Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Substance-K receptor (Homo sapiens (Human)) | BDBM50256882 (6-((4-(2-(4-tert-butylphenyl)-1H-benzo[d]imidazol-...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 330 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Wyeth Research Curated by ChEMBL | Assay Description Inhibition of human neurokinin NK2 receptor | J Med Chem 52: 2148-52 (2009) Article DOI: 10.1021/jm801572m BindingDB Entry DOI: 10.7270/Q2ZC82RT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine H2 receptor (Homo sapiens (Human)) | BDBM50256882 (6-((4-(2-(4-tert-butylphenyl)-1H-benzo[d]imidazol-...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 850 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Wyeth Research Curated by ChEMBL | Assay Description Inhibition of human histamine H2 receptor | J Med Chem 52: 2148-52 (2009) Article DOI: 10.1021/jm801572m BindingDB Entry DOI: 10.7270/Q2ZC82RT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Gonadotropin-releasing hormone receptor (Homo sapiens (Human)) | BDBM50256836 (7-((4-(2-(4-tert-butylphenyl)-1H-benzo[d]imidazol-...) | PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.80 | n/a | n/a | n/a | n/a | n/a | n/a |
Wyeth Research Curated by ChEMBL | Assay Description Displacement of [D-Trp6]-GnRH from human recombinant GnRH receptor | J Med Chem 52: 2148-52 (2009) Article DOI: 10.1021/jm801572m BindingDB Entry DOI: 10.7270/Q2ZC82RT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Gonadotropin-releasing hormone receptor (Homo sapiens (Human)) | BDBM50256834 (7-((4-(2-(4-tert-butylphenyl)-1H-benzo[d]imidazol-...) | PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 3.5 | n/a | n/a | n/a | n/a | n/a | n/a |
Wyeth Research Curated by ChEMBL | Assay Description Displacement of [D-Trp6]-GnRH from human recombinant GnRH receptor | J Med Chem 52: 2148-52 (2009) Article DOI: 10.1021/jm801572m BindingDB Entry DOI: 10.7270/Q2ZC82RT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Gonadotropin-releasing hormone receptor (Homo sapiens (Human)) | BDBM50244211 (6-((4-(2-(4-tert-butylphenyl)-1H-benzo[d]imidazol-...) | PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 4.90 | n/a | n/a | n/a | n/a | n/a | n/a |
Wyeth Research Curated by ChEMBL | Assay Description Displacement of [D-Trp6]-GnRH from human recombinant GnRH receptor | J Med Chem 52: 2148-52 (2009) Article DOI: 10.1021/jm801572m BindingDB Entry DOI: 10.7270/Q2ZC82RT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Gonadotropin-releasing hormone receptor (Homo sapiens (Human)) | BDBM50256835 (7-((4-(2-(4-tert-butylphenyl)-1H-benzo[d]imidazol-...) | PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 5.60 | n/a | n/a | n/a | n/a | n/a | n/a |
Wyeth Research Curated by ChEMBL | Assay Description Displacement of [D-Trp6]-GnRH from human recombinant GnRH receptor | J Med Chem 52: 2148-52 (2009) Article DOI: 10.1021/jm801572m BindingDB Entry DOI: 10.7270/Q2ZC82RT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Gonadotropin-releasing hormone receptor (Homo sapiens (Human)) | BDBM50256834 (7-((4-(2-(4-tert-butylphenyl)-1H-benzo[d]imidazol-...) | PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 7.40 | n/a | n/a | n/a | n/a | n/a | n/a |
Wyeth Research Curated by ChEMBL | Assay Description Antagonist activity at human GnRH receptor assessed as inhibition of [D-Trp6]-GnRH-stimulated [3H]IP reduction | J Med Chem 52: 2148-52 (2009) Article DOI: 10.1021/jm801572m BindingDB Entry DOI: 10.7270/Q2ZC82RT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Gonadotropin-releasing hormone receptor (Homo sapiens (Human)) | BDBM50244211 (6-((4-(2-(4-tert-butylphenyl)-1H-benzo[d]imidazol-...) | PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 9.40 | n/a | n/a | n/a | n/a | n/a | n/a |
Wyeth Research Curated by ChEMBL | Assay Description Antagonist activity at human GnRH receptor assessed as inhibition of [D-Trp6]-GnRH-stimulated [3H]IP reduction | J Med Chem 52: 2148-52 (2009) Article DOI: 10.1021/jm801572m BindingDB Entry DOI: 10.7270/Q2ZC82RT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Gonadotropin-releasing hormone receptor (Homo sapiens (Human)) | BDBM50256836 (7-((4-(2-(4-tert-butylphenyl)-1H-benzo[d]imidazol-...) | PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 9.70 | n/a | n/a | n/a | n/a | n/a | n/a |
Wyeth Research Curated by ChEMBL | Assay Description Antagonist activity at human GnRH receptor assessed as inhibition of [D-Trp6]-GnRH-stimulated [3H]IP reduction | J Med Chem 52: 2148-52 (2009) Article DOI: 10.1021/jm801572m BindingDB Entry DOI: 10.7270/Q2ZC82RT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Gonadotropin-releasing hormone receptor (Homo sapiens (Human)) | BDBM50256882 (6-((4-(2-(4-tert-butylphenyl)-1H-benzo[d]imidazol-...) | PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 12 | n/a | n/a | n/a | n/a | n/a | n/a |
Wyeth Research Curated by ChEMBL | Assay Description Displacement of [D-Trp6]-GnRH from human recombinant GnRH receptor | J Med Chem 52: 2148-52 (2009) Article DOI: 10.1021/jm801572m BindingDB Entry DOI: 10.7270/Q2ZC82RT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Gonadotropin-releasing hormone receptor (Homo sapiens (Human)) | BDBM50256835 (7-((4-(2-(4-tert-butylphenyl)-1H-benzo[d]imidazol-...) | PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 14 | n/a | n/a | n/a | n/a | n/a | n/a |
Wyeth Research Curated by ChEMBL | Assay Description Antagonist activity at human GnRH receptor assessed as inhibition of [D-Trp6]-GnRH-stimulated [3H]IP reduction | J Med Chem 52: 2148-52 (2009) Article DOI: 10.1021/jm801572m BindingDB Entry DOI: 10.7270/Q2ZC82RT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Gonadotropin-releasing hormone receptor (Homo sapiens (Human)) | BDBM50256881 (6-((4-(2-(4-tert-butylphenyl)-1H-benzo[d]imidazol-...) | PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents | Article PubMed | n/a | n/a | 16 | n/a | n/a | n/a | n/a | n/a | n/a |
Wyeth Research Curated by ChEMBL | Assay Description Displacement of [D-Trp6]-GnRH from human recombinant GnRH receptor | J Med Chem 52: 2148-52 (2009) Article DOI: 10.1021/jm801572m BindingDB Entry DOI: 10.7270/Q2ZC82RT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Gonadotropin-releasing hormone receptor (Homo sapiens (Human)) | BDBM50256881 (6-((4-(2-(4-tert-butylphenyl)-1H-benzo[d]imidazol-...) | PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents | Article PubMed | n/a | n/a | 16 | n/a | n/a | n/a | n/a | n/a | n/a |
Wyeth Research Curated by ChEMBL | Assay Description Antagonist activity at human GnRH receptor assessed as inhibition of [D-Trp6]-GnRH-stimulated [3H]IP reduction | J Med Chem 52: 2148-52 (2009) Article DOI: 10.1021/jm801572m BindingDB Entry DOI: 10.7270/Q2ZC82RT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Gonadotropin-releasing hormone receptor (Rattus norvegicus) | BDBM50256834 (7-((4-(2-(4-tert-butylphenyl)-1H-benzo[d]imidazol-...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 17 | n/a | n/a | n/a | n/a | n/a | n/a |
Wyeth Research Curated by ChEMBL | Assay Description Displacement of [D-Trp6]-GnRH from rat recombinant GnRH receptor | J Med Chem 52: 2148-52 (2009) Article DOI: 10.1021/jm801572m BindingDB Entry DOI: 10.7270/Q2ZC82RT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Gonadotropin-releasing hormone receptor (Homo sapiens (Human)) | BDBM50256883 (6-((4-(2-(4-tert-butylphenyl)-1H-benzo[d]imidazol-...) | PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 21 | n/a | n/a | n/a | n/a | n/a | n/a |
Wyeth Research Curated by ChEMBL | Assay Description Displacement of [D-Trp6]-GnRH from human recombinant GnRH receptor | J Med Chem 52: 2148-52 (2009) Article DOI: 10.1021/jm801572m BindingDB Entry DOI: 10.7270/Q2ZC82RT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Gonadotropin-releasing hormone receptor (Homo sapiens (Human)) | BDBM50256884 (7-((4-(2-(4-tert-butylphenyl)-1H-benzo[d]imidazol-...) | PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 24 | n/a | n/a | n/a | n/a | n/a | n/a |
Wyeth Research Curated by ChEMBL | Assay Description Displacement of [D-Trp6]-GnRH from human recombinant GnRH receptor | J Med Chem 52: 2148-52 (2009) Article DOI: 10.1021/jm801572m BindingDB Entry DOI: 10.7270/Q2ZC82RT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Gonadotropin-releasing hormone receptor (Rattus norvegicus) | BDBM50244211 (6-((4-(2-(4-tert-butylphenyl)-1H-benzo[d]imidazol-...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 25 | n/a | n/a | n/a | n/a | n/a | n/a |
Wyeth Research Curated by ChEMBL | Assay Description Antagonist activity at rat recombinant GnRH receptor assessed as inhibition of [D-Trp6]-GnRH-stimulated LH release from rat pituitary cells | J Med Chem 52: 2148-52 (2009) Article DOI: 10.1021/jm801572m BindingDB Entry DOI: 10.7270/Q2ZC82RT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Gonadotropin-releasing hormone receptor (Homo sapiens (Human)) | BDBM50256939 (5-((4-(2-(4-tert-butylphenyl)-1H-benzo[d]imidazol-...) | PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 26 | n/a | n/a | n/a | n/a | n/a | n/a |
Wyeth Research Curated by ChEMBL | Assay Description Displacement of [D-Trp6]-GnRH from human recombinant GnRH receptor | J Med Chem 52: 2148-52 (2009) Article DOI: 10.1021/jm801572m BindingDB Entry DOI: 10.7270/Q2ZC82RT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Gonadotropin-releasing hormone receptor (Homo sapiens (Human)) | BDBM50256882 (6-((4-(2-(4-tert-butylphenyl)-1H-benzo[d]imidazol-...) | PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 28 | n/a | n/a | n/a | n/a | n/a | n/a |
Wyeth Research Curated by ChEMBL | Assay Description Antagonist activity at human GnRH receptor assessed as inhibition of [D-Trp6]-GnRH-stimulated [3H]IP reduction | J Med Chem 52: 2148-52 (2009) Article DOI: 10.1021/jm801572m BindingDB Entry DOI: 10.7270/Q2ZC82RT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Gonadotropin-releasing hormone receptor (Rattus norvegicus) | BDBM50256836 (7-((4-(2-(4-tert-butylphenyl)-1H-benzo[d]imidazol-...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 33 | n/a | n/a | n/a | n/a | n/a | n/a |
Wyeth Research Curated by ChEMBL | Assay Description Displacement of [D-Trp6]-GnRH from rat recombinant GnRH receptor | J Med Chem 52: 2148-52 (2009) Article DOI: 10.1021/jm801572m BindingDB Entry DOI: 10.7270/Q2ZC82RT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Gonadotropin-releasing hormone receptor (Rattus norvegicus) | BDBM50244211 (6-((4-(2-(4-tert-butylphenyl)-1H-benzo[d]imidazol-...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 40 | n/a | n/a | n/a | n/a | n/a | n/a |
Wyeth Research Curated by ChEMBL | Assay Description Displacement of [D-Trp6]-GnRH from rat recombinant GnRH receptor | J Med Chem 52: 2148-52 (2009) Article DOI: 10.1021/jm801572m BindingDB Entry DOI: 10.7270/Q2ZC82RT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Gonadotropin-releasing hormone receptor (Rattus norvegicus) | BDBM50256834 (7-((4-(2-(4-tert-butylphenyl)-1H-benzo[d]imidazol-...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 44 | n/a | n/a | n/a | n/a | n/a | n/a |
Wyeth Research Curated by ChEMBL | Assay Description Antagonist activity at rat recombinant GnRH receptor assessed as inhibition of [D-Trp6]-GnRH-stimulated LH release from rat pituitary cells | J Med Chem 52: 2148-52 (2009) Article DOI: 10.1021/jm801572m BindingDB Entry DOI: 10.7270/Q2ZC82RT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Gonadotropin-releasing hormone receptor (Rattus norvegicus) | BDBM50256835 (7-((4-(2-(4-tert-butylphenyl)-1H-benzo[d]imidazol-...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 47 | n/a | n/a | n/a | n/a | n/a | n/a |
Wyeth Research Curated by ChEMBL | Assay Description Displacement of [D-Trp6]-GnRH from rat recombinant GnRH receptor | J Med Chem 52: 2148-52 (2009) Article DOI: 10.1021/jm801572m BindingDB Entry DOI: 10.7270/Q2ZC82RT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Gonadotropin-releasing hormone receptor (Homo sapiens (Human)) | BDBM50256883 (6-((4-(2-(4-tert-butylphenyl)-1H-benzo[d]imidazol-...) | PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 64 | n/a | n/a | n/a | n/a | n/a | n/a |
Wyeth Research Curated by ChEMBL | Assay Description Antagonist activity at human GnRH receptor assessed as inhibition of [D-Trp6]-GnRH-stimulated [3H]IP reduction | J Med Chem 52: 2148-52 (2009) Article DOI: 10.1021/jm801572m BindingDB Entry DOI: 10.7270/Q2ZC82RT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Gonadotropin-releasing hormone receptor (Rattus norvegicus) | BDBM50256835 (7-((4-(2-(4-tert-butylphenyl)-1H-benzo[d]imidazol-...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 69 | n/a | n/a | n/a | n/a | n/a | n/a |
Wyeth Research Curated by ChEMBL | Assay Description Antagonist activity at rat recombinant GnRH receptor assessed as inhibition of [D-Trp6]-GnRH-stimulated LH release from rat pituitary cells | J Med Chem 52: 2148-52 (2009) Article DOI: 10.1021/jm801572m BindingDB Entry DOI: 10.7270/Q2ZC82RT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Gonadotropin-releasing hormone receptor (Rattus norvegicus) | BDBM50256882 (6-((4-(2-(4-tert-butylphenyl)-1H-benzo[d]imidazol-...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 71 | n/a | n/a | n/a | n/a | n/a | n/a |
Wyeth Research Curated by ChEMBL | Assay Description Displacement of [D-Trp6]-GnRH from rat recombinant GnRH receptor | J Med Chem 52: 2148-52 (2009) Article DOI: 10.1021/jm801572m BindingDB Entry DOI: 10.7270/Q2ZC82RT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Gonadotropin-releasing hormone receptor (Rattus norvegicus) | BDBM50256881 (6-((4-(2-(4-tert-butylphenyl)-1H-benzo[d]imidazol-...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents | Article PubMed | n/a | n/a | 87 | n/a | n/a | n/a | n/a | n/a | n/a |
Wyeth Research Curated by ChEMBL | Assay Description Displacement of [D-Trp6]-GnRH from rat recombinant GnRH receptor | J Med Chem 52: 2148-52 (2009) Article DOI: 10.1021/jm801572m BindingDB Entry DOI: 10.7270/Q2ZC82RT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Gonadotropin-releasing hormone receptor (Rattus norvegicus) | BDBM50256881 (6-((4-(2-(4-tert-butylphenyl)-1H-benzo[d]imidazol-...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents | Article PubMed | n/a | n/a | 120 | n/a | n/a | n/a | n/a | n/a | n/a |
Wyeth Research Curated by ChEMBL | Assay Description Antagonist activity at rat recombinant GnRH receptor assessed as inhibition of [D-Trp6]-GnRH-stimulated LH release from rat pituitary cells | J Med Chem 52: 2148-52 (2009) Article DOI: 10.1021/jm801572m BindingDB Entry DOI: 10.7270/Q2ZC82RT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Gonadotropin-releasing hormone receptor (Homo sapiens (Human)) | BDBM50256884 (7-((4-(2-(4-tert-butylphenyl)-1H-benzo[d]imidazol-...) | PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 140 | n/a | n/a | n/a | n/a | n/a | n/a |
Wyeth Research Curated by ChEMBL | Assay Description Antagonist activity at human GnRH receptor assessed as inhibition of [D-Trp6]-GnRH-stimulated [3H]IP reduction | J Med Chem 52: 2148-52 (2009) Article DOI: 10.1021/jm801572m BindingDB Entry DOI: 10.7270/Q2ZC82RT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Gonadotropin-releasing hormone receptor (Rattus norvegicus) | BDBM50256836 (7-((4-(2-(4-tert-butylphenyl)-1H-benzo[d]imidazol-...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 240 | n/a | n/a | n/a | n/a | n/a | n/a |
Wyeth Research Curated by ChEMBL | Assay Description Antagonist activity at rat recombinant GnRH receptor assessed as inhibition of [D-Trp6]-GnRH-stimulated LH release from rat pituitary cells | J Med Chem 52: 2148-52 (2009) Article DOI: 10.1021/jm801572m BindingDB Entry DOI: 10.7270/Q2ZC82RT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Gonadotropin-releasing hormone receptor (Rattus norvegicus) | BDBM50256882 (6-((4-(2-(4-tert-butylphenyl)-1H-benzo[d]imidazol-...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 320 | n/a | n/a | n/a | n/a | n/a | n/a |
Wyeth Research Curated by ChEMBL | Assay Description Antagonist activity at rat recombinant GnRH receptor assessed as inhibition of [D-Trp6]-GnRH-stimulated LH release from rat pituitary cells | J Med Chem 52: 2148-52 (2009) Article DOI: 10.1021/jm801572m BindingDB Entry DOI: 10.7270/Q2ZC82RT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Gonadotropin-releasing hormone receptor (Homo sapiens (Human)) | BDBM50256939 (5-((4-(2-(4-tert-butylphenyl)-1H-benzo[d]imidazol-...) | PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 400 | n/a | n/a | n/a | n/a | n/a | n/a |
Wyeth Research Curated by ChEMBL | Assay Description Antagonist activity at human GnRH receptor assessed as inhibition of [D-Trp6]-GnRH-stimulated [3H]IP reduction | J Med Chem 52: 2148-52 (2009) Article DOI: 10.1021/jm801572m BindingDB Entry DOI: 10.7270/Q2ZC82RT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Gonadotropin-releasing hormone receptor (Rattus norvegicus) | BDBM50256884 (7-((4-(2-(4-tert-butylphenyl)-1H-benzo[d]imidazol-...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 540 | n/a | n/a | n/a | n/a | n/a | n/a |
Wyeth Research Curated by ChEMBL | Assay Description Antagonist activity at rat recombinant GnRH receptor assessed as inhibition of [D-Trp6]-GnRH-stimulated LH release from rat pituitary cells | J Med Chem 52: 2148-52 (2009) Article DOI: 10.1021/jm801572m BindingDB Entry DOI: 10.7270/Q2ZC82RT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Gonadotropin-releasing hormone receptor (Rattus norvegicus) | BDBM50256883 (6-((4-(2-(4-tert-butylphenyl)-1H-benzo[d]imidazol-...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 830 | n/a | n/a | n/a | n/a | n/a | n/a |
Wyeth Research Curated by ChEMBL | Assay Description Antagonist activity at rat recombinant GnRH receptor assessed as inhibition of [D-Trp6]-GnRH-stimulated LH release from rat pituitary cells | J Med Chem 52: 2148-52 (2009) Article DOI: 10.1021/jm801572m BindingDB Entry DOI: 10.7270/Q2ZC82RT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Gonadotropin-releasing hormone receptor (Rattus norvegicus) | BDBM50256939 (5-((4-(2-(4-tert-butylphenyl)-1H-benzo[d]imidazol-...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 5.90E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Wyeth Research Curated by ChEMBL | Assay Description Antagonist activity at rat recombinant GnRH receptor assessed as inhibition of [D-Trp6]-GnRH-stimulated LH release from rat pituitary cells | J Med Chem 52: 2148-52 (2009) Article DOI: 10.1021/jm801572m BindingDB Entry DOI: 10.7270/Q2ZC82RT | |||||||||||
More data for this Ligand-Target Pair |