Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Microtubule-associated protein 2 (Homo sapiens (Human)) | BDBM50234032 (CHEMBL4060668) | KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | 38 | n/a | n/a | n/a | n/a | n/a | n/a |
Merck KGaA Curated by ChEMBL | Assay Description Inhibition of recombinant human N-terminal His tagged MetAP-2 using tripeptide Met-Ala-Ser as substrate preincubated for 15 mins followed by substrat... | Bioorg Med Chem Lett 27: 551-556 (2017) Article DOI: 10.1016/j.bmcl.2016.12.019 BindingDB Entry DOI: 10.7270/Q2V98BB4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Microtubule-associated protein 2 (Homo sapiens (Human)) | BDBM50234031 (CHEMBL4082542) | KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 110 | n/a | n/a | n/a | n/a | n/a | n/a |
Merck KGaA Curated by ChEMBL | Assay Description Inhibition of recombinant human N-terminal His tagged MetAP-2 using tripeptide Met-Ala-Ser as substrate preincubated for 15 mins followed by substrat... | Bioorg Med Chem Lett 27: 551-556 (2017) Article DOI: 10.1016/j.bmcl.2016.12.019 BindingDB Entry DOI: 10.7270/Q2V98BB4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Microtubule-associated protein 2 (Homo sapiens (Human)) | BDBM50234025 (CHEMBL4093791) | KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 230 | n/a | n/a | n/a | n/a | n/a | n/a |
Merck KGaA Curated by ChEMBL | Assay Description Inhibition of recombinant human N-terminal His tagged MetAP-2 using tripeptide Met-Ala-Ser as substrate preincubated for 15 mins followed by substrat... | Bioorg Med Chem Lett 27: 551-556 (2017) Article DOI: 10.1016/j.bmcl.2016.12.019 BindingDB Entry DOI: 10.7270/Q2V98BB4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Microtubule-associated protein 2 (Homo sapiens (Human)) | BDBM50234035 (CHEMBL4070008) | KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 450 | n/a | n/a | n/a | n/a | n/a | n/a |
Merck KGaA Curated by ChEMBL | Assay Description Inhibition of recombinant human N-terminal His tagged MetAP-2 using tripeptide Met-Ala-Ser as substrate preincubated for 15 mins followed by substrat... | Bioorg Med Chem Lett 27: 551-556 (2017) Article DOI: 10.1016/j.bmcl.2016.12.019 BindingDB Entry DOI: 10.7270/Q2V98BB4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Microtubule-associated protein 2 (Homo sapiens (Human)) | BDBM50234037 (CHEMBL4083510) | KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 560 | n/a | n/a | n/a | n/a | n/a | n/a |
Merck KGaA Curated by ChEMBL | Assay Description Inhibition of recombinant human N-terminal His tagged MetAP-2 using tripeptide Met-Ala-Ser as substrate preincubated for 15 mins followed by substrat... | Bioorg Med Chem Lett 27: 551-556 (2017) Article DOI: 10.1016/j.bmcl.2016.12.019 BindingDB Entry DOI: 10.7270/Q2V98BB4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Microtubule-associated protein 2 (Homo sapiens (Human)) | BDBM50234024 (CHEMBL4097198) | KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 700 | n/a | n/a | n/a | n/a | n/a | n/a |
Merck KGaA Curated by ChEMBL | Assay Description Inhibition of recombinant human N-terminal His tagged MetAP-2 using tripeptide Met-Ala-Ser as substrate preincubated for 15 mins followed by substrat... | Bioorg Med Chem Lett 27: 551-556 (2017) Article DOI: 10.1016/j.bmcl.2016.12.019 BindingDB Entry DOI: 10.7270/Q2V98BB4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Microtubule-associated protein 2 (Homo sapiens (Human)) | BDBM50234033 (CHEMBL4078213) | KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents | Article PubMed | n/a | n/a | 1.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Merck KGaA Curated by ChEMBL | Assay Description Inhibition of recombinant human N-terminal His tagged MetAP-2 using tripeptide Met-Ala-Ser as substrate preincubated for 15 mins followed by substrat... | Bioorg Med Chem Lett 27: 551-556 (2017) Article DOI: 10.1016/j.bmcl.2016.12.019 BindingDB Entry DOI: 10.7270/Q2V98BB4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Microtubule-associated protein 2 (Homo sapiens (Human)) | BDBM50234022 (CHEMBL4066295) | KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.30E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Merck KGaA Curated by ChEMBL | Assay Description Inhibition of recombinant human N-terminal His tagged MetAP-2 using tripeptide Met-Ala-Ser as substrate preincubated for 15 mins followed by substrat... | Bioorg Med Chem Lett 27: 551-556 (2017) Article DOI: 10.1016/j.bmcl.2016.12.019 BindingDB Entry DOI: 10.7270/Q2V98BB4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Microtubule-associated protein 2 (Homo sapiens (Human)) | BDBM50234020 (CHEMBL4101592) | KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.60E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Merck KGaA Curated by ChEMBL | Assay Description Inhibition of recombinant human N-terminal His tagged MetAP-2 using tripeptide Met-Ala-Ser as substrate preincubated for 15 mins followed by substrat... | Bioorg Med Chem Lett 27: 551-556 (2017) Article DOI: 10.1016/j.bmcl.2016.12.019 BindingDB Entry DOI: 10.7270/Q2V98BB4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Microtubule-associated protein 2 (Homo sapiens (Human)) | BDBM50234030 (CHEMBL4101510) | KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.80E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Merck KGaA Curated by ChEMBL | Assay Description Inhibition of recombinant human N-terminal His tagged MetAP-2 using tripeptide Met-Ala-Ser as substrate preincubated for 15 mins followed by substrat... | Bioorg Med Chem Lett 27: 551-556 (2017) Article DOI: 10.1016/j.bmcl.2016.12.019 BindingDB Entry DOI: 10.7270/Q2V98BB4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Microtubule-associated protein 2 (Homo sapiens (Human)) | BDBM50234021 (CHEMBL4074903) | KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 2.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Merck KGaA Curated by ChEMBL | Assay Description Inhibition of recombinant human N-terminal His tagged MetAP-2 using tripeptide Met-Ala-Ser as substrate preincubated for 15 mins followed by substrat... | Bioorg Med Chem Lett 27: 551-556 (2017) Article DOI: 10.1016/j.bmcl.2016.12.019 BindingDB Entry DOI: 10.7270/Q2V98BB4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Microtubule-associated protein 2 (Homo sapiens (Human)) | BDBM50234027 (CHEMBL4086033) | KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 2.20E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Merck KGaA Curated by ChEMBL | Assay Description Inhibition of recombinant human N-terminal His tagged MetAP-2 using tripeptide Met-Ala-Ser as substrate preincubated for 15 mins followed by substrat... | Bioorg Med Chem Lett 27: 551-556 (2017) Article DOI: 10.1016/j.bmcl.2016.12.019 BindingDB Entry DOI: 10.7270/Q2V98BB4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Microtubule-associated protein 2 (Homo sapiens (Human)) | BDBM50234028 (CHEMBL4063448) | KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 2.80E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Merck KGaA Curated by ChEMBL | Assay Description Inhibition of recombinant human N-terminal His tagged MetAP-2 using tripeptide Met-Ala-Ser as substrate preincubated for 15 mins followed by substrat... | Bioorg Med Chem Lett 27: 551-556 (2017) Article DOI: 10.1016/j.bmcl.2016.12.019 BindingDB Entry DOI: 10.7270/Q2V98BB4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Microtubule-associated protein 2 (Homo sapiens (Human)) | BDBM50234034 (CHEMBL4093860) | KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 3.80E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Merck KGaA Curated by ChEMBL | Assay Description Inhibition of recombinant human N-terminal His tagged MetAP-2 using tripeptide Met-Ala-Ser as substrate preincubated for 15 mins followed by substrat... | Bioorg Med Chem Lett 27: 551-556 (2017) Article DOI: 10.1016/j.bmcl.2016.12.019 BindingDB Entry DOI: 10.7270/Q2V98BB4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Microtubule-associated protein 2 (Homo sapiens (Human)) | BDBM50234036 (CHEMBL4064507) | KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | 8.60E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Merck KGaA Curated by ChEMBL | Assay Description Inhibition of recombinant human N-terminal His tagged MetAP-2 using tripeptide Met-Ala-Ser as substrate preincubated for 15 mins followed by substrat... | Bioorg Med Chem Lett 27: 551-556 (2017) Article DOI: 10.1016/j.bmcl.2016.12.019 BindingDB Entry DOI: 10.7270/Q2V98BB4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Microtubule-associated protein 2 (Homo sapiens (Human)) | BDBM50234026 (CHEMBL4073089) | KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >5.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Merck KGaA Curated by ChEMBL | Assay Description Inhibition of recombinant human N-terminal His tagged MetAP-2 using tripeptide Met-Ala-Ser as substrate preincubated for 15 mins followed by substrat... | Bioorg Med Chem Lett 27: 551-556 (2017) Article DOI: 10.1016/j.bmcl.2016.12.019 BindingDB Entry DOI: 10.7270/Q2V98BB4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Microtubule-associated protein 2 (Homo sapiens (Human)) | BDBM50234019 (CHEMBL4096268) | KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >5.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Merck KGaA Curated by ChEMBL | Assay Description Inhibition of recombinant human N-terminal His tagged MetAP-2 using tripeptide Met-Ala-Ser as substrate preincubated for 15 mins followed by substrat... | Bioorg Med Chem Lett 27: 551-556 (2017) Article DOI: 10.1016/j.bmcl.2016.12.019 BindingDB Entry DOI: 10.7270/Q2V98BB4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Microtubule-associated protein 2 (Homo sapiens (Human)) | BDBM50234029 (CHEMBL4091303) | KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >5.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Merck KGaA Curated by ChEMBL | Assay Description Inhibition of recombinant human N-terminal His tagged MetAP-2 using tripeptide Met-Ala-Ser as substrate preincubated for 15 mins followed by substrat... | Bioorg Med Chem Lett 27: 551-556 (2017) Article DOI: 10.1016/j.bmcl.2016.12.019 BindingDB Entry DOI: 10.7270/Q2V98BB4 | |||||||||||
More data for this Ligand-Target Pair |