Compile Data Set for Download or QSAR

Found 60 hits Enz. Inhib. hit(s) with all data for entry = 50047266   

Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kJ/mole	IC50 nM	Kd nM	EC50/IC50 nM	koff s-1	kon M-1s-1	pH	Temp °C
Serine/threonine-protein kinase pim-1 (Homo sapiens (Human))	BDBM50161840 (CHEMBL3792425) Show SMILES Nc1cc(nc(n1)C(F)(F)F)-c1ccncc1NC(=O)c1nc(ccc1N)-c1c(F)cccc1F Show InChI InChI=1S/C22H14F5N7O/c23-11-2-1-3-12(24)18(11)14-5-4-13(28)19(31-14)20(35)32-16-9-30-7-6-10(16)15-8-17(29)34-21(33-15)22(25,26)27/h1-9H,28H2,(H,32,35)(H2,29,33,34)	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem	Article PubMed	<1	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Novartis Institutes for Biomedical Research Curated by ChEMBL					Assay Description Inhibition of Pim1 (unknown origin) using BAD peptide preincubated for 15 mins followed by ATP addition measured after 60 to 100 mins by Kinase-Glo r...				Bioorg Med Chem Lett 26: 2328-32 (2016) Article DOI: 10.1016/j.bmcl.2016.03.037 BindingDB Entry DOI: 10.7270/Q2WD42F0
					More data for this Ligand-Target Pair
Serine/threonine-protein kinase pim-1 (Homo sapiens (Human))	BDBM50161839 (CHEMBL3792736) Show SMILES Nc1cc(nc(n1)C(F)(F)F)-c1ccncc1NC(=O)c1nc(ccc1N)-c1nccs1 Show InChI InChI=1S/C19H13F3N8OS/c20-19(21,22)18-29-12(7-14(24)30-18)9-3-4-25-8-13(9)28-16(31)15-10(23)1-2-11(27-15)17-26-5-6-32-17/h1-8H,23H2,(H,28,31)(H2,24,29,30)	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	<1	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Novartis Institutes for Biomedical Research Curated by ChEMBL					Assay Description Inhibition of Pim1 (unknown origin) using BAD peptide preincubated for 15 mins followed by ATP addition measured after 60 to 100 mins by Kinase-Glo r...				Bioorg Med Chem Lett 26: 2328-32 (2016) Article DOI: 10.1016/j.bmcl.2016.03.037 BindingDB Entry DOI: 10.7270/Q2WD42F0
					More data for this Ligand-Target Pair
Serine/threonine-protein kinase pim-1 (Homo sapiens (Human))	BDBM50161838 (CHEMBL3792922) Show SMILES Cc1cc(nc(N)n1)-c1ccncc1NC(=O)c1nc(ccc1N)-c1nccs1 Show InChI InChI=1S/C19H16N8OS/c1-10-8-14(27-19(21)24-10)11-4-5-22-9-15(11)26-17(28)16-12(20)2-3-13(25-16)18-23-6-7-29-18/h2-9H,20H2,1H3,(H,26,28)(H2,21,24,27)	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	<1	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Novartis Institutes for Biomedical Research Curated by ChEMBL					Assay Description Inhibition of Pim1 (unknown origin) using BAD peptide preincubated for 15 mins followed by ATP addition measured after 60 to 100 mins by Kinase-Glo r...				Bioorg Med Chem Lett 26: 2328-32 (2016) Article DOI: 10.1016/j.bmcl.2016.03.037 BindingDB Entry DOI: 10.7270/Q2WD42F0
					More data for this Ligand-Target Pair
Serine/threonine-protein kinase pim-3 (Homo sapiens (Human))	BDBM106896 (US8592455, 96) Show SMILES C[C@H]1CN(C[C@@H](N)[C@@H]1O)c1ccncc1NC(=O)c1ccc(F)c(n1)-c1c(F)cccc1F |r,wU:7.8,wD:1.0,5.5,(-6,2.69,;-4.67,1.93,;-4.67,.38,;-3.33,-.38,;-2,.38,;-2,1.93,;-.67,2.69,;-3.33,2.69,;-3.33,4.23,;-3.33,-1.93,;-4.67,-2.69,;-4.67,-4.23,;-3.33,-5,;-2,-4.23,;-2,-2.69,;-.67,-1.93,;.67,-2.69,;.67,-4.23,;2,-1.93,;3.33,-2.69,;4.67,-1.93,;4.67,-.38,;6,.38,;3.33,.38,;2,-.38,;3.33,1.93,;4.67,2.69,;6,1.93,;4.67,4.23,;3.33,5,;2,4.23,;2,2.69,;.67,1.93,)| Show InChI InChI=1S/C23H22F3N5O2/c1-12-10-31(11-16(27)22(12)32)19-7-8-28-9-18(19)30-23(33)17-6-5-15(26)21(29-17)20-13(24)3-2-4-14(20)25/h2-9,12,16,22,32H,10-11,27H2,1H3,(H,30,33)/t12-,16+,22+/m0/s1	KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	Purchase MCE PC cid PC sid PDB UniChem Similars	Article PubMed	<1	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Novartis Institutes for Biomedical Research Curated by ChEMBL					Assay Description Inhibition of Pim3 (unknown origin) using BAD peptide preincubated for 15 mins followed by ATP addition measured after 60 to 100 mins by Kinase-Glo r...				Bioorg Med Chem Lett 26: 2328-32 (2016) Article DOI: 10.1016/j.bmcl.2016.03.037 BindingDB Entry DOI: 10.7270/Q2WD42F0
					More data for this Ligand-Target Pair
Serine/threonine-protein kinase pim-1 (Homo sapiens (Human))	BDBM50160995 (CHEMBL3793938) Show SMILES Cc1nc(N)cc(n1)-c1ccncc1NC(=O)c1nc(ccc1N)-c1c(F)cccc1F Show InChI InChI=1S/C22H17F2N7O/c1-11-28-17(9-19(26)29-11)12-7-8-27-10-18(12)31-22(32)21-15(25)5-6-16(30-21)20-13(23)3-2-4-14(20)24/h2-10H,25H2,1H3,(H,31,32)(H2,26,28,29)	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	<1	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Novartis Institutes for Biomedical Research Curated by ChEMBL					Assay Description Inhibition of Pim1 (unknown origin) using BAD peptide preincubated for 15 mins followed by ATP addition measured after 60 to 100 mins by Kinase-Glo r...				Bioorg Med Chem Lett 26: 2328-32 (2016) Article DOI: 10.1016/j.bmcl.2016.03.037 BindingDB Entry DOI: 10.7270/Q2WD42F0
					More data for this Ligand-Target Pair
Serine/threonine-protein kinase pim-1 (Homo sapiens (Human))	BDBM106896 (US8592455, 96) Show SMILES C[C@H]1CN(C[C@@H](N)[C@@H]1O)c1ccncc1NC(=O)c1ccc(F)c(n1)-c1c(F)cccc1F |r,wU:7.8,wD:1.0,5.5,(-6,2.69,;-4.67,1.93,;-4.67,.38,;-3.33,-.38,;-2,.38,;-2,1.93,;-.67,2.69,;-3.33,2.69,;-3.33,4.23,;-3.33,-1.93,;-4.67,-2.69,;-4.67,-4.23,;-3.33,-5,;-2,-4.23,;-2,-2.69,;-.67,-1.93,;.67,-2.69,;.67,-4.23,;2,-1.93,;3.33,-2.69,;4.67,-1.93,;4.67,-.38,;6,.38,;3.33,.38,;2,-.38,;3.33,1.93,;4.67,2.69,;6,1.93,;4.67,4.23,;3.33,5,;2,4.23,;2,2.69,;.67,1.93,)| Show InChI InChI=1S/C23H22F3N5O2/c1-12-10-31(11-16(27)22(12)32)19-7-8-28-9-18(19)30-23(33)17-6-5-15(26)21(29-17)20-13(24)3-2-4-14(20)25/h2-9,12,16,22,32H,10-11,27H2,1H3,(H,30,33)/t12-,16+,22+/m0/s1	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	Purchase MCE PC cid PC sid PDB UniChem Similars	Article PubMed	<1	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Novartis Institutes for Biomedical Research Curated by ChEMBL					Assay Description Inhibition of Pim1 (unknown origin) using BAD peptide preincubated for 15 mins followed by ATP addition measured after 60 to 100 mins by Kinase-Glo r...				Bioorg Med Chem Lett 26: 2328-32 (2016) Article DOI: 10.1016/j.bmcl.2016.03.037 BindingDB Entry DOI: 10.7270/Q2WD42F0
					More data for this Ligand-Target Pair
Serine/threonine-protein kinase pim-1 (Homo sapiens (Human))	BDBM50162818 (CHEMBL3793067) Show SMILES Cc1cc(cc(N)n1)-c1ccncc1NC(=O)c1nc(ccc1N)-c1c(F)cccc1F Show InChI InChI=1S/C23H18F2N6O/c1-12-9-13(10-20(27)29-12)14-7-8-28-11-19(14)31-23(32)22-17(26)5-6-18(30-22)21-15(24)3-2-4-16(21)25/h2-11H,26H2,1H3,(H2,27,29)(H,31,32)	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Patents Similars	Article PubMed	<1	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Novartis Institutes for Biomedical Research Curated by ChEMBL					Assay Description Inhibition of Pim1 (unknown origin) using BAD peptide preincubated for 15 mins followed by ATP addition measured after 60 to 100 mins by Kinase-Glo r...				Bioorg Med Chem Lett 26: 2328-32 (2016) Article DOI: 10.1016/j.bmcl.2016.03.037 BindingDB Entry DOI: 10.7270/Q2WD42F0
					More data for this Ligand-Target Pair
Serine/threonine-protein kinase pim-1 (Homo sapiens (Human))	BDBM50005209 (CHEMBL3103867) Show SMILES N[C@H]1CCCN(C1)c1ccncc1NC(=O)c1nc(ccc1N)-c1ccccc1F |r| Show InChI InChI=1S/C22H23FN6O/c23-16-6-2-1-5-15(16)18-8-7-17(25)21(27-18)22(30)28-19-12-26-10-9-20(19)29-11-3-4-14(24)13-29/h1-2,5-10,12,14H,3-4,11,13,24-25H2,(H,28,30)/t14-/m0/s1	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	<1	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Novartis Institutes for Biomedical Research Curated by ChEMBL					Assay Description Inhibition of Pim1 (unknown origin) using BAD peptide preincubated for 15 mins followed by ATP addition measured after 60 to 100 mins by Kinase-Glo r...				Bioorg Med Chem Lett 26: 2328-32 (2016) Article DOI: 10.1016/j.bmcl.2016.03.037 BindingDB Entry DOI: 10.7270/Q2WD42F0
					More data for this Ligand-Target Pair
Serine/threonine-protein kinase pim-1 (Homo sapiens (Human))	BDBM50162815 (CHEMBL3793035) Show SMILES Cc1cc(nc(N)n1)-c1ccncc1NC(=O)c1nc(ccc1N)-c1ccccc1F Show InChI InChI=1S/C22H18FN7O/c1-12-10-18(30-22(25)27-12)14-8-9-26-11-19(14)29-21(31)20-16(24)6-7-17(28-20)13-4-2-3-5-15(13)23/h2-11H,24H2,1H3,(H,29,31)(H2,25,27,30)	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Patents Similars	Article PubMed	<1	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Novartis Institutes for Biomedical Research Curated by ChEMBL					Assay Description Inhibition of Pim1 (unknown origin) using BAD peptide preincubated for 15 mins followed by ATP addition measured after 60 to 100 mins by Kinase-Glo r...				Bioorg Med Chem Lett 26: 2328-32 (2016) Article DOI: 10.1016/j.bmcl.2016.03.037 BindingDB Entry DOI: 10.7270/Q2WD42F0
					More data for this Ligand-Target Pair
Serine/threonine-protein kinase pim-2 (Homo sapiens (Human))	BDBM106896 (US8592455, 96) Show SMILES C[C@H]1CN(C[C@@H](N)[C@@H]1O)c1ccncc1NC(=O)c1ccc(F)c(n1)-c1c(F)cccc1F |r,wU:7.8,wD:1.0,5.5,(-6,2.69,;-4.67,1.93,;-4.67,.38,;-3.33,-.38,;-2,.38,;-2,1.93,;-.67,2.69,;-3.33,2.69,;-3.33,4.23,;-3.33,-1.93,;-4.67,-2.69,;-4.67,-4.23,;-3.33,-5,;-2,-4.23,;-2,-2.69,;-.67,-1.93,;.67,-2.69,;.67,-4.23,;2,-1.93,;3.33,-2.69,;4.67,-1.93,;4.67,-.38,;6,.38,;3.33,.38,;2,-.38,;3.33,1.93,;4.67,2.69,;6,1.93,;4.67,4.23,;3.33,5,;2,4.23,;2,2.69,;.67,1.93,)| Show InChI InChI=1S/C23H22F3N5O2/c1-12-10-31(11-16(27)22(12)32)19-7-8-28-9-18(19)30-23(33)17-6-5-15(26)21(29-17)20-13(24)3-2-4-14(20)25/h2-9,12,16,22,32H,10-11,27H2,1H3,(H,30,33)/t12-,16+,22+/m0/s1	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	Purchase MCE PC cid PC sid PDB UniChem Similars	Article PubMed	<1	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Novartis Institutes for Biomedical Research Curated by ChEMBL					Assay Description Inhibition of Pim2 (unknown origin) using BAD peptide preincubated for 15 mins followed by ATP addition measured after 60 to 100 mins by Kinase-Glo r...				Bioorg Med Chem Lett 26: 2328-32 (2016) Article DOI: 10.1016/j.bmcl.2016.03.037 BindingDB Entry DOI: 10.7270/Q2WD42F0
					More data for this Ligand-Target Pair
Serine/threonine-protein kinase pim-1 (Homo sapiens (Human))	BDBM50161843 (CHEMBL3794146) Show SMILES COc1cc(cc(N)n1)-c1ccncc1NC(=O)c1nc(ccc1N)-c1c(F)cccc1F Show InChI InChI=1S/C23H18F2N6O2/c1-33-20-10-12(9-19(27)31-20)13-7-8-28-11-18(13)30-23(32)22-16(26)5-6-17(29-22)21-14(24)3-2-4-15(21)25/h2-11H,26H2,1H3,(H2,27,31)(H,30,32)	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	<1	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Novartis Institutes for Biomedical Research Curated by ChEMBL					Assay Description Inhibition of Pim1 (unknown origin) using BAD peptide preincubated for 15 mins followed by ATP addition measured after 60 to 100 mins by Kinase-Glo r...				Bioorg Med Chem Lett 26: 2328-32 (2016) Article DOI: 10.1016/j.bmcl.2016.03.037 BindingDB Entry DOI: 10.7270/Q2WD42F0
					More data for this Ligand-Target Pair
Serine/threonine-protein kinase pim-1 (Homo sapiens (Human))	BDBM50161002 (CHEMBL3792742) Show SMILES Cc1cc(cc(N)n1)-c1ccncc1NC(=O)c1nc(ccc1N)-c1ccccc1F Show InChI InChI=1S/C23H19FN6O/c1-13-10-14(11-21(26)28-13)15-8-9-27-12-20(15)30-23(31)22-18(25)6-7-19(29-22)16-4-2-3-5-17(16)24/h2-12H,25H2,1H3,(H2,26,28)(H,30,31)	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid PDB UniChem Similars	Article PubMed	<1	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Novartis Institutes for Biomedical Research Curated by ChEMBL					Assay Description Inhibition of Pim1 (unknown origin) using BAD peptide preincubated for 15 mins followed by ATP addition measured after 60 to 100 mins by Kinase-Glo r...				Bioorg Med Chem Lett 26: 2328-32 (2016) Article DOI: 10.1016/j.bmcl.2016.03.037 BindingDB Entry DOI: 10.7270/Q2WD42F0
					More data for this Ligand-Target Pair
Serine/threonine-protein kinase pim-1 (Homo sapiens (Human))	BDBM50156374 (CHEMBL3792428) Show SMILES Nc1cc(ccn1)-c1ccncc1NC(=O)c1nc(ccc1N)-c1ccccc1F Show InChI InChI=1S/C22H17FN6O/c23-16-4-2-1-3-15(16)18-6-5-17(24)21(28-18)22(30)29-19-12-26-9-8-14(19)13-7-10-27-20(25)11-13/h1-12H,24H2,(H2,25,27)(H,29,30)	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Patents Similars	Article PubMed	<1	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Novartis Institutes for Biomedical Research Curated by ChEMBL					Assay Description Inhibition of Pim1 (unknown origin) using BAD peptide preincubated for 15 mins followed by ATP addition measured after 60 to 100 mins by Kinase-Glo r...				Bioorg Med Chem Lett 26: 2328-32 (2016) Article DOI: 10.1016/j.bmcl.2016.03.037 BindingDB Entry DOI: 10.7270/Q2WD42F0
					More data for this Ligand-Target Pair
Serine/threonine-protein kinase pim-1 (Homo sapiens (Human))	BDBM50156380 (CHEMBL3793927) Show SMILES Nc1cc(ccn1)-c1ccncc1NC(=O)c1nc(ccc1N)-c1c(F)cccc1F Show InChI InChI=1S/C22H16F2N6O/c23-14-2-1-3-15(24)20(14)17-5-4-16(25)21(29-17)22(31)30-18-11-27-8-7-13(18)12-6-9-28-19(26)10-12/h1-11H,25H2,(H2,26,28)(H,30,31)	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Patents Similars	Article PubMed	2	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Novartis Institutes for Biomedical Research Curated by ChEMBL					Assay Description Inhibition of Pim1 (unknown origin) using BAD peptide preincubated for 15 mins followed by ATP addition measured after 60 to 100 mins by Kinase-Glo r...				Bioorg Med Chem Lett 26: 2328-32 (2016) Article DOI: 10.1016/j.bmcl.2016.03.037 BindingDB Entry DOI: 10.7270/Q2WD42F0
					More data for this Ligand-Target Pair
Serine/threonine-protein kinase pim-3 (Homo sapiens (Human))	BDBM50161843 (CHEMBL3794146) Show SMILES COc1cc(cc(N)n1)-c1ccncc1NC(=O)c1nc(ccc1N)-c1c(F)cccc1F Show InChI InChI=1S/C23H18F2N6O2/c1-33-20-10-12(9-19(27)31-20)13-7-8-28-11-18(13)30-23(32)22-16(26)5-6-17(29-22)21-14(24)3-2-4-15(21)25/h2-11H,26H2,1H3,(H2,27,31)(H,30,32)	KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	<3	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Novartis Institutes for Biomedical Research Curated by ChEMBL					Assay Description Inhibition of Pim3 (unknown origin) using BAD peptide preincubated for 15 mins followed by ATP addition measured after 60 to 100 mins by Kinase-Glo r...				Bioorg Med Chem Lett 26: 2328-32 (2016) Article DOI: 10.1016/j.bmcl.2016.03.037 BindingDB Entry DOI: 10.7270/Q2WD42F0
					More data for this Ligand-Target Pair
Serine/threonine-protein kinase pim-2 (Homo sapiens (Human))	BDBM50162818 (CHEMBL3793067) Show SMILES Cc1cc(cc(N)n1)-c1ccncc1NC(=O)c1nc(ccc1N)-c1c(F)cccc1F Show InChI InChI=1S/C23H18F2N6O/c1-12-9-13(10-20(27)29-12)14-7-8-28-11-19(14)31-23(32)22-17(26)5-6-18(30-22)21-15(24)3-2-4-16(21)25/h2-11H,26H2,1H3,(H2,27,29)(H,31,32)	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Patents Similars	Article PubMed	<3	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Novartis Institutes for Biomedical Research Curated by ChEMBL					Assay Description Inhibition of Pim2 (unknown origin) using BAD peptide preincubated for 15 mins followed by ATP addition measured after 60 to 100 mins by Kinase-Glo r...				Bioorg Med Chem Lett 26: 2328-32 (2016) Article DOI: 10.1016/j.bmcl.2016.03.037 BindingDB Entry DOI: 10.7270/Q2WD42F0
					More data for this Ligand-Target Pair
Serine/threonine-protein kinase pim-2 (Homo sapiens (Human))	BDBM50161838 (CHEMBL3792922) Show SMILES Cc1cc(nc(N)n1)-c1ccncc1NC(=O)c1nc(ccc1N)-c1nccs1 Show InChI InChI=1S/C19H16N8OS/c1-10-8-14(27-19(21)24-10)11-4-5-22-9-15(11)26-17(28)16-12(20)2-3-13(25-16)18-23-6-7-29-18/h2-9H,20H2,1H3,(H,26,28)(H2,21,24,27)	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	<3	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Novartis Institutes for Biomedical Research Curated by ChEMBL					Assay Description Inhibition of Pim2 (unknown origin) using BAD peptide preincubated for 15 mins followed by ATP addition measured after 60 to 100 mins by Kinase-Glo r...				Bioorg Med Chem Lett 26: 2328-32 (2016) Article DOI: 10.1016/j.bmcl.2016.03.037 BindingDB Entry DOI: 10.7270/Q2WD42F0
					More data for this Ligand-Target Pair
Serine/threonine-protein kinase pim-2 (Homo sapiens (Human))	BDBM50162815 (CHEMBL3793035) Show SMILES Cc1cc(nc(N)n1)-c1ccncc1NC(=O)c1nc(ccc1N)-c1ccccc1F Show InChI InChI=1S/C22H18FN7O/c1-12-10-18(30-22(25)27-12)14-8-9-26-11-19(14)29-21(31)20-16(24)6-7-17(28-20)13-4-2-3-5-15(13)23/h2-11H,24H2,1H3,(H,29,31)(H2,25,27,30)	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Patents Similars	Article PubMed	<3	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Novartis Institutes for Biomedical Research Curated by ChEMBL					Assay Description Inhibition of Pim2 (unknown origin) using BAD peptide preincubated for 15 mins followed by ATP addition measured after 60 to 100 mins by Kinase-Glo r...				Bioorg Med Chem Lett 26: 2328-32 (2016) Article DOI: 10.1016/j.bmcl.2016.03.037 BindingDB Entry DOI: 10.7270/Q2WD42F0
					More data for this Ligand-Target Pair
Serine/threonine-protein kinase pim-2 (Homo sapiens (Human))	BDBM50161839 (CHEMBL3792736) Show SMILES Nc1cc(nc(n1)C(F)(F)F)-c1ccncc1NC(=O)c1nc(ccc1N)-c1nccs1 Show InChI InChI=1S/C19H13F3N8OS/c20-19(21,22)18-29-12(7-14(24)30-18)9-3-4-25-8-13(9)28-16(31)15-10(23)1-2-11(27-15)17-26-5-6-32-17/h1-8H,23H2,(H,28,31)(H2,24,29,30)	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	<3	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Novartis Institutes for Biomedical Research Curated by ChEMBL					Assay Description Inhibition of Pim2 (unknown origin) using BAD peptide preincubated for 15 mins followed by ATP addition measured after 60 to 100 mins by Kinase-Glo r...				Bioorg Med Chem Lett 26: 2328-32 (2016) Article DOI: 10.1016/j.bmcl.2016.03.037 BindingDB Entry DOI: 10.7270/Q2WD42F0
					More data for this Ligand-Target Pair
Serine/threonine-protein kinase pim-2 (Homo sapiens (Human))	BDBM50005209 (CHEMBL3103867) Show SMILES N[C@H]1CCCN(C1)c1ccncc1NC(=O)c1nc(ccc1N)-c1ccccc1F |r| Show InChI InChI=1S/C22H23FN6O/c23-16-6-2-1-5-15(16)18-8-7-17(25)21(27-18)22(30)28-19-12-26-10-9-20(19)29-11-3-4-14(24)13-29/h1-2,5-10,12,14H,3-4,11,13,24-25H2,(H,28,30)/t14-/m0/s1	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	<3	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Novartis Institutes for Biomedical Research Curated by ChEMBL					Assay Description Inhibition of Pim2 (unknown origin) using BAD peptide preincubated for 15 mins followed by ATP addition measured after 60 to 100 mins by Kinase-Glo r...				Bioorg Med Chem Lett 26: 2328-32 (2016) Article DOI: 10.1016/j.bmcl.2016.03.037 BindingDB Entry DOI: 10.7270/Q2WD42F0
					More data for this Ligand-Target Pair
Serine/threonine-protein kinase pim-3 (Homo sapiens (Human))	BDBM50156374 (CHEMBL3792428) Show SMILES Nc1cc(ccn1)-c1ccncc1NC(=O)c1nc(ccc1N)-c1ccccc1F Show InChI InChI=1S/C22H17FN6O/c23-16-4-2-1-3-15(16)18-6-5-17(24)21(28-18)22(30)29-19-12-26-9-8-14(19)13-7-10-27-20(25)11-13/h1-12H,24H2,(H2,25,27)(H,29,30)	KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Patents Similars	Article PubMed	3	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Novartis Institutes for Biomedical Research Curated by ChEMBL					Assay Description Inhibition of Pim3 (unknown origin) using BAD peptide preincubated for 15 mins followed by ATP addition measured after 60 to 100 mins by Kinase-Glo r...				Bioorg Med Chem Lett 26: 2328-32 (2016) Article DOI: 10.1016/j.bmcl.2016.03.037 BindingDB Entry DOI: 10.7270/Q2WD42F0
					More data for this Ligand-Target Pair
Serine/threonine-protein kinase pim-2 (Homo sapiens (Human))	BDBM50161840 (CHEMBL3792425) Show SMILES Nc1cc(nc(n1)C(F)(F)F)-c1ccncc1NC(=O)c1nc(ccc1N)-c1c(F)cccc1F Show InChI InChI=1S/C22H14F5N7O/c23-11-2-1-3-12(24)18(11)14-5-4-13(28)19(31-14)20(35)32-16-9-30-7-6-10(16)15-8-17(29)34-21(33-15)22(25,26)27/h1-9H,28H2,(H,32,35)(H2,29,33,34)	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem	Article PubMed	<3	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Novartis Institutes for Biomedical Research Curated by ChEMBL					Assay Description Inhibition of Pim2 (unknown origin) using BAD peptide preincubated for 15 mins followed by ATP addition measured after 60 to 100 mins by Kinase-Glo r...				Bioorg Med Chem Lett 26: 2328-32 (2016) Article DOI: 10.1016/j.bmcl.2016.03.037 BindingDB Entry DOI: 10.7270/Q2WD42F0
					More data for this Ligand-Target Pair
Serine/threonine-protein kinase pim-3 (Homo sapiens (Human))	BDBM50005209 (CHEMBL3103867) Show SMILES N[C@H]1CCCN(C1)c1ccncc1NC(=O)c1nc(ccc1N)-c1ccccc1F |r| Show InChI InChI=1S/C22H23FN6O/c23-16-6-2-1-5-15(16)18-8-7-17(25)21(27-18)22(30)28-19-12-26-10-9-20(19)29-11-3-4-14(24)13-29/h1-2,5-10,12,14H,3-4,11,13,24-25H2,(H,28,30)/t14-/m0/s1	KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	<3	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Novartis Institutes for Biomedical Research Curated by ChEMBL					Assay Description Inhibition of Pim3 (unknown origin) using BAD peptide preincubated for 15 mins followed by ATP addition measured after 60 to 100 mins by Kinase-Glo r...				Bioorg Med Chem Lett 26: 2328-32 (2016) Article DOI: 10.1016/j.bmcl.2016.03.037 BindingDB Entry DOI: 10.7270/Q2WD42F0
					More data for this Ligand-Target Pair
Serine/threonine-protein kinase pim-1 (Homo sapiens (Human))	BDBM50156379 (CHEMBL3792474) Show SMILES Nc1cncc(n1)-c1ccncc1NC(=O)c1nc(ccc1N)-c1ccccc1F Show InChI InChI=1S/C21H16FN7O/c22-14-4-2-1-3-12(14)16-6-5-15(23)20(28-16)21(30)29-18-9-25-8-7-13(18)17-10-26-11-19(24)27-17/h1-11H,23H2,(H2,24,27)(H,29,30)	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Patents Similars	Article PubMed	3	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Novartis Institutes for Biomedical Research Curated by ChEMBL					Assay Description Inhibition of Pim1 (unknown origin) using BAD peptide preincubated for 15 mins followed by ATP addition measured after 60 to 100 mins by Kinase-Glo r...				Bioorg Med Chem Lett 26: 2328-32 (2016) Article DOI: 10.1016/j.bmcl.2016.03.037 BindingDB Entry DOI: 10.7270/Q2WD42F0
					More data for this Ligand-Target Pair
Serine/threonine-protein kinase pim-3 (Homo sapiens (Human))	BDBM50156380 (CHEMBL3793927) Show SMILES Nc1cc(ccn1)-c1ccncc1NC(=O)c1nc(ccc1N)-c1c(F)cccc1F Show InChI InChI=1S/C22H16F2N6O/c23-14-2-1-3-15(24)20(14)17-5-4-16(25)21(29-17)22(31)30-18-11-27-8-7-13(18)12-6-9-28-19(26)10-12/h1-11H,25H2,(H2,26,28)(H,30,31)	KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Patents Similars	Article PubMed	<3	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Novartis Institutes for Biomedical Research Curated by ChEMBL					Assay Description Inhibition of Pim3 (unknown origin) using BAD peptide preincubated for 15 mins followed by ATP addition measured after 60 to 100 mins by Kinase-Glo r...				Bioorg Med Chem Lett 26: 2328-32 (2016) Article DOI: 10.1016/j.bmcl.2016.03.037 BindingDB Entry DOI: 10.7270/Q2WD42F0
					More data for this Ligand-Target Pair
Serine/threonine-protein kinase pim-3 (Homo sapiens (Human))	BDBM50160995 (CHEMBL3793938) Show SMILES Cc1nc(N)cc(n1)-c1ccncc1NC(=O)c1nc(ccc1N)-c1c(F)cccc1F Show InChI InChI=1S/C22H17F2N7O/c1-11-28-17(9-19(26)29-11)12-7-8-27-10-18(12)31-22(32)21-15(25)5-6-16(30-21)20-13(23)3-2-4-14(20)24/h2-10H,25H2,1H3,(H,31,32)(H2,26,28,29)	KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	<3	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Novartis Institutes for Biomedical Research Curated by ChEMBL					Assay Description Inhibition of Pim3 (unknown origin) using BAD peptide preincubated for 15 mins followed by ATP addition measured after 60 to 100 mins by Kinase-Glo r...				Bioorg Med Chem Lett 26: 2328-32 (2016) Article DOI: 10.1016/j.bmcl.2016.03.037 BindingDB Entry DOI: 10.7270/Q2WD42F0
					More data for this Ligand-Target Pair
Serine/threonine-protein kinase pim-3 (Homo sapiens (Human))	BDBM50162815 (CHEMBL3793035) Show SMILES Cc1cc(nc(N)n1)-c1ccncc1NC(=O)c1nc(ccc1N)-c1ccccc1F Show InChI InChI=1S/C22H18FN7O/c1-12-10-18(30-22(25)27-12)14-8-9-26-11-19(14)29-21(31)20-16(24)6-7-17(28-20)13-4-2-3-5-15(13)23/h2-11H,24H2,1H3,(H,29,31)(H2,25,27,30)	KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Patents Similars	Article PubMed	<3	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Novartis Institutes for Biomedical Research Curated by ChEMBL					Assay Description Inhibition of Pim3 (unknown origin) using BAD peptide preincubated for 15 mins followed by ATP addition measured after 60 to 100 mins by Kinase-Glo r...				Bioorg Med Chem Lett 26: 2328-32 (2016) Article DOI: 10.1016/j.bmcl.2016.03.037 BindingDB Entry DOI: 10.7270/Q2WD42F0
					More data for this Ligand-Target Pair
Serine/threonine-protein kinase pim-3 (Homo sapiens (Human))	BDBM50162818 (CHEMBL3793067) Show SMILES Cc1cc(cc(N)n1)-c1ccncc1NC(=O)c1nc(ccc1N)-c1c(F)cccc1F Show InChI InChI=1S/C23H18F2N6O/c1-12-9-13(10-20(27)29-12)14-7-8-28-11-19(14)31-23(32)22-17(26)5-6-18(30-22)21-15(24)3-2-4-16(21)25/h2-11H,26H2,1H3,(H2,27,29)(H,31,32)	KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Patents Similars	Article PubMed	<3	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Novartis Institutes for Biomedical Research Curated by ChEMBL					Assay Description Inhibition of Pim3 (unknown origin) using BAD peptide preincubated for 15 mins followed by ATP addition measured after 60 to 100 mins by Kinase-Glo r...				Bioorg Med Chem Lett 26: 2328-32 (2016) Article DOI: 10.1016/j.bmcl.2016.03.037 BindingDB Entry DOI: 10.7270/Q2WD42F0
					More data for this Ligand-Target Pair
Serine/threonine-protein kinase pim-3 (Homo sapiens (Human))	BDBM50161002 (CHEMBL3792742) Show SMILES Cc1cc(cc(N)n1)-c1ccncc1NC(=O)c1nc(ccc1N)-c1ccccc1F Show InChI InChI=1S/C23H19FN6O/c1-13-10-14(11-21(26)28-13)15-8-9-27-12-20(15)30-23(31)22-18(25)6-7-19(29-22)16-4-2-3-5-17(16)24/h2-12H,25H2,1H3,(H2,26,28)(H,30,31)	KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid PDB UniChem Similars	Article PubMed	<3	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Novartis Institutes for Biomedical Research Curated by ChEMBL					Assay Description Inhibition of Pim3 (unknown origin) using BAD peptide preincubated for 15 mins followed by ATP addition measured after 60 to 100 mins by Kinase-Glo r...				Bioorg Med Chem Lett 26: 2328-32 (2016) Article DOI: 10.1016/j.bmcl.2016.03.037 BindingDB Entry DOI: 10.7270/Q2WD42F0
					More data for this Ligand-Target Pair
Serine/threonine-protein kinase pim-2 (Homo sapiens (Human))	BDBM50160995 (CHEMBL3793938) Show SMILES Cc1nc(N)cc(n1)-c1ccncc1NC(=O)c1nc(ccc1N)-c1c(F)cccc1F Show InChI InChI=1S/C22H17F2N7O/c1-11-28-17(9-19(26)29-11)12-7-8-27-10-18(12)31-22(32)21-15(25)5-6-16(30-21)20-13(23)3-2-4-14(20)24/h2-10H,25H2,1H3,(H,31,32)(H2,26,28,29)	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	<3	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Novartis Institutes for Biomedical Research Curated by ChEMBL					Assay Description Inhibition of Pim2 (unknown origin) using BAD peptide preincubated for 15 mins followed by ATP addition measured after 60 to 100 mins by Kinase-Glo r...				Bioorg Med Chem Lett 26: 2328-32 (2016) Article DOI: 10.1016/j.bmcl.2016.03.037 BindingDB Entry DOI: 10.7270/Q2WD42F0
					More data for this Ligand-Target Pair
Serine/threonine-protein kinase pim-3 (Homo sapiens (Human))	BDBM50161840 (CHEMBL3792425) Show SMILES Nc1cc(nc(n1)C(F)(F)F)-c1ccncc1NC(=O)c1nc(ccc1N)-c1c(F)cccc1F Show InChI InChI=1S/C22H14F5N7O/c23-11-2-1-3-12(24)18(11)14-5-4-13(28)19(31-14)20(35)32-16-9-30-7-6-10(16)15-8-17(29)34-21(33-15)22(25,26)27/h1-9H,28H2,(H,32,35)(H2,29,33,34)	KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem	Article PubMed	<3	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Novartis Institutes for Biomedical Research Curated by ChEMBL					Assay Description Inhibition of Pim3 (unknown origin) using BAD peptide preincubated for 15 mins followed by ATP addition measured after 60 to 100 mins by Kinase-Glo r...				Bioorg Med Chem Lett 26: 2328-32 (2016) Article DOI: 10.1016/j.bmcl.2016.03.037 BindingDB Entry DOI: 10.7270/Q2WD42F0
					More data for this Ligand-Target Pair
Serine/threonine-protein kinase pim-3 (Homo sapiens (Human))	BDBM50161839 (CHEMBL3792736) Show SMILES Nc1cc(nc(n1)C(F)(F)F)-c1ccncc1NC(=O)c1nc(ccc1N)-c1nccs1 Show InChI InChI=1S/C19H13F3N8OS/c20-19(21,22)18-29-12(7-14(24)30-18)9-3-4-25-8-13(9)28-16(31)15-10(23)1-2-11(27-15)17-26-5-6-32-17/h1-8H,23H2,(H,28,31)(H2,24,29,30)	KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	<3	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Novartis Institutes for Biomedical Research Curated by ChEMBL					Assay Description Inhibition of Pim3 (unknown origin) using BAD peptide preincubated for 15 mins followed by ATP addition measured after 60 to 100 mins by Kinase-Glo r...				Bioorg Med Chem Lett 26: 2328-32 (2016) Article DOI: 10.1016/j.bmcl.2016.03.037 BindingDB Entry DOI: 10.7270/Q2WD42F0
					More data for this Ligand-Target Pair
Serine/threonine-protein kinase pim-3 (Homo sapiens (Human))	BDBM50161838 (CHEMBL3792922) Show SMILES Cc1cc(nc(N)n1)-c1ccncc1NC(=O)c1nc(ccc1N)-c1nccs1 Show InChI InChI=1S/C19H16N8OS/c1-10-8-14(27-19(21)24-10)11-4-5-22-9-15(11)26-17(28)16-12(20)2-3-13(25-16)18-23-6-7-29-18/h2-9H,20H2,1H3,(H,26,28)(H2,21,24,27)	KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	<3	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Novartis Institutes for Biomedical Research Curated by ChEMBL					Assay Description Inhibition of Pim3 (unknown origin) using BAD peptide preincubated for 15 mins followed by ATP addition measured after 60 to 100 mins by Kinase-Glo r...				Bioorg Med Chem Lett 26: 2328-32 (2016) Article DOI: 10.1016/j.bmcl.2016.03.037 BindingDB Entry DOI: 10.7270/Q2WD42F0
					More data for this Ligand-Target Pair
Serine/threonine-protein kinase pim-1 (Homo sapiens (Human))	BDBM50160997 (CHEMBL3793221) Show SMILES Nc1cc(ncn1)-c1ccncc1NC(=O)c1nc(ccc1N)-c1c(F)cccc1F Show InChI InChI=1S/C21H15F2N7O/c22-12-2-1-3-13(23)19(12)15-5-4-14(24)20(29-15)21(31)30-17-9-26-7-6-11(17)16-8-18(25)28-10-27-16/h1-10H,24H2,(H,30,31)(H2,25,27,28)	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	4	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Novartis Institutes for Biomedical Research Curated by ChEMBL					Assay Description Inhibition of Pim1 (unknown origin) using BAD peptide preincubated for 15 mins followed by ATP addition measured after 60 to 100 mins by Kinase-Glo r...				Bioorg Med Chem Lett 26: 2328-32 (2016) Article DOI: 10.1016/j.bmcl.2016.03.037 BindingDB Entry DOI: 10.7270/Q2WD42F0
					More data for this Ligand-Target Pair
Serine/threonine-protein kinase pim-1 (Homo sapiens (Human))	BDBM50156376 (CHEMBL3793600) Show SMILES Nc1ccc(cn1)-c1ccncc1NC(=O)c1nc(ccc1N)-c1ccccc1F Show InChI InChI=1S/C22H17FN6O/c23-16-4-2-1-3-15(16)18-7-6-17(24)21(28-18)22(30)29-19-12-26-10-9-14(19)13-5-8-20(25)27-11-13/h1-12H,24H2,(H2,25,27)(H,29,30)	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Patents Similars	Article PubMed	4	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Novartis Institutes for Biomedical Research Curated by ChEMBL					Assay Description Inhibition of Pim1 (unknown origin) using BAD peptide preincubated for 15 mins followed by ATP addition measured after 60 to 100 mins by Kinase-Glo r...				Bioorg Med Chem Lett 26: 2328-32 (2016) Article DOI: 10.1016/j.bmcl.2016.03.037 BindingDB Entry DOI: 10.7270/Q2WD42F0
					More data for this Ligand-Target Pair
Serine/threonine-protein kinase pim-2 (Homo sapiens (Human))	BDBM50161002 (CHEMBL3792742) Show SMILES Cc1cc(cc(N)n1)-c1ccncc1NC(=O)c1nc(ccc1N)-c1ccccc1F Show InChI InChI=1S/C23H19FN6O/c1-13-10-14(11-21(26)28-13)15-8-9-27-12-20(15)30-23(31)22-18(25)6-7-19(29-22)16-4-2-3-5-17(16)24/h2-12H,25H2,1H3,(H2,26,28)(H,30,31)	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid PDB UniChem Similars	Article PubMed	4	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Novartis Institutes for Biomedical Research Curated by ChEMBL					Assay Description Inhibition of Pim2 (unknown origin) using BAD peptide preincubated for 15 mins followed by ATP addition measured after 60 to 100 mins by Kinase-Glo r...				Bioorg Med Chem Lett 26: 2328-32 (2016) Article DOI: 10.1016/j.bmcl.2016.03.037 BindingDB Entry DOI: 10.7270/Q2WD42F0
					More data for this Ligand-Target Pair
Serine/threonine-protein kinase pim-2 (Homo sapiens (Human))	BDBM50161843 (CHEMBL3794146) Show SMILES COc1cc(cc(N)n1)-c1ccncc1NC(=O)c1nc(ccc1N)-c1c(F)cccc1F Show InChI InChI=1S/C23H18F2N6O2/c1-33-20-10-12(9-19(27)31-20)13-7-8-28-11-18(13)30-23(32)22-16(26)5-6-17(29-22)21-14(24)3-2-4-15(21)25/h2-11H,26H2,1H3,(H2,27,31)(H,30,32)	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	4	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Novartis Institutes for Biomedical Research Curated by ChEMBL					Assay Description Inhibition of Pim2 (unknown origin) using BAD peptide preincubated for 15 mins followed by ATP addition measured after 60 to 100 mins by Kinase-Glo r...				Bioorg Med Chem Lett 26: 2328-32 (2016) Article DOI: 10.1016/j.bmcl.2016.03.037 BindingDB Entry DOI: 10.7270/Q2WD42F0
					More data for this Ligand-Target Pair
Serine/threonine-protein kinase pim-3 (Homo sapiens (Human))	BDBM50160997 (CHEMBL3793221) Show SMILES Nc1cc(ncn1)-c1ccncc1NC(=O)c1nc(ccc1N)-c1c(F)cccc1F Show InChI InChI=1S/C21H15F2N7O/c22-12-2-1-3-13(23)19(12)15-5-4-14(24)20(29-15)21(31)30-17-9-26-7-6-11(17)16-8-18(25)28-10-27-16/h1-10H,24H2,(H,30,31)(H2,25,27,28)	KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	5	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Novartis Institutes for Biomedical Research Curated by ChEMBL					Assay Description Inhibition of Pim3 (unknown origin) using BAD peptide preincubated for 15 mins followed by ATP addition measured after 60 to 100 mins by Kinase-Glo r...				Bioorg Med Chem Lett 26: 2328-32 (2016) Article DOI: 10.1016/j.bmcl.2016.03.037 BindingDB Entry DOI: 10.7270/Q2WD42F0
					More data for this Ligand-Target Pair
Serine/threonine-protein kinase pim-3 (Homo sapiens (Human))	BDBM50160996 (CHEMBL3793267) Show SMILES Nc1nccc(n1)-c1ccncc1NC(=O)c1nc(ccc1N)-c1c(F)cccc1F Show InChI InChI=1S/C21H15F2N7O/c22-12-2-1-3-13(23)18(12)16-5-4-14(24)19(28-16)20(31)29-17-10-26-8-6-11(17)15-7-9-27-21(25)30-15/h1-10H,24H2,(H,29,31)(H2,25,27,30)	KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	5	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Novartis Institutes for Biomedical Research Curated by ChEMBL					Assay Description Inhibition of Pim3 (unknown origin) using BAD peptide preincubated for 15 mins followed by ATP addition measured after 60 to 100 mins by Kinase-Glo r...				Bioorg Med Chem Lett 26: 2328-32 (2016) Article DOI: 10.1016/j.bmcl.2016.03.037 BindingDB Entry DOI: 10.7270/Q2WD42F0
					More data for this Ligand-Target Pair
Serine/threonine-protein kinase pim-1 (Homo sapiens (Human))	BDBM50160996 (CHEMBL3793267) Show SMILES Nc1nccc(n1)-c1ccncc1NC(=O)c1nc(ccc1N)-c1c(F)cccc1F Show InChI InChI=1S/C21H15F2N7O/c22-12-2-1-3-13(23)18(12)16-5-4-14(24)19(28-16)20(31)29-17-10-26-8-6-11(17)15-7-9-27-21(25)30-15/h1-10H,24H2,(H,29,31)(H2,25,27,30)	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	6	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Novartis Institutes for Biomedical Research Curated by ChEMBL					Assay Description Inhibition of Pim1 (unknown origin) using BAD peptide preincubated for 15 mins followed by ATP addition measured after 60 to 100 mins by Kinase-Glo r...				Bioorg Med Chem Lett 26: 2328-32 (2016) Article DOI: 10.1016/j.bmcl.2016.03.037 BindingDB Entry DOI: 10.7270/Q2WD42F0
					More data for this Ligand-Target Pair
Serine/threonine-protein kinase pim-3 (Homo sapiens (Human))	BDBM50156379 (CHEMBL3792474) Show SMILES Nc1cncc(n1)-c1ccncc1NC(=O)c1nc(ccc1N)-c1ccccc1F Show InChI InChI=1S/C21H16FN7O/c22-14-4-2-1-3-12(14)16-6-5-15(23)20(28-16)21(30)29-18-9-25-8-7-13(18)17-10-26-11-19(24)27-17/h1-11H,23H2,(H2,24,27)(H,29,30)	KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Patents Similars	Article PubMed	6	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Novartis Institutes for Biomedical Research Curated by ChEMBL					Assay Description Inhibition of Pim3 (unknown origin) using BAD peptide preincubated for 15 mins followed by ATP addition measured after 60 to 100 mins by Kinase-Glo r...				Bioorg Med Chem Lett 26: 2328-32 (2016) Article DOI: 10.1016/j.bmcl.2016.03.037 BindingDB Entry DOI: 10.7270/Q2WD42F0
					More data for this Ligand-Target Pair
Serine/threonine-protein kinase pim-2 (Homo sapiens (Human))	BDBM50156380 (CHEMBL3793927) Show SMILES Nc1cc(ccn1)-c1ccncc1NC(=O)c1nc(ccc1N)-c1c(F)cccc1F Show InChI InChI=1S/C22H16F2N6O/c23-14-2-1-3-15(24)20(14)17-5-4-16(25)21(29-17)22(31)30-18-11-27-8-7-13(18)12-6-9-28-19(26)10-12/h1-11H,25H2,(H2,26,28)(H,30,31)	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Patents Similars	Article PubMed	8	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Novartis Institutes for Biomedical Research Curated by ChEMBL					Assay Description Inhibition of Pim2 (unknown origin) using BAD peptide preincubated for 15 mins followed by ATP addition measured after 60 to 100 mins by Kinase-Glo r...				Bioorg Med Chem Lett 26: 2328-32 (2016) Article DOI: 10.1016/j.bmcl.2016.03.037 BindingDB Entry DOI: 10.7270/Q2WD42F0
					More data for this Ligand-Target Pair
Serine/threonine-protein kinase pim-1 (Homo sapiens (Human))	BDBM50156373 (CHEMBL3793440) Show SMILES Nc1ccc(nc1C(=O)Nc1cnccc1-c1ccncc1)-c1ccccc1F Show InChI InChI=1S/C22H16FN5O/c23-17-4-2-1-3-16(17)19-6-5-18(24)21(27-19)22(29)28-20-13-26-12-9-15(20)14-7-10-25-11-8-14/h1-13H,24H2,(H,28,29)	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Patents Similars	Article PubMed	8	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Novartis Institutes for Biomedical Research Curated by ChEMBL					Assay Description Inhibition of Pim1 (unknown origin) using BAD peptide preincubated for 15 mins followed by ATP addition measured after 60 to 100 mins by Kinase-Glo r...				Bioorg Med Chem Lett 26: 2328-32 (2016) Article DOI: 10.1016/j.bmcl.2016.03.037 BindingDB Entry DOI: 10.7270/Q2WD42F0
					More data for this Ligand-Target Pair
Serine/threonine-protein kinase pim-3 (Homo sapiens (Human))	BDBM50156376 (CHEMBL3793600) Show SMILES Nc1ccc(cn1)-c1ccncc1NC(=O)c1nc(ccc1N)-c1ccccc1F Show InChI InChI=1S/C22H17FN6O/c23-16-4-2-1-3-15(16)18-7-6-17(24)21(28-18)22(30)29-19-12-26-10-9-14(19)13-5-8-20(25)27-11-13/h1-12H,24H2,(H2,25,27)(H,29,30)	KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Patents Similars	Article PubMed	12	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Novartis Institutes for Biomedical Research Curated by ChEMBL					Assay Description Inhibition of Pim3 (unknown origin) using BAD peptide preincubated for 15 mins followed by ATP addition measured after 60 to 100 mins by Kinase-Glo r...				Bioorg Med Chem Lett 26: 2328-32 (2016) Article DOI: 10.1016/j.bmcl.2016.03.037 BindingDB Entry DOI: 10.7270/Q2WD42F0
					More data for this Ligand-Target Pair
Serine/threonine-protein kinase pim-3 (Homo sapiens (Human))	BDBM50161842 (CHEMBL3792905) Show SMILES Nc1cc(nc(N)n1)-c1ccncc1NC(=O)c1nc(ccc1N)-c1ccccc1F Show InChI InChI=1S/C21H17FN8O/c22-13-4-2-1-3-11(13)15-6-5-14(23)19(27-15)20(31)28-17-10-26-8-7-12(17)16-9-18(24)30-21(25)29-16/h1-10H,23H2,(H,28,31)(H4,24,25,29,30)	KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem	Article PubMed	15	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Novartis Institutes for Biomedical Research Curated by ChEMBL					Assay Description Inhibition of Pim3 (unknown origin) using BAD peptide preincubated for 15 mins followed by ATP addition measured after 60 to 100 mins by Kinase-Glo r...				Bioorg Med Chem Lett 26: 2328-32 (2016) Article DOI: 10.1016/j.bmcl.2016.03.037 BindingDB Entry DOI: 10.7270/Q2WD42F0
					More data for this Ligand-Target Pair
Serine/threonine-protein kinase pim-1 (Homo sapiens (Human))	BDBM50161842 (CHEMBL3792905) Show SMILES Nc1cc(nc(N)n1)-c1ccncc1NC(=O)c1nc(ccc1N)-c1ccccc1F Show InChI InChI=1S/C21H17FN8O/c22-13-4-2-1-3-11(13)15-6-5-14(23)19(27-15)20(31)28-17-10-26-8-7-12(17)16-9-18(24)30-21(25)29-16/h1-10H,23H2,(H,28,31)(H4,24,25,29,30)	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem	Article PubMed	17	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Novartis Institutes for Biomedical Research Curated by ChEMBL					Assay Description Inhibition of Pim1 (unknown origin) using BAD peptide preincubated for 15 mins followed by ATP addition measured after 60 to 100 mins by Kinase-Glo r...				Bioorg Med Chem Lett 26: 2328-32 (2016) Article DOI: 10.1016/j.bmcl.2016.03.037 BindingDB Entry DOI: 10.7270/Q2WD42F0
					More data for this Ligand-Target Pair
Serine/threonine-protein kinase pim-3 (Homo sapiens (Human))	BDBM50156373 (CHEMBL3793440) Show SMILES Nc1ccc(nc1C(=O)Nc1cnccc1-c1ccncc1)-c1ccccc1F Show InChI InChI=1S/C22H16FN5O/c23-17-4-2-1-3-16(17)19-6-5-18(24)21(27-19)22(29)28-20-13-26-12-9-15(20)14-7-10-25-11-8-14/h1-13H,24H2,(H,28,29)	KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Patents Similars	Article PubMed	21	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Novartis Institutes for Biomedical Research Curated by ChEMBL					Assay Description Inhibition of Pim3 (unknown origin) using BAD peptide preincubated for 15 mins followed by ATP addition measured after 60 to 100 mins by Kinase-Glo r...				Bioorg Med Chem Lett 26: 2328-32 (2016) Article DOI: 10.1016/j.bmcl.2016.03.037 BindingDB Entry DOI: 10.7270/Q2WD42F0
					More data for this Ligand-Target Pair
Serine/threonine-protein kinase pim-2 (Homo sapiens (Human))	BDBM50160997 (CHEMBL3793221) Show SMILES Nc1cc(ncn1)-c1ccncc1NC(=O)c1nc(ccc1N)-c1c(F)cccc1F Show InChI InChI=1S/C21H15F2N7O/c22-12-2-1-3-13(23)19(12)15-5-4-14(24)20(29-15)21(31)30-17-9-26-7-6-11(17)16-8-18(25)28-10-27-16/h1-10H,24H2,(H,30,31)(H2,25,27,28)	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	27	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Novartis Institutes for Biomedical Research Curated by ChEMBL					Assay Description Inhibition of Pim2 (unknown origin) using BAD peptide preincubated for 15 mins followed by ATP addition measured after 60 to 100 mins by Kinase-Glo r...				Bioorg Med Chem Lett 26: 2328-32 (2016) Article DOI: 10.1016/j.bmcl.2016.03.037 BindingDB Entry DOI: 10.7270/Q2WD42F0
					More data for this Ligand-Target Pair
Serine/threonine-protein kinase pim-1 (Homo sapiens (Human))	BDBM50156378 (CHEMBL3792552) Show SMILES Nc1ccc(nc1C(=O)Nc1cnccc1-c1cccnc1N)-c1c(F)cccc1F Show InChI InChI=1S/C22H16F2N6O/c23-14-4-1-5-15(24)19(14)17-7-6-16(25)20(29-17)22(31)30-18-11-27-10-8-12(18)13-3-2-9-28-21(13)26/h1-11H,25H2,(H2,26,28)(H,30,31)	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Patents Similars	Article PubMed	28	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Novartis Institutes for Biomedical Research Curated by ChEMBL					Assay Description Inhibition of Pim1 (unknown origin) using BAD peptide preincubated for 15 mins followed by ATP addition measured after 60 to 100 mins by Kinase-Glo r...				Bioorg Med Chem Lett 26: 2328-32 (2016) Article DOI: 10.1016/j.bmcl.2016.03.037 BindingDB Entry DOI: 10.7270/Q2WD42F0
					More data for this Ligand-Target Pair
Serine/threonine-protein kinase pim-2 (Homo sapiens (Human))	BDBM50156374 (CHEMBL3792428) Show SMILES Nc1cc(ccn1)-c1ccncc1NC(=O)c1nc(ccc1N)-c1ccccc1F Show InChI InChI=1S/C22H17FN6O/c23-16-4-2-1-3-15(16)18-6-5-17(24)21(28-18)22(30)29-19-12-26-9-8-14(19)13-7-10-27-20(25)11-13/h1-12H,24H2,(H2,25,27)(H,29,30)	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Patents Similars	Article PubMed	35	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Novartis Institutes for Biomedical Research Curated by ChEMBL					Assay Description Inhibition of Pim2 (unknown origin) using BAD peptide preincubated for 15 mins followed by ATP addition measured after 60 to 100 mins by Kinase-Glo r...				Bioorg Med Chem Lett 26: 2328-32 (2016) Article DOI: 10.1016/j.bmcl.2016.03.037 BindingDB Entry DOI: 10.7270/Q2WD42F0
					More data for this Ligand-Target Pair

Displayed 1 to 50 (of 60 total )  |  Next  |  Last  >>

Jump to: