) | BDBM50173430 ((3R,3aS,4S,4aR,8aS,9aR)-4-{(E)-2-[5-(3-Bromo-pheny...) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 25 | n/a | n/a | n/a | n/a | n/a | n/a |
Schering-Plough Research Institute Curated by ChEMBL | Assay Description In vitro inhibitory concentration aganist human protease activated receptor 1 using [3H]-haTRAP as radioligand | J Med Chem 48: 5884-7 (2005) Article DOI: 10.1021/jm0502236 BindingDB Entry DOI: 10.7270/Q2V69J5Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Proteinase-activated receptor 1 (Homo sapiens (Human)) | BDBM50173447 ((3R,3aS,4S,4aR,8aS,9aR)-4-{(E)-2-[5-(2-Chloro-phen...) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 26 | n/a | n/a | n/a | n/a | n/a | n/a |
Schering-Plough Research Institute Curated by ChEMBL | Assay Description In vitro inhibitory concentration aganist human protease activated receptor 1 using [3H]-haTRAP as radioligand | J Med Chem 48: 5884-7 (2005) Article DOI: 10.1021/jm0502236 BindingDB Entry DOI: 10.7270/Q2V69J5Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Proteinase-activated receptor 1 (Homo sapiens (Human)) | BDBM50173421 ((3R,3aS,4S,4aR,8aS,9aR)-3-Methyl-4-[(E)-2-(5-pheny...) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 27 | n/a | n/a | n/a | n/a | n/a | n/a |
Schering-Plough Research Institute Curated by ChEMBL | Assay Description In vitro inhibitory concentration aganist human protease activated receptor 1 using [3H]-haTRAP as radioligand | J Med Chem 48: 5884-7 (2005) Article DOI: 10.1021/jm0502236 BindingDB Entry DOI: 10.7270/Q2V69J5Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Proteinase-activated receptor 1 (Homo sapiens (Human)) | BDBM50173446 ((3R,3aS,4S,4aR,8aS,9aR)-4-{(E)-2-[5-(3-Methoxy-phe...) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 28 | n/a | n/a | n/a | n/a | n/a | n/a |
Schering-Plough Research Institute Curated by ChEMBL | Assay Description In vitro inhibitory concentration aganist human protease activated receptor 1 using [3H]-haTRAP as radioligand | J Med Chem 48: 5884-7 (2005) Article DOI: 10.1021/jm0502236 BindingDB Entry DOI: 10.7270/Q2V69J5Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Proteinase-activated receptor 1 (Homo sapiens (Human)) | BDBM50173445 ((3R,3aS,4S,4aR,8aS,9aR)-4-{(E)-2-[5-(3-Fluoro-phen...) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 35 | n/a | n/a | n/a | n/a | n/a | n/a |
Schering-Plough Research Institute Curated by ChEMBL | Assay Description In vitro inhibitory concentration aganist human protease activated receptor 1 using [3H]-haTRAP as radioligand | J Med Chem 48: 5884-7 (2005) Article DOI: 10.1021/jm0502236 BindingDB Entry DOI: 10.7270/Q2V69J5Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Proteinase-activated receptor 1 (Homo sapiens (Human)) | BDBM50173419 ((3R,3aS,4S,4aR,8aS,9aR)-3-Methyl-4-{(E)-2-[5-(3-tr...) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 44 | n/a | n/a | n/a | n/a | n/a | n/a |
Schering-Plough Research Institute Curated by ChEMBL | Assay Description In vitro inhibitory concentration aganist human protease activated receptor 1 using [3H]-haTRAP as radioligand | J Med Chem 48: 5884-7 (2005) Article DOI: 10.1021/jm0502236 BindingDB Entry DOI: 10.7270/Q2V69J5Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Proteinase-activated receptor 1 (Homo sapiens (Human)) | BDBM50173434 (2-{6-[(E)-2-((3R,3aS,4S,4aR,8aS,9aR)-3-Methyl-1-ox...) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 44 | n/a | n/a | n/a | n/a | n/a | n/a |
Schering-Plough Research Institute Curated by ChEMBL | Assay Description In vitro inhibitory concentration aganist human protease activated receptor 1 using [3H]-haTRAP as radioligand | J Med Chem 48: 5884-7 (2005) Article DOI: 10.1021/jm0502236 BindingDB Entry DOI: 10.7270/Q2V69J5Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Proteinase-activated receptor 1 (Homo sapiens (Human)) | BDBM50173450 ((3R,3aS,4S,4aR,8aS,9aR)-3-Methyl-4-{(E)-2-[5-(2-tr...) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 46 | n/a | n/a | n/a | n/a | n/a | n/a |
Schering-Plough Research Institute Curated by ChEMBL | Assay Description In vitro inhibitory concentration aganist human protease activated receptor 1 using [3H]-haTRAP as radioligand | J Med Chem 48: 5884-7 (2005) Article DOI: 10.1021/jm0502236 BindingDB Entry DOI: 10.7270/Q2V69J5Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Proteinase-activated receptor 1 (Homo sapiens (Human)) | BDBM50173417 ((3R,3aS,4S,4aR,8aS,9aR)-4-(2-(6-ethylpyridin-2-yl)...) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 85 | n/a | n/a | n/a | n/a | n/a | n/a |
Schering-Plough Research Institute Curated by ChEMBL | Assay Description In vitro inhibitory concentration aganist human protease activated receptor 1 using [3H]-haTRAP as radioligand | J Med Chem 48: 5884-7 (2005) Article DOI: 10.1021/jm0502236 BindingDB Entry DOI: 10.7270/Q2V69J5Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Proteinase-activated receptor 1 (Homo sapiens (Human)) | BDBM50173417 ((3R,3aS,4S,4aR,8aS,9aR)-4-(2-(6-ethylpyridin-2-yl)...) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 85 | n/a | n/a | n/a | n/a | n/a | n/a |
Schering-Plough Research Institute Curated by ChEMBL | Assay Description In vitro inhibitory concentration aganist human protease activated receptor 1 using [3H]-haTRAP as radioligand | J Med Chem 48: 5884-7 (2005) Article DOI: 10.1021/jm0502236 BindingDB Entry DOI: 10.7270/Q2V69J5Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Proteinase-activated receptor 1 (Homo sapiens (Human)) | BDBM50173431 (3-{6-[(E)-2-((3R,3aS,4S,4aR,8aS,9aR)-3-Methyl-1-ox...) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | 100 | n/a | n/a | n/a | n/a | n/a | n/a |
Schering-Plough Research Institute Curated by ChEMBL | Assay Description In vitro inhibitory concentration aganist human protease activated receptor 1 using [3H]-haTRAP as radioligand | J Med Chem 48: 5884-7 (2005) Article DOI: 10.1021/jm0502236 BindingDB Entry DOI: 10.7270/Q2V69J5Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Proteinase-activated receptor 1 (Homo sapiens (Human)) | BDBM50173415 ((3R,3aS,4S,4aR,8aS,9aR)-4-[(E)-2-(6-Butyl-pyridin-...) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 143 | n/a | n/a | n/a | n/a | n/a | n/a |
Schering-Plough Research Institute Curated by ChEMBL | Assay Description In vitro inhibitory concentration aganist human protease activated receptor 1 using [3H]-haTRAP as radioligand | J Med Chem 48: 5884-7 (2005) Article DOI: 10.1021/jm0502236 BindingDB Entry DOI: 10.7270/Q2V69J5Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Proteinase-activated receptor 1 (Homo sapiens (Human)) | BDBM50173424 ((3R,3aS,4S,4aR,8aS,9aR)-3-Methyl-4-[(E)-2-(6-vinyl...) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 150 | n/a | n/a | n/a | n/a | n/a | n/a |
Schering-Plough Research Institute Curated by ChEMBL | Assay Description In vitro inhibitory concentration aganist human protease activated receptor 1 using [3H]-haTRAP as radioligand | J Med Chem 48: 5884-7 (2005) Article DOI: 10.1021/jm0502236 BindingDB Entry DOI: 10.7270/Q2V69J5Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Proteinase-activated receptor 1 (Homo sapiens (Human)) | BDBM50173426 ((3R,3aS,4S,4aR,8aS,9aR)-4-{(E)-2-[5-(4-Methoxy-phe...) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 204 | n/a | n/a | n/a | n/a | n/a | n/a |
Schering-Plough Research Institute Curated by ChEMBL | Assay Description In vitro inhibitory concentration aganist human protease activated receptor 1 using [3H]-haTRAP as radioligand | J Med Chem 48: 5884-7 (2005) Article DOI: 10.1021/jm0502236 BindingDB Entry DOI: 10.7270/Q2V69J5Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Proteinase-activated receptor 1 (Homo sapiens (Human)) | BDBM50173427 ((3R,3aS,4S,4aR,8aS,9aR)-4-[(E)-2-(6-Cyclopropyl-py...) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 210 | n/a | n/a | n/a | n/a | n/a | n/a |
Schering-Plough Research Institute Curated by ChEMBL | Assay Description In vitro inhibitory concentration aganist human protease activated receptor 1 using [3H]-haTRAP as radioligand | J Med Chem 48: 5884-7 (2005) Article DOI: 10.1021/jm0502236 BindingDB Entry DOI: 10.7270/Q2V69J5Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Proteinase-activated receptor 1 (Homo sapiens (Human)) | BDBM50173449 ((3R,3aS,4S,4aR,8aS,9aR)-3-Methyl-4-[(E)-2-(6-propy...) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 250 | n/a | n/a | n/a | n/a | n/a | n/a |
Schering-Plough Research Institute Curated by ChEMBL | Assay Description In vitro inhibitory concentration aganist human protease activated receptor 1 using [3H]-haTRAP as radioligand | J Med Chem 48: 5884-7 (2005) Article DOI: 10.1021/jm0502236 BindingDB Entry DOI: 10.7270/Q2V69J5Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Proteinase-activated receptor 1 (Homo sapiens (Human)) | BDBM50173425 ((3R,3aS,4S,4aR,8aS,9aR)-3-Methyl-4-[(E)-2-(6-methy...) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 300 | n/a | n/a | n/a | n/a | n/a | n/a |
Schering-Plough Research Institute Curated by ChEMBL | Assay Description In vitro inhibitory concentration aganist human protease activated receptor 1 using [3H]-haTRAP as radioligand | J Med Chem 48: 5884-7 (2005) Article DOI: 10.1021/jm0502236 BindingDB Entry DOI: 10.7270/Q2V69J5Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Proteinase-activated receptor 1 (Homo sapiens (Human)) | BDBM50173425 ((3R,3aS,4S,4aR,8aS,9aR)-3-Methyl-4-[(E)-2-(6-methy...) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 300 | n/a | n/a | n/a | n/a | n/a | n/a |
Schering-Plough Research Institute Curated by ChEMBL | Assay Description In vitro inhibitory concentration aganist human protease activated receptor 1 using [3H]-haTRAP as radioligand | J Med Chem 48: 5884-7 (2005) Article DOI: 10.1021/jm0502236 BindingDB Entry DOI: 10.7270/Q2V69J5Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Proteinase-activated receptor 1 (Homo sapiens (Human)) | BDBM50173412 ((3R,3aS,4S,4aR,8aS,9aR)-3-Methyl-4-{(E)-2-[5-(4-tr...) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >300 | n/a | n/a | n/a | n/a | n/a | n/a |
Schering-Plough Research Institute Curated by ChEMBL | Assay Description In vitro inhibitory concentration aganist human protease activated receptor 1 using [3H]-haTRAP as radioligand | J Med Chem 48: 5884-7 (2005) Article DOI: 10.1021/jm0502236 BindingDB Entry DOI: 10.7270/Q2V69J5Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Proteinase-activated receptor 1 (Homo sapiens (Human)) | BDBM50173414 ((3R,3aS,4S,4aR,8aS,9aR)-4-[(E)-2-(5-Methoxy-pyridi...) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 325 | n/a | n/a | n/a | n/a | n/a | n/a |
Schering-Plough Research Institute Curated by ChEMBL | Assay Description In vitro inhibitory concentration aganist human protease activated receptor 1 using [3H]-haTRAP as radioligand | J Med Chem 48: 5884-7 (2005) Article DOI: 10.1021/jm0502236 BindingDB Entry DOI: 10.7270/Q2V69J5Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Proteinase-activated receptor 1 (Homo sapiens (Human)) | BDBM50173420 ((3R,3aS,4S,4aR,8aS,9aR)-3-Methyl-4-[(E)-2-(5-p-tol...) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 325 | n/a | n/a | n/a | n/a | n/a | n/a |
Schering-Plough Research Institute Curated by ChEMBL | Assay Description In vitro inhibitory concentration aganist human protease activated receptor 1 using [3H]-haTRAP as radioligand | J Med Chem 48: 5884-7 (2005) Article DOI: 10.1021/jm0502236 BindingDB Entry DOI: 10.7270/Q2V69J5Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Proteinase-activated receptor 1 (Homo sapiens (Human)) | BDBM50173411 ((3S,3aR,4R,4aS,8aR,9aS)-4-[(E)-2-(6-Ethyl-pyridin-...) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 400 | n/a | n/a | n/a | n/a | n/a | n/a |
Schering-Plough Research Institute Curated by ChEMBL | Assay Description In vitro inhibitory concentration aganist human protease activated receptor 1 using [3H]-haTRAP as radioligand | J Med Chem 48: 5884-7 (2005) Article DOI: 10.1021/jm0502236 BindingDB Entry DOI: 10.7270/Q2V69J5Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Proteinase-activated receptor 1 (Homo sapiens (Human)) | BDBM50173443 ((3R,3aS,4S,4aR,8aS,9aR)-4-{(E)-2-[5-(4-Fluoro-phen...) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 467 | n/a | n/a | n/a | n/a | n/a | n/a |
Schering-Plough Research Institute Curated by ChEMBL | Assay Description In vitro inhibitory concentration aganist human protease activated receptor 1 using [3H]-haTRAP as radioligand | J Med Chem 48: 5884-7 (2005) Article DOI: 10.1021/jm0502236 BindingDB Entry DOI: 10.7270/Q2V69J5Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Proteinase-activated receptor 1 (Homo sapiens (Human)) | BDBM50173422 ((3R,3aS,4S,4aR,8aS,9aR)-4-[(E)-2-(6-Isobutyl-pyrid...) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 550 | n/a | n/a | n/a | n/a | n/a | n/a |
Schering-Plough Research Institute Curated by ChEMBL | Assay Description In vitro inhibitory concentration aganist human protease activated receptor 1 using [3H]-haTRAP as radioligand | J Med Chem 48: 5884-7 (2005) Article DOI: 10.1021/jm0502236 BindingDB Entry DOI: 10.7270/Q2V69J5Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Proteinase-activated receptor 1 (Homo sapiens (Human)) | BDBM50173439 ((3R,3aS,4S,4aR,8aS,9aR)-4-[(E)-2-(6-Isopropyl-pyri...) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 725 | n/a | n/a | n/a | n/a | n/a | n/a |
Schering-Plough Research Institute Curated by ChEMBL | Assay Description In vitro inhibitory concentration aganist human protease activated receptor 1 using [3H]-haTRAP as radioligand | J Med Chem 48: 5884-7 (2005) Article DOI: 10.1021/jm0502236 BindingDB Entry DOI: 10.7270/Q2V69J5Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Proteinase-activated receptor 1 (Homo sapiens (Human)) | BDBM50173440 ((3R,3aS,4S,4aR,8aS,9aR)-4-[(E)-2-(6-Methoxymethyl-...) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 850 | n/a | n/a | n/a | n/a | n/a | n/a |
Schering-Plough Research Institute Curated by ChEMBL | Assay Description In vitro inhibitory concentration aganist human protease activated receptor 1 using [3H]-haTRAP as radioligand | J Med Chem 48: 5884-7 (2005) Article DOI: 10.1021/jm0502236 BindingDB Entry DOI: 10.7270/Q2V69J5Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Proteinase-activated receptor 1 (Homo sapiens (Human)) | BDBM50173444 ((3R,3aS,4S,4aR,8aS,9aR)-4-[(E)-2-(6-Benzyl-pyridin...) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 900 | n/a | n/a | n/a | n/a | n/a | n/a |
Schering-Plough Research Institute Curated by ChEMBL | Assay Description In vitro inhibitory concentration aganist human protease activated receptor 1 using [3H]-haTRAP as radioligand | J Med Chem 48: 5884-7 (2005) Article DOI: 10.1021/jm0502236 BindingDB Entry DOI: 10.7270/Q2V69J5Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Proteinase-activated receptor 1 (Homo sapiens (Human)) | BDBM50173432 ((3R,3aS,4S,4aR,8aS,9aR)-4-{(E)-2-[5-(4-Chloro-phen...) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Schering-Plough Research Institute Curated by ChEMBL | Assay Description In vitro inhibitory concentration aganist human protease activated receptor 1 using [3H]-haTRAP as radioligand | J Med Chem 48: 5884-7 (2005) Article DOI: 10.1021/jm0502236 BindingDB Entry DOI: 10.7270/Q2V69J5Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Proteinase-activated receptor 1 (Homo sapiens (Human)) | BDBM50173429 ((3R,3aS,4S,4aR,8aS,9aR)-3-Methyl-4-[(E)-2-(5-methy...) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 1.10E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Schering-Plough Research Institute Curated by ChEMBL | Assay Description In vitro inhibitory concentration aganist human protease activated receptor 1 using [3H]-haTRAP as radioligand | J Med Chem 48: 5884-7 (2005) Article DOI: 10.1021/jm0502236 BindingDB Entry DOI: 10.7270/Q2V69J5Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Proteinase-activated receptor 1 (Homo sapiens (Human)) | BDBM50173441 ((3R,3aS,4S,4aR,8aS,9aR)-3-Methyl-4-[(E)-2-(6-methy...) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.25E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Schering-Plough Research Institute Curated by ChEMBL | Assay Description In vitro inhibitory concentration aganist human protease activated receptor 1 using [3H]-haTRAP as radioligand | J Med Chem 48: 5884-7 (2005) Article DOI: 10.1021/jm0502236 BindingDB Entry DOI: 10.7270/Q2V69J5Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Proteinase-activated receptor 1 (Homo sapiens (Human)) | BDBM50173442 ((3S,3aR,4R,4aS,8aR,9aS)-3-Methyl-4-[(E)-2-(6-methy...) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.50E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Schering-Plough Research Institute Curated by ChEMBL | Assay Description In vitro inhibitory concentration aganist human protease activated receptor 1 using [3H]-haTRAP as radioligand | J Med Chem 48: 5884-7 (2005) Article DOI: 10.1021/jm0502236 BindingDB Entry DOI: 10.7270/Q2V69J5Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Proteinase-activated receptor 1 (Homo sapiens (Human)) | BDBM50173428 ((3R,3aS,4S,4aR,8aS,9aR)-4-[(E)-2-(6-Hydroxymethyl-...) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.50E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Schering-Plough Research Institute Curated by ChEMBL | Assay Description In vitro inhibitory concentration aganist human protease activated receptor 1 using [3H]-haTRAP as radioligand | J Med Chem 48: 5884-7 (2005) Article DOI: 10.1021/jm0502236 BindingDB Entry DOI: 10.7270/Q2V69J5Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Proteinase-activated receptor 1 (Homo sapiens (Human)) | BDBM50173413 ((3R,3aS,4S,4aR,8aS,9aR)-3-Methyl-4-[(E)-2-(4-methy...) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 2.10E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Schering-Plough Research Institute Curated by ChEMBL | Assay Description In vitro inhibitory concentration aganist human protease activated receptor 1 using [3H]-haTRAP as radioligand | J Med Chem 48: 5884-7 (2005) Article DOI: 10.1021/jm0502236 BindingDB Entry DOI: 10.7270/Q2V69J5Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Proteinase-activated receptor 1 (Homo sapiens (Human)) | BDBM50173435 ((3R,3aS,4S,4aR,8aS,9aR)-4-[(E)-2-(6-Hexyl-pyridin-...) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 3.50E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Schering-Plough Research Institute Curated by ChEMBL | Assay Description In vitro inhibitory concentration aganist human protease activated receptor 1 using [3H]-haTRAP as radioligand | J Med Chem 48: 5884-7 (2005) Article DOI: 10.1021/jm0502236 BindingDB Entry DOI: 10.7270/Q2V69J5Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Proteinase-activated receptor 1 (Homo sapiens (Human)) | BDBM50173448 ((3R,3aS,4S,4aR,8aS,9aR)-4-[(E)-2-(5-Benzyl-pyridin...) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 3.68E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Schering-Plough Research Institute Curated by ChEMBL | Assay Description In vitro inhibitory concentration aganist human protease activated receptor 1 using [3H]-haTRAP as radioligand | J Med Chem 48: 5884-7 (2005) Article DOI: 10.1021/jm0502236 BindingDB Entry DOI: 10.7270/Q2V69J5Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Proteinase-activated receptor 1 (Homo sapiens (Human)) | BDBM50173416 ((3R,3aS,4S,4aR,8aS,9aR)-3-Methyl-4-((E)-2-pyridin-...) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 4.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Schering-Plough Research Institute Curated by ChEMBL | Assay Description In vitro inhibitory concentration aganist human protease activated receptor 1 using [3H]-haTRAP as radioligand | J Med Chem 48: 5884-7 (2005) Article DOI: 10.1021/jm0502236 BindingDB Entry DOI: 10.7270/Q2V69J5Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Proteinase-activated receptor 1 (Homo sapiens (Human)) | BDBM50173423 ((3R,3aS,4S,4aR,8aS,9aR)-3-Methyl-4-[(E)-2-(3-methy...) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >5.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Schering-Plough Research Institute Curated by ChEMBL | Assay Description In vitro inhibitory concentration aganist human protease activated receptor 1 using [3H]-haTRAP as radioligand | J Med Chem 48: 5884-7 (2005) Article DOI: 10.1021/jm0502236 BindingDB Entry DOI: 10.7270/Q2V69J5Q | |||||||||||
More data for this Ligand-Target Pair |