Compile Data Set for Download or QSAR

Found 274 hits Enz. Inhib. hit(s) with all data for entry = 827   

Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kJ/mole	IC50 nM	Kd nM	EC50/IC50 nM	koff s-1	kon M-1s-1	pH	Temp °C
Lysine-specific demethylase 4C (Homo sapiens (Human))	BDBM293670 (3-({[(1R)-6-[methyl(pyridin-3-yl)amino]-1,2,3,4- |...) Show SMILES CN(c1cccnc1)c1ccc2[C@H](CNc3cnccc3C(O)=O)CCCc2c1 |r| Show InChI InChI=1S/C23H24N4O2/c1-27(19-6-3-10-24-14-19)18-7-8-20-16(12-18)4-2-5-17(20)13-26-22-15-25-11-9-21(22)23(28)29/h3,6-12,14-15,17,26H,2,4-5,13H2,1H3,(H,28,29)/t17-/m0/s1	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<100	n/a	n/a	n/a	n/a	n/a	25
Celgene Quanticel Research, Inc. US Patent					Assay Description The ability of test compounds to inhibit the activity of JMJD2C was determined in 384-well plate format under the following reaction conditions: 0.3 ...				US Patent US10106534 (2018) BindingDB Entry DOI: 10.7270/Q2JW8GZX
					More data for this Ligand-Target Pair
Lysine-specific demethylase 6B (Homo sapiens (Human))	BDBM293686 (3-({[7-(furan-3-yl)-3,4-dihydro-2H-1-benzopyran-4-...) Show SMILES OC(=O)c1ccncc1NCC1CCOc2cc(ccc12)-c1ccoc1 Show InChI InChI=1S/C20H18N2O4/c23-20(24)17-3-6-21-11-18(17)22-10-14-5-8-26-19-9-13(1-2-16(14)19)15-4-7-25-12-15/h1-4,6-7,9,11-12,14,22H,5,8,10H2,(H,23,24)	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<100	n/a	n/a	n/a	n/a	n/a	25
Celgene Quanticel Research, Inc. US Patent					Assay Description The enzymatic assay of JMJD3 activity is based upon Time Resolved-Fluorescence Resonance Energy Transfer (TR-FRET) detection. The ability of test com...				US Patent US10106534 (2018) BindingDB Entry DOI: 10.7270/Q2JW8GZX
					More data for this Ligand-Target Pair
Lysine-specific demethylase 6B (Homo sapiens (Human))	BDBM293691 (3-({[(4S)-7-(thiophen-3-yl)-3,4-dihydro-2H-1-benzo...) Show SMILES OC(=O)c1ccncc1NC[C@H]1CCOc2cc(ccc12)-c1ccsc1 |r| Show InChI InChI=1S/C20H18N2O3S/c23-20(24)17-3-6-21-11-18(17)22-10-14-4-7-25-19-9-13(1-2-16(14)19)15-5-8-26-12-15/h1-3,5-6,8-9,11-12,14,22H,4,7,10H2,(H,23,24)/t14-/m1/s1	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<100	n/a	n/a	n/a	n/a	n/a	25
Celgene Quanticel Research, Inc. US Patent					Assay Description The enzymatic assay of JMJD3 activity is based upon Time Resolved-Fluorescence Resonance Energy Transfer (TR-FRET) detection. The ability of test com...				US Patent US10106534 (2018) BindingDB Entry DOI: 10.7270/Q2JW8GZX
					More data for this Ligand-Target Pair
Lysine-specific demethylase 4C (Homo sapiens (Human))	BDBM293863 (3-({[(4R)-7-{methyl[4-(1-methylpiperidin-4-yl)phen...) Show SMILES CN(c1ccc(cc1)C1CCN(C)CC1)c1ccc2[C@H](CNc3cnccc3C(O)=O)CCOc2c1 |r| Show InChI InChI=1S/C29H34N4O3/c1-32-14-10-21(11-15-32)20-3-5-23(6-4-20)33(2)24-7-8-25-22(12-16-36-28(25)17-24)18-31-27-19-30-13-9-26(27)29(34)35/h3-9,13,17,19,21-22,31H,10-12,14-16,18H2,1-2H3,(H,34,35)/t22-/m0/s1	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<100	n/a	n/a	n/a	n/a	n/a	25
Celgene Quanticel Research, Inc. US Patent					Assay Description The ability of test compounds to inhibit the activity of JMJD2C was determined in 384-well plate format under the following reaction conditions: 0.3 ...				US Patent US10106534 (2018) BindingDB Entry DOI: 10.7270/Q2JW8GZX
					More data for this Ligand-Target Pair
Lysine-specific demethylase 4C (Homo sapiens (Human))	BDBM293831 (3-({[(1R)-6-[methyl(pyridin-4-yl)amino]-1,2,3,4- |...) Show SMILES CN(c1ccncc1)c1ccc2[C@H](CNc3cnccc3C(O)=O)CCCc2c1 |r| Show InChI InChI=1S/C23H24N4O2/c1-27(18-7-10-24-11-8-18)19-5-6-20-16(13-19)3-2-4-17(20)14-26-22-15-25-12-9-21(22)23(28)29/h5-13,15,17,26H,2-4,14H2,1H3,(H,28,29)/t17-/m0/s1	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<100	n/a	n/a	n/a	n/a	n/a	25
Celgene Quanticel Research, Inc. US Patent					Assay Description The ability of test compounds to inhibit the activity of JMJD2C was determined in 384-well plate format under the following reaction conditions: 0.3 ...				US Patent US10106534 (2018) BindingDB Entry DOI: 10.7270/Q2JW8GZX
					More data for this Ligand-Target Pair
Lysine-specific demethylase 4C (Homo sapiens (Human))	BDBM293836 (3-({[(4R)-7-[(4-methoxyphenyl)(methyl)amino]-3,4-d...) Show SMILES COc1ccc(cc1)N(C)c1ccc2[C@H](CNc3cnccc3C(O)=O)CCOc2c1 |r| Show InChI InChI=1S/C24H25N3O4/c1-27(17-3-6-19(30-2)7-4-17)18-5-8-20-16(10-12-31-23(20)13-18)14-26-22-15-25-11-9-21(22)24(28)29/h3-9,11,13,15-16,26H,10,12,14H2,1-2H3,(H,28,29)/t16-/m0/s1	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<100	n/a	n/a	n/a	n/a	n/a	25
Celgene Quanticel Research, Inc. US Patent					Assay Description The ability of test compounds to inhibit the activity of JMJD2C was determined in 384-well plate format under the following reaction conditions: 0.3 ...				US Patent US10106534 (2018) BindingDB Entry DOI: 10.7270/Q2JW8GZX
					More data for this Ligand-Target Pair
Lysine-specific demethylase 4C (Homo sapiens (Human))	BDBM293862 (3-({[(4R)-7-{methyl[4-(1-methyl-1,2,3,6-tetrahydro...) Show SMILES CN(c1ccc(cc1)C1=CCN(C)CC1)c1ccc2[C@H](CNc3cnccc3C(O)=O)CCOc2c1 |r,t:9| Show InChI InChI=1S/C29H32N4O3/c1-32-14-10-21(11-15-32)20-3-5-23(6-4-20)33(2)24-7-8-25-22(12-16-36-28(25)17-24)18-31-27-19-30-13-9-26(27)29(34)35/h3-10,13,17,19,22,31H,11-12,14-16,18H2,1-2H3,(H,34,35)/t22-/m0/s1	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<100	n/a	n/a	n/a	n/a	n/a	25
Celgene Quanticel Research, Inc. US Patent					Assay Description The ability of test compounds to inhibit the activity of JMJD2C was determined in 384-well plate format under the following reaction conditions: 0.3 ...				US Patent US10106534 (2018) BindingDB Entry DOI: 10.7270/Q2JW8GZX
					More data for this Ligand-Target Pair
Lysine-specific demethylase 4C (Homo sapiens (Human))	BDBM293803 (3-({[(4R)-7-[methyl(5-methylpyridin-2-yl)amino]-3,...) Show SMILES CN(c1ccc2[C@H](CNc3cnccc3C(O)=O)CCOc2c1)c1ccc(C)cn1 |r| Show InChI InChI=1S/C23H24N4O3/c1-15-3-6-22(26-12-15)27(2)17-4-5-18-16(8-10-30-21(18)11-17)13-25-20-14-24-9-7-19(20)23(28)29/h3-7,9,11-12,14,16,25H,8,10,13H2,1-2H3,(H,28,29)/t16-/m0/s1	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	<100	n/a	n/a	n/a	n/a	n/a	25
Celgene Quanticel Research, Inc. US Patent					Assay Description The ability of test compounds to inhibit the activity of JMJD2C was determined in 384-well plate format under the following reaction conditions: 0.3 ...				US Patent US10106534 (2018) BindingDB Entry DOI: 10.7270/Q2JW8GZX
					More data for this Ligand-Target Pair
Lysine-specific demethylase 4C (Homo sapiens (Human))	BDBM293660 (3-({[(1S)-6-[methyl(phenyl)amino]-1,2,3,4-tetrahyd...) Show SMILES CN(c1ccccc1)c1ccc2[C@H](CNc3cnccc3C(O)=O)CCCc2c1 |r| Show InChI InChI=1S/C24H25N3O2/c1-27(19-8-3-2-4-9-19)20-10-11-21-17(14-20)6-5-7-18(21)15-26-23-16-25-13-12-22(23)24(28)29/h2-4,8-14,16,18,26H,5-7,15H2,1H3,(H,28,29)/t18-/m0/s1	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	Purchase MCE PC cid PC sid PDB UniChem	US Patent	n/a	n/a	550	n/a	n/a	n/a	n/a	n/a	25
Celgene Quanticel Research, Inc. US Patent					Assay Description The ability of test compounds to inhibit the activity of JMJD2C was determined in 384-well plate format under the following reaction conditions: 0.3 ...				US Patent US10106534 (2018) BindingDB Entry DOI: 10.7270/Q2JW8GZX
					More data for this Ligand-Target Pair
Lysine-specific demethylase 4C (Homo sapiens (Human))	BDBM293661 (3-({[6-(2-oxopyrrolidin-1-yl)-1,2,3,4-tetrahydrona...) Show SMILES OC(=O)c1ccncc1NCC1CCCc2cc(ccc12)N1CCCC1=O Show InChI InChI=1S/C21H23N3O3/c25-20-5-2-10-24(20)16-6-7-17-14(11-16)3-1-4-15(17)12-23-19-13-22-9-8-18(19)21(26)27/h6-9,11,13,15,23H,1-5,10,12H2,(H,26,27)	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	550	n/a	n/a	n/a	n/a	n/a	25
Celgene Quanticel Research, Inc. US Patent					Assay Description The ability of test compounds to inhibit the activity of JMJD2C was determined in 384-well plate format under the following reaction conditions: 0.3 ...				US Patent US10106534 (2018) BindingDB Entry DOI: 10.7270/Q2JW8GZX
					More data for this Ligand-Target Pair
Lysine-specific demethylase 4C (Homo sapiens (Human))	BDBM293664 (3-({[(1R)-6-[(2-fluorophenyl)(methyl)amino]-1,2,3,...) Show SMILES CN(c1ccc2[C@H](CNc3cnccc3C(O)=O)CCCc2c1)c1ccccc1F |r| Show InChI InChI=1S/C24H24FN3O2/c1-28(23-8-3-2-7-21(23)25)18-9-10-19-16(13-18)5-4-6-17(19)14-27-22-15-26-12-11-20(22)24(29)30/h2-3,7-13,15,17,27H,4-6,14H2,1H3,(H,29,30)/t17-/m0/s1	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	550	n/a	n/a	n/a	n/a	n/a	25
Celgene Quanticel Research, Inc. US Patent					Assay Description The ability of test compounds to inhibit the activity of JMJD2C was determined in 384-well plate format under the following reaction conditions: 0.3 ...				US Patent US10106534 (2018) BindingDB Entry DOI: 10.7270/Q2JW8GZX
					More data for this Ligand-Target Pair
Lysine-specific demethylase 4C (Homo sapiens (Human))	BDBM293665 (3-({[(1R)-6-[(3-fluorophenyl)(methyl)amino]-1,2,3,...) Show SMILES CN(c1cccc(F)c1)c1ccc2[C@H](CNc3cnccc3C(O)=O)CCCc2c1 |r| Show InChI InChI=1S/C24H24FN3O2/c1-28(19-7-3-6-18(25)13-19)20-8-9-21-16(12-20)4-2-5-17(21)14-27-23-15-26-11-10-22(23)24(29)30/h3,6-13,15,17,27H,2,4-5,14H2,1H3,(H,29,30)/t17-/m0/s1	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	550	n/a	n/a	n/a	n/a	n/a	25
Celgene Quanticel Research, Inc. US Patent					Assay Description The ability of test compounds to inhibit the activity of JMJD2C was determined in 384-well plate format under the following reaction conditions: 0.3 ...				US Patent US10106534 (2018) BindingDB Entry DOI: 10.7270/Q2JW8GZX
					More data for this Ligand-Target Pair
Lysine-specific demethylase 4C (Homo sapiens (Human))	BDBM293666 (3-({[(1R)-6-[(4-fluorophenyl)(methyl)amino]-1,2,3,...) Show SMILES CN(c1ccc(F)cc1)c1ccc2[C@H](CNc3cnccc3C(O)=O)CCCc2c1 |r| Show InChI InChI=1S/C24H24FN3O2/c1-28(19-7-5-18(25)6-8-19)20-9-10-21-16(13-20)3-2-4-17(21)14-27-23-15-26-12-11-22(23)24(29)30/h5-13,15,17,27H,2-4,14H2,1H3,(H,29,30)/t17-/m0/s1	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	550	n/a	n/a	n/a	n/a	n/a	25
Celgene Quanticel Research, Inc. US Patent					Assay Description The ability of test compounds to inhibit the activity of JMJD2C was determined in 384-well plate format under the following reaction conditions: 0.3 ...				US Patent US10106534 (2018) BindingDB Entry DOI: 10.7270/Q2JW8GZX
					More data for this Ligand-Target Pair
Lysine-specific demethylase 4C (Homo sapiens (Human))	BDBM293668 (3-({[(1R)-6-[ethyl(phenyl)amino]-1,2,3,4-tetrahydr...) Show SMILES CCN(c1ccccc1)c1ccc2[C@H](CNc3cnccc3C(O)=O)CCCc2c1 |r| Show InChI InChI=1S/C25H27N3O2/c1-2-28(20-9-4-3-5-10-20)21-11-12-22-18(15-21)7-6-8-19(22)16-27-24-17-26-14-13-23(24)25(29)30/h3-5,9-15,17,19,27H,2,6-8,16H2,1H3,(H,29,30)/t19-/m0/s1	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	550	n/a	n/a	n/a	n/a	n/a	25
Celgene Quanticel Research, Inc. US Patent					Assay Description The ability of test compounds to inhibit the activity of JMJD2C was determined in 384-well plate format under the following reaction conditions: 0.3 ...				US Patent US10106534 (2018) BindingDB Entry DOI: 10.7270/Q2JW8GZX
					More data for this Ligand-Target Pair
Lysine-specific demethylase 4C (Homo sapiens (Human))	BDBM293669 (3-({[(1R)-6-[methyl(pyridin-2-yl)amino]-1,2,3,4- |...) Show SMILES CN(c1ccc2[C@H](CNc3cnccc3C(O)=O)CCCc2c1)c1ccccn1 |r| Show InChI InChI=1S/C23H24N4O2/c1-27(22-7-2-3-11-25-22)18-8-9-19-16(13-18)5-4-6-17(19)14-26-21-15-24-12-10-20(21)23(28)29/h2-3,7-13,15,17,26H,4-6,14H2,1H3,(H,28,29)/t17-/m0/s1	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	550	n/a	n/a	n/a	n/a	n/a	25
Celgene Quanticel Research, Inc. US Patent					Assay Description The ability of test compounds to inhibit the activity of JMJD2C was determined in 384-well plate format under the following reaction conditions: 0.3 ...				US Patent US10106534 (2018) BindingDB Entry DOI: 10.7270/Q2JW8GZX
					More data for this Ligand-Target Pair
Lysine-specific demethylase 4C (Homo sapiens (Human))	BDBM293672 (3-{[(7-bromo-3,4-dihydro-2H-1-benzopyran-4- | US10...) Show SMILES OC(=O)c1ccncc1NCC1CCOc2cc(Br)ccc12 Show InChI InChI=1S/C16H15BrN2O3/c17-11-1-2-12-10(4-6-22-15(12)7-11)8-19-14-9-18-5-3-13(14)16(20)21/h1-3,5,7,9-10,19H,4,6,8H2,(H,20,21)	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	550	n/a	n/a	n/a	n/a	n/a	25
Celgene Quanticel Research, Inc. US Patent					Assay Description The ability of test compounds to inhibit the activity of JMJD2C was determined in 384-well plate format under the following reaction conditions: 0.3 ...				US Patent US10106534 (2018) BindingDB Entry DOI: 10.7270/Q2JW8GZX
					More data for this Ligand-Target Pair
Lysine-specific demethylase 4C (Homo sapiens (Human))	BDBM293673 (3-({[7-(phenylamino)-3,4-dihydro-2H-1-benzopyran-4...) Show SMILES OC(=O)c1ccncc1NCC1CCOc2cc(Nc3ccccc3)ccc12 Show InChI InChI=1S/C22H21N3O3/c26-22(27)19-8-10-23-14-20(19)24-13-15-9-11-28-21-12-17(6-7-18(15)21)25-16-4-2-1-3-5-16/h1-8,10,12,14-15,24-25H,9,11,13H2,(H,26,27)	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	550	n/a	n/a	n/a	n/a	n/a	25
Celgene Quanticel Research, Inc. US Patent					Assay Description The ability of test compounds to inhibit the activity of JMJD2C was determined in 384-well plate format under the following reaction conditions: 0.3 ...				US Patent US10106534 (2018) BindingDB Entry DOI: 10.7270/Q2JW8GZX
					More data for this Ligand-Target Pair
Lysine-specific demethylase 4C (Homo sapiens (Human))	BDBM293674 (3-({[7-(1,2,3,4-tetrahydroquinolin-1-yl)-3,4-dihyd...) Show SMILES OC(=O)c1ccncc1NCC1CCOc2cc(ccc12)N1CCCc2ccccc12 Show InChI InChI=1S/C25H25N3O3/c29-25(30)21-9-11-26-16-22(21)27-15-18-10-13-31-24-14-19(7-8-20(18)24)28-12-3-5-17-4-1-2-6-23(17)28/h1-2,4,6-9,11,14,16,18,27H,3,5,10,12-13,15H2,(H,29,30)	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	550	n/a	n/a	n/a	n/a	n/a	25
Celgene Quanticel Research, Inc. US Patent					Assay Description The ability of test compounds to inhibit the activity of JMJD2C was determined in 384-well plate format under the following reaction conditions: 0.3 ...				US Patent US10106534 (2018) BindingDB Entry DOI: 10.7270/Q2JW8GZX
					More data for this Ligand-Target Pair
Lysine-specific demethylase 4C (Homo sapiens (Human))	BDBM293675 (3-({[7-(2,3-dihydro-1H-indol-1-yl)-3,4-dihydro-2H-...) Show SMILES OC(=O)c1ccncc1NCC1CCOc2cc(ccc12)N1CCc2ccccc12 Show InChI InChI=1S/C24H23N3O3/c28-24(29)20-7-10-25-15-21(20)26-14-17-9-12-30-23-13-18(5-6-19(17)23)27-11-8-16-3-1-2-4-22(16)27/h1-7,10,13,15,17,26H,8-9,11-12,14H2,(H,28,29)	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	550	n/a	n/a	n/a	n/a	n/a	25
Celgene Quanticel Research, Inc. US Patent					Assay Description The ability of test compounds to inhibit the activity of JMJD2C was determined in 384-well plate format under the following reaction conditions: 0.3 ...				US Patent US10106534 (2018) BindingDB Entry DOI: 10.7270/Q2JW8GZX
					More data for this Ligand-Target Pair
Lysine-specific demethylase 4C (Homo sapiens (Human))	BDBM293676 (3-({[(4R)-7-[methyl(phenyl)amino]-3,4-dihydro-2H-1...) Show SMILES CN(c1ccccc1)c1ccc2[C@H](CNc3cnccc3C(O)=O)CCOc2c1 |r| Show InChI InChI=1S/C23H23N3O3/c1-26(17-5-3-2-4-6-17)18-7-8-19-16(10-12-29-22(19)13-18)14-25-21-15-24-11-9-20(21)23(27)28/h2-9,11,13,15-16,25H,10,12,14H2,1H3,(H,27,28)/t16-/m0/s1	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	550	n/a	n/a	n/a	n/a	n/a	25
Celgene Quanticel Research, Inc. US Patent					Assay Description The ability of test compounds to inhibit the activity of JMJD2C was determined in 384-well plate format under the following reaction conditions: 0.3 ...				US Patent US10106534 (2018) BindingDB Entry DOI: 10.7270/Q2JW8GZX
					More data for this Ligand-Target Pair
Lysine-specific demethylase 6B (Homo sapiens (Human))	BDBM293676 (3-({[(4R)-7-[methyl(phenyl)amino]-3,4-dihydro-2H-1...) Show SMILES CN(c1ccccc1)c1ccc2[C@H](CNc3cnccc3C(O)=O)CCOc2c1 |r| Show InChI InChI=1S/C23H23N3O3/c1-26(17-5-3-2-4-6-17)18-7-8-19-16(10-12-29-22(19)13-18)14-25-21-15-24-11-9-20(21)23(27)28/h2-9,11,13,15-16,25H,10,12,14H2,1H3,(H,27,28)/t16-/m0/s1	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	550	n/a	n/a	n/a	n/a	n/a	25
Celgene Quanticel Research, Inc. US Patent					Assay Description The enzymatic assay of JMJD3 activity is based upon Time Resolved-Fluorescence Resonance Energy Transfer (TR-FRET) detection. The ability of test com...				US Patent US10106534 (2018) BindingDB Entry DOI: 10.7270/Q2JW8GZX
					More data for this Ligand-Target Pair
Lysine-specific demethylase 4C (Homo sapiens (Human))	BDBM293677 (3-({[(4R)-7-[(2-fluorophenyl)(methyl)amino]-3,4-di...) Show SMILES CN(c1ccc2[C@H](CNc3cnccc3C(O)=O)CCOc2c1)c1ccccc1F |r| Show InChI InChI=1S/C23H22FN3O3/c1-27(21-5-3-2-4-19(21)24)16-6-7-17-15(9-11-30-22(17)12-16)13-26-20-14-25-10-8-18(20)23(28)29/h2-8,10,12,14-15,26H,9,11,13H2,1H3,(H,28,29)/t15-/m0/s1	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	550	n/a	n/a	n/a	n/a	n/a	25
Celgene Quanticel Research, Inc. US Patent					Assay Description The ability of test compounds to inhibit the activity of JMJD2C was determined in 384-well plate format under the following reaction conditions: 0.3 ...				US Patent US10106534 (2018) BindingDB Entry DOI: 10.7270/Q2JW8GZX
					More data for this Ligand-Target Pair
Lysine-specific demethylase 4C (Homo sapiens (Human))	BDBM293678 (3-({[(4R)-7-[(3-fluorophenyl)(methyl)amino]-3,4-di...) Show SMILES CN(c1cccc(F)c1)c1ccc2[C@H](CNc3cnccc3C(O)=O)CCOc2c1 |r| Show InChI InChI=1S/C23H22FN3O3/c1-27(17-4-2-3-16(24)11-17)18-5-6-19-15(8-10-30-22(19)12-18)13-26-21-14-25-9-7-20(21)23(28)29/h2-7,9,11-12,14-15,26H,8,10,13H2,1H3,(H,28,29)/t15-/m0/s1	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	550	n/a	n/a	n/a	n/a	n/a	25
Celgene Quanticel Research, Inc. US Patent					Assay Description The ability of test compounds to inhibit the activity of JMJD2C was determined in 384-well plate format under the following reaction conditions: 0.3 ...				US Patent US10106534 (2018) BindingDB Entry DOI: 10.7270/Q2JW8GZX
					More data for this Ligand-Target Pair
Lysine-specific demethylase 4C (Homo sapiens (Human))	BDBM293679 (3-({[(4R)-7-[(4-fluorophenyl)(methyl)amino]-3,4-di...) Show SMILES CN(c1ccc(F)cc1)c1ccc2[C@H](CNc3cnccc3C(O)=O)CCOc2c1 |r| Show InChI InChI=1S/C23H22FN3O3/c1-27(17-4-2-16(24)3-5-17)18-6-7-19-15(9-11-30-22(19)12-18)13-26-21-14-25-10-8-20(21)23(28)29/h2-8,10,12,14-15,26H,9,11,13H2,1H3,(H,28,29)/t15-/m0/s1	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	550	n/a	n/a	n/a	n/a	n/a	25
Celgene Quanticel Research, Inc. US Patent					Assay Description The ability of test compounds to inhibit the activity of JMJD2C was determined in 384-well plate format under the following reaction conditions: 0.3 ...				US Patent US10106534 (2018) BindingDB Entry DOI: 10.7270/Q2JW8GZX
					More data for this Ligand-Target Pair
Lysine-specific demethylase 4C (Homo sapiens (Human))	BDBM293680 (3-({[(4R)-7-[methyl(4-methylphenyl)amino]-3,4-dihy...) Show SMILES CN(c1ccc(C)cc1)c1ccc2[C@H](CNc3cnccc3C(O)=O)CCOc2c1 |r| Show InChI InChI=1S/C24H25N3O3/c1-16-3-5-18(6-4-16)27(2)19-7-8-20-17(10-12-30-23(20)13-19)14-26-22-15-25-11-9-21(22)24(28)29/h3-9,11,13,15,17,26H,10,12,14H2,1-2H3,(H,28,29)/t17-/m0/s1	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	550	n/a	n/a	n/a	n/a	n/a	25
Celgene Quanticel Research, Inc. US Patent					Assay Description The ability of test compounds to inhibit the activity of JMJD2C was determined in 384-well plate format under the following reaction conditions: 0.3 ...				US Patent US10106534 (2018) BindingDB Entry DOI: 10.7270/Q2JW8GZX
					More data for this Ligand-Target Pair
Lysine-specific demethylase 4C (Homo sapiens (Human))	BDBM293681 (3-({[(4R)-7-[(4-chlorophenyl)(methyl)amino]-3,4-di...) Show SMILES CN(c1ccc(Cl)cc1)c1ccc2[C@H](CNc3cnccc3C(O)=O)CCOc2c1 |r| Show InChI InChI=1S/C23H22ClN3O3/c1-27(17-4-2-16(24)3-5-17)18-6-7-19-15(9-11-30-22(19)12-18)13-26-21-14-25-10-8-20(21)23(28)29/h2-8,10,12,14-15,26H,9,11,13H2,1H3,(H,28,29)/t15-/m0/s1	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	550	n/a	n/a	n/a	n/a	n/a	25
Celgene Quanticel Research, Inc. US Patent					Assay Description The ability of test compounds to inhibit the activity of JMJD2C was determined in 384-well plate format under the following reaction conditions: 0.3 ...				US Patent US10106534 (2018) BindingDB Entry DOI: 10.7270/Q2JW8GZX
					More data for this Ligand-Target Pair
Lysine-specific demethylase 4C (Homo sapiens (Human))	BDBM293682 (3-({[(4R)-7-[ethyl(phenyl)amino]-3,4-dihydro-2H-1-...) Show SMILES CCN(c1ccccc1)c1ccc2[C@H](CNc3cnccc3C(O)=O)CCOc2c1 |r| Show InChI InChI=1S/C24H25N3O3/c1-2-27(18-6-4-3-5-7-18)19-8-9-20-17(11-13-30-23(20)14-19)15-26-22-16-25-12-10-21(22)24(28)29/h3-10,12,14,16-17,26H,2,11,13,15H2,1H3,(H,28,29)/t17-/m0/s1	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	550	n/a	n/a	n/a	n/a	n/a	25
Celgene Quanticel Research, Inc. US Patent					Assay Description The ability of test compounds to inhibit the activity of JMJD2C was determined in 384-well plate format under the following reaction conditions: 0.3 ...				US Patent US10106534 (2018) BindingDB Entry DOI: 10.7270/Q2JW8GZX
					More data for this Ligand-Target Pair
Lysine-specific demethylase 4C (Homo sapiens (Human))	BDBM293683 (3-{[(2-phenyl-5,6,7,8-tetrahydroquinolin-5- | US10...) Show SMILES OC(=O)c1ccncc1NCC1CCCc2nc(ccc12)-c1ccccc1 Show InChI InChI=1S/C22H21N3O2/c26-22(27)18-11-12-23-14-21(18)24-13-16-7-4-8-20-17(16)9-10-19(25-20)15-5-2-1-3-6-15/h1-3,5-6,9-12,14,16,24H,4,7-8,13H2,(H,26,27)	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	550	n/a	n/a	n/a	n/a	n/a	25
Celgene Quanticel Research, Inc. US Patent					Assay Description The ability of test compounds to inhibit the activity of JMJD2C was determined in 384-well plate format under the following reaction conditions: 0.3 ...				US Patent US10106534 (2018) BindingDB Entry DOI: 10.7270/Q2JW8GZX
					More data for this Ligand-Target Pair
Lysine-specific demethylase 6B (Homo sapiens (Human))	BDBM293683 (3-{[(2-phenyl-5,6,7,8-tetrahydroquinolin-5- | US10...) Show SMILES OC(=O)c1ccncc1NCC1CCCc2nc(ccc12)-c1ccccc1 Show InChI InChI=1S/C22H21N3O2/c26-22(27)18-11-12-23-14-21(18)24-13-16-7-4-8-20-17(16)9-10-19(25-20)15-5-2-1-3-6-15/h1-3,5-6,9-12,14,16,24H,4,7-8,13H2,(H,26,27)	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	550	n/a	n/a	n/a	n/a	n/a	25
Celgene Quanticel Research, Inc. US Patent					Assay Description The enzymatic assay of JMJD3 activity is based upon Time Resolved-Fluorescence Resonance Energy Transfer (TR-FRET) detection. The ability of test com...				US Patent US10106534 (2018) BindingDB Entry DOI: 10.7270/Q2JW8GZX
					More data for this Ligand-Target Pair
Lysine-specific demethylase 4C (Homo sapiens (Human))	BDBM293684 (3-[({2-[methyl(phenyl)amino]-5,6,7,8-tetrahydroqui...) Show SMILES CN(c1ccccc1)c1ccc2C(CNc3cnccc3C(O)=O)CCCc2n1 Show InChI InChI=1S/C23H24N4O2/c1-27(17-7-3-2-4-8-17)22-11-10-18-16(6-5-9-20(18)26-22)14-25-21-15-24-13-12-19(21)23(28)29/h2-4,7-8,10-13,15-16,25H,5-6,9,14H2,1H3,(H,28,29)	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	550	n/a	n/a	n/a	n/a	n/a	25
Celgene Quanticel Research, Inc. US Patent					Assay Description The ability of test compounds to inhibit the activity of JMJD2C was determined in 384-well plate format under the following reaction conditions: 0.3 ...				US Patent US10106534 (2018) BindingDB Entry DOI: 10.7270/Q2JW8GZX
					More data for this Ligand-Target Pair
Lysine-specific demethylase 6B (Homo sapiens (Human))	BDBM293687 (3-({[(4S)-7-(3-methylphenyl)-3,4-dihydro-2H-1-benz...) Show SMILES Cc1cccc(c1)-c1ccc2[C@@H](CNc3cnccc3C(O)=O)CCOc2c1 |r| Show InChI InChI=1S/C23H22N2O3/c1-15-3-2-4-16(11-15)17-5-6-19-18(8-10-28-22(19)12-17)13-25-21-14-24-9-7-20(21)23(26)27/h2-7,9,11-12,14,18,25H,8,10,13H2,1H3,(H,26,27)/t18-/m1/s1	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	550	n/a	n/a	n/a	n/a	n/a	25
Celgene Quanticel Research, Inc. US Patent					Assay Description The enzymatic assay of JMJD3 activity is based upon Time Resolved-Fluorescence Resonance Energy Transfer (TR-FRET) detection. The ability of test com...				US Patent US10106534 (2018) BindingDB Entry DOI: 10.7270/Q2JW8GZX
					More data for this Ligand-Target Pair
Lysine-specific demethylase 4C (Homo sapiens (Human))	BDBM293688 (3-({[(4R)-7-(3-methylphenyl)-3,4-dihydro-2H-1-benz...) Show SMILES Cc1cccc(c1)-c1ccc2[C@H](CNc3cnccc3C(O)=O)CCOc2c1 |r| Show InChI InChI=1S/C23H22N2O3/c1-15-3-2-4-16(11-15)17-5-6-19-18(8-10-28-22(19)12-17)13-25-21-14-24-9-7-20(21)23(26)27/h2-7,9,11-12,14,18,25H,8,10,13H2,1H3,(H,26,27)/t18-/m0/s1	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	550	n/a	n/a	n/a	n/a	n/a	25
Celgene Quanticel Research, Inc. US Patent					Assay Description The ability of test compounds to inhibit the activity of JMJD2C was determined in 384-well plate format under the following reaction conditions: 0.3 ...				US Patent US10106534 (2018) BindingDB Entry DOI: 10.7270/Q2JW8GZX
					More data for this Ligand-Target Pair
Lysine-specific demethylase 6B (Homo sapiens (Human))	BDBM293689 (3-({[(4S)-7-(4-methylphenyl)-3,4-dihydro-2H-1-benz...) Show SMILES Cc1ccc(cc1)-c1ccc2[C@@H](CNc3cnccc3C(O)=O)CCOc2c1 |r| Show InChI InChI=1S/C23H22N2O3/c1-15-2-4-16(5-3-15)17-6-7-19-18(9-11-28-22(19)12-17)13-25-21-14-24-10-8-20(21)23(26)27/h2-8,10,12,14,18,25H,9,11,13H2,1H3,(H,26,27)/t18-/m1/s1	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	550	n/a	n/a	n/a	n/a	n/a	25
Celgene Quanticel Research, Inc. US Patent					Assay Description The enzymatic assay of JMJD3 activity is based upon Time Resolved-Fluorescence Resonance Energy Transfer (TR-FRET) detection. The ability of test com...				US Patent US10106534 (2018) BindingDB Entry DOI: 10.7270/Q2JW8GZX
					More data for this Ligand-Target Pair
Lysine-specific demethylase 4C (Homo sapiens (Human))	BDBM293690 (3-({[(4R)-7-(4-methylphenyl)-3,4-dihydro-2H-1-benz...) Show SMILES Cc1ccc(cc1)-c1ccc2[C@H](CNc3cnccc3C(O)=O)CCOc2c1 |r| Show InChI InChI=1S/C23H22N2O3/c1-15-2-4-16(5-3-15)17-6-7-19-18(9-11-28-22(19)12-17)13-25-21-14-24-10-8-20(21)23(26)27/h2-8,10,12,14,18,25H,9,11,13H2,1H3,(H,26,27)/t18-/m0/s1	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	550	n/a	n/a	n/a	n/a	n/a	25
Celgene Quanticel Research, Inc. US Patent					Assay Description The ability of test compounds to inhibit the activity of JMJD2C was determined in 384-well plate format under the following reaction conditions: 0.3 ...				US Patent US10106534 (2018) BindingDB Entry DOI: 10.7270/Q2JW8GZX
					More data for this Ligand-Target Pair
Lysine-specific demethylase 4C (Homo sapiens (Human))	BDBM293692 (3-({[(4R)-7-(thiophen-3-yl)-3,4-dihydro-2H-1-benzo...) Show SMILES OC(=O)c1ccncc1NC[C@@H]1CCOc2cc(ccc12)-c1ccsc1 |r| Show InChI InChI=1S/C20H18N2O3S/c23-20(24)17-3-6-21-11-18(17)22-10-14-4-7-25-19-9-13(1-2-16(14)19)15-5-8-26-12-15/h1-3,5-6,8-9,11-12,14,22H,4,7,10H2,(H,23,24)/t14-/m0/s1	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	550	n/a	n/a	n/a	n/a	n/a	25
Celgene Quanticel Research, Inc. US Patent					Assay Description The ability of test compounds to inhibit the activity of JMJD2C was determined in 384-well plate format under the following reaction conditions: 0.3 ...				US Patent US10106534 (2018) BindingDB Entry DOI: 10.7270/Q2JW8GZX
					More data for this Ligand-Target Pair
Lysine-specific demethylase 4C (Homo sapiens (Human))	BDBM293693 (3-({[(4R)-7-cyclohexyl-3,4-dihydro-2H-1-benzopyran...) Show SMILES OC(=O)c1ccncc1NCC1CCOc2cc(ccc12)C1CCCCC1 Show InChI InChI=1S/C22H26N2O3/c25-22(26)19-8-10-23-14-20(19)24-13-17-9-11-27-21-12-16(6-7-18(17)21)15-4-2-1-3-5-15/h6-8,10,12,14-15,17,24H,1-5,9,11,13H2,(H,25,26)	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	550	n/a	n/a	n/a	n/a	n/a	25
Celgene Quanticel Research, Inc. US Patent					Assay Description The ability of test compounds to inhibit the activity of JMJD2C was determined in 384-well plate format under the following reaction conditions: 0.3 ...				US Patent US10106534 (2018) BindingDB Entry DOI: 10.7270/Q2JW8GZX
					More data for this Ligand-Target Pair
Lysine-specific demethylase 6B (Homo sapiens (Human))	BDBM293694 (3-({[(4S)-7-(2-methylthiophen-3-yl)-3,4-dihydro-2H...) Show SMILES Cc1sccc1-c1ccc2[C@@H](CNc3cnccc3C(O)=O)CCOc2c1 |r| Show InChI InChI=1S/C21H20N2O3S/c1-13-16(6-9-27-13)14-2-3-17-15(5-8-26-20(17)10-14)11-23-19-12-22-7-4-18(19)21(24)25/h2-4,6-7,9-10,12,15,23H,5,8,11H2,1H3,(H,24,25)/t15-/m1/s1	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	550	n/a	n/a	n/a	n/a	n/a	25
Celgene Quanticel Research, Inc. US Patent					Assay Description The enzymatic assay of JMJD3 activity is based upon Time Resolved-Fluorescence Resonance Energy Transfer (TR-FRET) detection. The ability of test com...				US Patent US10106534 (2018) BindingDB Entry DOI: 10.7270/Q2JW8GZX
					More data for this Ligand-Target Pair
Lysine-specific demethylase 4C (Homo sapiens (Human))	BDBM293696 (3-({[7-(3-methylbut-1-yn-1-yl)-3,4-dihydro-2H-1-be...) Show SMILES CC(C)C#Cc1ccc2C(CNc3cnccc3C(O)=O)CCOc2c1 Show InChI InChI=1S/C21H22N2O3/c1-14(2)3-4-15-5-6-17-16(8-10-26-20(17)11-15)12-23-19-13-22-9-7-18(19)21(24)25/h5-7,9,11,13-14,16,23H,8,10,12H2,1-2H3,(H,24,25)	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	550	n/a	n/a	n/a	n/a	n/a	25
Celgene Quanticel Research, Inc. US Patent					Assay Description The ability of test compounds to inhibit the activity of JMJD2C was determined in 384-well plate format under the following reaction conditions: 0.3 ...				US Patent US10106534 (2018) BindingDB Entry DOI: 10.7270/Q2JW8GZX
					More data for this Ligand-Target Pair
Lysine-specific demethylase 6B (Homo sapiens (Human))	BDBM293697 (3-({[(4S)-7-(2-chlorophenyl)-3,4-dihydro-2H-1-benz...) Show SMILES OC(=O)c1ccncc1NC[C@H]1CCOc2cc(ccc12)-c1ccccc1Cl |r| Show InChI InChI=1S/C22H19ClN2O3/c23-19-4-2-1-3-16(19)14-5-6-17-15(8-10-28-21(17)11-14)12-25-20-13-24-9-7-18(20)22(26)27/h1-7,9,11,13,15,25H,8,10,12H2,(H,26,27)/t15-/m1/s1	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	550	n/a	n/a	n/a	n/a	n/a	25
Celgene Quanticel Research, Inc. US Patent					Assay Description The enzymatic assay of JMJD3 activity is based upon Time Resolved-Fluorescence Resonance Energy Transfer (TR-FRET) detection. The ability of test com...				US Patent US10106534 (2018) BindingDB Entry DOI: 10.7270/Q2JW8GZX
					More data for this Ligand-Target Pair
Lysine-specific demethylase 4C (Homo sapiens (Human))	BDBM293698 (3-({[(4R)-7-(2-chlorophenyl)-3,4-dihydro-2H-1-benz...) Show SMILES OC(=O)c1ccncc1NC[C@@H]1CCOc2cc(ccc12)-c1ccccc1Cl |r| Show InChI InChI=1S/C22H19ClN2O3/c23-19-4-2-1-3-16(19)14-5-6-17-15(8-10-28-21(17)11-14)12-25-20-13-24-9-7-18(20)22(26)27/h1-7,9,11,13,15,25H,8,10,12H2,(H,26,27)/t15-/m0/s1	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	550	n/a	n/a	n/a	n/a	n/a	25
Celgene Quanticel Research, Inc. US Patent					Assay Description The ability of test compounds to inhibit the activity of JMJD2C was determined in 384-well plate format under the following reaction conditions: 0.3 ...				US Patent US10106534 (2018) BindingDB Entry DOI: 10.7270/Q2JW8GZX
					More data for this Ligand-Target Pair
Lysine-specific demethylase 4C (Homo sapiens (Human))	BDBM293700 (3-({[(4R)-7-(3-fluoro-2-methylphenyl)-3,4-dihydro-...) Show SMILES Cc1c(F)cccc1-c1ccc2[C@H](CNc3cnccc3C(O)=O)CCOc2c1 |r| Show InChI InChI=1S/C23H21FN2O3/c1-14-17(3-2-4-20(14)24)15-5-6-18-16(8-10-29-22(18)11-15)12-26-21-13-25-9-7-19(21)23(27)28/h2-7,9,11,13,16,26H,8,10,12H2,1H3,(H,27,28)/t16-/m0/s1	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	550	n/a	n/a	n/a	n/a	n/a	25
Celgene Quanticel Research, Inc. US Patent					Assay Description The ability of test compounds to inhibit the activity of JMJD2C was determined in 384-well plate format under the following reaction conditions: 0.3 ...				US Patent US10106534 (2018) BindingDB Entry DOI: 10.7270/Q2JW8GZX
					More data for this Ligand-Target Pair
Lysine-specific demethylase 4C (Homo sapiens (Human))	BDBM293702 (3-({[(4R)-7-(2-chloro-3-fluorophenyl)-3,4-dihydro-...) Show SMILES OC(=O)c1ccncc1NC[C@@H]1CCOc2cc(ccc12)-c1cccc(F)c1Cl |r| Show InChI InChI=1S/C22H18ClFN2O3/c23-21-16(2-1-3-18(21)24)13-4-5-15-14(7-9-29-20(15)10-13)11-26-19-12-25-8-6-17(19)22(27)28/h1-6,8,10,12,14,26H,7,9,11H2,(H,27,28)/t14-/m0/s1	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	550	n/a	n/a	n/a	n/a	n/a	25
Celgene Quanticel Research, Inc. US Patent					Assay Description The ability of test compounds to inhibit the activity of JMJD2C was determined in 384-well plate format under the following reaction conditions: 0.3 ...				US Patent US10106534 (2018) BindingDB Entry DOI: 10.7270/Q2JW8GZX
					More data for this Ligand-Target Pair
Lysine-specific demethylase 4C (Homo sapiens (Human))	BDBM293703 (3-({[(4R)-7-(2-chloro-5-fluorophenyl)-3,4-dihydro-...) Show SMILES OC(=O)c1ccncc1NC[C@@H]1CCOc2cc(ccc12)-c1cc(F)ccc1Cl |r| Show InChI InChI=1S/C22H18ClFN2O3/c23-19-4-2-15(24)10-18(19)13-1-3-16-14(6-8-29-21(16)9-13)11-26-20-12-25-7-5-17(20)22(27)28/h1-5,7,9-10,12,14,26H,6,8,11H2,(H,27,28)/t14-/m0/s1	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	550	n/a	n/a	n/a	n/a	n/a	25
Celgene Quanticel Research, Inc. US Patent					Assay Description The ability of test compounds to inhibit the activity of JMJD2C was determined in 384-well plate format under the following reaction conditions: 0.3 ...				US Patent US10106534 (2018) BindingDB Entry DOI: 10.7270/Q2JW8GZX
					More data for this Ligand-Target Pair
Lysine-specific demethylase 4C (Homo sapiens (Human))	BDBM293704 (3-({[(4R)-7-[2-(trifluoromethyl)phenyl]-3,4-dihydr...) Show SMILES OC(=O)c1ccncc1NC[C@@H]1CCOc2cc(ccc12)-c1ccccc1[B](F)(F)F |r| Show InChI InChI=1S/C23H19F3N2O3/c24-23(25,26)19-4-2-1-3-16(19)14-5-6-17-15(8-10-31-21(17)11-14)12-28-20-13-27-9-7-18(20)22(29)30/h1-7,9,11,13,15,28H,8,10,12H2,(H,29,30)/t15-/m0/s1	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	550	n/a	n/a	n/a	n/a	n/a	25
Celgene Quanticel Research, Inc. US Patent					Assay Description The ability of test compounds to inhibit the activity of JMJD2C was determined in 384-well plate format under the following reaction conditions: 0.3 ...				US Patent US10106534 (2018) BindingDB Entry DOI: 10.7270/Q2JW8GZX
					More data for this Ligand-Target Pair
Lysine-specific demethylase 4C (Homo sapiens (Human))	BDBM293706 (3-({[(4R)-7-phenoxy-3,4-dihydro-2H-1-benzopyran-4-...) Show SMILES OC(=O)c1ccncc1NC[C@@H]1CCOc2cc(Oc3ccccc3)ccc12 |r| Show InChI InChI=1S/C22H20N2O4/c25-22(26)19-8-10-23-14-20(19)24-13-15-9-11-27-21-12-17(6-7-18(15)21)28-16-4-2-1-3-5-16/h1-8,10,12,14-15,24H,9,11,13H2,(H,25,26)/t15-/m0/s1	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	550	n/a	n/a	n/a	n/a	n/a	25
Celgene Quanticel Research, Inc. US Patent					Assay Description The ability of test compounds to inhibit the activity of JMJD2C was determined in 384-well plate format under the following reaction conditions: 0.3 ...				US Patent US10106534 (2018) BindingDB Entry DOI: 10.7270/Q2JW8GZX
					More data for this Ligand-Target Pair
Lysine-specific demethylase 4C (Homo sapiens (Human))	BDBM293707 (3-({[7-(thiophen-2-ylsulfanyl)-3,4-dihydro-2H-1-be...) Show SMILES OC(=O)c1ccncc1NCC1CCOc2cc(Sc3cccs3)ccc12 Show InChI InChI=1S/C20H18N2O3S2/c23-20(24)16-5-7-21-12-17(16)22-11-13-6-8-25-18-10-14(3-4-15(13)18)27-19-2-1-9-26-19/h1-5,7,9-10,12-13,22H,6,8,11H2,(H,23,24)	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	550	n/a	n/a	n/a	n/a	n/a	25
Celgene Quanticel Research, Inc. US Patent					Assay Description The ability of test compounds to inhibit the activity of JMJD2C was determined in 384-well plate format under the following reaction conditions: 0.3 ...				US Patent US10106534 (2018) BindingDB Entry DOI: 10.7270/Q2JW8GZX
					More data for this Ligand-Target Pair
Lysine-specific demethylase 6B (Homo sapiens (Human))	BDBM293710 (3-({[(4S)-7-[(3-fluorophenyl)sulfanyl]-3,4-dihydro...) Show SMILES OC(=O)c1ccncc1NC[C@H]1CCOc2cc(Sc3cccc(F)c3)ccc12 |r| Show InChI InChI=1S/C22H19FN2O3S/c23-15-2-1-3-16(10-15)29-17-4-5-18-14(7-9-28-21(18)11-17)12-25-20-13-24-8-6-19(20)22(26)27/h1-6,8,10-11,13-14,25H,7,9,12H2,(H,26,27)/t14-/m1/s1	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	550	n/a	n/a	n/a	n/a	n/a	25
Celgene Quanticel Research, Inc. US Patent					Assay Description The enzymatic assay of JMJD3 activity is based upon Time Resolved-Fluorescence Resonance Energy Transfer (TR-FRET) detection. The ability of test com...				US Patent US10106534 (2018) BindingDB Entry DOI: 10.7270/Q2JW8GZX
					More data for this Ligand-Target Pair
Lysine-specific demethylase 4C (Homo sapiens (Human))	BDBM293711 (3-({[(4R)-7-[(3-fluorophenyl)sulfanyl]-3,4-dihydro...) Show SMILES OC(=O)c1ccncc1NC[C@@H]1CCOc2cc(Sc3cccc(F)c3)ccc12 |r| Show InChI InChI=1S/C22H19FN2O3S/c23-15-2-1-3-16(10-15)29-17-4-5-18-14(7-9-28-21(18)11-17)12-25-20-13-24-8-6-19(20)22(26)27/h1-6,8,10-11,13-14,25H,7,9,12H2,(H,26,27)/t14-/m0/s1	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	550	n/a	n/a	n/a	n/a	n/a	25
Celgene Quanticel Research, Inc. US Patent					Assay Description The ability of test compounds to inhibit the activity of JMJD2C was determined in 384-well plate format under the following reaction conditions: 0.3 ...				US Patent US10106534 (2018) BindingDB Entry DOI: 10.7270/Q2JW8GZX
					More data for this Ligand-Target Pair
Lysine-specific demethylase 6B (Homo sapiens (Human))	BDBM293712 (3-({[(4S)-7-[(4-fluorophenyl)sulfanyl]-3,4-dihydro...) Show SMILES OC(=O)c1ccncc1NC[C@H]1CCOc2cc(Sc3ccc(F)cc3)ccc12 |r| Show InChI InChI=1S/C22H19FN2O3S/c23-15-1-3-16(4-2-15)29-17-5-6-18-14(8-10-28-21(18)11-17)12-25-20-13-24-9-7-19(20)22(26)27/h1-7,9,11,13-14,25H,8,10,12H2,(H,26,27)/t14-/m1/s1	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	550	n/a	n/a	n/a	n/a	n/a	25
Celgene Quanticel Research, Inc. US Patent					Assay Description The enzymatic assay of JMJD3 activity is based upon Time Resolved-Fluorescence Resonance Energy Transfer (TR-FRET) detection. The ability of test com...				US Patent US10106534 (2018) BindingDB Entry DOI: 10.7270/Q2JW8GZX
					More data for this Ligand-Target Pair
Lysine-specific demethylase 4C (Homo sapiens (Human))	BDBM293713 (3-({[(4R)-7-[(4-fluorophenyl)sulfanyl]-3,4-dihydro...) Show SMILES OC(=O)c1ccncc1NC[C@@H]1CCOc2cc(Sc3ccc(F)cc3)ccc12 |r| Show InChI InChI=1S/C22H19FN2O3S/c23-15-1-3-16(4-2-15)29-17-5-6-18-14(8-10-28-21(18)11-17)12-25-20-13-24-9-7-19(20)22(26)27/h1-7,9,11,13-14,25H,8,10,12H2,(H,26,27)/t14-/m0/s1	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	550	n/a	n/a	n/a	n/a	n/a	25
Celgene Quanticel Research, Inc. US Patent					Assay Description The ability of test compounds to inhibit the activity of JMJD2C was determined in 384-well plate format under the following reaction conditions: 0.3 ...				US Patent US10106534 (2018) BindingDB Entry DOI: 10.7270/Q2JW8GZX
					More data for this Ligand-Target Pair

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