Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Sodium-dependent serotonin transporter (Homo sapiens (Human)) | BDBM50310662 ((S)-2,4-dichloro-N-isobutyl-N-(pyrrolidin-3-yl)ben...) | PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Displacement of [3H]5HT from human 5HT transporter expressed in HEK293 cells by scintillation counting | Bioorg Med Chem Lett 19: 5078-81 (2009) Article DOI: 10.1016/j.bmcl.2009.07.049 BindingDB Entry DOI: 10.7270/Q2JQ115V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sodium-dependent serotonin transporter (Homo sapiens (Human)) | BDBM50310647 ((S)-2,3-dichloro-N-phenyl-N-(pyrrolidin-3-yl)benza...) | PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | 3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Displacement of [3H]5HT from human 5HT transporter expressed in HEK293 cells by scintillation counting | Bioorg Med Chem Lett 19: 5078-81 (2009) Article DOI: 10.1016/j.bmcl.2009.07.049 BindingDB Entry DOI: 10.7270/Q2JQ115V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sodium-dependent serotonin transporter (Homo sapiens (Human)) | BDBM50310652 ((S)-3-chloro-N-isobutyl-2-methyl-N-(pyrrolidin-3-y...) | PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Displacement of [3H]5HT from human 5HT transporter expressed in HEK293 cells by scintillation counting | Bioorg Med Chem Lett 19: 5078-81 (2009) Article DOI: 10.1016/j.bmcl.2009.07.049 BindingDB Entry DOI: 10.7270/Q2JQ115V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sodium-dependent serotonin transporter (Homo sapiens (Human)) | BDBM50310661 ((S)-2,3-dichloro-N-neopentyl-N-(pyrrolidin-3-yl)be...) | PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Displacement of [3H]5HT from human 5HT transporter expressed in HEK293 cells by scintillation counting | Bioorg Med Chem Lett 19: 5078-81 (2009) Article DOI: 10.1016/j.bmcl.2009.07.049 BindingDB Entry DOI: 10.7270/Q2JQ115V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sodium-dependent serotonin transporter (Homo sapiens (Human)) | BDBM50310650 ((S)-3,4-dichloro-N-isobutyl-N-(pyrrolidin-3-yl)ben...) | PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Displacement of [3H]5HT from human 5HT transporter expressed in HEK293 cells by scintillation counting | Bioorg Med Chem Lett 19: 5078-81 (2009) Article DOI: 10.1016/j.bmcl.2009.07.049 BindingDB Entry DOI: 10.7270/Q2JQ115V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sodium-dependent serotonin transporter (Homo sapiens (Human)) | BDBM84745 (CAS_136434-34-9 | DULOXETINE | LY-248686 | LY24868...) | PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | Purchase DrugBank MCE PC cid PC sid PDB UniChem Patents Similars | DrugBank Article PubMed | 5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Displacement of [3H]5HT from human 5HT transporter expressed in HEK293 cells by scintillation counting | Bioorg Med Chem Lett 19: 5078-81 (2009) Article DOI: 10.1016/j.bmcl.2009.07.049 BindingDB Entry DOI: 10.7270/Q2JQ115V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sodium-dependent serotonin transporter (Homo sapiens (Human)) | BDBM50310644 ((S)-2,3-dichloro-N-cyclopentyl-N-(pyrrolidin-3-yl)...) | PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 6 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Displacement of [3H]5HT from human 5HT transporter expressed in HEK293 cells by scintillation counting | Bioorg Med Chem Lett 19: 5078-81 (2009) Article DOI: 10.1016/j.bmcl.2009.07.049 BindingDB Entry DOI: 10.7270/Q2JQ115V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sodium-dependent serotonin transporter (Homo sapiens (Human)) | BDBM50310649 ((S)-3,5-dichloro-N-isobutyl-N-(pyrrolidin-3-yl)ben...) | PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 6 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Displacement of [3H]5HT from human 5HT transporter expressed in HEK293 cells by scintillation counting | Bioorg Med Chem Lett 19: 5078-81 (2009) Article DOI: 10.1016/j.bmcl.2009.07.049 BindingDB Entry DOI: 10.7270/Q2JQ115V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sodium-dependent serotonin transporter (Homo sapiens (Human)) | BDBM50310646 ((S)-2,3-dichloro-N-(2H-pyran-4-yl)-N-(pyrrolidin-3...) | PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | 6 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Displacement of [3H]5HT from human 5HT transporter expressed in HEK293 cells by scintillation counting | Bioorg Med Chem Lett 19: 5078-81 (2009) Article DOI: 10.1016/j.bmcl.2009.07.049 BindingDB Entry DOI: 10.7270/Q2JQ115V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sodium-dependent serotonin transporter (Homo sapiens (Human)) | BDBM50310656 ((S)-2,3-dichloro-N-isobutyl-N-(pyrrolidin-3-yl)ben...) | PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL MCE PC cid PC sid UniChem Patents Similars | Article PubMed | 6 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Displacement of [3H]5HT from human 5HT transporter expressed in HEK293 cells by scintillation counting | Bioorg Med Chem Lett 19: 5078-81 (2009) Article DOI: 10.1016/j.bmcl.2009.07.049 BindingDB Entry DOI: 10.7270/Q2JQ115V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sodium-dependent serotonin transporter (Homo sapiens (Human)) | BDBM50310666 ((S)-2-chloro-4-fluoro-N-isobutyl-N-(pyrrolidin-3-y...) | PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 7 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Displacement of [3H]5HT from human 5HT transporter expressed in HEK293 cells by scintillation counting | Bioorg Med Chem Lett 19: 5078-81 (2009) Article DOI: 10.1016/j.bmcl.2009.07.049 BindingDB Entry DOI: 10.7270/Q2JQ115V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sodium-dependent serotonin transporter (Homo sapiens (Human)) | BDBM50262411 ((S)-N-(2,3-dichlorobenzyl)-N-(pyrrolidin-3-yl)isob...) | PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 9 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Displacement of [3H]5HT from human 5HT transporter expressed in HEK293 cells by scintillation counting | Bioorg Med Chem Lett 19: 5078-81 (2009) Article DOI: 10.1016/j.bmcl.2009.07.049 BindingDB Entry DOI: 10.7270/Q2JQ115V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sodium-dependent serotonin transporter (Homo sapiens (Human)) | BDBM50310653 ((S)-3-chloro-2-fluoro-N-isobutyl-N-(pyrrolidin-3-y...) | PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 10 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Displacement of [3H]5HT from human 5HT transporter expressed in HEK293 cells by scintillation counting | Bioorg Med Chem Lett 19: 5078-81 (2009) Article DOI: 10.1016/j.bmcl.2009.07.049 BindingDB Entry DOI: 10.7270/Q2JQ115V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sodium-dependent noradrenaline transporter (Homo sapiens (Human)) | BDBM50310646 ((S)-2,3-dichloro-N-(2H-pyran-4-yl)-N-(pyrrolidin-3...) | Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | 10 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Displacement of [3H]noradrenaline from human NET receptor expressed in HEK293 cells by scintillation counting | Bioorg Med Chem Lett 19: 5078-81 (2009) Article DOI: 10.1016/j.bmcl.2009.07.049 BindingDB Entry DOI: 10.7270/Q2JQ115V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sodium-dependent serotonin transporter (Homo sapiens (Human)) | BDBM50310651 ((S)-2-chloro-N-isobutyl-N-(pyrrolidin-3-yl)-3-(tri...) | PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 11 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Displacement of [3H]5HT from human 5HT transporter expressed in HEK293 cells by scintillation counting | Bioorg Med Chem Lett 19: 5078-81 (2009) Article DOI: 10.1016/j.bmcl.2009.07.049 BindingDB Entry DOI: 10.7270/Q2JQ115V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sodium-dependent noradrenaline transporter (Homo sapiens (Human)) | BDBM50310647 ((S)-2,3-dichloro-N-phenyl-N-(pyrrolidin-3-yl)benza...) | Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | 11 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Displacement of [3H]noradrenaline from human NET receptor expressed in HEK293 cells by scintillation counting | Bioorg Med Chem Lett 19: 5078-81 (2009) Article DOI: 10.1016/j.bmcl.2009.07.049 BindingDB Entry DOI: 10.7270/Q2JQ115V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sodium-dependent noradrenaline transporter (Homo sapiens (Human)) | BDBM50310644 ((S)-2,3-dichloro-N-cyclopentyl-N-(pyrrolidin-3-yl)...) | Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 11 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Displacement of [3H]noradrenaline from human NET receptor expressed in HEK293 cells by scintillation counting | Bioorg Med Chem Lett 19: 5078-81 (2009) Article DOI: 10.1016/j.bmcl.2009.07.049 BindingDB Entry DOI: 10.7270/Q2JQ115V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sodium-dependent serotonin transporter (Homo sapiens (Human)) | BDBM50310664 ((S)-3-fluoro-N-isobutyl-2-methyl-N-(pyrrolidin-3-y...) | PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 13 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Displacement of [3H]5HT from human 5HT transporter expressed in HEK293 cells by scintillation counting | Bioorg Med Chem Lett 19: 5078-81 (2009) Article DOI: 10.1016/j.bmcl.2009.07.049 BindingDB Entry DOI: 10.7270/Q2JQ115V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sodium-dependent serotonin transporter (Homo sapiens (Human)) | BDBM50310667 ((R)-2,3-dichloro-N-isobutyl-N-(pyrrolidin-3-yl)ben...) | PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 13 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Displacement of [3H]5HT from human 5HT transporter expressed in HEK293 cells by scintillation counting | Bioorg Med Chem Lett 19: 5078-81 (2009) Article DOI: 10.1016/j.bmcl.2009.07.049 BindingDB Entry DOI: 10.7270/Q2JQ115V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sodium-dependent noradrenaline transporter (Homo sapiens (Human)) | BDBM50310661 ((S)-2,3-dichloro-N-neopentyl-N-(pyrrolidin-3-yl)be...) | Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 13 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Displacement of [3H]noradrenaline from human NET receptor expressed in HEK293 cells by scintillation counting | Bioorg Med Chem Lett 19: 5078-81 (2009) Article DOI: 10.1016/j.bmcl.2009.07.049 BindingDB Entry DOI: 10.7270/Q2JQ115V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sodium-dependent serotonin transporter (Homo sapiens (Human)) | BDBM50310665 ((S)-2-chloro-3-fluoro-N-isobutyl-N-(pyrrolidin-3-y...) | PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 15 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Displacement of [3H]5HT from human 5HT transporter expressed in HEK293 cells by scintillation counting | Bioorg Med Chem Lett 19: 5078-81 (2009) Article DOI: 10.1016/j.bmcl.2009.07.049 BindingDB Entry DOI: 10.7270/Q2JQ115V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sodium-dependent serotonin transporter (Homo sapiens (Human)) | BDBM50310660 ((S)-2,3-dichloro-N-(2-cyclopropylethyl)-N-(pyrroli...) | PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 15 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Displacement of [3H]5HT from human 5HT transporter expressed in HEK293 cells by scintillation counting | Bioorg Med Chem Lett 19: 5078-81 (2009) Article DOI: 10.1016/j.bmcl.2009.07.049 BindingDB Entry DOI: 10.7270/Q2JQ115V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sodium-dependent serotonin transporter (Homo sapiens (Human)) | BDBM50310658 ((S)-2,3-dichloro-N-propyl-N-(pyrrolidin-3-yl)benza...) | PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 16 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Displacement of [3H]5HT from human 5HT transporter expressed in HEK293 cells by scintillation counting | Bioorg Med Chem Lett 19: 5078-81 (2009) Article DOI: 10.1016/j.bmcl.2009.07.049 BindingDB Entry DOI: 10.7270/Q2JQ115V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sodium-dependent serotonin transporter (Homo sapiens (Human)) | BDBM50310663 ((S)-3-chloro-N-isobutyl-N-(pyrrolidin-3-yl)benzami...) | PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 19 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Displacement of [3H]5HT from human 5HT transporter expressed in HEK293 cells by scintillation counting | Bioorg Med Chem Lett 19: 5078-81 (2009) Article DOI: 10.1016/j.bmcl.2009.07.049 BindingDB Entry DOI: 10.7270/Q2JQ115V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sodium-dependent serotonin transporter (Homo sapiens (Human)) | BDBM50310645 ((S)-2,3-dichloro-N-(pentan-3-yl)-N-(pyrrolidin-3-y...) | PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 20 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Displacement of [3H]5HT from human 5HT transporter expressed in HEK293 cells by scintillation counting | Bioorg Med Chem Lett 19: 5078-81 (2009) Article DOI: 10.1016/j.bmcl.2009.07.049 BindingDB Entry DOI: 10.7270/Q2JQ115V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sodium-dependent noradrenaline transporter (Homo sapiens (Human)) | BDBM50310656 ((S)-2,3-dichloro-N-isobutyl-N-(pyrrolidin-3-yl)ben...) | Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL MCE PC cid PC sid UniChem Patents Similars | Article PubMed | 21 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Displacement of [3H]noradrenaline from human NET receptor expressed in HEK293 cells by scintillation counting | Bioorg Med Chem Lett 19: 5078-81 (2009) Article DOI: 10.1016/j.bmcl.2009.07.049 BindingDB Entry DOI: 10.7270/Q2JQ115V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sodium-dependent noradrenaline transporter (Homo sapiens (Human)) | BDBM50310660 ((S)-2,3-dichloro-N-(2-cyclopropylethyl)-N-(pyrroli...) | Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 24 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Displacement of [3H]noradrenaline from human NET receptor expressed in HEK293 cells by scintillation counting | Bioorg Med Chem Lett 19: 5078-81 (2009) Article DOI: 10.1016/j.bmcl.2009.07.049 BindingDB Entry DOI: 10.7270/Q2JQ115V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sodium-dependent serotonin transporter (Homo sapiens (Human)) | BDBM50310654 ((S)-3-fluoro-N-isobutyl-N-(pyrrolidin-3-yl)-2-(tri...) | PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 25 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Displacement of [3H]5HT from human 5HT transporter expressed in HEK293 cells by scintillation counting | Bioorg Med Chem Lett 19: 5078-81 (2009) Article DOI: 10.1016/j.bmcl.2009.07.049 BindingDB Entry DOI: 10.7270/Q2JQ115V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sodium-dependent noradrenaline transporter (Homo sapiens (Human)) | BDBM50310654 ((S)-3-fluoro-N-isobutyl-N-(pyrrolidin-3-yl)-2-(tri...) | Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 26 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Displacement of [3H]noradrenaline from human NET receptor expressed in HEK293 cells by scintillation counting | Bioorg Med Chem Lett 19: 5078-81 (2009) Article DOI: 10.1016/j.bmcl.2009.07.049 BindingDB Entry DOI: 10.7270/Q2JQ115V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sodium-dependent noradrenaline transporter (Homo sapiens (Human)) | BDBM50310652 ((S)-3-chloro-N-isobutyl-2-methyl-N-(pyrrolidin-3-y...) | Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 29 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Displacement of [3H]noradrenaline from human NET receptor expressed in HEK293 cells by scintillation counting | Bioorg Med Chem Lett 19: 5078-81 (2009) Article DOI: 10.1016/j.bmcl.2009.07.049 BindingDB Entry DOI: 10.7270/Q2JQ115V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sodium-dependent serotonin transporter (Homo sapiens (Human)) | BDBM50310657 ((S)-2,3-dichloro-N-ethyl-N-(pyrrolidin-3-yl)benzam...) | PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 29 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Displacement of [3H]5HT from human 5HT transporter expressed in HEK293 cells by scintillation counting | Bioorg Med Chem Lett 19: 5078-81 (2009) Article DOI: 10.1016/j.bmcl.2009.07.049 BindingDB Entry DOI: 10.7270/Q2JQ115V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sodium-dependent noradrenaline transporter (Homo sapiens (Human)) | BDBM50310658 ((S)-2,3-dichloro-N-propyl-N-(pyrrolidin-3-yl)benza...) | Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 36 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Displacement of [3H]noradrenaline from human NET receptor expressed in HEK293 cells by scintillation counting | Bioorg Med Chem Lett 19: 5078-81 (2009) Article DOI: 10.1016/j.bmcl.2009.07.049 BindingDB Entry DOI: 10.7270/Q2JQ115V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sodium-dependent noradrenaline transporter (Homo sapiens (Human)) | BDBM50310645 ((S)-2,3-dichloro-N-(pentan-3-yl)-N-(pyrrolidin-3-y...) | Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 37 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Displacement of [3H]noradrenaline from human NET receptor expressed in HEK293 cells by scintillation counting | Bioorg Med Chem Lett 19: 5078-81 (2009) Article DOI: 10.1016/j.bmcl.2009.07.049 BindingDB Entry DOI: 10.7270/Q2JQ115V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sodium-dependent noradrenaline transporter (Homo sapiens (Human)) | BDBM50310662 ((S)-2,4-dichloro-N-isobutyl-N-(pyrrolidin-3-yl)ben...) | Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 37 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Displacement of [3H]noradrenaline from human NET receptor expressed in HEK293 cells by scintillation counting | Bioorg Med Chem Lett 19: 5078-81 (2009) Article DOI: 10.1016/j.bmcl.2009.07.049 BindingDB Entry DOI: 10.7270/Q2JQ115V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sodium-dependent serotonin transporter (Homo sapiens (Human)) | BDBM50310659 ((S)-2,3-dichloro-N-(pyrrolidin-3-yl)-N-(2,2,2-trif...) | PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 39 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Displacement of [3H]5HT from human 5HT transporter expressed in HEK293 cells by scintillation counting | Bioorg Med Chem Lett 19: 5078-81 (2009) Article DOI: 10.1016/j.bmcl.2009.07.049 BindingDB Entry DOI: 10.7270/Q2JQ115V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sodium-dependent noradrenaline transporter (Homo sapiens (Human)) | BDBM50310649 ((S)-3,5-dichloro-N-isobutyl-N-(pyrrolidin-3-yl)ben...) | Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 43 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Displacement of [3H]noradrenaline from human NET receptor expressed in HEK293 cells by scintillation counting | Bioorg Med Chem Lett 19: 5078-81 (2009) Article DOI: 10.1016/j.bmcl.2009.07.049 BindingDB Entry DOI: 10.7270/Q2JQ115V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sodium-dependent noradrenaline transporter (Homo sapiens (Human)) | BDBM84745 (CAS_136434-34-9 | DULOXETINE | LY-248686 | LY24868...) | Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | Purchase DrugBank MCE PC cid PC sid PDB UniChem Patents Similars | DrugBank Article PubMed | 45 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Displacement of [3H]noradrenaline from human NET receptor expressed in HEK293 cells by scintillation counting | Bioorg Med Chem Lett 19: 5078-81 (2009) Article DOI: 10.1016/j.bmcl.2009.07.049 BindingDB Entry DOI: 10.7270/Q2JQ115V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sodium-dependent noradrenaline transporter (Homo sapiens (Human)) | BDBM50310650 ((S)-3,4-dichloro-N-isobutyl-N-(pyrrolidin-3-yl)ben...) | Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 50 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Displacement of [3H]noradrenaline from human NET receptor expressed in HEK293 cells by scintillation counting | Bioorg Med Chem Lett 19: 5078-81 (2009) Article DOI: 10.1016/j.bmcl.2009.07.049 BindingDB Entry DOI: 10.7270/Q2JQ115V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sodium-dependent noradrenaline transporter (Homo sapiens (Human)) | BDBM50262411 ((S)-N-(2,3-dichlorobenzyl)-N-(pyrrolidin-3-yl)isob...) | Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 52 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Displacement of [3H]noradrenaline from human NET receptor expressed in HEK293 cells by scintillation counting | Bioorg Med Chem Lett 19: 5078-81 (2009) Article DOI: 10.1016/j.bmcl.2009.07.049 BindingDB Entry DOI: 10.7270/Q2JQ115V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sodium-dependent serotonin transporter (Homo sapiens (Human)) | BDBM50310648 ((S)-2,5-dichloro-N-isobutyl-N-(pyrrolidin-3-yl)ben...) | PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 54 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Displacement of [3H]5HT from human 5HT transporter expressed in HEK293 cells by scintillation counting | Bioorg Med Chem Lett 19: 5078-81 (2009) Article DOI: 10.1016/j.bmcl.2009.07.049 BindingDB Entry DOI: 10.7270/Q2JQ115V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sodium-dependent noradrenaline transporter (Homo sapiens (Human)) | BDBM50310655 ((S)-N-isobutyl-2-isopropyl-N-(pyrrolidin-3-yl)benz...) | Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 65 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Displacement of [3H]noradrenaline from human NET receptor expressed in HEK293 cells by scintillation counting | Bioorg Med Chem Lett 19: 5078-81 (2009) Article DOI: 10.1016/j.bmcl.2009.07.049 BindingDB Entry DOI: 10.7270/Q2JQ115V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sodium-dependent noradrenaline transporter (Homo sapiens (Human)) | BDBM50310665 ((S)-2-chloro-3-fluoro-N-isobutyl-N-(pyrrolidin-3-y...) | Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 67 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Displacement of [3H]noradrenaline from human NET receptor expressed in HEK293 cells by scintillation counting | Bioorg Med Chem Lett 19: 5078-81 (2009) Article DOI: 10.1016/j.bmcl.2009.07.049 BindingDB Entry DOI: 10.7270/Q2JQ115V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sodium-dependent noradrenaline transporter (Homo sapiens (Human)) | BDBM50310664 ((S)-3-fluoro-N-isobutyl-2-methyl-N-(pyrrolidin-3-y...) | Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 69 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Displacement of [3H]noradrenaline from human NET receptor expressed in HEK293 cells by scintillation counting | Bioorg Med Chem Lett 19: 5078-81 (2009) Article DOI: 10.1016/j.bmcl.2009.07.049 BindingDB Entry DOI: 10.7270/Q2JQ115V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sodium-dependent noradrenaline transporter (Homo sapiens (Human)) | BDBM50310659 ((S)-2,3-dichloro-N-(pyrrolidin-3-yl)-N-(2,2,2-trif...) | Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 95 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Displacement of [3H]noradrenaline from human NET receptor expressed in HEK293 cells by scintillation counting | Bioorg Med Chem Lett 19: 5078-81 (2009) Article DOI: 10.1016/j.bmcl.2009.07.049 BindingDB Entry DOI: 10.7270/Q2JQ115V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sodium-dependent noradrenaline transporter (Homo sapiens (Human)) | BDBM50310651 ((S)-2-chloro-N-isobutyl-N-(pyrrolidin-3-yl)-3-(tri...) | Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 103 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Displacement of [3H]noradrenaline from human NET receptor expressed in HEK293 cells by scintillation counting | Bioorg Med Chem Lett 19: 5078-81 (2009) Article DOI: 10.1016/j.bmcl.2009.07.049 BindingDB Entry DOI: 10.7270/Q2JQ115V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sodium-dependent noradrenaline transporter (Homo sapiens (Human)) | BDBM50310663 ((S)-3-chloro-N-isobutyl-N-(pyrrolidin-3-yl)benzami...) | Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 135 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Displacement of [3H]noradrenaline from human NET receptor expressed in HEK293 cells by scintillation counting | Bioorg Med Chem Lett 19: 5078-81 (2009) Article DOI: 10.1016/j.bmcl.2009.07.049 BindingDB Entry DOI: 10.7270/Q2JQ115V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sodium-dependent noradrenaline transporter (Homo sapiens (Human)) | BDBM50310653 ((S)-3-chloro-2-fluoro-N-isobutyl-N-(pyrrolidin-3-y...) | Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 139 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Displacement of [3H]noradrenaline from human NET receptor expressed in HEK293 cells by scintillation counting | Bioorg Med Chem Lett 19: 5078-81 (2009) Article DOI: 10.1016/j.bmcl.2009.07.049 BindingDB Entry DOI: 10.7270/Q2JQ115V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sodium-dependent noradrenaline transporter (Homo sapiens (Human)) | BDBM50310667 ((R)-2,3-dichloro-N-isobutyl-N-(pyrrolidin-3-yl)ben...) | Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 169 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Displacement of [3H]noradrenaline from human NET receptor expressed in HEK293 cells by scintillation counting | Bioorg Med Chem Lett 19: 5078-81 (2009) Article DOI: 10.1016/j.bmcl.2009.07.049 BindingDB Entry DOI: 10.7270/Q2JQ115V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sodium-dependent noradrenaline transporter (Homo sapiens (Human)) | BDBM50310648 ((S)-2,5-dichloro-N-isobutyl-N-(pyrrolidin-3-yl)ben...) | Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 198 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Displacement of [3H]noradrenaline from human NET receptor expressed in HEK293 cells by scintillation counting | Bioorg Med Chem Lett 19: 5078-81 (2009) Article DOI: 10.1016/j.bmcl.2009.07.049 BindingDB Entry DOI: 10.7270/Q2JQ115V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sodium-dependent noradrenaline transporter (Homo sapiens (Human)) | BDBM50310657 ((S)-2,3-dichloro-N-ethyl-N-(pyrrolidin-3-yl)benzam...) | Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 217 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Displacement of [3H]noradrenaline from human NET receptor expressed in HEK293 cells by scintillation counting | Bioorg Med Chem Lett 19: 5078-81 (2009) Article DOI: 10.1016/j.bmcl.2009.07.049 BindingDB Entry DOI: 10.7270/Q2JQ115V | |||||||||||
More data for this Ligand-Target Pair |
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