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Compile Data Set for Download or QSAR

Found 331 hits Enz. Inhib. hit(s) with all data for assayid = 1 entry = 2449   
Target/Host
(Institution)
LigandTarget/Host
Links
Ligand
Links
Trg + Lig
Links
Ki
nM
ΔG°
kJ/mole
IC50
nM
Kd
nM
EC50/IC50
nM
koff
s-1
kon
M-1s-1
pHTemp
°C
3-phosphoinositide-dependent protein kinase 1 (PDK1)


(Homo sapiens (Human))
BDBM366233
PNG
(US9873693, Compound 156)
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PC sid
UniChem
Article
n/an/a<500n/an/an/an/an/an/a



Duquesne University





J Med Chem 51: 68-76 (2008)


Article DOI: 10.1021/jm701052u
More data for this
Ligand-Target Pair
3-phosphoinositide-dependent protein kinase 1 (PDK1)


(Homo sapiens (Human))
BDBM366234
PNG
(US9873693, Compound 157)
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
n/an/a<500n/an/an/an/an/an/a



Duquesne University





J Med Chem 51: 68-76 (2008)


Article DOI: 10.1021/jm701052u
More data for this
Ligand-Target Pair
3-phosphoinositide-dependent protein kinase 1 (PDK1)


(Homo sapiens (Human))
BDBM366236
PNG
(US9873693, Compound 159)
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
n/an/a<500n/an/an/an/an/an/a



Duquesne University





J Med Chem 51: 68-76 (2008)


Article DOI: 10.1021/jm701052u
More data for this
Ligand-Target Pair
3-phosphoinositide-dependent protein kinase 1 (PDK1)


(Homo sapiens (Human))
BDBM366237
PNG
(US9873693, Compound 160)
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
n/an/a<500n/an/an/an/an/an/a



Duquesne University





J Med Chem 51: 68-76 (2008)


Article DOI: 10.1021/jm701052u
More data for this
Ligand-Target Pair
3-phosphoinositide-dependent protein kinase 1 (PDK1)


(Homo sapiens (Human))
BDBM366238
PNG
(US9873693, Compound 161)
GoogleScholar
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PC sid
UniChem
Article
n/an/a<500n/an/an/an/an/an/a



Duquesne University





J Med Chem 51: 68-76 (2008)


Article DOI: 10.1021/jm701052u
More data for this
Ligand-Target Pair
3-phosphoinositide-dependent protein kinase 1 (PDK1)


(Homo sapiens (Human))
BDBM366328
PNG
(US9873693, Compound 255)
GoogleScholar
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PC sid
UniChem
Article
n/an/a<500n/an/an/an/an/an/a



Duquesne University





J Med Chem 51: 68-76 (2008)


Article DOI: 10.1021/jm701052u
More data for this
Ligand-Target Pair
3-phosphoinositide-dependent protein kinase 1 (PDK1)


(Homo sapiens (Human))
BDBM366330
PNG
(US9873693, Compound 257)
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
n/an/a<500n/an/an/an/an/an/a



Duquesne University





J Med Chem 51: 68-76 (2008)


Article DOI: 10.1021/jm701052u
More data for this
Ligand-Target Pair
3-phosphoinositide-dependent protein kinase 1 (PDK1)


(Homo sapiens (Human))
BDBM366331
PNG
(US9873693, Compound 258)
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
n/an/a<500n/an/an/an/an/an/a



Duquesne University





J Med Chem 51: 68-76 (2008)


Article DOI: 10.1021/jm701052u
More data for this
Ligand-Target Pair
3-phosphoinositide-dependent protein kinase 1 (PDK1)


(Homo sapiens (Human))
BDBM366332
PNG
(US9873693, Compound 259)
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
n/an/a<500n/an/an/an/an/an/a



Duquesne University





J Med Chem 51: 68-76 (2008)


Article DOI: 10.1021/jm701052u
More data for this
Ligand-Target Pair
3-phosphoinositide-dependent protein kinase 1 (PDK1)


(Homo sapiens (Human))
BDBM366183
PNG
(US9873693, Compound 106 | US9873693, Compound 260)
GoogleScholar
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PC sid
UniChem
Article
n/an/a<500n/an/an/an/an/an/a



Duquesne University





J Med Chem 51: 68-76 (2008)


Article DOI: 10.1021/jm701052u
More data for this
Ligand-Target Pair
3-phosphoinositide-dependent protein kinase 1 (PDK1)


(Homo sapiens (Human))
BDBM366335
PNG
(US9873693, Compound 262)
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
n/an/a<500n/an/an/an/an/an/a



Duquesne University





J Med Chem 51: 68-76 (2008)


Article DOI: 10.1021/jm701052u
More data for this
Ligand-Target Pair
3-phosphoinositide-dependent protein kinase 1 (PDK1)


(Homo sapiens (Human))
BDBM366336
PNG
(US9873693, Compound 263)
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
n/an/a<500n/an/an/an/an/an/a



Duquesne University





J Med Chem 51: 68-76 (2008)


Article DOI: 10.1021/jm701052u
More data for this
Ligand-Target Pair
3-phosphoinositide-dependent protein kinase 1 (PDK1)


(Homo sapiens (Human))
BDBM366186
PNG
(US9873693, Compound 109 | US9873693, Compound 264)
GoogleScholar
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PC sid
UniChem
Article
n/an/a<500n/an/an/an/an/an/a



Duquesne University





J Med Chem 51: 68-76 (2008)


Article DOI: 10.1021/jm701052u
More data for this
Ligand-Target Pair
3-phosphoinositide-dependent protein kinase 1 (PDK1)


(Homo sapiens (Human))
BDBM366098
PNG
(US9873693, Compound 21)
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
n/an/a<500n/an/an/an/an/an/a



Duquesne University





J Med Chem 51: 68-76 (2008)


Article DOI: 10.1021/jm701052u
More data for this
Ligand-Target Pair
3-phosphoinositide-dependent protein kinase 1 (PDK1)


(Homo sapiens (Human))
BDBM366099
PNG
(US9873693, Compound 22)
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
n/an/a<500n/an/an/an/an/an/a



Duquesne University





J Med Chem 51: 68-76 (2008)


Article DOI: 10.1021/jm701052u
More data for this
Ligand-Target Pair
3-phosphoinositide-dependent protein kinase 1 (PDK1)


(Homo sapiens (Human))
BDBM366100
PNG
(US9873693, Compound 23)
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
n/an/a<500n/an/an/an/an/an/a



Duquesne University





J Med Chem 51: 68-76 (2008)


Article DOI: 10.1021/jm701052u
More data for this
Ligand-Target Pair
3-phosphoinositide-dependent protein kinase 1 (PDK1)


(Homo sapiens (Human))
BDBM366101
PNG
(US9873693, Compound 24)
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
n/an/a<500n/an/an/an/an/an/a



Duquesne University





J Med Chem 51: 68-76 (2008)


Article DOI: 10.1021/jm701052u
More data for this
Ligand-Target Pair
3-phosphoinositide-dependent protein kinase 1 (PDK1)


(Homo sapiens (Human))
BDBM366102
PNG
(US9873693, Compound 25)
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
n/an/a<500n/an/an/an/an/an/a



Duquesne University





J Med Chem 51: 68-76 (2008)


Article DOI: 10.1021/jm701052u
More data for this
Ligand-Target Pair
3-phosphoinositide-dependent protein kinase 1 (PDK1)


(Homo sapiens (Human))
BDBM366103
PNG
(US9873693, Compound 26)
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
n/an/a<500n/an/an/an/an/an/a



Duquesne University





J Med Chem 51: 68-76 (2008)


Article DOI: 10.1021/jm701052u
More data for this
Ligand-Target Pair
3-phosphoinositide-dependent protein kinase 1 (PDK1)


(Homo sapiens (Human))
BDBM366216
PNG
(US9873693, Compound 139)
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
n/an/a<500n/an/an/an/an/an/a



Duquesne University





J Med Chem 51: 68-76 (2008)


Article DOI: 10.1021/jm701052u
More data for this
Ligand-Target Pair
3-phosphoinositide-dependent protein kinase 1 (PDK1)


(Homo sapiens (Human))
BDBM366217
PNG
(US9873693, Compound 140)
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
n/an/a<500n/an/an/an/an/an/a



Duquesne University





J Med Chem 51: 68-76 (2008)


Article DOI: 10.1021/jm701052u
More data for this
Ligand-Target Pair
3-phosphoinositide-dependent protein kinase 1 (PDK1)


(Homo sapiens (Human))
BDBM366218
PNG
(US9873693, Compound 141)
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
n/an/a<500n/an/an/an/an/an/a



Duquesne University





J Med Chem 51: 68-76 (2008)


Article DOI: 10.1021/jm701052u
More data for this
Ligand-Target Pair
3-phosphoinositide-dependent protein kinase 1 (PDK1)


(Homo sapiens (Human))
BDBM366219
PNG
(US9873693, Compound 142)
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
n/an/a<500n/an/an/an/an/an/a



Duquesne University





J Med Chem 51: 68-76 (2008)


Article DOI: 10.1021/jm701052u
More data for this
Ligand-Target Pair
3-phosphoinositide-dependent protein kinase 1 (PDK1)


(Homo sapiens (Human))
BDBM366220
PNG
(US9873693, Compound 143)
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
n/an/a<500n/an/an/an/an/an/a



Duquesne University





J Med Chem 51: 68-76 (2008)


Article DOI: 10.1021/jm701052u
More data for this
Ligand-Target Pair
3-phosphoinositide-dependent protein kinase 1 (PDK1)


(Homo sapiens (Human))
BDBM50361645
PNG
(CHEMBL1234429 | US9873693, Compound 144)
Show SMILES Fc1ccc(Cn2cccc(C(=O)N[C@@H](COc3ccc4[nH]c(=O)[nH]c4c3)c3ccccc3)c2=O)cc1F |r|
Show InChI InChI=1S/C28H22F2N4O4/c29-21-10-8-17(13-22(21)30)15-34-12-4-7-20(27(34)36)26(35)31-25(18-5-2-1-3-6-18)16-38-19-9-11-23-24(14-19)33-28(37)32-23/h1-14,25H,15-16H2,(H,31,35)(H2,32,33,37)/t25-/m0/s1
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Article
n/an/a<500n/an/an/an/an/an/a



Duquesne University





J Med Chem 51: 68-76 (2008)


Article DOI: 10.1021/jm701052u
More data for this
Ligand-Target Pair
3-phosphoinositide-dependent protein kinase 1 (PDK1)


(Homo sapiens (Human))
BDBM366222
PNG
(US9873693, Compound 145)
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
n/an/a<500n/an/an/an/an/an/a



Duquesne University





J Med Chem 51: 68-76 (2008)


Article DOI: 10.1021/jm701052u
More data for this
Ligand-Target Pair
3-phosphoinositide-dependent protein kinase 1 (PDK1)


(Homo sapiens (Human))
BDBM366223
PNG
(US9873693, Compound 146)
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
n/an/a<500n/an/an/an/an/an/a



Duquesne University





J Med Chem 51: 68-76 (2008)


Article DOI: 10.1021/jm701052u
More data for this
Ligand-Target Pair
3-phosphoinositide-dependent protein kinase 1 (PDK1)


(Homo sapiens (Human))
BDBM366092
PNG
(US9873693, Compound 15 | US9873693, Compound 234)
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
n/an/a<500n/an/an/an/an/an/a



Duquesne University





J Med Chem 51: 68-76 (2008)


Article DOI: 10.1021/jm701052u
More data for this
Ligand-Target Pair
3-phosphoinositide-dependent protein kinase 1 (PDK1)


(Homo sapiens (Human))
BDBM366312
PNG
(US9873693, Compound 237)
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
n/an/a<500n/an/an/an/an/an/a



Duquesne University





J Med Chem 51: 68-76 (2008)


Article DOI: 10.1021/jm701052u
More data for this
Ligand-Target Pair
3-phosphoinositide-dependent protein kinase 1 (PDK1)


(Homo sapiens (Human))
BDBM366313
PNG
(US9873693, Compound 238)
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
n/an/a<500n/an/an/an/an/an/a



Duquesne University





J Med Chem 51: 68-76 (2008)


Article DOI: 10.1021/jm701052u
More data for this
Ligand-Target Pair
3-phosphoinositide-dependent protein kinase 1 (PDK1)


(Homo sapiens (Human))
BDBM366314
PNG
(US9873693, Compound 239)
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
n/an/a<500n/an/an/an/an/an/a



Duquesne University





J Med Chem 51: 68-76 (2008)


Article DOI: 10.1021/jm701052u
More data for this
Ligand-Target Pair
3-phosphoinositide-dependent protein kinase 1 (PDK1)


(Homo sapiens (Human))
BDBM366104
PNG
(US9873693, Compound 27)
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
n/an/a<500n/an/an/an/an/an/a



Duquesne University





J Med Chem 51: 68-76 (2008)


Article DOI: 10.1021/jm701052u
More data for this
Ligand-Target Pair
3-phosphoinositide-dependent protein kinase 1 (PDK1)


(Homo sapiens (Human))
BDBM366105
PNG
(US9873693, Compound 28)
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
n/an/a<500n/an/an/an/an/an/a



Duquesne University





J Med Chem 51: 68-76 (2008)


Article DOI: 10.1021/jm701052u
More data for this
Ligand-Target Pair
3-phosphoinositide-dependent protein kinase 1 (PDK1)


(Homo sapiens (Human))
BDBM366106
PNG
(US9873693, Compound 29)
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
n/an/a<500n/an/an/an/an/an/a



Duquesne University





J Med Chem 51: 68-76 (2008)


Article DOI: 10.1021/jm701052u
More data for this
Ligand-Target Pair
3-phosphoinositide-dependent protein kinase 1 (PDK1)


(Homo sapiens (Human))
BDBM366107
PNG
(US9873693, Compound 30)
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
n/an/a<500n/an/an/an/an/an/a



Duquesne University





J Med Chem 51: 68-76 (2008)


Article DOI: 10.1021/jm701052u
More data for this
Ligand-Target Pair
3-phosphoinositide-dependent protein kinase 1 (PDK1)


(Homo sapiens (Human))
BDBM366108
PNG
(US9873693, Compound 31)
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
n/an/a<500n/an/an/an/an/an/a



Duquesne University





J Med Chem 51: 68-76 (2008)


Article DOI: 10.1021/jm701052u
More data for this
Ligand-Target Pair
3-phosphoinositide-dependent protein kinase 1 (PDK1)


(Homo sapiens (Human))
BDBM366109
PNG
(US9873693, Compound 32)
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
n/an/a<500n/an/an/an/an/an/a



Duquesne University





J Med Chem 51: 68-76 (2008)


Article DOI: 10.1021/jm701052u
More data for this
Ligand-Target Pair
3-phosphoinositide-dependent protein kinase 1 (PDK1)


(Homo sapiens (Human))
BDBM366110
PNG
(US9873693, Compound 33)
GoogleScholar
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PC cid
PC sid
UniChem
Article
n/an/a<500n/an/an/an/an/an/a



Duquesne University





J Med Chem 51: 68-76 (2008)


Article DOI: 10.1021/jm701052u
More data for this
Ligand-Target Pair
3-phosphoinositide-dependent protein kinase 1 (PDK1)


(Homo sapiens (Human))
BDBM366111
PNG
(US9873693, Compound 34)
GoogleScholar
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PC sid
UniChem
Article
n/an/a<500n/an/an/an/an/an/a



Duquesne University





J Med Chem 51: 68-76 (2008)


Article DOI: 10.1021/jm701052u
More data for this
Ligand-Target Pair
3-phosphoinositide-dependent protein kinase 1 (PDK1)


(Homo sapiens (Human))
BDBM366140
PNG
(US9873693, Compound 63)
GoogleScholar
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PC sid
UniChem
Article
n/an/a<500n/an/an/an/an/an/a



Duquesne University





J Med Chem 51: 68-76 (2008)


Article DOI: 10.1021/jm701052u
More data for this
Ligand-Target Pair
3-phosphoinositide-dependent protein kinase 1 (PDK1)


(Homo sapiens (Human))
BDBM366141
PNG
(US9873693, Compound 64)
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
n/an/a<500n/an/an/an/an/an/a



Duquesne University





J Med Chem 51: 68-76 (2008)


Article DOI: 10.1021/jm701052u
More data for this
Ligand-Target Pair
3-phosphoinositide-dependent protein kinase 1 (PDK1)


(Homo sapiens (Human))
BDBM366142
PNG
(US9873693, Compound 65)
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
n/an/a<500n/an/an/an/an/an/a



Duquesne University





J Med Chem 51: 68-76 (2008)


Article DOI: 10.1021/jm701052u
More data for this
Ligand-Target Pair
3-phosphoinositide-dependent protein kinase 1 (PDK1)


(Homo sapiens (Human))
BDBM366143
PNG
(US9873693, Compound 66)
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
n/an/a<500n/an/an/an/an/an/a



Duquesne University





J Med Chem 51: 68-76 (2008)


Article DOI: 10.1021/jm701052u
More data for this
Ligand-Target Pair
3-phosphoinositide-dependent protein kinase 1 (PDK1)


(Homo sapiens (Human))
BDBM366144
PNG
(US9873693, Compound 67)
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
n/an/a<500n/an/an/an/an/an/a



Duquesne University





J Med Chem 51: 68-76 (2008)


Article DOI: 10.1021/jm701052u
More data for this
Ligand-Target Pair
3-phosphoinositide-dependent protein kinase 1 (PDK1)


(Homo sapiens (Human))
BDBM366145
PNG
(US9873693, Compound 68)
GoogleScholar
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PC sid
UniChem
Article
n/an/a<500n/an/an/an/an/an/a



Duquesne University





J Med Chem 51: 68-76 (2008)


Article DOI: 10.1021/jm701052u
More data for this
Ligand-Target Pair
3-phosphoinositide-dependent protein kinase 1 (PDK1)


(Homo sapiens (Human))
BDBM366146
PNG
(US9873693, Compound 69)
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
n/an/a<500n/an/an/an/an/an/a



Duquesne University





J Med Chem 51: 68-76 (2008)


Article DOI: 10.1021/jm701052u
More data for this
Ligand-Target Pair
3-phosphoinositide-dependent protein kinase 1 (PDK1)


(Homo sapiens (Human))
BDBM366147
PNG
(US9873693, Compound 70)
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
n/an/a<500n/an/an/an/an/an/a



Duquesne University





J Med Chem 51: 68-76 (2008)


Article DOI: 10.1021/jm701052u
More data for this
Ligand-Target Pair
3-phosphoinositide-dependent protein kinase 1 (PDK1)


(Homo sapiens (Human))
BDBM366148
PNG
(US9873693, Compound 71)
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
n/an/a<500n/an/an/an/an/an/a



Duquesne University





J Med Chem 51: 68-76 (2008)


Article DOI: 10.1021/jm701052u
More data for this
Ligand-Target Pair
3-phosphoinositide-dependent protein kinase 1 (PDK1)


(Homo sapiens (Human))
BDBM366224
PNG
(US9873693, Compound 147)
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
n/an/a<500n/an/an/an/an/an/a



Duquesne University





J Med Chem 51: 68-76 (2008)


Article DOI: 10.1021/jm701052u
More data for this
Ligand-Target Pair
3-phosphoinositide-dependent protein kinase 1 (PDK1)


(Homo sapiens (Human))
BDBM366225
PNG
(US9873693, Compound 148)
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
n/an/a<500n/an/an/an/an/an/a



Duquesne University





J Med Chem 51: 68-76 (2008)


Article DOI: 10.1021/jm701052u
More data for this
Ligand-Target Pair
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