Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Solute carrier family 13 member 5 (Homo sapiens (Human)) | BDBM50149291 (CHEMBL3770609) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 110 | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Inc. Curated by ChEMBL | Assay Description Inhibition of NaCT (unknown origin) expressed in HEK293 cells assessed as inhibition of [14C]citrate uptake by microbeta plate reader analysis | J Med Chem 59: 1165-75 (2016) Article DOI: 10.1021/acs.jmedchem.5b01752 BindingDB Entry DOI: 10.7270/Q2ZW1NRC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Solute carrier family 13 member 5 (Homo sapiens (Human)) | BDBM50149290 (CHEMBL3771175) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem | Article PubMed | n/a | n/a | 110 | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Inc. Curated by ChEMBL | Assay Description Inhibition of NaCT (unknown origin) expressed in HEK293 cells assessed as inhibition of [14C]citrate uptake by microbeta plate reader analysis | J Med Chem 59: 1165-75 (2016) Article DOI: 10.1021/acs.jmedchem.5b01752 BindingDB Entry DOI: 10.7270/Q2ZW1NRC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Solute carrier family 13 member 5 (Homo sapiens (Human)) | BDBM50149291 (CHEMBL3770609) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 110 | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Inc. Curated by ChEMBL | Assay Description Inhibition of NaCT (unknown origin) expressed in HEK293 cells assessed as inhibition of [14C]citrate uptake by microbeta plate reader analysis | J Med Chem 59: 1165-75 (2016) Article DOI: 10.1021/acs.jmedchem.5b01752 BindingDB Entry DOI: 10.7270/Q2ZW1NRC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Solute carrier family 13 member 5 (Homo sapiens (Human)) | BDBM50149290 (CHEMBL3771175) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem | Article PubMed | n/a | n/a | 110 | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Inc. Curated by ChEMBL | Assay Description Inhibition of NaCT (unknown origin) expressed in HEK293 cells assessed as inhibition of [14C]citrate uptake by microbeta plate reader analysis | J Med Chem 59: 1165-75 (2016) Article DOI: 10.1021/acs.jmedchem.5b01752 BindingDB Entry DOI: 10.7270/Q2ZW1NRC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Solute carrier family 13 member 5 (Rattus norvegicus) | BDBM50149244 (CHEMBL3771118) | UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL MCE KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 120 | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Inc. Curated by ChEMBL | Assay Description Inhibition of NaCT in rat hepatocytes assessed as [14C]-citrate uptake after 30 mins by scintillation counting method | J Med Chem 59: 1165-75 (2016) Article DOI: 10.1021/acs.jmedchem.5b01752 BindingDB Entry DOI: 10.7270/Q2ZW1NRC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Solute carrier family 13 member 5 (Rattus norvegicus) | BDBM50149244 (CHEMBL3771118) | UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL MCE KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 126 | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Inc. Curated by ChEMBL | Assay Description Inhibition of NaCT in rat hepatocytes assessed as [14C]-citrate uptake after 30 mins by scintillation counting method | J Med Chem 59: 1165-75 (2016) Article DOI: 10.1021/acs.jmedchem.5b01752 BindingDB Entry DOI: 10.7270/Q2ZW1NRC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Solute carrier family 13 member 5 (Homo sapiens (Human)) | BDBM50149289 (CHEMBL3770497) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 190 | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Inc. Curated by ChEMBL | Assay Description Inhibition of NaCT (unknown origin) expressed in HEK293 cells assessed as inhibition of [14C]citrate uptake by microbeta plate reader analysis | J Med Chem 59: 1165-75 (2016) Article DOI: 10.1021/acs.jmedchem.5b01752 BindingDB Entry DOI: 10.7270/Q2ZW1NRC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Solute carrier family 13 member 5 (Homo sapiens (Human)) | BDBM50149289 (CHEMBL3770497) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 200 | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Inc. Curated by ChEMBL | Assay Description Inhibition of NaCT (unknown origin) expressed in HEK293 cells assessed as inhibition of [14C]citrate uptake by microbeta plate reader analysis | J Med Chem 59: 1165-75 (2016) Article DOI: 10.1021/acs.jmedchem.5b01752 BindingDB Entry DOI: 10.7270/Q2ZW1NRC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Solute carrier family 13 member 5 (Mus musculus) | BDBM50149244 (CHEMBL3771118) | UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL MCE KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 210 | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Inc. Curated by ChEMBL | Assay Description Inhibition of NaCT in mouse hepatocytes assessed as [14C]-citrate uptake after 30 mins by scintillation counting method | J Med Chem 59: 1165-75 (2016) Article DOI: 10.1021/acs.jmedchem.5b01752 BindingDB Entry DOI: 10.7270/Q2ZW1NRC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Solute carrier family 13 member 5 (Mus musculus) | BDBM50149244 (CHEMBL3771118) | UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL MCE KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 214 | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Inc. Curated by ChEMBL | Assay Description Inhibition of NaCT in mouse hepatocytes assessed as [14C]-citrate uptake after 30 mins by scintillation counting method | J Med Chem 59: 1165-75 (2016) Article DOI: 10.1021/acs.jmedchem.5b01752 BindingDB Entry DOI: 10.7270/Q2ZW1NRC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Solute carrier family 13 member 5 (Homo sapiens (Human)) | BDBM50149293 (CHEMBL3770675) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 316 | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Inc. Curated by ChEMBL | Assay Description Inhibition of NaCT (unknown origin) expressed in HEK293 cells assessed as inhibition of [14C]citrate uptake by microbeta plate reader analysis | J Med Chem 59: 1165-75 (2016) Article DOI: 10.1021/acs.jmedchem.5b01752 BindingDB Entry DOI: 10.7270/Q2ZW1NRC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Solute carrier family 13 member 5 (Homo sapiens (Human)) | BDBM50149291 (CHEMBL3770609) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 316 | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Inc. Curated by ChEMBL | Assay Description Inhibition of NaCT in human hepatocytes assessed as [14C]-citrate uptake after 30 mins by scintillation counting method | J Med Chem 59: 1165-75 (2016) Article DOI: 10.1021/acs.jmedchem.5b01752 BindingDB Entry DOI: 10.7270/Q2ZW1NRC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Solute carrier family 13 member 5 (Homo sapiens (Human)) | BDBM50149291 (CHEMBL3770609) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 330 | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Inc. Curated by ChEMBL | Assay Description Inhibition of NaCT in human hepatocytes assessed as [14C]-citrate uptake after 30 mins by scintillation counting method | J Med Chem 59: 1165-75 (2016) Article DOI: 10.1021/acs.jmedchem.5b01752 BindingDB Entry DOI: 10.7270/Q2ZW1NRC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Solute carrier family 13 member 5 (Homo sapiens (Human)) | BDBM50149293 (CHEMBL3770675) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 330 | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Inc. Curated by ChEMBL | Assay Description Inhibition of NaCT (unknown origin) expressed in HEK293 cells assessed as inhibition of [14C]citrate uptake by microbeta plate reader analysis | J Med Chem 59: 1165-75 (2016) Article DOI: 10.1021/acs.jmedchem.5b01752 BindingDB Entry DOI: 10.7270/Q2ZW1NRC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Solute carrier family 13 member 5 (Homo sapiens (Human)) | BDBM50149294 (CHEMBL3769578) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL MCE KEGG PC cid PC sid PDB UniChem Similars | PDB Article PubMed | n/a | n/a | 501 | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Inc. Curated by ChEMBL | Assay Description Inhibition of NaCT (unknown origin) expressed in HEK293 cells assessed as inhibition of [14C]citrate uptake by microbeta plate reader analysis | J Med Chem 59: 1165-75 (2016) Article DOI: 10.1021/acs.jmedchem.5b01752 BindingDB Entry DOI: 10.7270/Q2ZW1NRC | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
Solute carrier family 13 member 5 (Homo sapiens (Human)) | BDBM50149294 (CHEMBL3769578) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL MCE KEGG PC cid PC sid PDB UniChem Similars | PDB Article PubMed | n/a | n/a | 501 | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Inc. Curated by ChEMBL | Assay Description Inhibition of NaCT (unknown origin) expressed in HEK293 cells assessed as inhibition of [14C]citrate uptake by microbeta plate reader analysis | J Med Chem 59: 1165-75 (2016) Article DOI: 10.1021/acs.jmedchem.5b01752 BindingDB Entry DOI: 10.7270/Q2ZW1NRC | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
Solute carrier family 13 member 5 (Homo sapiens (Human)) | BDBM50149244 (CHEMBL3771118) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL MCE KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 501 | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Inc. Curated by ChEMBL | Assay Description Inhibition of NaCT (unknown origin) expressed in HEK293 cells assessed as inhibition of [14C]citrate uptake by microbeta plate reader analysis | J Med Chem 59: 1165-75 (2016) Article DOI: 10.1021/acs.jmedchem.5b01752 BindingDB Entry DOI: 10.7270/Q2ZW1NRC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Solute carrier family 13 member 5 (Homo sapiens (Human)) | BDBM50149244 (CHEMBL3771118) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL MCE KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 510 | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Inc. Curated by ChEMBL | Assay Description Inhibition of NaCT (unknown origin) expressed in HEK293 cells assessed as inhibition of [14C]citrate uptake by microbeta plate reader analysis | J Med Chem 59: 1165-75 (2016) Article DOI: 10.1021/acs.jmedchem.5b01752 BindingDB Entry DOI: 10.7270/Q2ZW1NRC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Solute carrier family 13 member 5 (Homo sapiens (Human)) | BDBM50149236 (CHEMBL3770370) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 650 | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Inc. Curated by ChEMBL | Assay Description Inhibition of NaCT (unknown origin) expressed in HEK293 cells assessed as inhibition of [14C]citrate uptake by microbeta plate reader analysis | J Med Chem 59: 1165-75 (2016) Article DOI: 10.1021/acs.jmedchem.5b01752 BindingDB Entry DOI: 10.7270/Q2ZW1NRC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Solute carrier family 13 member 5 (Homo sapiens (Human)) | BDBM50149236 (CHEMBL3770370) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 650 | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Inc. Curated by ChEMBL | Assay Description Inhibition of NaCT (unknown origin) expressed in HEK293 cells assessed as inhibition of [14C]citrate uptake by microbeta plate reader analysis | J Med Chem 59: 1165-75 (2016) Article DOI: 10.1021/acs.jmedchem.5b01752 BindingDB Entry DOI: 10.7270/Q2ZW1NRC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Solute carrier family 13 member 5 (Homo sapiens (Human)) | BDBM50149244 (CHEMBL3771118) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL MCE KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 740 | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Inc. Curated by ChEMBL | Assay Description Inhibition of NaCT in human hepatocytes assessed as [14C]-citrate uptake after 30 mins by scintillation counting method | J Med Chem 59: 1165-75 (2016) Article DOI: 10.1021/acs.jmedchem.5b01752 BindingDB Entry DOI: 10.7270/Q2ZW1NRC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Solute carrier family 13 member 5 (Homo sapiens (Human)) | BDBM50149215 (CHEMBL3769514) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL KEGG MMDB PC cid PC sid PDB UniChem Patents Similars | Article PubMed | n/a | n/a | 794 | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Inc. Curated by ChEMBL | Assay Description Inhibition of NaCT (unknown origin) expressed in HEK293 cells assessed as inhibition of [14C]citrate uptake by microbeta plate reader analysis | J Med Chem 59: 1165-75 (2016) Article DOI: 10.1021/acs.jmedchem.5b01752 BindingDB Entry DOI: 10.7270/Q2ZW1NRC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Solute carrier family 13 member 5 (Homo sapiens (Human)) | BDBM50149244 (CHEMBL3771118) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL MCE KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 794 | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Inc. Curated by ChEMBL | Assay Description Inhibition of NaCT in human hepatocytes assessed as [14C]-citrate uptake after 30 mins by scintillation counting method | J Med Chem 59: 1165-75 (2016) Article DOI: 10.1021/acs.jmedchem.5b01752 BindingDB Entry DOI: 10.7270/Q2ZW1NRC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Solute carrier family 13 member 5 (Homo sapiens (Human)) | BDBM50149215 (CHEMBL3769514) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL KEGG MMDB PC cid PC sid PDB UniChem Patents Similars | Article PubMed | n/a | n/a | 800 | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Inc. Curated by ChEMBL | Assay Description Inhibition of NaCT (unknown origin) expressed in HEK293 cells assessed as inhibition of [14C]citrate uptake by microbeta plate reader analysis | J Med Chem 59: 1165-75 (2016) Article DOI: 10.1021/acs.jmedchem.5b01752 BindingDB Entry DOI: 10.7270/Q2ZW1NRC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Solute carrier family 13 member 5 (Homo sapiens (Human)) | BDBM50149233 (CHEMBL3769911) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.59E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Inc. Curated by ChEMBL | Assay Description Inhibition of NaCT (unknown origin) expressed in HEK293 cells assessed as inhibition of [14C]citrate uptake by microbeta plate reader analysis | J Med Chem 59: 1165-75 (2016) Article DOI: 10.1021/acs.jmedchem.5b01752 BindingDB Entry DOI: 10.7270/Q2ZW1NRC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Solute carrier family 13 member 5 (Homo sapiens (Human)) | BDBM50149233 (CHEMBL3769911) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.65E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Inc. Curated by ChEMBL | Assay Description Inhibition of NaCT (unknown origin) expressed in HEK293 cells assessed as inhibition of [14C]citrate uptake by microbeta plate reader analysis | J Med Chem 59: 1165-75 (2016) Article DOI: 10.1021/acs.jmedchem.5b01752 BindingDB Entry DOI: 10.7270/Q2ZW1NRC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Solute carrier family 13 member 5 (Homo sapiens (Human)) | BDBM50149247 (CHEMBL3769766) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem | Article PubMed | n/a | n/a | 3.16E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Inc. Curated by ChEMBL | Assay Description Inhibition of NaCT (unknown origin) expressed in HEK293 cells assessed as inhibition of [14C]citrate uptake by microbeta plate reader analysis | J Med Chem 59: 1165-75 (2016) Article DOI: 10.1021/acs.jmedchem.5b01752 BindingDB Entry DOI: 10.7270/Q2ZW1NRC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Solute carrier family 13 member 5 (Homo sapiens (Human)) | BDBM50149247 (CHEMBL3769766) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem | Article PubMed | n/a | n/a | 3.37E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Inc. Curated by ChEMBL | Assay Description Inhibition of NaCT (unknown origin) expressed in HEK293 cells assessed as inhibition of [14C]citrate uptake by microbeta plate reader analysis | J Med Chem 59: 1165-75 (2016) Article DOI: 10.1021/acs.jmedchem.5b01752 BindingDB Entry DOI: 10.7270/Q2ZW1NRC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Solute carrier family 13 member 2 (Homo sapiens (Human)) | BDBM50149244 (CHEMBL3771118) | UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL MCE KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.32E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Inc. Curated by ChEMBL | Assay Description Inhibition of NaDC1 (unknown origin) expressed in HEK293 cells assessed as inhibition of [14C]citrate uptake by microbeta plate reader analysis | J Med Chem 59: 1165-75 (2016) Article DOI: 10.1021/acs.jmedchem.5b01752 BindingDB Entry DOI: 10.7270/Q2ZW1NRC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Solute carrier family 13 member 2 (Homo sapiens (Human)) | BDBM50149244 (CHEMBL3771118) | UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL MCE KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.32E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Inc. Curated by ChEMBL | Assay Description Inhibition of NaDC1 (unknown origin) expressed in HEK293 cells assessed as inhibition of [14C]citrate uptake by microbeta plate reader analysis | J Med Chem 59: 1165-75 (2016) Article DOI: 10.1021/acs.jmedchem.5b01752 BindingDB Entry DOI: 10.7270/Q2ZW1NRC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Solute carrier family 13 member 3 (Homo sapiens (Human)) | BDBM50149244 (CHEMBL3771118) | UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL MCE KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.41E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Inc. Curated by ChEMBL | Assay Description Inhibition of NaDC3 (unknown origin) expressed in HEK293 cells assessed as inhibition of [14C]citrate uptake by microbeta plate reader analysis | J Med Chem 59: 1165-75 (2016) Article DOI: 10.1021/acs.jmedchem.5b01752 BindingDB Entry DOI: 10.7270/Q2ZW1NRC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Solute carrier family 13 member 3 (Homo sapiens (Human)) | BDBM50149244 (CHEMBL3771118) | UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL MCE KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.41E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Inc. Curated by ChEMBL | Assay Description Inhibition of NaDC3 (unknown origin) expressed in HEK293 cells assessed as inhibition of [14C]citrate uptake by microbeta plate reader analysis | J Med Chem 59: 1165-75 (2016) Article DOI: 10.1021/acs.jmedchem.5b01752 BindingDB Entry DOI: 10.7270/Q2ZW1NRC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Solute carrier family 13 member 5 (Homo sapiens (Human)) | BDBM50149294 (CHEMBL3769578) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL MCE KEGG PC cid PC sid PDB UniChem Similars | PDB Article PubMed | n/a | n/a | 1.58E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Inc. Curated by ChEMBL | Assay Description Inhibition of NaCT in human hepatocytes assessed as [14C]-citrate uptake after 30 mins by scintillation counting method | J Med Chem 59: 1165-75 (2016) Article DOI: 10.1021/acs.jmedchem.5b01752 BindingDB Entry DOI: 10.7270/Q2ZW1NRC | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
Solute carrier family 13 member 5 (Homo sapiens (Human)) | BDBM50149294 (CHEMBL3769578) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL MCE KEGG PC cid PC sid PDB UniChem Similars | PDB Article PubMed | n/a | n/a | 1.62E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Inc. Curated by ChEMBL | Assay Description Inhibition of NaCT in human hepatocytes assessed as [14C]-citrate uptake after 30 mins by scintillation counting method | J Med Chem 59: 1165-75 (2016) Article DOI: 10.1021/acs.jmedchem.5b01752 BindingDB Entry DOI: 10.7270/Q2ZW1NRC | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
Solute carrier family 13 member 5 (Homo sapiens (Human)) | BDBM50149223 (CHEMBL3770439) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >1.70E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Inc. Curated by ChEMBL | Assay Description Inhibition of NaCT (unknown origin) expressed in HEK293 cells assessed as inhibition of [14C]citrate uptake by microbeta plate reader analysis | J Med Chem 59: 1165-75 (2016) Article DOI: 10.1021/acs.jmedchem.5b01752 BindingDB Entry DOI: 10.7270/Q2ZW1NRC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Solute carrier family 13 member 5 (Homo sapiens (Human)) | BDBM50149246 (CHEMBL3769920) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Patents | Article PubMed | n/a | n/a | >1.80E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Inc. Curated by ChEMBL | Assay Description Inhibition of NaCT (unknown origin) expressed in HEK293 cells assessed as inhibition of [14C]citrate uptake by microbeta plate reader analysis | J Med Chem 59: 1165-75 (2016) Article DOI: 10.1021/acs.jmedchem.5b01752 BindingDB Entry DOI: 10.7270/Q2ZW1NRC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Solute carrier family 13 member 5 (Homo sapiens (Human)) | BDBM50149292 (CHEMBL3771155) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | >2.50E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Inc. Curated by ChEMBL | Assay Description Inhibition of NaCT (unknown origin) expressed in HEK293 cells assessed as inhibition of [14C]citrate uptake by microbeta plate reader analysis | J Med Chem 59: 1165-75 (2016) Article DOI: 10.1021/acs.jmedchem.5b01752 BindingDB Entry DOI: 10.7270/Q2ZW1NRC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Solute carrier family 13 member 5 (Homo sapiens (Human)) | BDBM50149292 (CHEMBL3771155) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | >3.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Inc. Curated by ChEMBL | Assay Description Inhibition of NaCT in human hepatocytes assessed as [14C]-citrate uptake after 30 mins by scintillation counting method | J Med Chem 59: 1165-75 (2016) Article DOI: 10.1021/acs.jmedchem.5b01752 BindingDB Entry DOI: 10.7270/Q2ZW1NRC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Solute carrier family 13 member 2 (Homo sapiens (Human)) | BDBM50149294 (CHEMBL3769578) | UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL MCE KEGG PC cid PC sid PDB UniChem Similars | Article PubMed | n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Inc. Curated by ChEMBL | Assay Description Inhibition of NaDC1 (unknown origin) expressed in HEK293 cells assessed as inhibition of [14C]citrate uptake by microbeta plate reader analysis | J Med Chem 59: 1165-75 (2016) Article DOI: 10.1021/acs.jmedchem.5b01752 BindingDB Entry DOI: 10.7270/Q2ZW1NRC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Solute carrier family 13 member 3 (Homo sapiens (Human)) | BDBM50149294 (CHEMBL3769578) | UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL MCE KEGG PC cid PC sid PDB UniChem Similars | Article PubMed | n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Inc. Curated by ChEMBL | Assay Description Inhibition of NaDC3 (unknown origin) expressed in HEK293 cells assessed as inhibition of [14C]citrate uptake by microbeta plate reader analysis | J Med Chem 59: 1165-75 (2016) Article DOI: 10.1021/acs.jmedchem.5b01752 BindingDB Entry DOI: 10.7270/Q2ZW1NRC | |||||||||||
More data for this Ligand-Target Pair |