Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Androgen receptor (Rattus norvegicus (Rat)) | BDBM18161 ((1S,2S,7S,10R,11S,14S,15S)-14-hydroxy-2,15-dimethy...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase CHEMBL KEGG MMDB PC cid PC sid PDB UniChem Patents Similars | PDB PubMed | 0.690 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
The University of Michigan Medical School Curated by ChEMBL | Assay Description Inhibitory constant against rat prostate cytosol androgen receptor using [3H]mibolerone | J Med Chem 43: 3344-7 (2000) BindingDB Entry DOI: 10.7270/Q2GQ6ZFW | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
Androgen receptor (Rattus norvegicus (Rat)) | BDBM50091401 (4-[3-(4-Hydroxy-butyl)-4,4-dimethyl-5-oxo-2-thioxo...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 0.710 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
The University of Michigan Medical School Curated by ChEMBL | Assay Description Inhibitory constant against rat prostate cytosol androgen receptor using [3H]mibolerone | J Med Chem 43: 3344-7 (2000) BindingDB Entry DOI: 10.7270/Q2GQ6ZFW | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Androgen receptor (Rattus norvegicus (Rat)) | BDBM26258 ((1S,2R,9R,10R,11S,14S,15S)-14-hydroxy-9,14,15-trim...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase KEGG PC cid PC sid UniChem Patents Similars | PubMed | 0.75 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
The University of Michigan Medical School Curated by ChEMBL | Assay Description Inhibitory constant against rat prostate cytosol androgen receptor using [3H]mibolerone | J Med Chem 43: 3344-7 (2000) BindingDB Entry DOI: 10.7270/Q2GQ6ZFW | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Androgen receptor (Rattus norvegicus (Rat)) | BDBM8885 ((1S,2R,10R,11S,14S,15S)-14-hydroxy-2,15-dimethylte...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase DrugBank KEGG MMDB PC cid PC sid PDB UniChem Similars | PDB PubMed | 1.40 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
The University of Michigan Medical School Curated by ChEMBL | Assay Description Inhibitory constant against rat prostate cytosol androgen receptor using [3H]mibolerone | J Med Chem 43: 3344-7 (2000) BindingDB Entry DOI: 10.7270/Q2GQ6ZFW | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
Androgen receptor (Rattus norvegicus (Rat)) | BDBM50091400 (4-(3-(4-hydroxybutyl)-4,4-dimethyl-5-oxo-2-thioxoi...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Patents Similars | PubMed | 2.20 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
The University of Michigan Medical School Curated by ChEMBL | Assay Description Inhibitory constant against rat prostate cytosol androgen receptor using [3H]mibolerone | J Med Chem 43: 3344-7 (2000) BindingDB Entry DOI: 10.7270/Q2GQ6ZFW | |||||||||||
More data for this Ligand-Target Pair |