BindingDB PrimarySearch

Found 6 hits Enz. Inhib. hit(s) with all data for entry = 50047263
Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kJ/mole	IC50 nM	Kd nM	EC50/IC50 nM	k_off s^-1	k_on M^-1s^-1	pH	Temp °C
Casein kinase II subunit alpha (Homo sapiens (Human))	BDBM50156669 (4,5,6,7-TETRABROMO-BENZIMIDAZOLE \| 4,5,6,7-tetrabr...) Show SMILES Brc1c(Br)c(Br)c2[nH]cnc2c1Br Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	Purchase CHEMBL MCE MMDB PC cid PC sid PDB UniChem Patents Similars	Article PubMed	45	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Colorado State University Curated by ChEMBL					Assay Description Inhibition of human wild type CK2alpha				J Med Chem 59: 1655-70 (2016) Article DOI: 10.1021/acs.jmedchem.5b00997 BindingDB Entry DOI: 10.7270/Q24T6M70
Colorado State University Curated by ChEMBL					More data for this Ligand-Target Pair
Casein kinase II subunit alpha (Homo sapiens (Human))	BDBM50156368 (CHEMBL608394) Show SMILES Brc1c(Br)c(Br)c2[nH]c(=S)[nH]c2c1Br Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid PDB UniChem Patents Similars	Article PubMed	70	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Colorado State University Curated by ChEMBL					Assay Description Inhibition of human wild type CK2alpha				J Med Chem 59: 1655-70 (2016) Article DOI: 10.1021/acs.jmedchem.5b00997 BindingDB Entry DOI: 10.7270/Q24T6M70
Colorado State University Curated by ChEMBL					More data for this Ligand-Target Pair
Casein kinase II subunit alpha (Homo sapiens (Human))	BDBM50156367 (CHEMBL3793598) Show SMILES Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Patents Similars	Article PubMed	150	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Colorado State University Curated by ChEMBL					Assay Description Competitive inhibition of human wild type CK2alpha by Dixon plot analysis				J Med Chem 59: 1655-70 (2016) Article DOI: 10.1021/acs.jmedchem.5b00997 BindingDB Entry DOI: 10.7270/Q24T6M70
Colorado State University Curated by ChEMBL					More data for this Ligand-Target Pair
Casein kinase II subunit alpha (Homo sapiens (Human))	BDBM34045 (iodinated benzimidazole, 8a) Show SMILES Cc1nc2c(I)c(Cl)c(Cl)c(I)c2[nH]1 Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem Similars	Article PubMed	200	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Colorado State University Curated by ChEMBL					Assay Description Competitive inhibition of human wild type CK2alpha by Dixon plot analysis				J Med Chem 59: 1655-70 (2016) Article DOI: 10.1021/acs.jmedchem.5b00997 BindingDB Entry DOI: 10.7270/Q24T6M70
Colorado State University Curated by ChEMBL					More data for this Ligand-Target Pair
Casein kinase II subunit alpha (Homo sapiens (Human))	BDBM34041 (iodinated benzimidazole, 4a) Show SMILES Clc1c(Cl)c(I)c2[nH]cnc2c1I Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem Similars	Article PubMed	300	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Colorado State University Curated by ChEMBL					Assay Description Competitive inhibition of human wild type CK2alpha by Dixon plot analysis				J Med Chem 59: 1655-70 (2016) Article DOI: 10.1021/acs.jmedchem.5b00997 BindingDB Entry DOI: 10.7270/Q24T6M70
Colorado State University Curated by ChEMBL					More data for this Ligand-Target Pair
Casein kinase II subunit alpha (Homo sapiens (Human))	BDBM50156369 (CHEMBL227370) Show SMILES Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Patents Similars	Article PubMed	400	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Colorado State University Curated by ChEMBL					Assay Description Inhibition of CK2alpha (unknown origin)				J Med Chem 59: 1655-70 (2016) Article DOI: 10.1021/acs.jmedchem.5b00997 BindingDB Entry DOI: 10.7270/Q24T6M70
Colorado State University Curated by ChEMBL					More data for this Ligand-Target Pair