Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Progesterone receptor (Homo sapiens (Human)) | BDBM50065585 (5-(4-Chloro-3-methyl-phenyl)-9-fluoro-2,2,4-trimet...) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | 0.400 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Ligand Pharmaceuticals Inc. Curated by ChEMBL | Assay Description Binding affinity for human progesterone receptor isoform A expressed in CV-1 cells | J Med Chem 41: 2779-85 (1998) Article DOI: 10.1021/jm980190c BindingDB Entry DOI: 10.7270/Q2CV4JFM | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Progesterone receptor (Homo sapiens (Human)) | BDBM50065585 (5-(4-Chloro-3-methyl-phenyl)-9-fluoro-2,2,4-trimet...) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | 0.400 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Ligand Pharmaceuticals Inc. Curated by ChEMBL | Assay Description Binding affinity for human progesterone receptor isoform A expressed in CV-1 cells | J Med Chem 41: 2779-85 (1998) Article DOI: 10.1021/jm980190c BindingDB Entry DOI: 10.7270/Q2CV4JFM | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Progesterone receptor (Homo sapiens (Human)) | BDBM50062430 (9-Chloro-5-(3-chloro-phenyl)-2,2,4-trimethyl-2,5-d...) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 0.480 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Ligand Pharmaceuticals Inc. Curated by ChEMBL | Assay Description Binding affinity for human progesterone receptor isoform A expressed in CV-1 cells | J Med Chem 41: 2779-85 (1998) Article DOI: 10.1021/jm980190c BindingDB Entry DOI: 10.7270/Q2CV4JFM | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Progesterone receptor (Homo sapiens (Human)) | BDBM50062429 (5-(4-Chloro-3-methyl-phenyl)-9-fluoro-2,2,4-trimet...) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 0.490 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Ligand Pharmaceuticals Inc. Curated by ChEMBL | Assay Description Binding affinity for human progesterone receptor isoform A expressed in CV-1 cells | J Med Chem 41: 2779-85 (1998) Article DOI: 10.1021/jm980190c BindingDB Entry DOI: 10.7270/Q2CV4JFM | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Progesterone receptor (Homo sapiens (Human)) | BDBM50062439 (9-Chloro-5-(4-chloro-3-methyl-phenyl)-2,2,4-trimet...) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 0.5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Ligand Pharmaceuticals Inc. Curated by ChEMBL | Assay Description Binding affinity for human progesterone receptor isoform A expressed in CV-1 cells | J Med Chem 41: 2779-85 (1998) Article DOI: 10.1021/jm980190c BindingDB Entry DOI: 10.7270/Q2CV4JFM | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Progesterone receptor (Homo sapiens (Human)) | BDBM8903 ((1S,2R,10S,11S,14S,15S)-14-acetyl-2,15-dimethyltet...) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL DrugBank MCE KEGG MMDB PC cid PC sid PDB UniChem Similars | DrugBank Article PubMed | 3.80 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Ligand Pharmaceuticals Inc. Curated by ChEMBL | Assay Description Binding affinity for human progesterone receptor isoform A expressed in CV-1 cells | J Med Chem 41: 2779-85 (1998) Article DOI: 10.1021/jm980190c BindingDB Entry DOI: 10.7270/Q2CV4JFM | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucocorticoid receptor (Homo sapiens (Human)) | BDBM50062430 (9-Chloro-5-(3-chloro-phenyl)-2,2,4-trimethyl-2,5-d...) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 6.30 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Ligand Pharmaceuticals Inc. Curated by ChEMBL | Assay Description Binding affinity for human glucocorticoid receptor expressed in CV-1 cells | J Med Chem 41: 2779-85 (1998) Article DOI: 10.1021/jm980190c BindingDB Entry DOI: 10.7270/Q2CV4JFM | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucocorticoid receptor (Homo sapiens (Human)) | BDBM50062439 (9-Chloro-5-(4-chloro-3-methyl-phenyl)-2,2,4-trimet...) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 14 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Ligand Pharmaceuticals Inc. Curated by ChEMBL | Assay Description Binding affinity for human glucocorticoid receptor expressed in CV-1 cells | J Med Chem 41: 2779-85 (1998) Article DOI: 10.1021/jm980190c BindingDB Entry DOI: 10.7270/Q2CV4JFM | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Progesterone receptor (Homo sapiens (Human)) | BDBM50062432 (5-(3-Chloro-phenyl)-9-fluoro-2,2,4-trimethyl-2,5-d...) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 30 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Ligand Pharmaceuticals Inc. Curated by ChEMBL | Assay Description Binding affinity for human progesterone receptor isoform A expressed in CV-1 cells | J Med Chem 41: 2779-85 (1998) Article DOI: 10.1021/jm980190c BindingDB Entry DOI: 10.7270/Q2CV4JFM | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Progesterone receptor (Homo sapiens (Human)) | BDBM50062432 (5-(3-Chloro-phenyl)-9-fluoro-2,2,4-trimethyl-2,5-d...) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 30 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Ligand Pharmaceuticals Inc. Curated by ChEMBL | Assay Description Binding affinity for human progesterone receptor isoform A expressed in CV-1 cells | J Med Chem 41: 2779-85 (1998) Article DOI: 10.1021/jm980190c BindingDB Entry DOI: 10.7270/Q2CV4JFM | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucocorticoid receptor (Homo sapiens (Human)) | BDBM50062432 (5-(3-Chloro-phenyl)-9-fluoro-2,2,4-trimethyl-2,5-d...) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 133 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Ligand Pharmaceuticals Inc. Curated by ChEMBL | Assay Description Binding affinity for human glucocorticoid receptor expressed in CV-1 cells | J Med Chem 41: 2779-85 (1998) Article DOI: 10.1021/jm980190c BindingDB Entry DOI: 10.7270/Q2CV4JFM | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucocorticoid receptor (Homo sapiens (Human)) | BDBM50062429 (5-(4-Chloro-3-methyl-phenyl)-9-fluoro-2,2,4-trimet...) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 210 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Ligand Pharmaceuticals Inc. Curated by ChEMBL | Assay Description Binding affinity for human glucocorticoid receptor expressed in CV-1 cells | J Med Chem 41: 2779-85 (1998) Article DOI: 10.1021/jm980190c BindingDB Entry DOI: 10.7270/Q2CV4JFM | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Progesterone receptor (Homo sapiens (Human)) | BDBM8903 ((1S,2R,10S,11S,14S,15S)-14-acetyl-2,15-dimethyltet...) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL DrugBank MCE KEGG MMDB PC cid PC sid PDB UniChem Similars | DrugBank Article PubMed | n/a | n/a | n/a | n/a | 1.5 | n/a | n/a | n/a | n/a |
Ligand Pharmaceuticals Inc. Curated by ChEMBL | Assay Description Effective concentration for half-maximal activation of human progesterone receptor expressed in CV-1 cells | J Med Chem 41: 2779-85 (1998) Article DOI: 10.1021/jm980190c BindingDB Entry DOI: 10.7270/Q2CV4JFM | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Progesterone receptor (Homo sapiens (Human)) | BDBM50062439 (9-Chloro-5-(4-chloro-3-methyl-phenyl)-2,2,4-trimet...) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 9.40 | n/a | n/a | n/a | n/a |
Ligand Pharmaceuticals Inc. Curated by ChEMBL | Assay Description Effective concentration for half-maximal activation of human progesterone receptor expressed in CV-1 cells | J Med Chem 41: 2779-85 (1998) Article DOI: 10.1021/jm980190c BindingDB Entry DOI: 10.7270/Q2CV4JFM | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Progesterone receptor (Homo sapiens (Human)) | BDBM50062432 (5-(3-Chloro-phenyl)-9-fluoro-2,2,4-trimethyl-2,5-d...) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 1.30 | n/a | n/a | n/a | n/a |
Ligand Pharmaceuticals Inc. Curated by ChEMBL | Assay Description Effective concentration for half-maximal activation of human progesterone receptor expressed in CV-1 cells | J Med Chem 41: 2779-85 (1998) Article DOI: 10.1021/jm980190c BindingDB Entry DOI: 10.7270/Q2CV4JFM | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Progesterone receptor (Homo sapiens (Human)) | BDBM50065585 (5-(4-Chloro-3-methyl-phenyl)-9-fluoro-2,2,4-trimet...) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 2.40 | n/a | n/a | n/a | n/a |
Ligand Pharmaceuticals Inc. Curated by ChEMBL | Assay Description Effective concentration for half-maximal activation of human progesterone receptor expressed in CV-1 cells | J Med Chem 41: 2779-85 (1998) Article DOI: 10.1021/jm980190c BindingDB Entry DOI: 10.7270/Q2CV4JFM | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Progesterone receptor (Homo sapiens (Human)) | BDBM50062429 (5-(4-Chloro-3-methyl-phenyl)-9-fluoro-2,2,4-trimet...) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | 2.70 | n/a | n/a | n/a | n/a |
Ligand Pharmaceuticals Inc. Curated by ChEMBL | Assay Description Effective concentration for half-maximal activation of human progesterone receptor expressed in CV-1 cells | J Med Chem 41: 2779-85 (1998) Article DOI: 10.1021/jm980190c BindingDB Entry DOI: 10.7270/Q2CV4JFM | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Progesterone receptor (Homo sapiens (Human)) | BDBM50062430 (9-Chloro-5-(3-chloro-phenyl)-2,2,4-trimethyl-2,5-d...) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 3.60 | n/a | n/a | n/a | n/a |
Ligand Pharmaceuticals Inc. Curated by ChEMBL | Assay Description Effective concentration for half-maximal activation of human progesterone receptor expressed in CV-1 cells | J Med Chem 41: 2779-85 (1998) Article DOI: 10.1021/jm980190c BindingDB Entry DOI: 10.7270/Q2CV4JFM | |||||||||||
More data for this Ligand-Target Pair |