Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
C-X-C chemokine receptor type 3 (Homo sapiens (Human)) | BDBM50198419 (1-(1-(((1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 16 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
UCB Inflammation Discovery Curated by ChEMBL | Assay Description Binding affinity to human CXCR3 receptor expressed in CHO membrane by ITAC-stimulated GTP gammaS assay | Bioorg Med Chem Lett 17: 6806-10 (2007) Article DOI: 10.1016/j.bmcl.2007.10.029 BindingDB Entry DOI: 10.7270/Q24F1QGP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C-X-C chemokine receptor type 3 (Homo sapiens (Human)) | BDBM50225715 (3-(3,5-bis(trifluoromethyl)phenyl)-1-(1-(((1R,5S)-...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 26 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
UCB Inflammation Discovery Curated by ChEMBL | Assay Description Binding affinity to human CXCR3 receptor expressed in CHO membrane by ITAC-stimulated GTP gammaS assay | Bioorg Med Chem Lett 17: 6806-10 (2007) Article DOI: 10.1016/j.bmcl.2007.10.029 BindingDB Entry DOI: 10.7270/Q24F1QGP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C-X-C chemokine receptor type 3 (Homo sapiens (Human)) | BDBM50225718 (1-(1-(((1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 100 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
UCB Inflammation Discovery Curated by ChEMBL | Assay Description Binding affinity to human CXCR3 receptor expressed in CHO membrane by ITAC-stimulated GTP gammaS assay | Bioorg Med Chem Lett 17: 6806-10 (2007) Article DOI: 10.1016/j.bmcl.2007.10.029 BindingDB Entry DOI: 10.7270/Q24F1QGP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C-X-C chemokine receptor type 3 (Homo sapiens (Human)) | BDBM50225729 (3-(4-chloro-3-(trifluoromethyl)phenyl)-1-(1-(((1R,...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 120 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
UCB Inflammation Discovery Curated by ChEMBL | Assay Description Binding affinity to human CXCR3 receptor expressed in CHO membrane by ITAC-stimulated GTP gammaS assay | Bioorg Med Chem Lett 17: 6806-10 (2007) Article DOI: 10.1016/j.bmcl.2007.10.029 BindingDB Entry DOI: 10.7270/Q24F1QGP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C-X-C chemokine receptor type 3 (Homo sapiens (Human)) | BDBM50225725 (6-bromo-N-(1-(((1R,5S)-6,6-dimethylbicyclo[3.1.1]h...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 130 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
UCB Inflammation Discovery Curated by ChEMBL | Assay Description Binding affinity to human CXCR3 receptor expressed in CHO membrane by ITAC-stimulated GTP gammaS assay | Bioorg Med Chem Lett 17: 6806-10 (2007) Article DOI: 10.1016/j.bmcl.2007.10.029 BindingDB Entry DOI: 10.7270/Q24F1QGP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C-X-C chemokine receptor type 3 (Homo sapiens (Human)) | BDBM50225711 (CHEMBL437776 | N-(1-(((1R,5S)-6,6-dimethylbicyclo[...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 140 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
UCB Inflammation Discovery Curated by ChEMBL | Assay Description Binding affinity to human CXCR3 receptor expressed in CHO membrane by ITAC-stimulated GTP gammaS assay | Bioorg Med Chem Lett 17: 6806-10 (2007) Article DOI: 10.1016/j.bmcl.2007.10.029 BindingDB Entry DOI: 10.7270/Q24F1QGP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C-X-C chemokine receptor type 3 (Homo sapiens (Human)) | BDBM50225726 (4-bromo-N-(1-(((1R,5S)-6,6-dimethylbicyclo[3.1.1]h...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 150 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
UCB Inflammation Discovery Curated by ChEMBL | Assay Description Binding affinity to human CXCR3 receptor expressed in CHO membrane by ITAC-stimulated GTP gammaS assay | Bioorg Med Chem Lett 17: 6806-10 (2007) Article DOI: 10.1016/j.bmcl.2007.10.029 BindingDB Entry DOI: 10.7270/Q24F1QGP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C-X-C chemokine receptor type 3 (Homo sapiens (Human)) | BDBM50225731 (1-(3,5-bis(trifluoromethyl)phenyl)-3-(1-(((1R,5S)-...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 170 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
UCB Inflammation Discovery Curated by ChEMBL | Assay Description Binding affinity to human CXCR3 receptor expressed in CHO membrane by ITAC-stimulated GTP gammaS assay | Bioorg Med Chem Lett 17: 6806-10 (2007) Article DOI: 10.1016/j.bmcl.2007.10.029 BindingDB Entry DOI: 10.7270/Q24F1QGP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C-X-C chemokine receptor type 3 (Homo sapiens (Human)) | BDBM50225733 (6-chloro-N-(1-(((1R,5S)-6,6-dimethylbicyclo[3.1.1]...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 170 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
UCB Inflammation Discovery Curated by ChEMBL | Assay Description Binding affinity to human CXCR3 receptor expressed in CHO membrane by ITAC-stimulated GTP gammaS assay | Bioorg Med Chem Lett 17: 6806-10 (2007) Article DOI: 10.1016/j.bmcl.2007.10.029 BindingDB Entry DOI: 10.7270/Q24F1QGP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C-X-C chemokine receptor type 3 (Homo sapiens (Human)) | BDBM50225732 (1-(1-(((1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 180 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
UCB Inflammation Discovery Curated by ChEMBL | Assay Description Binding affinity to human CXCR3 receptor expressed in CHO membrane by ITAC-stimulated GTP gammaS assay | Bioorg Med Chem Lett 17: 6806-10 (2007) Article DOI: 10.1016/j.bmcl.2007.10.029 BindingDB Entry DOI: 10.7270/Q24F1QGP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C-X-C chemokine receptor type 3 (Homo sapiens (Human)) | BDBM50225714 (1-(1-(((1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 200 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
UCB Inflammation Discovery Curated by ChEMBL | Assay Description Binding affinity to human CXCR3 receptor expressed in CHO membrane by ITAC-stimulated GTP gammaS assay | Bioorg Med Chem Lett 17: 6806-10 (2007) Article DOI: 10.1016/j.bmcl.2007.10.029 BindingDB Entry DOI: 10.7270/Q24F1QGP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C-X-C chemokine receptor type 3 (Homo sapiens (Human)) | BDBM50225710 (1-(1-(((1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 220 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
UCB Inflammation Discovery Curated by ChEMBL | Assay Description Binding affinity to human CXCR3 receptor expressed in CHO membrane by ITAC-stimulated GTP gammaS assay | Bioorg Med Chem Lett 17: 6806-10 (2007) Article DOI: 10.1016/j.bmcl.2007.10.029 BindingDB Entry DOI: 10.7270/Q24F1QGP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C-X-C chemokine receptor type 3 (Homo sapiens (Human)) | BDBM50225724 (CHEMBL250658 | N-(4-(3,5-bis(trifluoromethyl)pheny...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 260 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
UCB Inflammation Discovery Curated by ChEMBL | Assay Description Binding affinity to human CXCR3 receptor expressed in CHO membrane by ITAC-stimulated GTP gammaS assay | Bioorg Med Chem Lett 17: 6806-10 (2007) Article DOI: 10.1016/j.bmcl.2007.10.029 BindingDB Entry DOI: 10.7270/Q24F1QGP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C-X-C chemokine receptor type 3 (Homo sapiens (Human)) | BDBM50225728 (CHEMBL250483 | N-(3-(3,5-bis(trifluoromethyl)pheny...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | 270 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
UCB Inflammation Discovery Curated by ChEMBL | Assay Description Binding affinity to human CXCR3 receptor expressed in CHO membrane by ITAC-stimulated GTP gammaS assay | Bioorg Med Chem Lett 17: 6806-10 (2007) Article DOI: 10.1016/j.bmcl.2007.10.029 BindingDB Entry DOI: 10.7270/Q24F1QGP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C-X-C chemokine receptor type 3 (Homo sapiens (Human)) | BDBM50225722 (5-chloro-N-(1-(((1R,5S)-6,6-dimethylbicyclo[3.1.1]...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 290 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
UCB Inflammation Discovery Curated by ChEMBL | Assay Description Binding affinity to human CXCR3 receptor expressed in CHO membrane by ITAC-stimulated GTP gammaS assay | Bioorg Med Chem Lett 17: 6806-10 (2007) Article DOI: 10.1016/j.bmcl.2007.10.029 BindingDB Entry DOI: 10.7270/Q24F1QGP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C-X-C chemokine receptor type 3 (Homo sapiens (Human)) | BDBM50225717 (CHEMBL249016 | N-(1-(((1R,5S)-6,6-dimethylbicyclo[...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 350 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
UCB Inflammation Discovery Curated by ChEMBL | Assay Description Binding affinity to human CXCR3 receptor expressed in CHO membrane by ITAC-stimulated GTP gammaS assay | Bioorg Med Chem Lett 17: 6806-10 (2007) Article DOI: 10.1016/j.bmcl.2007.10.029 BindingDB Entry DOI: 10.7270/Q24F1QGP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C-X-C chemokine receptor type 3 (Homo sapiens (Human)) | BDBM50225716 (1-(1-(((1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 380 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
UCB Inflammation Discovery Curated by ChEMBL | Assay Description Binding affinity to human CXCR3 receptor expressed in CHO membrane by ITAC-stimulated GTP gammaS assay | Bioorg Med Chem Lett 17: 6806-10 (2007) Article DOI: 10.1016/j.bmcl.2007.10.029 BindingDB Entry DOI: 10.7270/Q24F1QGP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C-X-C chemokine receptor type 3 (Homo sapiens (Human)) | BDBM50225720 (CHEMBL250657 | N-(4-(3,4-dichlorophenyl)thiazol-2-...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 460 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
UCB Inflammation Discovery Curated by ChEMBL | Assay Description Binding affinity to human CXCR3 receptor expressed in CHO membrane by ITAC-stimulated GTP gammaS assay | Bioorg Med Chem Lett 17: 6806-10 (2007) Article DOI: 10.1016/j.bmcl.2007.10.029 BindingDB Entry DOI: 10.7270/Q24F1QGP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C-X-C chemokine receptor type 3 (Homo sapiens (Human)) | BDBM50225712 (4-chloro-N-(1-(((1R,5S)-6,6-dimethylbicyclo[3.1.1]...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 460 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
UCB Inflammation Discovery Curated by ChEMBL | Assay Description Binding affinity to human CXCR3 receptor expressed in CHO membrane by ITAC-stimulated GTP gammaS assay | Bioorg Med Chem Lett 17: 6806-10 (2007) Article DOI: 10.1016/j.bmcl.2007.10.029 BindingDB Entry DOI: 10.7270/Q24F1QGP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C-X-C chemokine receptor type 3 (Homo sapiens (Human)) | BDBM50225721 (7-chloro-N-(1-(((1R,5S)-6,6-dimethylbicyclo[3.1.1]...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 620 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
UCB Inflammation Discovery Curated by ChEMBL | Assay Description Binding affinity to human CXCR3 receptor expressed in CHO membrane by ITAC-stimulated GTP gammaS assay | Bioorg Med Chem Lett 17: 6806-10 (2007) Article DOI: 10.1016/j.bmcl.2007.10.029 BindingDB Entry DOI: 10.7270/Q24F1QGP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C-X-C chemokine receptor type 3 (Homo sapiens (Human)) | BDBM50225709 (CHEMBL249612 | N-(1-(((1R,5S)-6,6-dimethylbicyclo[...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 680 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
UCB Inflammation Discovery Curated by ChEMBL | Assay Description Binding affinity to human CXCR3 receptor expressed in CHO membrane by ITAC-stimulated GTP gammaS assay | Bioorg Med Chem Lett 17: 6806-10 (2007) Article DOI: 10.1016/j.bmcl.2007.10.029 BindingDB Entry DOI: 10.7270/Q24F1QGP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C-X-C chemokine receptor type 3 (Homo sapiens (Human)) | BDBM50225723 (CHEMBL249014 | N-(1-(((1R,5S)-6,6-dimethylbicyclo[...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 720 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
UCB Inflammation Discovery Curated by ChEMBL | Assay Description Binding affinity to human CXCR3 receptor expressed in CHO membrane by ITAC-stimulated GTP gammaS assay | Bioorg Med Chem Lett 17: 6806-10 (2007) Article DOI: 10.1016/j.bmcl.2007.10.029 BindingDB Entry DOI: 10.7270/Q24F1QGP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C-X-C chemokine receptor type 3 (Homo sapiens (Human)) | BDBM50225719 (1-(1-(((1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 750 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
UCB Inflammation Discovery Curated by ChEMBL | Assay Description Binding affinity to human CXCR3 receptor expressed in CHO membrane by ITAC-stimulated GTP gammaS assay | Bioorg Med Chem Lett 17: 6806-10 (2007) Article DOI: 10.1016/j.bmcl.2007.10.029 BindingDB Entry DOI: 10.7270/Q24F1QGP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C-X-C chemokine receptor type 3 (Homo sapiens (Human)) | BDBM50225734 (1-(((1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 880 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
UCB Inflammation Discovery Curated by ChEMBL | Assay Description Binding affinity to human CXCR3 receptor expressed in CHO membrane by ITAC-stimulated GTP gammaS assay | Bioorg Med Chem Lett 17: 6806-10 (2007) Article DOI: 10.1016/j.bmcl.2007.10.029 BindingDB Entry DOI: 10.7270/Q24F1QGP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C-X-C chemokine receptor type 3 (Homo sapiens (Human)) | BDBM50225727 (CHEMBL248632 | N-(1-(((1R,5S)-6,6-dimethylbicyclo[...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | 950 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
UCB Inflammation Discovery Curated by ChEMBL | Assay Description Binding affinity to human CXCR3 receptor expressed in CHO membrane by ITAC-stimulated GTP gammaS assay | Bioorg Med Chem Lett 17: 6806-10 (2007) Article DOI: 10.1016/j.bmcl.2007.10.029 BindingDB Entry DOI: 10.7270/Q24F1QGP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C-X-C chemokine receptor type 3 (Homo sapiens (Human)) | BDBM50225730 (3-(1-(((1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 3.50E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
UCB Inflammation Discovery Curated by ChEMBL | Assay Description Binding affinity to human CXCR3 receptor expressed in CHO membrane by ITAC-stimulated GTP gammaS assay | Bioorg Med Chem Lett 17: 6806-10 (2007) Article DOI: 10.1016/j.bmcl.2007.10.029 BindingDB Entry DOI: 10.7270/Q24F1QGP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C-X-C chemokine receptor type 3 (Homo sapiens (Human)) | BDBM50225713 (1-(1-(((1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 3.60E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
UCB Inflammation Discovery Curated by ChEMBL | Assay Description Binding affinity to human CXCR3 receptor expressed in CHO membrane by ITAC-stimulated GTP gammaS assay | Bioorg Med Chem Lett 17: 6806-10 (2007) Article DOI: 10.1016/j.bmcl.2007.10.029 BindingDB Entry DOI: 10.7270/Q24F1QGP | |||||||||||
More data for this Ligand-Target Pair |