BindingDB PrimarySearch

Found 29 hits Enz. Inhib. hit(s) with all data for entry = 50028427
Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kJ/mole	IC50 nM	Kd nM	EC50/IC50 nM	k_off s^-1	k_on M^-1s^-1	pH	Temp °C
Potassium voltage-gated channel subfamily A member 3 (Homo sapiens (Human))	BDBM50279106 (4-(4-phenoxybutoxy)-7H-furo[3,2-g]chromen-7-one \| ...) Show SMILES O=c1ccc2c(OCCCCOc3ccccc3)c3ccoc3cc2o1 Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	Purchase CHEMBL MCE PC cid PC sid UniChem Patents Similars	Article PubMed	n/a	n/a	10	n/a	n/a	n/a	n/a	n/a	n/a
4SC AG Curated by ChEMBL					Assay Description Inhibition of cloned Kv1.3 channel (unknown origin) expressed in mammalian cells by whole cell patch clamp assay				Bioorg Med Chem Lett 19: 2299-304 (2009) Article DOI: 10.1016/j.bmcl.2009.02.077 BindingDB Entry DOI: 10.7270/Q29K4B38
4SC AG Curated by ChEMBL					More data for this Ligand-Target Pair
Intermediate conductance calcium-activated potassium channel protein 4 (Homo sapiens (Human))	BDBM50279107 (1-((2-chlorophenyl)diphenylmethyl)-1H-pyrazole \| C...) Show SMILES Clc1ccccc1C(c1ccccc1)(c1ccccc1)n1cccn1 Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	Purchase CHEMBL MCE KEGG PC cid PC sid UniChem Patents	Article PubMed	n/a	n/a	20	n/a	n/a	n/a	n/a	n/a	n/a
4SC AG Curated by ChEMBL					Assay Description Inhibition of IK1 (unknown origin)				Bioorg Med Chem Lett 19: 2299-304 (2009) Article DOI: 10.1016/j.bmcl.2009.02.077 BindingDB Entry DOI: 10.7270/Q29K4B38
4SC AG Curated by ChEMBL					More data for this Ligand-Target Pair
Intermediate conductance calcium-activated potassium channel protein 4 (Homo sapiens (Human))	BDBM50279107 (1-((2-chlorophenyl)diphenylmethyl)-1H-pyrazole \| C...) Show SMILES Clc1ccccc1C(c1ccccc1)(c1ccccc1)n1cccn1 Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	Purchase CHEMBL MCE KEGG PC cid PC sid UniChem Patents	Article PubMed	n/a	n/a	20	n/a	n/a	n/a	n/a	n/a	n/a
4SC AG Curated by ChEMBL					Assay Description Inhibition of human cloned IK1 expressed in african green monkey COS7 cells by whole cell patch clamp assay				Bioorg Med Chem Lett 19: 2299-304 (2009) Article DOI: 10.1016/j.bmcl.2009.02.077 BindingDB Entry DOI: 10.7270/Q29K4B38
4SC AG Curated by ChEMBL					More data for this Ligand-Target Pair
Intermediate conductance calcium-activated potassium channel protein 4 (Homo sapiens (Human))	BDBM31774 (CHEMBL104 \| Canesten \| Clotrimazole \| Lotrimin \| M...) Show SMILES Clc1ccccc1C(c1ccccc1)(c1ccccc1)n1ccnc1 Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	Purchase CHEMBL DrugBank MCE KEGG MMDB PC cid PC sid PDB UniChem Patents Similars	DrugBank Article PubMed	n/a	n/a	70	n/a	n/a	n/a	n/a	n/a	n/a
4SC AG Curated by ChEMBL					Assay Description Inhibition of human cloned IK1 expressed in african green monkey COS7 cells by whole cell patch clamp assay				Bioorg Med Chem Lett 19: 2299-304 (2009) Article DOI: 10.1016/j.bmcl.2009.02.077 BindingDB Entry DOI: 10.7270/Q29K4B38
4SC AG Curated by ChEMBL					More data for this Ligand-Target Pair
Intermediate conductance calcium-activated potassium channel protein 4 (Homo sapiens (Human))	BDBM31774 (CHEMBL104 \| Canesten \| Clotrimazole \| Lotrimin \| M...) Show SMILES Clc1ccccc1C(c1ccccc1)(c1ccccc1)n1ccnc1 Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	Purchase CHEMBL DrugBank MCE KEGG MMDB PC cid PC sid PDB UniChem Patents Similars	DrugBank Article PubMed	n/a	n/a	70	n/a	n/a	n/a	n/a	n/a	n/a
4SC AG Curated by ChEMBL					Assay Description Inhibition of IK1 (unknown origin)				Bioorg Med Chem Lett 19: 2299-304 (2009) Article DOI: 10.1016/j.bmcl.2009.02.077 BindingDB Entry DOI: 10.7270/Q29K4B38
4SC AG Curated by ChEMBL					More data for this Ligand-Target Pair
Potassium voltage-gated channel subfamily A member 3 (Homo sapiens (Human))	BDBM50279024 ((1,3-dimethyl-1H-pyrazol-5-yl)(5-(furan-2-carbonyl...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem	Article PubMed	n/a	n/a	710	n/a	n/a	n/a	n/a	n/a	n/a
4SC AG Curated by ChEMBL					Assay Description Inhibition of cloned Kv1.3 channel (unknown origin) expressed in mammalian cells by whole cell patch clamp assay				Bioorg Med Chem Lett 19: 2299-304 (2009) Article DOI: 10.1016/j.bmcl.2009.02.077 BindingDB Entry DOI: 10.7270/Q29K4B38
4SC AG Curated by ChEMBL					More data for this Ligand-Target Pair
Potassium voltage-gated channel subfamily A member 3 (Homo sapiens (Human))	BDBM50278971 (2-(5-(furan-2-carbonyl)-5,6-dihydrophenanthridin-6...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	1.00E+3	n/a	n/a	n/a	n/a	n/a	n/a
4SC AG Curated by ChEMBL					Assay Description Inhibition of cloned Kv1.3 channel (unknown origin) expressed in mammalian cells by whole cell patch clamp assay				Bioorg Med Chem Lett 19: 2299-304 (2009) Article DOI: 10.1016/j.bmcl.2009.02.077 BindingDB Entry DOI: 10.7270/Q29K4B38
4SC AG Curated by ChEMBL					More data for this Ligand-Target Pair
Intermediate conductance calcium-activated potassium channel protein 4 (Homo sapiens (Human))	BDBM50279105 (5-(3-chlorobenzoyl)-5H-dibenzo[b,d]azepin-7(6H)-on...) Show SMILES Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	1.30E+3	n/a	n/a	n/a	n/a	n/a	n/a
4SC AG Curated by ChEMBL					Assay Description Inhibition of human cloned IK1 expressed in african green monkey COS7 cells by whole cell patch clamp assay				Bioorg Med Chem Lett 19: 2299-304 (2009) Article DOI: 10.1016/j.bmcl.2009.02.077 BindingDB Entry DOI: 10.7270/Q29K4B38
4SC AG Curated by ChEMBL					More data for this Ligand-Target Pair
Intermediate conductance calcium-activated potassium channel protein 4 (Homo sapiens (Human))	BDBM50279065 (5-(4-chlorophenylsulfonyl)-5H-dibenzo[b,d]azepin-7...) Show SMILES Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	1.40E+3	n/a	n/a	n/a	n/a	n/a	n/a
4SC AG Curated by ChEMBL					Assay Description Inhibition of human cloned IK1 expressed in african green monkey COS7 cells by whole cell patch clamp assay				Bioorg Med Chem Lett 19: 2299-304 (2009) Article DOI: 10.1016/j.bmcl.2009.02.077 BindingDB Entry DOI: 10.7270/Q29K4B38
4SC AG Curated by ChEMBL					More data for this Ligand-Target Pair
Potassium voltage-gated channel subfamily A member 3 (Homo sapiens (Human))	BDBM50278972 (CHEMBL500166 \| methyl 2-(5-(furan-2-carbonyl)-5,6-...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	1.40E+3	n/a	n/a	n/a	n/a	n/a	n/a
4SC AG Curated by ChEMBL					Assay Description Inhibition of cloned Kv1.3 channel (unknown origin) expressed in mammalian cells by whole cell patch clamp assay				Bioorg Med Chem Lett 19: 2299-304 (2009) Article DOI: 10.1016/j.bmcl.2009.02.077 BindingDB Entry DOI: 10.7270/Q29K4B38
4SC AG Curated by ChEMBL					More data for this Ligand-Target Pair
Potassium voltage-gated channel subfamily A member 3 (Homo sapiens (Human))	BDBM50278973 ((5-(furan-2-carbonyl)-5,6-dihydrophenanthridin-6-y...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	1.50E+3	n/a	n/a	n/a	n/a	n/a	n/a
4SC AG Curated by ChEMBL					Assay Description Inhibition of cloned Kv1.3 channel (unknown origin) expressed in mammalian cells by whole cell patch clamp assay				Bioorg Med Chem Lett 19: 2299-304 (2009) Article DOI: 10.1016/j.bmcl.2009.02.077 BindingDB Entry DOI: 10.7270/Q29K4B38
4SC AG Curated by ChEMBL					More data for this Ligand-Target Pair
Potassium voltage-gated channel subfamily A member 3 (Homo sapiens (Human))	BDBM50278994 (CHEMBL498728 \| phenanthridine-5,6(6H)-diylbis(fura...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	1.50E+3	n/a	n/a	n/a	n/a	n/a	n/a
4SC AG Curated by ChEMBL					Assay Description Inhibition of cloned Kv1.3 channel (unknown origin) expressed in mammalian cells by whole cell patch clamp assay				Bioorg Med Chem Lett 19: 2299-304 (2009) Article DOI: 10.1016/j.bmcl.2009.02.077 BindingDB Entry DOI: 10.7270/Q29K4B38
4SC AG Curated by ChEMBL					More data for this Ligand-Target Pair
Potassium voltage-gated channel subfamily A member 3 (Homo sapiens (Human))	BDBM50278938 (1-(5-(furan-2-carbonyl)-5,6-dihydrophenanthridin-6...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	1.90E+3	n/a	n/a	n/a	n/a	n/a	n/a
4SC AG Curated by ChEMBL					Assay Description Inhibition of cloned Kv1.3 channel (unknown origin) expressed in mammalian cells by whole cell patch clamp assay				Bioorg Med Chem Lett 19: 2299-304 (2009) Article DOI: 10.1016/j.bmcl.2009.02.077 BindingDB Entry DOI: 10.7270/Q29K4B38
4SC AG Curated by ChEMBL					More data for this Ligand-Target Pair
Intermediate conductance calcium-activated potassium channel protein 4 (Homo sapiens (Human))	BDBM50279063 (5-tosyl-5H-dibenzo[b,d]azepin-7(6H)-one \| CHEMBL49...) Show SMILES Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	2.10E+3	n/a	n/a	n/a	n/a	n/a	n/a
4SC AG Curated by ChEMBL					Assay Description Inhibition of human cloned IK1 expressed in african green monkey COS7 cells by whole cell patch clamp assay				Bioorg Med Chem Lett 19: 2299-304 (2009) Article DOI: 10.1016/j.bmcl.2009.02.077 BindingDB Entry DOI: 10.7270/Q29K4B38
4SC AG Curated by ChEMBL					More data for this Ligand-Target Pair
Intermediate conductance calcium-activated potassium channel protein 4 (Homo sapiens (Human))	BDBM50279103 (5-(thiophen-2-ylsulfonyl)-5H-dibenzo[b,d]azepin-7(...) Show SMILES Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	2.40E+3	n/a	n/a	n/a	n/a	n/a	n/a
4SC AG Curated by ChEMBL					Assay Description Inhibition of human cloned IK1 expressed in african green monkey COS7 cells by whole cell patch clamp assay				Bioorg Med Chem Lett 19: 2299-304 (2009) Article DOI: 10.1016/j.bmcl.2009.02.077 BindingDB Entry DOI: 10.7270/Q29K4B38
4SC AG Curated by ChEMBL					More data for this Ligand-Target Pair
Potassium voltage-gated channel subfamily A member 3 (Homo sapiens (Human))	BDBM50279105 (5-(3-chlorobenzoyl)-5H-dibenzo[b,d]azepin-7(6H)-on...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	3.40E+3	n/a	n/a	n/a	n/a	n/a	n/a
4SC AG Curated by ChEMBL					Assay Description Inhibition of cloned Kv1.3 channel (unknown origin) expressed in mammalian cells by whole cell patch clamp assay				Bioorg Med Chem Lett 19: 2299-304 (2009) Article DOI: 10.1016/j.bmcl.2009.02.077 BindingDB Entry DOI: 10.7270/Q29K4B38
4SC AG Curated by ChEMBL					More data for this Ligand-Target Pair
Potassium voltage-gated channel subfamily A member 3 (Homo sapiens (Human))	BDBM50279066 (5-(3-chlorophenylsulfonyl)-5H-dibenzo[b,d]azepin-7...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	3.60E+3	n/a	n/a	n/a	n/a	n/a	n/a
4SC AG Curated by ChEMBL					Assay Description Inhibition of cloned Kv1.3 channel (unknown origin) expressed in mammalian cells by whole cell patch clamp assay				Bioorg Med Chem Lett 19: 2299-304 (2009) Article DOI: 10.1016/j.bmcl.2009.02.077 BindingDB Entry DOI: 10.7270/Q29K4B38
4SC AG Curated by ChEMBL					More data for this Ligand-Target Pair
Potassium voltage-gated channel subfamily A member 3 (Homo sapiens (Human))	BDBM50279104 (5-(4-methylbenzoyl)-5H-dibenzo[b,d]azepin-7(6H)-on...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	4.00E+3	n/a	n/a	n/a	n/a	n/a	n/a
4SC AG Curated by ChEMBL					Assay Description Inhibition of cloned Kv1.3 channel (unknown origin) expressed in mammalian cells by whole cell patch clamp assay				Bioorg Med Chem Lett 19: 2299-304 (2009) Article DOI: 10.1016/j.bmcl.2009.02.077 BindingDB Entry DOI: 10.7270/Q29K4B38
4SC AG Curated by ChEMBL					More data for this Ligand-Target Pair
Potassium voltage-gated channel subfamily A member 3 (Homo sapiens (Human))	BDBM50278939 ((6-(cyclobutanecarbonyl)phenanthridin-5(6H)-yl)(fu...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	4.20E+3	n/a	n/a	n/a	n/a	n/a	n/a
4SC AG Curated by ChEMBL					Assay Description Inhibition of cloned Kv1.3 channel (unknown origin) expressed in mammalian cells by whole cell patch clamp assay				Bioorg Med Chem Lett 19: 2299-304 (2009) Article DOI: 10.1016/j.bmcl.2009.02.077 BindingDB Entry DOI: 10.7270/Q29K4B38
4SC AG Curated by ChEMBL					More data for this Ligand-Target Pair
Potassium voltage-gated channel subfamily A member 3 (Homo sapiens (Human))	BDBM50279107 (1-((2-chlorophenyl)diphenylmethyl)-1H-pyrazole \| C...) Show SMILES Clc1ccccc1C(c1ccccc1)(c1ccccc1)n1cccn1 Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	Purchase CHEMBL MCE KEGG PC cid PC sid UniChem Patents	Article PubMed	n/a	n/a	5.00E+3	n/a	n/a	n/a	n/a	n/a	n/a
4SC AG Curated by ChEMBL					Assay Description Inhibition of cloned Kv1.3 channel (unknown origin) expressed in mammalian cells by whole cell patch clamp assay				Bioorg Med Chem Lett 19: 2299-304 (2009) Article DOI: 10.1016/j.bmcl.2009.02.077 BindingDB Entry DOI: 10.7270/Q29K4B38
4SC AG Curated by ChEMBL					More data for this Ligand-Target Pair
Potassium voltage-gated channel subfamily A member 3 (Homo sapiens (Human))	BDBM50278936 (1-(6-(1H-indol-3-yl)phenanthridin-5(6H)-yl)ethanon...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem	Article PubMed	n/a	n/a	5.00E+3	n/a	n/a	n/a	n/a	n/a	n/a
4SC AG Curated by ChEMBL					Assay Description Inhibition of cloned Kv1.3 channel (unknown origin) expressed in mammalian cells by whole cell patch clamp assay				Bioorg Med Chem Lett 19: 2299-304 (2009) Article DOI: 10.1016/j.bmcl.2009.02.077 BindingDB Entry DOI: 10.7270/Q29K4B38
4SC AG Curated by ChEMBL					More data for this Ligand-Target Pair
Potassium voltage-gated channel subfamily A member 3 (Homo sapiens (Human))	BDBM50279063 (5-tosyl-5H-dibenzo[b,d]azepin-7(6H)-one \| CHEMBL49...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	5.80E+3	n/a	n/a	n/a	n/a	n/a	n/a
4SC AG Curated by ChEMBL					Assay Description Inhibition of cloned Kv1.3 channel (unknown origin) expressed in mammalian cells by whole cell patch clamp assay				Bioorg Med Chem Lett 19: 2299-304 (2009) Article DOI: 10.1016/j.bmcl.2009.02.077 BindingDB Entry DOI: 10.7270/Q29K4B38
4SC AG Curated by ChEMBL					More data for this Ligand-Target Pair
Potassium voltage-gated channel subfamily A member 3 (Homo sapiens (Human))	BDBM31774 (CHEMBL104 \| Canesten \| Clotrimazole \| Lotrimin \| M...) Show SMILES Clc1ccccc1C(c1ccccc1)(c1ccccc1)n1ccnc1 Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	Purchase CHEMBL DrugBank MCE KEGG MMDB PC cid PC sid PDB UniChem Patents Similars	Article PubMed	n/a	n/a	6.00E+3	n/a	n/a	n/a	n/a	n/a	n/a
4SC AG Curated by ChEMBL					Assay Description Inhibition of cloned Kv1.3 channel (unknown origin) expressed in mammalian cells by whole cell patch clamp assay				Bioorg Med Chem Lett 19: 2299-304 (2009) Article DOI: 10.1016/j.bmcl.2009.02.077 BindingDB Entry DOI: 10.7270/Q29K4B38
4SC AG Curated by ChEMBL					More data for this Ligand-Target Pair
Potassium voltage-gated channel subfamily A member 3 (Homo sapiens (Human))	BDBM50279065 (5-(4-chlorophenylsulfonyl)-5H-dibenzo[b,d]azepin-7...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	6.10E+3	n/a	n/a	n/a	n/a	n/a	n/a
4SC AG Curated by ChEMBL					Assay Description Inhibition of cloned Kv1.3 channel (unknown origin) expressed in mammalian cells by whole cell patch clamp assay				Bioorg Med Chem Lett 19: 2299-304 (2009) Article DOI: 10.1016/j.bmcl.2009.02.077 BindingDB Entry DOI: 10.7270/Q29K4B38
4SC AG Curated by ChEMBL					More data for this Ligand-Target Pair
Potassium voltage-gated channel subfamily A member 3 (Homo sapiens (Human))	BDBM50278937 (1-(5-(furan-2-carbonyl)-5,6-dihydrophenanthridin-6...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	7.40E+3	n/a	n/a	n/a	n/a	n/a	n/a
4SC AG Curated by ChEMBL					Assay Description Inhibition of cloned Kv1.3 channel (unknown origin) expressed in mammalian cells by whole cell patch clamp assay				Bioorg Med Chem Lett 19: 2299-304 (2009) Article DOI: 10.1016/j.bmcl.2009.02.077 BindingDB Entry DOI: 10.7270/Q29K4B38
4SC AG Curated by ChEMBL					More data for this Ligand-Target Pair
Intermediate conductance calcium-activated potassium channel protein 4 (Homo sapiens (Human))	BDBM50279106 (4-(4-phenoxybutoxy)-7H-furo[3,2-g]chromen-7-one \| ...) Show SMILES O=c1ccc2c(OCCCCOc3ccccc3)c3ccoc3cc2o1 Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	Purchase CHEMBL MCE PC cid PC sid UniChem Patents Similars	Article PubMed	n/a	n/a	1.00E+4	n/a	n/a	n/a	n/a	n/a	n/a
4SC AG Curated by ChEMBL					Assay Description Inhibition of human cloned IK1 expressed in african green monkey COS7 cells by whole cell patch clamp assay				Bioorg Med Chem Lett 19: 2299-304 (2009) Article DOI: 10.1016/j.bmcl.2009.02.077 BindingDB Entry DOI: 10.7270/Q29K4B38
4SC AG Curated by ChEMBL					More data for this Ligand-Target Pair
Potassium voltage-gated channel subfamily A member 3 (Homo sapiens (Human))	BDBM50279064 (5-(4-nitrophenylsulfonyl)-5H-dibenzo[b,d]azepin-7(...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	>1.00E+4	n/a	n/a	n/a	n/a	n/a	n/a
4SC AG Curated by ChEMBL					Assay Description Inhibition of cloned Kv1.3 channel (unknown origin) expressed in mammalian cells by whole cell patch clamp assay				Bioorg Med Chem Lett 19: 2299-304 (2009) Article DOI: 10.1016/j.bmcl.2009.02.077 BindingDB Entry DOI: 10.7270/Q29K4B38
4SC AG Curated by ChEMBL					More data for this Ligand-Target Pair
Potassium voltage-gated channel subfamily A member 3 (Homo sapiens (Human))	BDBM50279103 (5-(thiophen-2-ylsulfonyl)-5H-dibenzo[b,d]azepin-7(...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	1.30E+4	n/a	n/a	n/a	n/a	n/a	n/a
4SC AG Curated by ChEMBL					Assay Description Inhibition of cloned Kv1.3 channel (unknown origin) expressed in mammalian cells by whole cell patch clamp assay				Bioorg Med Chem Lett 19: 2299-304 (2009) Article DOI: 10.1016/j.bmcl.2009.02.077 BindingDB Entry DOI: 10.7270/Q29K4B38
4SC AG Curated by ChEMBL					More data for this Ligand-Target Pair
Intermediate conductance calcium-activated potassium channel protein 4 (Homo sapiens (Human))	BDBM50279104 (5-(4-methylbenzoyl)-5H-dibenzo[b,d]azepin-7(6H)-on...) Show SMILES Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	1.60E+4	n/a	n/a	n/a	n/a	n/a	n/a
4SC AG Curated by ChEMBL					Assay Description Inhibition of human cloned IK1 expressed in african green monkey COS7 cells by whole cell patch clamp assay				Bioorg Med Chem Lett 19: 2299-304 (2009) Article DOI: 10.1016/j.bmcl.2009.02.077 BindingDB Entry DOI: 10.7270/Q29K4B38
4SC AG Curated by ChEMBL					More data for this Ligand-Target Pair